Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Estrogen receptor beta (Homo sapiens (Human)) | BDBM312140 (6,8-dihydroxy-2-(4-hydroxyphenyl)-4-(4-methoxyphen...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 0.480 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
GTX, Inc. US Patent | Assay Description Recombinant ER-α or ER-β ligand binding domain (LBD) was combined with [3H]E2 (PerkinElmer, Waltham, Mass.) in buffer A (10 mM Tris, pH 7.4... | US Patent US9623021 (2017) BindingDB Entry DOI: 10.7270/Q20C4XV9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor beta (Homo sapiens (Human)) | BDBM312151 ((E)-6,8-dihydroxy-2-(4-hydroxyphenyl)-4-(prop-1-en...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 1.66 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
GTX, Inc. US Patent | Assay Description Recombinant ER-α or ER-β ligand binding domain (LBD) was combined with [3H]E2 (PerkinElmer, Waltham, Mass.) in buffer A (10 mM Tris, pH 7.4... | US Patent US9623021 (2017) BindingDB Entry DOI: 10.7270/Q20C4XV9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor beta (Homo sapiens (Human)) | BDBM312096 (4-bromo-6,8-dihydroxy-2-(4-hydroxyphenyl)isoquinol...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
GTX, Inc. US Patent | Assay Description Recombinant ER-α or ER-β ligand binding domain (LBD) was combined with [3H]E2 (PerkinElmer, Waltham, Mass.) in buffer A (10 mM Tris, pH 7.4... | US Patent US9623021 (2017) BindingDB Entry DOI: 10.7270/Q20C4XV9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor beta (Homo sapiens (Human)) | BDBM317457 (4-chloro-6,8-dihydroxy-2-(4-hydroxyphenyl)isoquino...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
GTX, Inc. US Patent | Assay Description Recombinant ER-α or ER-β ligand binding domain (LBD) was combined with [3H]E2 (PerkinElmer, Waltham, Mass.) in buffer A (10 mM Tris, pH 7.4... | US Patent US9623021 (2017) BindingDB Entry DOI: 10.7270/Q20C4XV9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor beta (Homo sapiens (Human)) | BDBM312149 (6,8-dihydroxy-2-(4-hydroxyphenyl)-4-(4-methoxyphen...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 3.03 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
GTX, Inc. US Patent | Assay Description Recombinant ER-α or ER-β ligand binding domain (LBD) was combined with [3H]E2 (PerkinElmer, Waltham, Mass.) in buffer A (10 mM Tris, pH 7.4... | US Patent US9623021 (2017) BindingDB Entry DOI: 10.7270/Q20C4XV9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor beta (Homo sapiens (Human)) | BDBM312139 (2-(3-fluoro-4-hydroxyphenyl)-6,8-dihydroxy-4-vinyl...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 3.96 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
GTX, Inc. US Patent | Assay Description Recombinant ER-α or ER-β ligand binding domain (LBD) was combined with [3H]E2 (PerkinElmer, Waltham, Mass.) in buffer A (10 mM Tris, pH 7.4... | US Patent US9623021 (2017) BindingDB Entry DOI: 10.7270/Q20C4XV9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor beta (Homo sapiens (Human)) | BDBM312136 (4-bromo-6-hydroxy-2-(4-hydroxyphenyl)-1-oxo-1,2-di...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 6 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
GTX, Inc. US Patent | Assay Description Recombinant ER-α or ER-β ligand binding domain (LBD) was combined with [3H]E2 (PerkinElmer, Waltham, Mass.) in buffer A (10 mM Tris, pH 7.4... | US Patent US9623021 (2017) BindingDB Entry DOI: 10.7270/Q20C4XV9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor beta (Homo sapiens (Human)) | BDBM317459 (6,8-dihydroxy-2-(4-hydroxyphenyl)-4-vinylisoquinol...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 7 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
GTX, Inc. US Patent | Assay Description Recombinant ER-α or ER-β ligand binding domain (LBD) was combined with [3H]E2 (PerkinElmer, Waltham, Mass.) in buffer A (10 mM Tris, pH 7.4... | US Patent US9623021 (2017) BindingDB Entry DOI: 10.7270/Q20C4XV9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor (Homo sapiens (Human)) | BDBM312096 (4-bromo-6,8-dihydroxy-2-(4-hydroxyphenyl)isoquinol...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 32 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
