Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Adenosine receptor A3 [I248L] (Homo sapiens (Human)) | BDBM191046 (US9181253, 109) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | 5.90 | -47.0 | n/a | n/a | n/a | n/a | n/a | 7.5 | 25 |
The United States of America, as represented by the Secretary, Department of Health and Human Services US Patent | Assay Description Radioligand binding assays at A1, A2A, and A3ARs were performed according to the procedures described previously. Each tube in the binding assay cont... | US Patent US9181253 (2015) BindingDB Entry DOI: 10.7270/Q2CV4GJ4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A3 [I248L] (Homo sapiens (Human)) | BDBM191068 (US9181253, 115) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | 6.60 | -46.7 | n/a | n/a | n/a | n/a | n/a | 7.5 | 25 |
The United States of America, as represented by the Secretary, Department of Health and Human Services US Patent | Assay Description Radioligand binding assays at A1, A2A, and A3ARs were performed according to the procedures described previously. Each tube in the binding assay cont... | US Patent US9181253 (2015) BindingDB Entry DOI: 10.7270/Q2CV4GJ4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A3 [I248L] (Homo sapiens (Human)) | BDBM191057 (US9181253, 119) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | 8.90 | -46.0 | n/a | n/a | n/a | n/a | n/a | 7.5 | 25 |
The United States of America, as represented by the Secretary, Department of Health and Human Services US Patent | Assay Description Radioligand binding assays at A1, A2A, and A3ARs were performed according to the procedures described previously. Each tube in the binding assay cont... | US Patent US9181253 (2015) BindingDB Entry DOI: 10.7270/Q2CV4GJ4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A3 [I248L] (Homo sapiens (Human)) | BDBM191061 (US9181253, 123) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | 10.3 | -45.6 | n/a | n/a | n/a | n/a | n/a | 7.5 | 25 |
The United States of America, as represented by the Secretary, Department of Health and Human Services US Patent | Assay Description Radioligand binding assays at A1, A2A, and A3ARs were performed according to the procedures described previously. Each tube in the binding assay cont... | US Patent US9181253 (2015) BindingDB Entry DOI: 10.7270/Q2CV4GJ4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A3 [I248L] (Homo sapiens (Human)) | BDBM191055 (US9181253, 117) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | 12 | -45.2 | n/a | n/a | n/a | n/a | n/a | 7.5 | 25 |
The United States of America, as represented by the Secretary, Department of Health and Human Services US Patent | Assay Description Radioligand binding assays at A1, A2A, and A3ARs were performed according to the procedures described previously. Each tube in the binding assay cont... | US Patent US9181253 (2015) BindingDB Entry DOI: 10.7270/Q2CV4GJ4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A3 [I248L] (Homo sapiens (Human)) | BDBM191045 (US9181253, 108) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | 12.1 | -45.2 | n/a | n/a | n/a | n/a | n/a | 7.5 | 25 |
The United States of America, as represented by the Secretary, Department of Health and Human Services US Patent | Assay Description Radioligand binding assays at A1, A2A, and A3ARs were performed according to the procedures described previously. Each tube in the binding assay cont... | US Patent US9181253 (2015) BindingDB Entry DOI: 10.7270/Q2CV4GJ4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A3 [I248L] (Homo sapiens (Human)) | BDBM191062 (US9181253, 124) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | 15.2 | -44.6 | n/a | n/a | n/a | n/a | n/a | 7.5 | 25 |
The United States of America, as represented by the Secretary, Department of Health and Human Services US Patent | Assay Description Radioligand binding assays at A1, A2A, and A3ARs were performed according to the procedures described previously. Each tube in the binding assay cont... | US Patent US9181253 (2015) BindingDB Entry DOI: 10.7270/Q2CV4GJ4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A3 [I248L] (Homo sapiens (Human)) | BDBM191064 (US9181253, 126) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | 16.5 | -44.4 | n/a | n/a | n/a | n/a | n/a | 7.5 | 25 |
The United States of America, as represented by the Secretary, Department of Health and Human Services US Patent | Assay Description Radioligand binding assays at A1, A2A, and A3ARs were performed according to the procedures described previously. Each tube in the binding assay cont... | US Patent US9181253 (2015) BindingDB Entry DOI: 10.7270/Q2CV4GJ4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A3 [I248L] (Homo sapiens (Human)) | BDBM191069 (US9181253, 116) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | 32.4 | -42.7 | n/a | n/a | n/a | n/a | n/a | 7.5 | 25 |
