Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Melanocortin receptor 3 (Mus musculus) | BDBM50029747 ((4S)-4-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-[({[(2S...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 2.14 | n/a | n/a | n/a | n/a |
University of Florida Curated by ChEMBL | Assay Description Agonist activity at mouse MC3R expressed in HEK293 cells assessed as forskolin-stimulated response by beta-galactosidase reporter gene assay | J Med Chem 51: 1423-31 (2008) Article DOI: 10.1021/jm701303z BindingDB Entry DOI: 10.7270/Q2KH0P61 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocyte-stimulating hormone receptor (Mus musculus) | BDBM50374114 (CHEMBL272437) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a |
University of Florida Curated by ChEMBL | Assay Description Agonist activity at mouse MC1R expressed in HEK293 cells assessed as forskolin-stimulated response by beta-galactosidase reporter gene assay | J Med Chem 51: 1423-31 (2008) Article DOI: 10.1021/jm701303z BindingDB Entry DOI: 10.7270/Q2KH0P61 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 3 (Mus musculus) | BDBM50374116 (CHEMBL270270) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 320 | n/a | n/a | n/a | n/a |
University of Florida Curated by ChEMBL | Assay Description Agonist activity at mouse MC3R expressed in HEK293 cells assessed as forskolin-stimulated response by beta-galactosidase reporter gene assay | J Med Chem 51: 1423-31 (2008) Article DOI: 10.1021/jm701303z BindingDB Entry DOI: 10.7270/Q2KH0P61 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 3 (Mus musculus) | BDBM50374117 (CHEMBL406651) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a |
University of Florida Curated by ChEMBL | Assay Description Agonist activity at mouse MC3R expressed in HEK293 cells assessed as forskolin-stimulated response by beta-galactosidase reporter gene assay | J Med Chem 51: 1423-31 (2008) Article DOI: 10.1021/jm701303z BindingDB Entry DOI: 10.7270/Q2KH0P61 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 5 (Mus musculus (Mouse)) | BDBM50374118 (CHEMBL270689) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a |
University of Florida Curated by ChEMBL | Assay Description Agonist activity at mouse MC5R expressed in HEK293 cells assessed as forskolin-stimulated response by beta-galactosidase reporter gene assay | J Med Chem 51: 1423-31 (2008) Article DOI: 10.1021/jm701303z BindingDB Entry DOI: 10.7270/Q2KH0P61 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 5 (Mus musculus (Mouse)) | BDBM50374114 (CHEMBL272437) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a |
University of Florida Curated by ChEMBL | Assay Description Agonist activity at mouse MC5R expressed in HEK293 cells assessed as forskolin-stimulated response by beta-galactosidase reporter gene assay | J Med Chem 51: 1423-31 (2008) Article DOI: 10.1021/jm701303z BindingDB Entry DOI: 10.7270/Q2KH0P61 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 5 (Mus musculus (Mouse)) | BDBM50374119 (CHEMBL410435) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a |
University of Florida Curated by ChEMBL | Assay Description Agonist activity at mouse MC5R expressed in HEK293 cells assessed as forskolin-stimulated response by beta-galactosidase reporter gene assay | J Med Chem 51: 1423-31 (2008) Article DOI: 10.1021/jm701303z BindingDB Entry DOI: 10.7270/Q2KH0P61 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 5 (Mus musculus (Mouse)) | BDBM50374120 (CHEMBL272843) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a |
University of Florida Curated by ChEMBL | Assay Description Agonist activity at mouse MC5R expressed in HEK293 cells assessed as forskolin-stimulated response by beta-galactosidase reporter gene assay | J Med Chem 51: 1423-31 (2008) Article DOI: 10.1021/jm701303z BindingDB Entry DOI: 10.7270/Q2KH0P61 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 5 (Mus musculus (Mouse)) | BDBM50374121 (CHEMBL272662) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a |
