Found 32 hits Enz. Inhib. hit(s) with all data for entry = 50033732 Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
Serine/threonine-protein kinase pim-1
(Homo sapiens (Human)) | BDBM50350423
(CHEMBL466154)Show InChI InChI=1S/C14H10O5/c1-6-2-7(15)4-10-12(6)14(18)13-9(17)3-8(16)5-11(13)19-10/h2-5,15-17H,1H3 | PDB MMDB
KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar AffyNet
| Purchase
CHEMBL MCE KEGG PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | 300 | n/a | n/a | n/a | n/a | n/a | n/a |
Heinrich-Heine-Universit£t
Curated by ChEMBL
| Assay Description Inhibition of recombinant PIM1 assessed as 33Pi incorporation after 60 mins by scintillation counting |
Bioorg Med Chem 19: 4644-51 (2011)
Article DOI: 10.1016/j.bmc.2011.06.013 BindingDB Entry DOI: 10.7270/Q2X92BNH |
More data for this Ligand-Target Pair | |
Serine/threonine-protein kinase pim-1
(Homo sapiens (Human)) | BDBM50350424
(CHEMBL454440)Show InChI InChI=1S/C14H10O6/c1-5-11-10(4-8(17)13(5)18)20-9-3-6(15)2-7(16)12(9)14(11)19/h2-4,15-18H,1H3 | PDB MMDB
KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar AffyNet
| Purchase
CHEMBL PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | 300 | n/a | n/a | n/a | n/a | n/a | n/a |
Heinrich-Heine-Universit£t
Curated by ChEMBL
| Assay Description Inhibition of recombinant PIM1 assessed as 33Pi incorporation after 60 mins by scintillation counting |
Bioorg Med Chem 19: 4644-51 (2011)
Article DOI: 10.1016/j.bmc.2011.06.013 BindingDB Entry DOI: 10.7270/Q2X92BNH |
More data for this Ligand-Target Pair | |
Aurora kinase B
(Homo sapiens (Human)) | BDBM50350424
(CHEMBL454440)Show InChI InChI=1S/C14H10O6/c1-5-11-10(4-8(17)13(5)18)20-9-3-6(15)2-7(16)12(9)14(11)19/h2-4,15-18H,1H3 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| Purchase
CHEMBL PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | 500 | n/a | n/a | n/a | n/a | n/a | n/a |
Heinrich-Heine-Universit£t
Curated by ChEMBL
| Assay Description Inhibition of recombinant Aurora-b assessed as 33Pi incorporation after 60 mins by scintillation counting |
Bioorg Med Chem 19: 4644-51 (2011)
Article DOI: 10.1016/j.bmc.2011.06.013 BindingDB Entry DOI: 10.7270/Q2X92BNH |
More data for this Ligand-Target Pair | |
Vascular endothelial growth factor receptor 2
(Homo sapiens (Human)) | BDBM50350424
(CHEMBL454440)Show InChI InChI=1S/C14H10O6/c1-5-11-10(4-8(17)13(5)18)20-9-3-6(15)2-7(16)12(9)14(11)19/h2-4,15-18H,1H3 | PDB MMDB
NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar AffyNet
| Purchase
CHEMBL PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | 800 | n/a | n/a | n/a | n/a | n/a | n/a |
Heinrich-Heine-Universit£t
Curated by ChEMBL
| Assay Description Inhibition of recombinant VEGF-R2 assessed as 33Pi incorporation after 60 mins by scintillation counting |
Bioorg Med Chem 19: 4644-51 (2011)
Article DOI: 10.1016/j.bmc.2011.06.013 BindingDB Entry DOI: 10.7270/Q2X92BNH |
More data for this Ligand-Target Pair | |
ALK tyrosine kinase receptor
(Homo sapiens (Human)) | BDBM50350424
(CHEMBL454440)Show InChI InChI=1S/C14H10O6/c1-5-11-10(4-8(17)13(5)18)20-9-3-6(15)2-7(16)12(9)14(11)19/h2-4,15-18H,1H3 | PDB
KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar AffyNet
| Purchase
