Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50186127 (CHEMBL378408 | N-[(R)-2-{4-[2-(acetyl-ethyl-amino)...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Lilly Research Laboratories Curated by ChEMBL | Assay Description Inhibition of [125]I-NDP-alpha-MSH binding to human MC4R transfected in HEK293 cells | Bioorg Med Chem Lett 16: 3449-53 (2006) Article DOI: 10.1016/j.bmcl.2006.04.002 BindingDB Entry DOI: 10.7270/Q2ST7PFS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50186127 (CHEMBL378408 | N-[(R)-2-{4-[2-(acetyl-ethyl-amino)...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Lilly Research Laboratories Curated by ChEMBL | Assay Description Inhibition of [125]I-NDP-alpha-MSH binding to human MC4R transfected in HEK293 cells | Bioorg Med Chem Lett 16: 3449-53 (2006) Article DOI: 10.1016/j.bmcl.2006.04.002 BindingDB Entry DOI: 10.7270/Q2ST7PFS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50186127 (CHEMBL378408 | N-[(R)-2-{4-[2-(acetyl-ethyl-amino)...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Lilly Research Laboratories Curated by ChEMBL | Assay Description Inhibition of [125]I-NDP-alpha-MSH binding to human MC4R transfected in HEK293 cells | Bioorg Med Chem Lett 16: 3449-53 (2006) Article DOI: 10.1016/j.bmcl.2006.04.002 BindingDB Entry DOI: 10.7270/Q2ST7PFS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50186121 ((R)-N-((R)-3-(4-chlorophenyl)-1-(4-(1-cyclopentyl-...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Lilly Research Laboratories Curated by ChEMBL | Assay Description Inhibition of [125]I-NDP-alpha-MSH binding to human MC4R transfected in HEK293 cells | Bioorg Med Chem Lett 16: 3449-53 (2006) Article DOI: 10.1016/j.bmcl.2006.04.002 BindingDB Entry DOI: 10.7270/Q2ST7PFS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50186131 ((R)-N-((R)-3-(4-chlorophenyl)-1-(4-(1-cyclohexyl-2...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Lilly Research Laboratories Curated by ChEMBL | Assay Description Inhibition of [125]I-NDP-alpha-MSH binding to human MC4R transfected in HEK293 cells | Bioorg Med Chem Lett 16: 3449-53 (2006) Article DOI: 10.1016/j.bmcl.2006.04.002 BindingDB Entry DOI: 10.7270/Q2ST7PFS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50186863 (CHEMBL379497 | N-((R)-3-(4-chlorophenyl)-1-(4-(1-c...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Lilly Research Laboratories Curated by ChEMBL | Assay Description Displacement of [125I]NDP-alpha-MSH from human MC4 receptor transfected in HEK293 cells | Bioorg Med Chem Lett 16: 3843-6 (2006) Article DOI: 10.1016/j.bmcl.2006.04.016 BindingDB Entry DOI: 10.7270/Q2SQ900D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50186128 (CHEMBL209990 | N-((R)-3-(4-chlorophenyl)-1-(4-(1-c...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Lilly Research Laboratories Curated by ChEMBL | Assay Description Inhibition of [125]I-NDP-alpha-MSH binding to human MC4R transfected in HEK293 cells | Bioorg Med Chem Lett 16: 3449-53 (2006) Article DOI: 10.1016/j.bmcl.2006.04.002 BindingDB Entry DOI: 10.7270/Q2ST7PFS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50186125 (CHEMBL377825 | N-((R)-3-(4-chlorophenyl)-1-(4-(3-c...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Lilly Research Laboratories Curated by ChEMBL | Assay Description Inhibition of [125]I-NDP-alpha-MSH binding to human MC4R transfected in HEK293 cells | Bioorg Med Chem Lett 16: 3449-53 (2006) Article DOI: 10.1016/j.bmcl.2006.04.002 BindingDB Entry DOI: 10.7270/Q2ST7PFS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50186128 (CHEMBL209990 | N-((R)-3-(4-chlorophenyl)-1-(4-(1-c...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Lilly Research Laboratories Curated by ChEMBL | Assay Description Inhibition of [125]I-NDP-alpha-MSH binding to human MC4R transfected in HEK293 cells | Bioorg Med Chem Lett 16: 3449-53 (2006) Article DOI: 10.1016/j.bmcl.2006.04.002 BindingDB Entry DOI: 10.7270/Q2ST7PFS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50177564 (CHEMBL380540 | N-((R)-3-(4-chlorophenyl)-1-(4-(2-(...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 5.80 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Lilly Research Laboratories Curated by ChEMBL | Assay Description Displacement of [125I]NDP-alpha-MSH from cloned human MC4R expressed in HEK293 cells | Bioorg Med Chem Lett 16: 2341-6 (2006) Article DOI: 10.1016/j.bmcl.2005.10.103 BindingDB Entry DOI: 10.7270/Q2NS0TF6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50186124 (CHEMBL410087 | N-((R)-3-(4-chlorophenyl)-1-(4-(1-c...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 6 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Lilly Research Laboratories Curated by ChEMBL | Assay Description Inhibition of [125]I-NDP-alpha-MSH binding to human MC4R transfected in HEK293 cells | Bioorg Med Chem Lett 16: 3449-53 (2006) Article DOI: 10.1016/j.bmcl.2006.04.002 BindingDB Entry DOI: 10.7270/Q2ST7PFS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50186124 (CHEMBL410087 | N-((R)-3-(4-chlorophenyl)-1-(4-(1-c...