GTX, Inc. US Patent | Assay Description Recombinant ER-α or ER-β ligand binding domain (LBD) was combined with [3H]E2 (PerkinElmer, Waltham, Mass.) in buffer A (10 mM Tris, pH 7.4... | US Patent US9623021 (2017) BindingDB Entry DOI: 10.7270/Q20C4XV9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor (Homo sapiens (Human)) | BDBM317457 (4-chloro-6,8-dihydroxy-2-(4-hydroxyphenyl)isoquino...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 40 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
GTX, Inc. US Patent | Assay Description Recombinant ER-α or ER-β ligand binding domain (LBD) was combined with [3H]E2 (PerkinElmer, Waltham, Mass.) in buffer A (10 mM Tris, pH 7.4... | US Patent US9623021 (2017) BindingDB Entry DOI: 10.7270/Q20C4XV9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor beta (Homo sapiens (Human)) | BDBM312134 (4-bromo-6-methoxy-2-(4-methoxyphenyl)-1-oxo-1,2-di...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 46 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
GTX, Inc. US Patent | Assay Description Recombinant ER-α or ER-β ligand binding domain (LBD) was combined with [3H]E2 (PerkinElmer, Waltham, Mass.) in buffer A (10 mM Tris, pH 7.4... | US Patent US9623021 (2017) BindingDB Entry DOI: 10.7270/Q20C4XV9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor beta (Homo sapiens (Human)) | BDBM310198 (4-bromo-6-hydroxy-2-(4-hydroxyphenyl)isoquinolin-1...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 49 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
GTX, Inc. US Patent | Assay Description Recombinant ER-α or ER-β ligand binding domain (LBD) was combined with [3H]E2 (PerkinElmer, Waltham, Mass.) in buffer A (10 mM Tris, pH 7.4... | US Patent US9623021 (2017) BindingDB Entry DOI: 10.7270/Q20C4XV9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor (Homo sapiens (Human)) | BDBM312140 (6,8-dihydroxy-2-(4-hydroxyphenyl)-4-(4-methoxyphen...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 70 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
GTX, Inc. US Patent | Assay Description Recombinant ER-α or ER-β ligand binding domain (LBD) was combined with [3H]E2 (PerkinElmer, Waltham, Mass.) in buffer A (10 mM Tris, pH 7.4... | US Patent US9623021 (2017) BindingDB Entry DOI: 10.7270/Q20C4XV9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor (Homo sapiens (Human)) | BDBM312136 (4-bromo-6-hydroxy-2-(4-hydroxyphenyl)-1-oxo-1,2-di...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 76 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
GTX, Inc. US Patent | Assay Description Recombinant ER-α or ER-β ligand binding domain (LBD) was combined with [3H]E2 (PerkinElmer, Waltham, Mass.) in buffer A (10 mM Tris, pH 7.4... | US Patent US9623021 (2017) BindingDB Entry DOI: 10.7270/Q20C4XV9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor (Homo sapiens (Human)) | BDBM317459 (6,8-dihydroxy-2-(4-hydroxyphenyl)-4-vinylisoquinol...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 94 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
GTX, Inc. US Patent | Assay Description Recombinant ER-α or ER-β ligand binding domain (LBD) was combined with [3H]E2 (PerkinElmer, Waltham, Mass.) in buffer A (10 mM Tris, pH 7.4... | US Patent US9623021 (2017) BindingDB Entry DOI: 10.7270/Q20C4XV9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor (Homo sapiens (Human)) | BDBM312151 ((E)-6,8-dihydroxy-2-(4-hydroxyphenyl)-4-(prop-1-en...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 102 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
GTX, Inc. US Patent | Assay Description Recombinant ER-α or ER-β ligand binding domain (LBD) was combined with [3H]E2 (PerkinElmer, Waltham, Mass.) in buffer A (10 mM Tris, pH 7.4... | US Patent US9623021 (2017) BindingDB Entry DOI: 10.7270/Q20C4XV9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor (Homo sapiens (Human)) | BDBM312149 (6,8-dihydroxy-2-(4-hydroxyphenyl)-4-(4-methoxyphen...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 124 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