The United States of America, as represented by the Secretary, Department of Health and Human Services US Patent | Assay Description Radioligand binding assays at A1, A2A, and A3ARs were performed according to the procedures described previously. Each tube in the binding assay cont... | US Patent US9181253 (2015) BindingDB Entry DOI: 10.7270/Q2CV4GJ4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A3 [I248L] (Homo sapiens (Human)) | BDBM191066 (US9181253, 128) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | 40.4 | -42.2 | n/a | n/a | n/a | n/a | n/a | 7.5 | 25 |
The United States of America, as represented by the Secretary, Department of Health and Human Services US Patent | Assay Description Radioligand binding assays at A1, A2A, and A3ARs were performed according to the procedures described previously. Each tube in the binding assay cont... | US Patent US9181253 (2015) BindingDB Entry DOI: 10.7270/Q2CV4GJ4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A3 [I248L] (Homo sapiens (Human)) | BDBM191060 (US9181253, 122) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | 41.5 | -42.1 | n/a | n/a | n/a | n/a | n/a | 7.5 | 25 |
The United States of America, as represented by the Secretary, Department of Health and Human Services US Patent | Assay Description Radioligand binding assays at A1, A2A, and A3ARs were performed according to the procedures described previously. Each tube in the binding assay cont... | US Patent US9181253 (2015) BindingDB Entry DOI: 10.7270/Q2CV4GJ4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A3 [I248L] (Homo sapiens (Human)) | BDBM191056 (US9181253, 118) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | 52 | -41.6 | n/a | n/a | n/a | n/a | n/a | 7.5 | 25 |
The United States of America, as represented by the Secretary, Department of Health and Human Services US Patent | Assay Description Radioligand binding assays at A1, A2A, and A3ARs were performed according to the procedures described previously. Each tube in the binding assay cont... | US Patent US9181253 (2015) BindingDB Entry DOI: 10.7270/Q2CV4GJ4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A3 [I248L] (Homo sapiens (Human)) | BDBM191065 (US9181253, 127) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | 83.2 | -40.4 | n/a | n/a | n/a | n/a | n/a | 7.5 | 25 |
The United States of America, as represented by the Secretary, Department of Health and Human Services US Patent | Assay Description Radioligand binding assays at A1, A2A, and A3ARs were performed according to the procedures described previously. Each tube in the binding assay cont... | US Patent US9181253 (2015) BindingDB Entry DOI: 10.7270/Q2CV4GJ4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A3 [I248L] (Homo sapiens (Human)) | BDBM191058 (US9181253, 120c) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | 110 | -39.7 | n/a | n/a | n/a | n/a | n/a | 7.5 | 25 |
The United States of America, as represented by the Secretary, Department of Health and Human Services US Patent | Assay Description Radioligand binding assays at A1, A2A, and A3ARs were performed according to the procedures described previously. Each tube in the binding assay cont... | US Patent US9181253 (2015) BindingDB Entry DOI: 10.7270/Q2CV4GJ4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A3 [I248L] (Homo sapiens (Human)) | BDBM191063 (US9181253, 125) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | 114 | -39.6 | n/a | n/a | n/a | n/a | n/a | 7.5 | 25 |
The United States of America, as represented by the Secretary, Department of Health and Human Services US Patent | Assay Description Radioligand binding assays at A1, A2A, and A3ARs were performed according to the procedures described previously. Each tube in the binding assay cont... | US Patent US9181253 (2015) BindingDB Entry DOI: 10.7270/Q2CV4GJ4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A3 [I248L] (Homo sapiens (Human)) | BDBM191067 (US9181253, 107) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | 160 | -38.8 | n/a | n/a | n/a | n/a | n/a | 7.5 | 25 |
The United States of America, as represented by the Secretary, Department of Health and Human Services US Patent | Assay Description Radioligand binding assays at A1, A2A, and A3ARs were performed according to the procedures described previously. Each tube in the binding assay cont... | US Patent US9181253 (2015) BindingDB Entry DOI: 10.7270/Q2CV4GJ4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A3 [I248L] (Homo sapiens (Human)) | BDBM191054 (US9181253, 114) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | 236 | -37.8 | n/a | n/a | n/a | n/a | n/a | 7.5 | 25 |