University of Florida Curated by ChEMBL | Assay Description Agonist activity at mouse MC5R expressed in HEK293 cells assessed as forskolin-stimulated response by beta-galactosidase reporter gene assay | J Med Chem 51: 1423-31 (2008) Article DOI: 10.1021/jm701303z BindingDB Entry DOI: 10.7270/Q2KH0P61 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocyte-stimulating hormone receptor (Mus musculus) | BDBM50029747 ((4S)-4-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-[({[(2S...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 0.700 | n/a | n/a | n/a | n/a |
University of Florida Curated by ChEMBL | Assay Description Agonist activity at mouse MC1R expressed in HEK293 cells assessed as forskolin-stimulated response by beta-galactosidase reporter gene assay | J Med Chem 51: 1423-31 (2008) Article DOI: 10.1021/jm701303z BindingDB Entry DOI: 10.7270/Q2KH0P61 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocyte-stimulating hormone receptor (Mus musculus) | BDBM50374122 (CHEMBL269837) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 6.90E+3 | n/a | n/a | n/a | n/a |
University of Florida Curated by ChEMBL | Assay Description Agonist activity at mouse MC1R expressed in HEK293 cells assessed as forskolin-stimulated response by beta-galactosidase reporter gene assay | J Med Chem 51: 1423-31 (2008) Article DOI: 10.1021/jm701303z BindingDB Entry DOI: 10.7270/Q2KH0P61 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocyte-stimulating hormone receptor (Mus musculus) | BDBM50374123 (CHEMBL273044) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 230 | n/a | n/a | n/a | n/a |
University of Florida Curated by ChEMBL | Assay Description Agonist activity at mouse MC1R expressed in HEK293 cells assessed as forskolin-stimulated response by beta-galactosidase reporter gene assay | J Med Chem 51: 1423-31 (2008) Article DOI: 10.1021/jm701303z BindingDB Entry DOI: 10.7270/Q2KH0P61 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocyte-stimulating hormone receptor (Mus musculus) | BDBM50374115 (CHEMBL270691) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 4.70E+3 | n/a | n/a | n/a | n/a |
University of Florida Curated by ChEMBL | Assay Description Agonist activity at mouse MC1R expressed in HEK293 cells assessed as forskolin-stimulated response by beta-galactosidase reporter gene assay | J Med Chem 51: 1423-31 (2008) Article DOI: 10.1021/jm701303z BindingDB Entry DOI: 10.7270/Q2KH0P61 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocyte-stimulating hormone receptor (Mus musculus) | BDBM50374116 (CHEMBL270270) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 48 | n/a | n/a | n/a | n/a |
University of Florida Curated by ChEMBL | Assay Description Agonist activity at mouse MC1R expressed in HEK293 cells assessed as forskolin-stimulated response by beta-galactosidase reporter gene assay | J Med Chem 51: 1423-31 (2008) Article DOI: 10.1021/jm701303z BindingDB Entry DOI: 10.7270/Q2KH0P61 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocyte-stimulating hormone receptor (Mus musculus) | BDBM50374119 (CHEMBL410435) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 2.16E+4 | n/a | n/a | n/a | n/a |
University of Florida Curated by ChEMBL | Assay Description Agonist activity at mouse MC1R expressed in HEK293 cells assessed as forskolin-stimulated response by beta-galactosidase reporter gene assay | J Med Chem 51: 1423-31 (2008) Article DOI: 10.1021/jm701303z BindingDB Entry DOI: 10.7270/Q2KH0P61 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocyte-stimulating hormone receptor (Mus musculus) | BDBM50374121 (CHEMBL272662) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.65E+4 | n/a | n/a | n/a | n/a |
University of Florida Curated by ChEMBL | Assay Description Agonist activity at mouse MC1R expressed in HEK293 cells assessed as forskolin-stimulated response by beta-galactosidase reporter gene assay | J Med Chem 51: 1423-31 (2008) Article DOI: 10.1021/jm701303z BindingDB Entry DOI: 10.7270/Q2KH0P61 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocyte-stimulating hormone receptor (Mus musculus) | BDBM50374117 (CHEMBL406651) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 3.29E+4 | n/a | n/a | n/a | n/a |