CHEMBL PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | 1.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Heinrich-Heine-Universit£t
Curated by ChEMBL
| Assay Description Inhibition of recombinant ALK assessed as 33Pi incorporation after 60 mins by scintillation counting |
Bioorg Med Chem 19: 4644-51 (2011)
Article DOI: 10.1016/j.bmc.2011.06.013 BindingDB Entry DOI: 10.7270/Q2X92BNH |
More data for this Ligand-Target Pair | |
Aurora kinase B
(Homo sapiens (Human)) | BDBM50350423
(CHEMBL466154)Show InChI InChI=1S/C14H10O5/c1-6-2-7(15)4-10-12(6)14(18)13-9(17)3-8(16)5-11(13)19-10/h2-5,15-17H,1H3 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| Purchase
CHEMBL MCE KEGG PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | 3.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Heinrich-Heine-Universit£t
Curated by ChEMBL
| Assay Description Inhibition of recombinant Aurora-b assessed as 33Pi incorporation after 60 mins by scintillation counting |
Bioorg Med Chem 19: 4644-51 (2011)
Article DOI: 10.1016/j.bmc.2011.06.013 BindingDB Entry DOI: 10.7270/Q2X92BNH |
More data for this Ligand-Target Pair | |
Hepatocyte growth factor receptor
(Homo sapiens (Human)) | BDBM50350424
(CHEMBL454440)Show InChI InChI=1S/C14H10O6/c1-5-11-10(4-8(17)13(5)18)20-9-3-6(15)2-7(16)12(9)14(11)19/h2-4,15-18H,1H3 | PDB MMDB
KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar AffyNet
| Purchase
CHEMBL PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | 4.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Heinrich-Heine-Universit£t
Curated by ChEMBL
| Assay Description Inhibition of wild type MET assessed as 33Pi incorporation after 60 mins by scintillation counting |
Bioorg Med Chem 19: 4644-51 (2011)
Article DOI: 10.1016/j.bmc.2011.06.013 BindingDB Entry DOI: 10.7270/Q2X92BNH |
More data for this Ligand-Target Pair | |
Tyrosine-protein kinase receptor UFO
(Homo sapiens (Human)) | BDBM50350424
(CHEMBL454440)Show InChI InChI=1S/C14H10O6/c1-5-11-10(4-8(17)13(5)18)20-9-3-6(15)2-7(16)12(9)14(11)19/h2-4,15-18H,1H3 | PDB
KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| Purchase
CHEMBL PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | 6.60E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Heinrich-Heine-Universit£t
Curated by ChEMBL
| Assay Description Inhibition of recombinant AXL assessed as 33Pi incorporation after 60 mins by scintillation counting |
Bioorg Med Chem 19: 4644-51 (2011)
Article DOI: 10.1016/j.bmc.2011.06.013 BindingDB Entry DOI: 10.7270/Q2X92BNH |
More data for this Ligand-Target Pair | |
Insulin-like growth factor 1 receptor
(Homo sapiens (Human)) | BDBM50350424
(CHEMBL454440)Show InChI InChI=1S/C14H10O6/c1-5-11-10(4-8(17)13(5)18)20-9-3-6(15)2-7(16)12(9)14(11)19/h2-4,15-18H,1H3 | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar AffyNet
| Purchase
CHEMBL PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | 8.60E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Heinrich-Heine-Universit£t
Curated by ChEMBL
| Assay Description Inhibition of recombinant IGF1-R assessed as 33Pi incorporation after 60 mins by scintillation counting |
Bioorg Med Chem 19: 4644-51 (2011)
Article DOI: 10.1016/j.bmc.2011.06.013 BindingDB Entry DOI: 10.7270/Q2X92BNH |
More data for this Ligand-Target Pair | |