The United States of America, as represented by the Secretary, Department of Health and Human Services US Patent | Assay Description Radioligand binding assays at A1, A2A, and A3ARs were performed according to the procedures described previously. Each tube in the binding assay cont... | US Patent US9181253 (2015) BindingDB Entry DOI: 10.7270/Q2CV4GJ4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A3 [I248L] (Homo sapiens (Human)) | BDBM191053 (US9181253, 113) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | 315 | -37.1 | n/a | n/a | n/a | n/a | n/a | 7.5 | 25 |
The United States of America, as represented by the Secretary, Department of Health and Human Services US Patent | Assay Description Radioligand binding assays at A1, A2A, and A3ARs were performed according to the procedures described previously. Each tube in the binding assay cont... | US Patent US9181253 (2015) BindingDB Entry DOI: 10.7270/Q2CV4GJ4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A3 [I248L] (Homo sapiens (Human)) | BDBM191059 (US9181253, 121) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | 470 | -36.1 | n/a | n/a | n/a | n/a | n/a | 7.5 | 25 |
The United States of America, as represented by the Secretary, Department of Health and Human Services US Patent | Assay Description Radioligand binding assays at A1, A2A, and A3ARs were performed according to the procedures described previously. Each tube in the binding assay cont... | US Patent US9181253 (2015) BindingDB Entry DOI: 10.7270/Q2CV4GJ4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A3 [I248L] (Homo sapiens (Human)) | BDBM191050 (US9181253, 110) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | 500 | -36.0 | n/a | n/a | n/a | n/a | n/a | 7.5 | 25 |
The United States of America, as represented by the Secretary, Department of Health and Human Services US Patent | Assay Description Radioligand binding assays at A1, A2A, and A3ARs were performed according to the procedures described previously. Each tube in the binding assay cont... | US Patent US9181253 (2015) BindingDB Entry DOI: 10.7270/Q2CV4GJ4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A3 [I248L] (Homo sapiens (Human)) | BDBM191051 (US9181253, 111) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | 560 | -35.7 | n/a | n/a | n/a | n/a | n/a | 7.5 | 25 |
The United States of America, as represented by the Secretary, Department of Health and Human Services US Patent | Assay Description Radioligand binding assays at A1, A2A, and A3ARs were performed according to the procedures described previously. Each tube in the binding assay cont... | US Patent US9181253 (2015) BindingDB Entry DOI: 10.7270/Q2CV4GJ4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A3 [I248L] (Homo sapiens (Human)) | BDBM175399 (1,3-Dimethyl-8-[{3-(2-(hexamethyleneimin-1-yl)-2-o...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 797 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Panjab University | Assay Description Dissociation constants at A1, A2A and A3 receptors (Ki-values) were determined in radioligand competition experiments as reported earlier [19,20]. Al... | Bioorg Chem 65: 26-37 (2016) Article DOI: 10.1016/j.bioorg.2016.01.003 BindingDB Entry DOI: 10.7270/Q2C53JN1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A3 [I248L] (Homo sapiens (Human)) | BDBM191052 (US9181253, 112) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | 1.53E+3 | -33.2 | n/a | n/a | n/a | n/a | n/a | 7.5 | 25 |
The United States of America, as represented by the Secretary, Department of Health and Human Services US Patent | Assay Description Radioligand binding assays at A1, A2A, and A3ARs were performed according to the procedures described previously. Each tube in the binding assay cont... | US Patent US9181253 (2015) BindingDB Entry DOI: 10.7270/Q2CV4GJ4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A3 [I248L] (Homo sapiens (Human)) | BDBM175398 (1,3-Dimethyl-8-[4-methoxy-3-{2-(piperidin-1-yl)-2-...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 1.97E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Panjab University | Assay Description Dissociation constants at A1, A2A and A3 receptors (Ki-values) were determined in radioligand competition experiments as reported earlier [19,20]. Al... | Bioorg Chem 65: 26-37 (2016) Article DOI: 10.1016/j.bioorg.2016.01.003 BindingDB Entry DOI: 10.7270/Q2C53JN1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A3 [I248L] (Homo sapiens (Human)) | BDBM175381 (1,3-Dimethyl-8-[3-{2-(hexamethyleneimin-1-yl)-2-ox...