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 6 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Lilly Research Laboratories Curated by ChEMBL | Assay Description Inhibition of [125]I-NDP-alpha-MSH binding to human MC4R transfected in HEK293 cells | Bioorg Med Chem Lett 16: 3449-53 (2006) Article DOI: 10.1016/j.bmcl.2006.04.002 BindingDB Entry DOI: 10.7270/Q2ST7PFS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50177560 (CHEMBL206042 | N-((R)-3-(4-chlorophenyl)-1-(4-(1-(...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 6.40 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Lilly Research Laboratories Curated by ChEMBL | Assay Description Displacement of [125I]NDP-alpha-MSH from cloned human MC4R expressed in HEK293 cells | Bioorg Med Chem Lett 16: 2341-6 (2006) Article DOI: 10.1016/j.bmcl.2005.10.103 BindingDB Entry DOI: 10.7270/Q2NS0TF6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50177560 (CHEMBL206042 | N-((R)-3-(4-chlorophenyl)-1-(4-(1-(...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 6.40 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Lilly Research Laboratories Curated by ChEMBL | Assay Description Displacement of [125I]NDP-alpha-MSH from cloned human MC4R expressed in HEK293 cells | Bioorg Med Chem Lett 16: 2341-6 (2006) Article DOI: 10.1016/j.bmcl.2005.10.103 BindingDB Entry DOI: 10.7270/Q2NS0TF6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50186868 (CHEMBL213340 | N-{(R)-1-(4-chloro-benzyl)-2-[4-(4-...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 6.80 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Lilly Research Laboratories Curated by ChEMBL | Assay Description Displacement of [125I]NDP-alpha-MSH from human MC4 receptor transfected in HEK293 cells | Bioorg Med Chem Lett 16: 3843-6 (2006) Article DOI: 10.1016/j.bmcl.2006.04.016 BindingDB Entry DOI: 10.7270/Q2SQ900D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50186138 (CHEMBL425609 | N-((R)-3-(4-chlorophenyl)-1-(4-(1-c...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | 7 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Lilly Research Laboratories Curated by ChEMBL | Assay Description Inhibition of [125]I-NDP-alpha-MSH binding to human MC4R transfected in HEK293 cells | Bioorg Med Chem Lett 16: 3449-53 (2006) Article DOI: 10.1016/j.bmcl.2006.04.002 BindingDB Entry DOI: 10.7270/Q2ST7PFS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50177563 (CHEMBL380855 | N-((R)-3-(4-chlorophenyl)-1-(4-(2-(...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 7.30 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Lilly Research Laboratories Curated by ChEMBL | Assay Description Displacement of [125I]NDP-alpha-MSH from cloned human MC4R expressed in HEK293 cells | Bioorg Med Chem Lett 16: 2341-6 (2006) Article DOI: 10.1016/j.bmcl.2005.10.103 BindingDB Entry DOI: 10.7270/Q2NS0TF6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50177557 (CHEMBL380365 | N-((R)-3-(4-chlorophenyl)-1-(4-(2-(...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Lilly Research Laboratories Curated by ChEMBL | Assay Description Displacement of [125I]NDP-alpha-MSH from cloned human MC4R expressed in HEK293 cells | Bioorg Med Chem Lett 16: 2341-6 (2006) Article DOI: 10.1016/j.bmcl.2005.10.103 BindingDB Entry DOI: 10.7270/Q2NS0TF6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50186122 (CHEMBL377313 | N-((R)-3-(4-chlorophenyl)-1-(4-(3-c...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Lilly Research Laboratories Curated by ChEMBL | Assay Description Inhibition of [125]I-NDP-alpha-MSH binding to human MC4R transfected in HEK293 cells | Bioorg Med Chem Lett 16: 3449-53 (2006) Article DOI: 10.1016/j.bmcl.2006.04.002 BindingDB Entry DOI: 10.7270/Q2ST7PFS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50186120 (CHEMBL380391 | N-((R)-3-(4-chlorophenyl)-1-(4-(1-(...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 12 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Lilly Research Laboratories Curated by ChEMBL | Assay Description Inhibition of [125]I-NDP-alpha-MSH binding to human MC4R transfected in HEK293 cells | Bioorg Med Chem Lett 16: 3449-53 (2006) Article DOI: 10.1016/j.bmcl.2006.04.002 BindingDB Entry DOI: 10.7270/Q2ST7PFS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50186874 (CHEMBL376999 | N-{(R)-1-(4-chloro-benzyl)-2-[4-(4-...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 13 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Lilly Research Laboratories Curated by ChEMBL | Assay Description Displacement of [125I]NDP-alpha-MSH from human MC4 receptor transfected in HEK293 cells | Bioorg Med Chem Lett 16: 3843-6 (2006) Article DOI: 10.1016/j.bmcl.2006.04.016 BindingDB Entry DOI: 10.7270/Q2SQ900D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50186862 (CHEMBL211260 | N-{(R)-1-(4-chloro-benzyl)-2-[4-(4-...