Serine/threonine-protein kinase PLK1
(Homo sapiens (Human)) | BDBM50350424
(CHEMBL454440)Show InChI InChI=1S/C14H10O6/c1-5-11-10(4-8(17)13(5)18)20-9-3-6(15)2-7(16)12(9)14(11)19/h2-4,15-18H,1H3 | PDB MMDB
NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar AffyNet
| Purchase
CHEMBL PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | 8.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Heinrich-Heine-Universit£t
Curated by ChEMBL
| Assay Description Inhibition of recombinant PLK1 assessed as 33Pi incorporation after 60 mins by scintillation counting |
Bioorg Med Chem 19: 4644-51 (2011)
Article DOI: 10.1016/j.bmc.2011.06.013 BindingDB Entry DOI: 10.7270/Q2X92BNH |
More data for this Ligand-Target Pair | |
Vascular endothelial growth factor receptor 2
(Homo sapiens (Human)) | BDBM50350423
(CHEMBL466154)Show InChI InChI=1S/C14H10O5/c1-6-2-7(15)4-10-12(6)14(18)13-9(17)3-8(16)5-11(13)19-10/h2-5,15-17H,1H3 | PDB MMDB
NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar AffyNet
| Purchase
CHEMBL MCE KEGG PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | 1.17E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Heinrich-Heine-Universit£t
Curated by ChEMBL
| Assay Description Inhibition of recombinant VEGF-R2 assessed as 33Pi incorporation after 60 mins by scintillation counting |
Bioorg Med Chem 19: 4644-51 (2011)
Article DOI: 10.1016/j.bmc.2011.06.013 BindingDB Entry DOI: 10.7270/Q2X92BNH |
More data for this Ligand-Target Pair | |
Proto-oncogene tyrosine-protein kinase Src
(Homo sapiens (Human)) | BDBM50350424
(CHEMBL454440)Show InChI InChI=1S/C14H10O6/c1-5-11-10(4-8(17)13(5)18)20-9-3-6(15)2-7(16)12(9)14(11)19/h2-4,15-18H,1H3 | PDB MMDB
KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar AffyNet
| Purchase
CHEMBL PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | 1.29E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Heinrich-Heine-Universit£t
Curated by ChEMBL
| Assay Description Inhibition of recombinant SRC assessed as 33Pi incorporation after 60 mins by scintillation counting |
Bioorg Med Chem 19: 4644-51 (2011)
Article DOI: 10.1016/j.bmc.2011.06.013 BindingDB Entry DOI: 10.7270/Q2X92BNH |
More data for this Ligand-Target Pair | |
Focal adhesion kinase 1
(Homo sapiens (Human)) | BDBM50350424
(CHEMBL454440)Show InChI InChI=1S/C14H10O6/c1-5-11-10(4-8(17)13(5)18)20-9-3-6(15)2-7(16)12(9)14(11)19/h2-4,15-18H,1H3 | PDB MMDB
NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar AffyNet
| Purchase
CHEMBL PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | 1.52E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Heinrich-Heine-Universit£t
Curated by ChEMBL
| Assay Description Inhibition of recombinant FAK assessed as 33Pi incorporation after 60 mins by scintillation counting |
Bioorg Med Chem 19: 4644-51 (2011)
Article DOI: 10.1016/j.bmc.2011.06.013 BindingDB Entry DOI: 10.7270/Q2X92BNH |
More data for this Ligand-Target Pair | |
NUAK family SNF1-like kinase 1
(Homo sapiens (Human)) | BDBM50350424
(CHEMBL454440)Show InChI InChI=1S/C14H10O6/c1-5-11-10(4-8(17)13(5)18)20-9-3-6(15)2-7(16)12(9)14(11)19/h2-4,15-18H,1H3 | KEGG
UniProtKB/SwissProt
antibodypedia GoogleScholar AffyNet
| Purchase