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 3.69E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Panjab University | Assay Description Dissociation constants at A1, A2A and A3 receptors (Ki-values) were determined in radioligand competition experiments as reported earlier [19,20]. Al... | Bioorg Chem 65: 26-37 (2016) Article DOI: 10.1016/j.bioorg.2016.01.003 BindingDB Entry DOI: 10.7270/Q2C53JN1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A3 [I248L] (Homo sapiens (Human)) | BDBM175365 (1,3-Dimethyl-8-[3-(2-methoxy-2-oxoethoxy)-phenyl]x...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 3.81E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Panjab University | Assay Description Dissociation constants at A1, A2A and A3 receptors (Ki-values) were determined in radioligand competition experiments as reported earlier [19,20]. Al... | Bioorg Chem 65: 26-37 (2016) Article DOI: 10.1016/j.bioorg.2016.01.003 BindingDB Entry DOI: 10.7270/Q2C53JN1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A3 [I248L] (Homo sapiens (Human)) | BDBM175402 (1,3-Dimethyl-8-[{3-(2-(imidazol-1-yl)-2-oxoethoxy)...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 4.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Panjab University | Assay Description Dissociation constants at A1, A2A and A3 receptors (Ki-values) were determined in radioligand competition experiments as reported earlier [19,20]. Al... | Bioorg Chem 65: 26-37 (2016) Article DOI: 10.1016/j.bioorg.2016.01.003 BindingDB Entry DOI: 10.7270/Q2C53JN1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A3 [I248L] (Homo sapiens (Human)) | BDBM175372 (1,3-Dimethyl-8-[4-{2-(hexamethyleneimin-1-yl)-2-ox...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 4.15E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Panjab University | Assay Description Dissociation constants at A1, A2A and A3 receptors (Ki-values) were determined in radioligand competition experiments as reported earlier [19,20]. Al... | Bioorg Chem 65: 26-37 (2016) Article DOI: 10.1016/j.bioorg.2016.01.003 BindingDB Entry DOI: 10.7270/Q2C53JN1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A3 [I248L] (Homo sapiens (Human)) | BDBM175380 (1,3-Dimethyl-8-[3-{2-(piperidin-1-yl)]-2-oxoethoxy...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 4.16E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Panjab University | Assay Description Dissociation constants at A1, A2A and A3 receptors (Ki-values) were determined in radioligand competition experiments as reported earlier [19,20]. Al... | Bioorg Chem 65: 26-37 (2016) Article DOI: 10.1016/j.bioorg.2016.01.003 BindingDB Entry DOI: 10.7270/Q2C53JN1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A3 [I248L] (Homo sapiens (Human)) | BDBM175379 (1,3-Dimethyl-8-[3-{2-(pyrrolidin-1-yl)-2-oxoethoxy...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 4.64E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Panjab University | Assay Description Dissociation constants at A1, A2A and A3 receptors (Ki-values) were determined in radioligand competition experiments as reported earlier [19,20]. Al... | Bioorg Chem 65: 26-37 (2016) Article DOI: 10.1016/j.bioorg.2016.01.003 BindingDB Entry DOI: 10.7270/Q2C53JN1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A3 [I248L] (Homo sapiens (Human)) | BDBM175384 (1,3-Dimethyl-8-[3-{2-(imidazol-1-yl)-2-oxoethoxy}-...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 4.89E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Panjab University | Assay Description Dissociation constants at A1, A2A and A3 receptors (Ki-values) were determined in radioligand competition experiments as reported earlier [19,20]. Al... | Bioorg Chem 65: 26-37 (2016) Article DOI: 10.1016/j.bioorg.2016.01.003 BindingDB Entry DOI: 10.7270/Q2C53JN1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A3 [I248L] (Homo sapiens (Human)) | BDBM175383 (1,3-Dimethyl-8-[3-{2-(1-methylpiperazin-4-yl)-2-ox...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 5.67E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Panjab University | Assay Description Dissociation constants at A1, A2A and A3 receptors (Ki-values) were determined in radioligand competition experiments as reported earlier [19,20]. Al... | Bioorg Chem 65: 26-37 (2016) Article DOI: 10.1016/j.bioorg.2016.01.003 BindingDB Entry DOI: 10.7270/Q2C53JN1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A3 [I248L] (Homo sapiens (Human)) | BDBM175370 (1,3-Dimethyl-8-[4-{2-(pyrrolidin-1-yl)-2-oxoethoxy...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 5.68E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Panjab University | Assay Description Dissociation constants at A1, A2A and A3 receptors (Ki-values) were determined in radioligand competition experiments as reported earlier [19,20]. Al... | Bioorg Chem 65: 26-37 (2016) Article DOI: 10.1016/j.bioorg.2016.01.003 BindingDB Entry DOI: 10.7270/Q2C53JN1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A3 [I248L] (Homo sapiens (Human)) | BDBM175364 (1,3-Dimethyl-8-[4-(2-methoxy-2-oxoethoxy)-phenyl]x...