University of Florida Curated by ChEMBL | Assay Description Agonist activity at mouse MC1R expressed in HEK293 cells assessed as forskolin-stimulated response by beta-galactosidase reporter gene assay | J Med Chem 51: 1423-31 (2008) Article DOI: 10.1021/jm701303z BindingDB Entry DOI: 10.7270/Q2KH0P61 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 3 (Mus musculus) | BDBM50374118 (CHEMBL270689) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a |
University of Florida Curated by ChEMBL | Assay Description Agonist activity at mouse MC3R expressed in HEK293 cells assessed as forskolin-stimulated response by beta-galactosidase reporter gene assay | J Med Chem 51: 1423-31 (2008) Article DOI: 10.1021/jm701303z BindingDB Entry DOI: 10.7270/Q2KH0P61 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 3 (Mus musculus) | BDBM50374114 (CHEMBL272437) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a |
University of Florida Curated by ChEMBL | Assay Description Agonist activity at mouse MC3R expressed in HEK293 cells assessed as forskolin-stimulated response by beta-galactosidase reporter gene assay | J Med Chem 51: 1423-31 (2008) Article DOI: 10.1021/jm701303z BindingDB Entry DOI: 10.7270/Q2KH0P61 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 3 (Mus musculus) | BDBM50374120 (CHEMBL272843) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a |
University of Florida Curated by ChEMBL | Assay Description Agonist activity at mouse MC3R expressed in HEK293 cells assessed as forskolin-stimulated response by beta-galactosidase reporter gene assay | J Med Chem 51: 1423-31 (2008) Article DOI: 10.1021/jm701303z BindingDB Entry DOI: 10.7270/Q2KH0P61 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 3 (Mus musculus) | BDBM50374121 (CHEMBL272662) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a |
University of Florida Curated by ChEMBL | Assay Description Agonist activity at mouse MC3R expressed in HEK293 cells assessed as forskolin-stimulated response by beta-galactosidase reporter gene assay | J Med Chem 51: 1423-31 (2008) Article DOI: 10.1021/jm701303z BindingDB Entry DOI: 10.7270/Q2KH0P61 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Mus musculus) | BDBM50029747 ((4S)-4-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-[({[(2S...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 2.56 | n/a | n/a | n/a | n/a |
University of Florida Curated by ChEMBL | Assay Description Agonist activity at mouse MC4R expressed in HEK293 cells assessed as forskolin-stimulated response by beta-galactosidase reporter gene assay | J Med Chem 51: 1423-31 (2008) Article DOI: 10.1021/jm701303z BindingDB Entry DOI: 10.7270/Q2KH0P61 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Mus musculus) | BDBM50374122 (CHEMBL269837) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 3.50E+4 | n/a | n/a | n/a | n/a |
University of Florida Curated by ChEMBL | Assay Description Agonist activity at mouse MC4R expressed in HEK293 cells assessed as forskolin-stimulated response by beta-galactosidase reporter gene assay | J Med Chem 51: 1423-31 (2008) Article DOI: 10.1021/jm701303z BindingDB Entry DOI: 10.7270/Q2KH0P61 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Mus musculus) | BDBM50374123 (CHEMBL273044) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.97E+3 | n/a | n/a | n/a | n/a |
University of Florida Curated by ChEMBL | Assay Description Agonist activity at mouse MC4R expressed in HEK293 cells assessed as forskolin-stimulated response by beta-galactosidase reporter gene assay | J Med Chem 51: 1423-31 (2008) Article DOI: 10.1021/jm701303z BindingDB Entry DOI: 10.7270/Q2KH0P61 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Mus musculus) | BDBM50374117 (CHEMBL406651) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a |
University of Florida Curated by ChEMBL | Assay Description Agonist activity at mouse MC4R expressed in HEK293 cells assessed as forskolin-stimulated response by beta-galactosidase reporter gene assay | J Med Chem 51: 1423-31 (2008) Article DOI: 10.1021/jm701303z BindingDB Entry DOI: 10.7270/Q2KH0P61 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Mus musculus) | BDBM50374118 (CHEMBL270689) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a |