CHEMBL PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | 1.56E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Heinrich-Heine-Universit£t
Curated by ChEMBL
| Assay Description Inhibition of recombinant ARK5 assessed as 33Pi incorporation after 60 mins by scintillation counting |
Bioorg Med Chem 19: 4644-51 (2011)
Article DOI: 10.1016/j.bmc.2011.06.013 BindingDB Entry DOI: 10.7270/Q2X92BNH |
More data for this Ligand-Target Pair | |
NUAK family SNF1-like kinase 1
(Homo sapiens (Human)) | BDBM50350423
(CHEMBL466154)Show InChI InChI=1S/C14H10O5/c1-6-2-7(15)4-10-12(6)14(18)13-9(17)3-8(16)5-11(13)19-10/h2-5,15-17H,1H3 | KEGG
UniProtKB/SwissProt
antibodypedia GoogleScholar AffyNet
| Purchase
CHEMBL MCE KEGG PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | 3.30E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Heinrich-Heine-Universit£t
Curated by ChEMBL
| Assay Description Inhibition of recombinant ARK5 assessed as 33Pi incorporation after 60 mins by scintillation counting |
Bioorg Med Chem 19: 4644-51 (2011)
Article DOI: 10.1016/j.bmc.2011.06.013 BindingDB Entry DOI: 10.7270/Q2X92BNH |
More data for this Ligand-Target Pair | |
Insulin-like growth factor 1 receptor
(Homo sapiens (Human)) | BDBM50350423
(CHEMBL466154)Show InChI InChI=1S/C14H10O5/c1-6-2-7(15)4-10-12(6)14(18)13-9(17)3-8(16)5-11(13)19-10/h2-5,15-17H,1H3 | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar AffyNet
| Purchase
CHEMBL MCE KEGG PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | 3.33E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Heinrich-Heine-Universit£t
Curated by ChEMBL
| Assay Description Inhibition of recombinant IGF1-R assessed as 33Pi incorporation after 60 mins by scintillation counting |
Bioorg Med Chem 19: 4644-51 (2011)
Article DOI: 10.1016/j.bmc.2011.06.013 BindingDB Entry DOI: 10.7270/Q2X92BNH |
More data for this Ligand-Target Pair | |
Proto-oncogene tyrosine-protein kinase Src
(Homo sapiens (Human)) | BDBM50350423
(CHEMBL466154)Show InChI InChI=1S/C14H10O5/c1-6-2-7(15)4-10-12(6)14(18)13-9(17)3-8(16)5-11(13)19-10/h2-5,15-17H,1H3 | PDB MMDB
KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar AffyNet
| Purchase
CHEMBL MCE KEGG PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | 3.50E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Heinrich-Heine-Universit£t
Curated by ChEMBL
| Assay Description Inhibition of recombinant SRC assessed as 33Pi incorporation after 60 mins by scintillation counting |
Bioorg Med Chem 19: 4644-51 (2011)
Article DOI: 10.1016/j.bmc.2011.06.013 BindingDB Entry DOI: 10.7270/Q2X92BNH |
More data for this Ligand-Target Pair | |
ALK tyrosine kinase receptor
(Homo sapiens (Human)) | BDBM50350423
(CHEMBL466154)Show InChI InChI=1S/C14H10O5/c1-6-2-7(15)4-10-12(6)14(18)13-9(17)3-8(16)5-11(13)19-10/h2-5,15-17H,1H3 | PDB
KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar AffyNet
| Purchase
CHEMBL MCE KEGG PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | 4.13E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Heinrich-Heine-Universit£t
Curated by ChEMBL
| Assay Description Inhibition of recombinant ALK assessed as 33Pi incorporation after 60 mins by scintillation counting |
Bioorg Med Chem 19: 4644-51 (2011)
Article DOI: 10.1016/j.bmc.2011.06.013 BindingDB Entry DOI: 10.7270/Q2X92BNH |
