Reaction Details | |||
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Target | Glucose-dependent insulinotropic receptor | ||
Ligand | BDBM50106217 | ||
Substrate/Competitor | n/a | ||
Meas. Tech. | ChEMBL_1506408 (CHEMBL3599704) | ||
EC50 | 49±n/a nM | ||
Citation | ![]() | ||
More Info.: | Get all data from this article, Assay Method | ||
Glucose-dependent insulinotropic receptor | |||
Name: | Glucose-dependent insulinotropic receptor | ||
Synonyms: | G-protein coupled receptor 119 (GPR119) | GP119_HUMAN | GPR119 | Glucose-dependent insulinotropic receptor | ||
Type: | Protein | ||
Mol. Mass.: | 36901.49 | ||
Organism: | Homo sapiens (Human) | ||
Description: | Q8TDV5 | ||
Residue: | 335 | ||
Sequence: |
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BDBM50106217 | |||
n/a | |||
Name | BDBM50106217 | ||
Synonyms: | CHEMBL3598110 | ||
Type | Small organic molecule | ||
Emp. Form. | C23H34F3N3O4S | ||
Mol. Mass. | 505.594 | ||
SMILES | CS(=O)(=O)c1cnc(O[C@H]2CC[C@@H](CC2)OC2CCN(CC3(CCCC3)C(F)(F)F)CC2)cn1 |r,wU:9.8,wD:12.15,(9.06,2.18,;8,1.56,;9.07,.95,;7.99,2.79,;6.67,.78,;6.67,-.76,;5.34,-1.53,;4,-.77,;2.67,-1.54,;1.33,-.77,;,-1.54,;-1.33,-.77,;-1.33,.77,;,1.54,;1.33,.77,;-2.67,1.54,;-2.66,3.08,;-4,3.86,;-3.99,5.4,;-2.65,6.16,;-2.65,7.7,;-1.31,8.47,;.05,9.12,;1.07,7.97,;.29,6.64,;-1.21,6.97,;-1.3,10.01,;-2.36,10.63,;-1.29,11.24,;-.23,10.62,;-1.32,5.39,;-1.33,3.85,;4,.77,;5.33,1.55,)| | ||
Structure | ![]() |