University of Florida Curated by ChEMBL | Assay Description Agonist activity at mouse MC4R expressed in HEK293 cells assessed as forskolin-stimulated response by beta-galactosidase reporter gene assay | J Med Chem 51: 1423-31 (2008) Article DOI: 10.1021/jm701303z BindingDB Entry DOI: 10.7270/Q2KH0P61 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Mus musculus) | BDBM50374119 (CHEMBL410435) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a |
University of Florida Curated by ChEMBL | Assay Description Agonist activity at mouse MC4R expressed in HEK293 cells assessed as forskolin-stimulated response by beta-galactosidase reporter gene assay | J Med Chem 51: 1423-31 (2008) Article DOI: 10.1021/jm701303z BindingDB Entry DOI: 10.7270/Q2KH0P61 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Mus musculus) | BDBM50374120 (CHEMBL272843) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a |
University of Florida Curated by ChEMBL | Assay Description Agonist activity at mouse MC4R expressed in HEK293 cells assessed as forskolin-stimulated response by beta-galactosidase reporter gene assay | J Med Chem 51: 1423-31 (2008) Article DOI: 10.1021/jm701303z BindingDB Entry DOI: 10.7270/Q2KH0P61 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Mus musculus) | BDBM50374121 (CHEMBL272662) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a |
University of Florida Curated by ChEMBL | Assay Description Agonist activity at mouse MC4R expressed in HEK293 cells assessed as forskolin-stimulated response by beta-galactosidase reporter gene assay | J Med Chem 51: 1423-31 (2008) Article DOI: 10.1021/jm701303z BindingDB Entry DOI: 10.7270/Q2KH0P61 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 5 (Mus musculus (Mouse)) | BDBM50029747 ((4S)-4-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-[({[(2S...) | UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 2 | n/a | n/a | n/a | n/a |
University of Florida Curated by ChEMBL | Assay Description Agonist activity at mouse MC5R expressed in HEK293 cells assessed as forskolin-stimulated response by beta-galactosidase reporter gene assay | J Med Chem 51: 1423-31 (2008) Article DOI: 10.1021/jm701303z BindingDB Entry DOI: 10.7270/Q2KH0P61 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 5 (Mus musculus (Mouse)) | BDBM50374115 (CHEMBL270691) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 4.35E+3 | n/a | n/a | n/a | n/a |
University of Florida Curated by ChEMBL | Assay Description Agonist activity at mouse MC5R expressed in HEK293 cells assessed as forskolin-stimulated response by beta-galactosidase reporter gene assay | J Med Chem 51: 1423-31 (2008) Article DOI: 10.1021/jm701303z BindingDB Entry DOI: 10.7270/Q2KH0P61 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 5 (Mus musculus (Mouse)) | BDBM50374116 (CHEMBL270270) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 87 | n/a | n/a | n/a | n/a |
University of Florida Curated by ChEMBL | Assay Description Agonist activity at mouse MC5R expressed in HEK293 cells assessed as forskolin-stimulated response by beta-galactosidase reporter gene assay | J Med Chem 51: 1423-31 (2008) Article DOI: 10.1021/jm701303z BindingDB Entry DOI: 10.7270/Q2KH0P61 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 5 (Mus musculus (Mouse)) | BDBM50374124 (CHEMBL272439) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.70E+4 | n/a | n/a | n/a | n/a |
University of Florida Curated by ChEMBL | Assay Description Agonist activity at mouse MC5R expressed in HEK293 cells assessed as forskolin-stimulated response by beta-galactosidase reporter gene assay | J Med Chem 51: 1423-31 (2008) Article DOI: 10.1021/jm701303z BindingDB Entry DOI: 10.7270/Q2KH0P61 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocyte-stimulating hormone receptor (Mus musculus) | BDBM50374125 (CHEMBL409222) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 3.40E+3 | n/a | n/a | n/a | n/a |
University of Florida Curated by ChEMBL | Assay Description Agonist activity at mouse MC1R expressed in HEK293 cells assessed as forskolin-stimulated response by beta-galactosidase reporter gene assay | J Med Chem 51: 1423-31 (2008) Article DOI: 10.1021/jm701303z BindingDB Entry DOI: 10.7270/Q2KH0P61 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocyte-stimulating hormone receptor (Mus musculus) | BDBM50374124 (CHEMBL272439) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.80E+3 | n/a | n/a | n/a | n/a |