More data for this Ligand-Target Pair | |
Serine/threonine-protein kinase N1
(Homo sapiens (Human)) | BDBM50350424
(CHEMBL454440)Show InChI InChI=1S/C14H10O6/c1-5-11-10(4-8(17)13(5)18)20-9-3-6(15)2-7(16)12(9)14(11)19/h2-4,15-18H,1H3 | PDB MMDB
NCI pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| Purchase
CHEMBL PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | 4.53E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Heinrich-Heine-Universit£t
Curated by ChEMBL
| Assay Description Inhibition of recombinant PRK1 assessed as 33Pi incorporation after 60 mins by scintillation counting |
Bioorg Med Chem 19: 4644-51 (2011)
Article DOI: 10.1016/j.bmc.2011.06.013 BindingDB Entry DOI: 10.7270/Q2X92BNH |
More data for this Ligand-Target Pair | |
Serine/threonine-protein kinase N1
(Homo sapiens (Human)) | BDBM50350423
(CHEMBL466154)Show InChI InChI=1S/C14H10O5/c1-6-2-7(15)4-10-12(6)14(18)13-9(17)3-8(16)5-11(13)19-10/h2-5,15-17H,1H3 | PDB MMDB
NCI pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| Purchase
CHEMBL MCE KEGG PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | 5.49E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Heinrich-Heine-Universit£t
Curated by ChEMBL
| Assay Description Inhibition of recombinant PRK1 assessed as 33Pi incorporation after 60 mins by scintillation counting |
Bioorg Med Chem 19: 4644-51 (2011)
Article DOI: 10.1016/j.bmc.2011.06.013 BindingDB Entry DOI: 10.7270/Q2X92BNH |
More data for this Ligand-Target Pair | |
Serine/threonine-protein kinase Nek6
(Homo sapiens (Human)) | BDBM50350424
(CHEMBL454440)Show InChI InChI=1S/C14H10O6/c1-5-11-10(4-8(17)13(5)18)20-9-3-6(15)2-7(16)12(9)14(11)19/h2-4,15-18H,1H3 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
antibodypedia GoogleScholar AffyNet
| Purchase
CHEMBL PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | 6.78E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Heinrich-Heine-Universit£t
Curated by ChEMBL
| Assay Description Inhibition of recombinant NEK6 assessed as 33Pi incorporation after 60 mins by scintillation counting |
Bioorg Med Chem 19: 4644-51 (2011)
Article DOI: 10.1016/j.bmc.2011.06.013 BindingDB Entry DOI: 10.7270/Q2X92BNH |
More data for this Ligand-Target Pair | |
Serine/threonine-protein kinase PLK1
(Homo sapiens (Human)) | BDBM50350423
(CHEMBL466154)Show InChI InChI=1S/C14H10O5/c1-6-2-7(15)4-10-12(6)14(18)13-9(17)3-8(16)5-11(13)19-10/h2-5,15-17H,1H3 | PDB MMDB
NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar AffyNet
| Purchase
CHEMBL MCE KEGG PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | 7.57E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Heinrich-Heine-Universit£t
Curated by ChEMBL
| Assay Description Inhibition of recombinant PLK1 assessed as 33Pi incorporation after 60 mins by scintillation counting |
Bioorg Med Chem 19: 4644-51 (2011)
Article DOI: 10.1016/j.bmc.2011.06.013 BindingDB Entry DOI: 10.7270/Q2X92BNH |
More data for this Ligand-Target Pair | |
Serine/threonine-protein kinase Nek2
(Homo sapiens (Human)) | BDBM50350424
(CHEMBL454440)Show InChI InChI=1S/C14H10O6/c1-5-11-10(4-8(17)13(5)18)20-9-3-6(15)2-7(16)12(9)14(11)19/h2-4,15-18H,1H3 | PDB
UniProtKB/SwissProt
antibodypedia GoogleScholar AffyNet