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 5.86E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Panjab University | Assay Description Dissociation constants at A1, A2A and A3 receptors (Ki-values) were determined in radioligand competition experiments as reported earlier [19,20]. Al... | Bioorg Chem 65: 26-37 (2016) Article DOI: 10.1016/j.bioorg.2016.01.003 BindingDB Entry DOI: 10.7270/Q2C53JN1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A3 [I248L] (Homo sapiens (Human)) | BDBM175376 (1,3-Dimethyl-8-[4-{2-(homoveratrylamino)-2-oxoetho...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 6.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Panjab University | Assay Description Dissociation constants at A1, A2A and A3 receptors (Ki-values) were determined in radioligand competition experiments as reported earlier [19,20]. Al... | Bioorg Chem 65: 26-37 (2016) Article DOI: 10.1016/j.bioorg.2016.01.003 BindingDB Entry DOI: 10.7270/Q2C53JN1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A3 [I248L] (Homo sapiens (Human)) | BDBM175373 (1,3-Dimethyl-8-[4-{2-(morpholin-1-yl)-2-oxoethoxy}...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 7.11E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Panjab University | Assay Description Dissociation constants at A1, A2A and A3 receptors (Ki-values) were determined in radioligand competition experiments as reported earlier [19,20]. Al... | Bioorg Chem 65: 26-37 (2016) Article DOI: 10.1016/j.bioorg.2016.01.003 BindingDB Entry DOI: 10.7270/Q2C53JN1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A3 [I248L] (Homo sapiens (Human)) | BDBM175382 (1,3-Dimethyl-8-[3-{2-(morpholin-1-yl)-2-oxoethoxy}...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 7.90E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Panjab University | Assay Description Dissociation constants at A1, A2A and A3 receptors (Ki-values) were determined in radioligand competition experiments as reported earlier [19,20]. Al... | Bioorg Chem 65: 26-37 (2016) Article DOI: 10.1016/j.bioorg.2016.01.003 BindingDB Entry DOI: 10.7270/Q2C53JN1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A3 [I248L] (Homo sapiens (Human)) | BDBM175369 (8-[4-{2-(Diethylaminoethylamino)-2-oxoethoxy}-phen...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 8.35E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Panjab University | Assay Description Dissociation constants at A1, A2A and A3 receptors (Ki-values) were determined in radioligand competition experiments as reported earlier [19,20]. Al... | Bioorg Chem 65: 26-37 (2016) Article DOI: 10.1016/j.bioorg.2016.01.003 BindingDB Entry DOI: 10.7270/Q2C53JN1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A3 [I248L] (Homo sapiens (Human)) | BDBM175378 (8-[3-{2-(Diethylaminoethylamino)-2-oxoethoxy}-phen...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 8.39E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Panjab University | Assay Description Dissociation constants at A1, A2A and A3 receptors (Ki-values) were determined in radioligand competition experiments as reported earlier [19,20]. Al... | Bioorg Chem 65: 26-37 (2016) Article DOI: 10.1016/j.bioorg.2016.01.003 BindingDB Entry DOI: 10.7270/Q2C53JN1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A3 [I248L] (Homo sapiens (Human)) | BDBM175377 (1,3-Dimethyl-8-[3-{2-(dimethylaminoethylamino)-2-o...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 8.97E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Panjab University | Assay Description Dissociation constants at A1, A2A and A3 receptors (Ki-values) were determined in radioligand competition experiments as reported earlier [19,20]. Al... | Bioorg Chem 65: 26-37 (2016) Article DOI: 10.1016/j.bioorg.2016.01.003 BindingDB Entry DOI: 10.7270/Q2C53JN1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A3 [I248L] (Homo sapiens (Human)) | BDBM175397 (1,3-Dimethyl-8-[4-methoxy-3-{2-(pyrrolidin-1-yl)-2...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 8.98E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Panjab University | Assay Description Dissociation constants at A1, A2A and A3 receptors (Ki-values) were determined in radioligand competition experiments as reported earlier [19,20]. Al... | Bioorg Chem 65: 26-37 (2016) Article DOI: 10.1016/j.bioorg.2016.01.003 BindingDB Entry DOI: 10.7270/Q2C53JN1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A3 [I248L] (Homo sapiens (Human)) | BDBM175390 (1,3-Dimethyl-8-[{4-(2-(hexamethyleneimin-1-yl)-2-o...