GTX, Inc. US Patent | Assay Description Recombinant ER-α or ER-β ligand binding domain (LBD) was combined with [3H]E2 (PerkinElmer, Waltham, Mass.) in buffer A (10 mM Tris, pH 7.4... | US Patent US9623021 (2017) BindingDB Entry DOI: 10.7270/Q20C4XV9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor beta (Homo sapiens (Human)) | BDBM317461 (4-bromo-6-hydroxy-2-(4-hydroxyphenyl)-1-oxo-1,2- d...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 130 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
GTX, Inc. US Patent | Assay Description Recombinant ER-α or ER-β ligand binding domain (LBD) was combined with [3H]E2 (PerkinElmer, Waltham, Mass.) in buffer A (10 mM Tris, pH 7.4... | US Patent US9623021 (2017) BindingDB Entry DOI: 10.7270/Q20C4XV9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor (Homo sapiens (Human)) | BDBM312139 (2-(3-fluoro-4-hydroxyphenyl)-6,8-dihydroxy-4-vinyl...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 205 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
GTX, Inc. US Patent | Assay Description Recombinant ER-α or ER-β ligand binding domain (LBD) was combined with [3H]E2 (PerkinElmer, Waltham, Mass.) in buffer A (10 mM Tris, pH 7.4... | US Patent US9623021 (2017) BindingDB Entry DOI: 10.7270/Q20C4XV9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor beta (Homo sapiens (Human)) | BDBM312137 (6-hydroxy-2-(4-hydroxyphenyl)-4-phenylisoquinolin-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 252 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
GTX, Inc. US Patent | Assay Description Recombinant ER-α or ER-β ligand binding domain (LBD) was combined with [3H]E2 (PerkinElmer, Waltham, Mass.) in buffer A (10 mM Tris, pH 7.4... | US Patent US9623021 (2017) BindingDB Entry DOI: 10.7270/Q20C4XV9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor (Homo sapiens (Human)) | BDBM312134 (4-bromo-6-methoxy-2-(4-methoxyphenyl)-1-oxo-1,2-di...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | >394 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
GTX, Inc. US Patent | Assay Description Recombinant ER-α or ER-β ligand binding domain (LBD) was combined with [3H]E2 (PerkinElmer, Waltham, Mass.) in buffer A (10 mM Tris, pH 7.4... | US Patent US9623021 (2017) BindingDB Entry DOI: 10.7270/Q20C4XV9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor (Homo sapiens (Human)) | BDBM310198 (4-bromo-6-hydroxy-2-(4-hydroxyphenyl)isoquinolin-1...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 998 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
GTX, Inc. US Patent | Assay Description Recombinant ER-α or ER-β ligand binding domain (LBD) was combined with [3H]E2 (PerkinElmer, Waltham, Mass.) in buffer A (10 mM Tris, pH 7.4... | US Patent US9623021 (2017) BindingDB Entry DOI: 10.7270/Q20C4XV9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor (Homo sapiens (Human)) | BDBM317461 (4-bromo-6-hydroxy-2-(4-hydroxyphenyl)-1-oxo-1,2- d...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 1.78E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
GTX, Inc. US Patent | Assay Description Recombinant ER-α or ER-β ligand binding domain (LBD) was combined with [3H]E2 (PerkinElmer, Waltham, Mass.) in buffer A (10 mM Tris, pH 7.4... | US Patent US9623021 (2017) BindingDB Entry DOI: 10.7270/Q20C4XV9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor (Homo sapiens (Human)) | BDBM312137 (6-hydroxy-2-(4-hydroxyphenyl)-4-phenylisoquinolin-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 2.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
GTX, Inc. US Patent | Assay Description Recombinant ER-α or ER-β ligand binding domain (LBD) was combined with [3H]E2 (PerkinElmer, Waltham, Mass.) in buffer A (10 mM Tris, pH 7.4... | US Patent US9623021 (2017) BindingDB Entry DOI: 10.7270/Q20C4XV9 | |||||||||||
More data for this Ligand-Target Pair |