| Purchase
CHEMBL PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | 8.39E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Heinrich-Heine-Universit£t
Curated by ChEMBL
| Assay Description Inhibition of recombinant NEK2 assessed as 33Pi incorporation after 60 mins by scintillation counting |
Bioorg Med Chem 19: 4644-51 (2011)
Article DOI: 10.1016/j.bmc.2011.06.013 BindingDB Entry DOI: 10.7270/Q2X92BNH |
More data for this Ligand-Target Pair | |
Dual specificity mitogen-activated protein kinase kinase 1
(Homo sapiens (Human)) | BDBM50350424
(CHEMBL454440)Show InChI InChI=1S/C14H10O6/c1-5-11-10(4-8(17)13(5)18)20-9-3-6(15)2-7(16)12(9)14(11)19/h2-4,15-18H,1H3 | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar AffyNet
| Purchase
CHEMBL PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Heinrich-Heine-Universit£t
Curated by ChEMBL
| Assay Description Inhibition of wild type MEK1 assessed as 33Pi incorporation after 60 mins by scintillation counting |
Bioorg Med Chem 19: 4644-51 (2011)
Article DOI: 10.1016/j.bmc.2011.06.013 BindingDB Entry DOI: 10.7270/Q2X92BNH |
More data for this Ligand-Target Pair | |
Tyrosine-protein kinase receptor UFO
(Homo sapiens (Human)) | BDBM50350423
(CHEMBL466154)Show InChI InChI=1S/C14H10O5/c1-6-2-7(15)4-10-12(6)14(18)13-9(17)3-8(16)5-11(13)19-10/h2-5,15-17H,1H3 | PDB
KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| Purchase
CHEMBL MCE KEGG PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Heinrich-Heine-Universit£t
Curated by ChEMBL
| Assay Description Inhibition of recombinant AXL assessed as 33Pi incorporation after 60 mins by scintillation counting |
Bioorg Med Chem 19: 4644-51 (2011)
Article DOI: 10.1016/j.bmc.2011.06.013 BindingDB Entry DOI: 10.7270/Q2X92BNH |
More data for this Ligand-Target Pair | |
Serine/threonine-protein kinase Nek6
(Homo sapiens (Human)) | BDBM50350423
(CHEMBL466154)Show InChI InChI=1S/C14H10O5/c1-6-2-7(15)4-10-12(6)14(18)13-9(17)3-8(16)5-11(13)19-10/h2-5,15-17H,1H3 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
antibodypedia GoogleScholar AffyNet
| Purchase
CHEMBL MCE KEGG PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Heinrich-Heine-Universit£t
Curated by ChEMBL
| Assay Description Inhibition of recombinant NEK6 assessed as 33Pi incorporation after 60 mins by scintillation counting |
Bioorg Med Chem 19: 4644-51 (2011)
Article DOI: 10.1016/j.bmc.2011.06.013 BindingDB Entry DOI: 10.7270/Q2X92BNH |
More data for this Ligand-Target Pair | |
Dual specificity mitogen-activated protein kinase kinase 1
(Homo sapiens (Human)) | BDBM50350423
(CHEMBL466154)Show InChI InChI=1S/C14H10O5/c1-6-2-7(15)4-10-12(6)14(18)13-9(17)3-8(16)5-11(13)19-10/h2-5,15-17H,1H3 | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar AffyNet
| Purchase
CHEMBL MCE KEGG PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Heinrich-Heine-Universit£t
Curated by ChEMBL
| Assay Description Inhibition of wild type MEK1 assessed as 33Pi incorporation after 60 mins by scintillation counting |
Bioorg Med Chem 19: 4644-51 (2011)
Article DOI: 10.1016/j.bmc.2011.06.013 BindingDB Entry DOI: 10.7270/Q2X92BNH |
More data for this Ligand-Target Pair | |
RAC-alpha serine/threonine-protein kinase
(Homo sapiens (Human)) | BDBM50350424