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 9.01E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Panjab University | Assay Description Dissociation constants at A1, A2A and A3 receptors (Ki-values) were determined in radioligand competition experiments as reported earlier [19,20]. Al... | Bioorg Chem 65: 26-37 (2016) Article DOI: 10.1016/j.bioorg.2016.01.003 BindingDB Entry DOI: 10.7270/Q2C53JN1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A3 [I248L] (Homo sapiens (Human)) | BDBM175385 (1,3-Dimethyl-8-[3-{2-(homoveratrylamino)-2-oxoetho...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 9.25E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Panjab University | Assay Description Dissociation constants at A1, A2A and A3 receptors (Ki-values) were determined in radioligand competition experiments as reported earlier [19,20]. Al... | Bioorg Chem 65: 26-37 (2016) Article DOI: 10.1016/j.bioorg.2016.01.003 BindingDB Entry DOI: 10.7270/Q2C53JN1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A3 [I248L] (Homo sapiens (Human)) | BDBM175386 (1,3-Dimethyl-8-[{4-(2-(dimethylaminoethylamino)-2-...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Panjab University | Assay Description Dissociation constants at A1, A2A and A3 receptors (Ki-values) were determined in radioligand competition experiments as reported earlier [19,20]. Al... | Bioorg Chem 65: 26-37 (2016) Article DOI: 10.1016/j.bioorg.2016.01.003 BindingDB Entry DOI: 10.7270/Q2C53JN1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A3 [I248L] (Homo sapiens (Human)) | BDBM175389 (1,3-Dimethyl-8-[3-methoxy-4-{2-(piperidin-1-yl)-2-...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Panjab University | Assay Description Dissociation constants at A1, A2A and A3 receptors (Ki-values) were determined in radioligand competition experiments as reported earlier [19,20]. Al... | Bioorg Chem 65: 26-37 (2016) Article DOI: 10.1016/j.bioorg.2016.01.003 BindingDB Entry DOI: 10.7270/Q2C53JN1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A3 [I248L] (Homo sapiens (Human)) | BDBM175401 (1,3-Dimethyl-8-[4-methoxy-3-{2-(1-methylpiperazin-...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Panjab University | Assay Description Dissociation constants at A1, A2A and A3 receptors (Ki-values) were determined in radioligand competition experiments as reported earlier [19,20]. Al... | Bioorg Chem 65: 26-37 (2016) Article DOI: 10.1016/j.bioorg.2016.01.003 BindingDB Entry DOI: 10.7270/Q2C53JN1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A3 [I248L] (Homo sapiens (Human)) | BDBM175366 (1,3-Dimethyl-8-[{4-(2-methoxy-2-oxoethoxy)-3-metho...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Panjab University | Assay Description Dissociation constants at A1, A2A and A3 receptors (Ki-values) were determined in radioligand competition experiments as reported earlier [19,20]. Al... | Bioorg Chem 65: 26-37 (2016) Article DOI: 10.1016/j.bioorg.2016.01.003 BindingDB Entry DOI: 10.7270/Q2C53JN1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A3 [I248L] (Homo sapiens (Human)) | BDBM175374 (1,3-Dimethyl-8-[4-{2-(1-methylpiperazin-4-yl)-2-ox...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 1.01E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Panjab University | Assay Description Dissociation constants at A1, A2A and A3 receptors (Ki-values) were determined in radioligand competition experiments as reported earlier [19,20]. Al... | Bioorg Chem 65: 26-37 (2016) Article DOI: 10.1016/j.bioorg.2016.01.003 BindingDB Entry DOI: 10.7270/Q2C53JN1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A3 [I248L] (Homo sapiens (Human)) | BDBM175368 (1,3-Dimethyl-8-[4-{2-(dimethylaminoethylamino)-2-o...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 1.05E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Panjab University | Assay Description Dissociation constants at A1, A2A and A3 receptors (Ki-values) were determined in radioligand competition experiments as reported earlier [19,20]. Al... | Bioorg Chem 65: 26-37 (2016) Article DOI: 10.1016/j.bioorg.2016.01.003 BindingDB Entry DOI: 10.7270/Q2C53JN1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A3 [I248L] (Homo sapiens (Human)) | BDBM175367 (1,3-Dimethyl-8-[{3-(2-methoxy-2-oxoethoxy)-4-metho...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 1.07E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Panjab University | Assay Description Dissociation constants at A1, A2A and A3 receptors (Ki-values) were determined in radioligand competition experiments as reported earlier [19,20]. Al... | Bioorg Chem 65: 26-37 (2016) Article DOI: 10.1016/j.bioorg.2016.01.003 BindingDB Entry DOI: 10.7270/Q2C53JN1 | |||||||||||
More data for this Ligand-Target Pair |
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