University of Florida Curated by ChEMBL | Assay Description Agonist activity at mouse MC1R expressed in HEK293 cells assessed as forskolin-stimulated response by beta-galactosidase reporter gene assay | J Med Chem 51: 1423-31 (2008) Article DOI: 10.1021/jm701303z BindingDB Entry DOI: 10.7270/Q2KH0P61 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 3 (Mus musculus) | BDBM50374123 (CHEMBL273044) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 4.16E+3 | n/a | n/a | n/a | n/a |
University of Florida Curated by ChEMBL | Assay Description Agonist activity at mouse MC3R expressed in HEK293 cells assessed as forskolin-stimulated response by beta-galactosidase reporter gene assay | J Med Chem 51: 1423-31 (2008) Article DOI: 10.1021/jm701303z BindingDB Entry DOI: 10.7270/Q2KH0P61 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 3 (Mus musculus) | BDBM50374124 (CHEMBL272439) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 3.07E+4 | n/a | n/a | n/a | n/a |
University of Florida Curated by ChEMBL | Assay Description Agonist activity at mouse MC3R expressed in HEK293 cells assessed as forskolin-stimulated response by beta-galactosidase reporter gene assay | J Med Chem 51: 1423-31 (2008) Article DOI: 10.1021/jm701303z BindingDB Entry DOI: 10.7270/Q2KH0P61 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 3 (Mus musculus) | BDBM50374119 (CHEMBL410435) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a |
University of Florida Curated by ChEMBL | Assay Description Agonist activity at mouse MC3R expressed in HEK293 cells assessed as forskolin-stimulated response by beta-galactosidase reporter gene assay | J Med Chem 51: 1423-31 (2008) Article DOI: 10.1021/jm701303z BindingDB Entry DOI: 10.7270/Q2KH0P61 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Mus musculus) | BDBM50374116 (CHEMBL270270) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 240 | n/a | n/a | n/a | n/a |
University of Florida Curated by ChEMBL | Assay Description Agonist activity at mouse MC4R expressed in HEK293 cells assessed as forskolin-stimulated response by beta-galactosidase reporter gene assay | J Med Chem 51: 1423-31 (2008) Article DOI: 10.1021/jm701303z BindingDB Entry DOI: 10.7270/Q2KH0P61 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Mus musculus) | BDBM50374114 (CHEMBL272437) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a |
University of Florida Curated by ChEMBL | Assay Description Agonist activity at mouse MC4R expressed in HEK293 cells assessed as forskolin-stimulated response by beta-galactosidase reporter gene assay | J Med Chem 51: 1423-31 (2008) Article DOI: 10.1021/jm701303z BindingDB Entry DOI: 10.7270/Q2KH0P61 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 5 (Mus musculus (Mouse)) | BDBM50374122 (CHEMBL269837) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 3.27E+3 | n/a | n/a | n/a | n/a |
University of Florida Curated by ChEMBL | Assay Description Agonist activity at mouse MC5R expressed in HEK293 cells assessed as forskolin-stimulated response by beta-galactosidase reporter gene assay | J Med Chem 51: 1423-31 (2008) Article DOI: 10.1021/jm701303z BindingDB Entry DOI: 10.7270/Q2KH0P61 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 5 (Mus musculus (Mouse)) | BDBM50374117 (CHEMBL406651) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a |
University of Florida Curated by ChEMBL | Assay Description Agonist activity at mouse MC5R expressed in HEK293 cells assessed as forskolin-stimulated response by beta-galactosidase reporter gene assay | J Med Chem 51: 1423-31 (2008) Article DOI: 10.1021/jm701303z BindingDB Entry DOI: 10.7270/Q2KH0P61 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 3 (Mus musculus) | BDBM50374115 (CHEMBL270691) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 2.33E+4 | n/a | n/a | n/a | n/a |
University of Florida Curated by ChEMBL | Assay Description Agonist activity at mouse MC3R expressed in HEK293 cells assessed as forskolin-stimulated response by beta-galactosidase reporter gene assay | J Med Chem 51: 1423-31 (2008) Article DOI: 10.1021/jm701303z BindingDB Entry DOI: 10.7270/Q2KH0P61 | |||||||||||
More data for this Ligand-Target Pair |