(CHEMBL454440)Show InChI InChI=1S/C14H10O6/c1-5-11-10(4-8(17)13(5)18)20-9-3-6(15)2-7(16)12(9)14(11)19/h2-4,15-18H,1H3 | PDB
UniProtKB/SwissProt
antibodypedia GoogleScholar AffyNet
| Purchase
CHEMBL PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Heinrich-Heine-Universit£t
Curated by ChEMBL
| Assay Description Inhibition of recombinant AKT1 assessed as 33Pi incorporation after 60 mins by scintillation counting |
Bioorg Med Chem 19: 4644-51 (2011)
Article DOI: 10.1016/j.bmc.2011.06.013 BindingDB Entry DOI: 10.7270/Q2X92BNH |
More data for this Ligand-Target Pair | |
RAC-alpha serine/threonine-protein kinase
(Homo sapiens (Human)) | BDBM50350423
(CHEMBL466154)Show InChI InChI=1S/C14H10O5/c1-6-2-7(15)4-10-12(6)14(18)13-9(17)3-8(16)5-11(13)19-10/h2-5,15-17H,1H3 | PDB
UniProtKB/SwissProt
antibodypedia GoogleScholar AffyNet
| Purchase
CHEMBL MCE KEGG PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Heinrich-Heine-Universit£t
Curated by ChEMBL
| Assay Description Inhibition of recombinant AKT1 assessed as 33Pi incorporation after 60 mins by scintillation counting |
Bioorg Med Chem 19: 4644-51 (2011)
Article DOI: 10.1016/j.bmc.2011.06.013 BindingDB Entry DOI: 10.7270/Q2X92BNH |
More data for this Ligand-Target Pair | |
Hepatocyte growth factor receptor
(Homo sapiens (Human)) | BDBM50350423
(CHEMBL466154)Show InChI InChI=1S/C14H10O5/c1-6-2-7(15)4-10-12(6)14(18)13-9(17)3-8(16)5-11(13)19-10/h2-5,15-17H,1H3 | PDB MMDB
KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar AffyNet
| Purchase
CHEMBL MCE KEGG PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Heinrich-Heine-Universit£t
Curated by ChEMBL
| Assay Description Inhibition of wild type MET assessed as 33Pi incorporation after 60 mins by scintillation counting |
Bioorg Med Chem 19: 4644-51 (2011)
Article DOI: 10.1016/j.bmc.2011.06.013 BindingDB Entry DOI: 10.7270/Q2X92BNH |
More data for this Ligand-Target Pair | |
Focal adhesion kinase 1
(Homo sapiens (Human)) | BDBM50350423
(CHEMBL466154)Show InChI InChI=1S/C14H10O5/c1-6-2-7(15)4-10-12(6)14(18)13-9(17)3-8(16)5-11(13)19-10/h2-5,15-17H,1H3 | PDB MMDB
NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar AffyNet
| Purchase
CHEMBL MCE KEGG PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Heinrich-Heine-Universit£t
Curated by ChEMBL
| Assay Description Inhibition of recombinant FAK assessed as 33Pi incorporation after 60 mins by scintillation counting |
Bioorg Med Chem 19: 4644-51 (2011)
Article DOI: 10.1016/j.bmc.2011.06.013 BindingDB Entry DOI: 10.7270/Q2X92BNH |
More data for this Ligand-Target Pair | |
Serine/threonine-protein kinase Nek2
(Homo sapiens (Human)) | BDBM50350423
(CHEMBL466154)Show InChI InChI=1S/C14H10O5/c1-6-2-7(15)4-10-12(6)14(18)13-9(17)3-8(16)5-11(13)19-10/h2-5,15-17H,1H3 | PDB
UniProtKB/SwissProt
antibodypedia GoogleScholar AffyNet
| Purchase
CHEMBL MCE KEGG PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Heinrich-Heine-Universit£t
Curated by ChEMBL
| Assay Description Inhibition of recombinant NEK2 assessed as 33Pi incorporation after 60 mins by scintillation counting |
Bioorg Med Chem 19: 4644-51 (2011)
Article DOI: 10.1016/j.bmc.2011.06.013 BindingDB Entry DOI: 10.7270/Q2X92BNH |
More data for this Ligand-Target Pair | |