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 13 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Lilly Research Laboratories Curated by ChEMBL | Assay Description Displacement of [125I]NDP-alpha-MSH from human MC4 receptor transfected in HEK293 cells | Bioorg Med Chem Lett 16: 3843-6 (2006) Article DOI: 10.1016/j.bmcl.2006.04.016 BindingDB Entry DOI: 10.7270/Q2SQ900D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50186135 ((R)-N-((R)-3-(4-chlorophenyl)-1-(4-(3-cyclohexyl-1...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 13 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Lilly Research Laboratories Curated by ChEMBL | Assay Description Inhibition of [125]I-NDP-alpha-MSH binding to human MC4R transfected in HEK293 cells | Bioorg Med Chem Lett 16: 3449-53 (2006) Article DOI: 10.1016/j.bmcl.2006.04.002 BindingDB Entry DOI: 10.7270/Q2ST7PFS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50186119 ((R)-N-((R)-3-(4-chlorophenyl)-1-(4-(1-cycloheptyl-...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 13 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Lilly Research Laboratories Curated by ChEMBL | Assay Description Inhibition of [125]I-NDP-alpha-MSH binding to human MC4R transfected in HEK293 cells | Bioorg Med Chem Lett 16: 3449-53 (2006) Article DOI: 10.1016/j.bmcl.2006.04.002 BindingDB Entry DOI: 10.7270/Q2ST7PFS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50186133 (3,4-Dihydro-1H-isoquinoline-2-carboxylic acid ((R)...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | 14 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Lilly Research Laboratories Curated by ChEMBL | Assay Description Inhibition of [125]I-NDP-alpha-MSH binding to human MC4R transfected in HEK293 cells | Bioorg Med Chem Lett 16: 3449-53 (2006) Article DOI: 10.1016/j.bmcl.2006.04.002 BindingDB Entry DOI: 10.7270/Q2ST7PFS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50174056 (CHEMBL381015 | Diethyl-[(S)-2-(2-fluoro-phenyl)-2-...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 14 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Lilly Research Laboratories Curated by ChEMBL | Assay Description Inhibition of [125I]-NDP MSH binding to human Melanocortin 4 receptor | Bioorg Med Chem Lett 15: 4973-8 (2005) Article DOI: 10.1016/j.bmcl.2005.08.018 BindingDB Entry DOI: 10.7270/Q2HT2NWT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50139027 ((R)-1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic a...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 14 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Lilly Research Laboratories Curated by ChEMBL | Assay Description Inhibition of [125I]-NDP MSH binding to human Melanocortin 4 receptor | Bioorg Med Chem Lett 15: 4973-8 (2005) Article DOI: 10.1016/j.bmcl.2005.08.018 BindingDB Entry DOI: 10.7270/Q2HT2NWT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50186865 (CHEMBL211202 | N-{(R)-1-(4-chloro-benzyl)-2-[4-(1-...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 16 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Lilly Research Laboratories Curated by ChEMBL | Assay Description Displacement of [125I]NDP-alpha-MSH from human MC4 receptor transfected in HEK293 cells | Bioorg Med Chem Lett 16: 3843-6 (2006) Article DOI: 10.1016/j.bmcl.2006.04.016 BindingDB Entry DOI: 10.7270/Q2SQ900D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50177565 (CHEMBL380858 | N-((R)-3-(4-chlorophenyl)-1-(4-(2-(...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 17 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Lilly Research Laboratories Curated by ChEMBL | Assay Description Displacement of [125I]NDP-alpha-MSH from cloned human MC4R expressed in HEK293 cells | Bioorg Med Chem Lett 16: 2341-6 (2006) Article DOI: 10.1016/j.bmcl.2005.10.103 BindingDB Entry DOI: 10.7270/Q2NS0TF6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50186132 (CHEMBL378411 | N-((R)-3-(4-chlorophenyl)-1-(4-(1-c...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 18 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Lilly Research Laboratories Curated by ChEMBL | Assay Description Inhibition of [125]I-NDP-alpha-MSH binding to human MC4R transfected in HEK293 cells | Bioorg Med Chem Lett 16: 3449-53 (2006) Article DOI: 10.1016/j.bmcl.2006.04.002 BindingDB Entry DOI: 10.7270/Q2ST7PFS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50186132 (CHEMBL378411 | N-((R)-3-(4-chlorophenyl)-1-(4-(1-c...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 18 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Lilly Research Laboratories Curated by ChEMBL | Assay Description Inhibition of [125]I-NDP-alpha-MSH binding to human MC4R transfected in HEK293 cells | Bioorg Med Chem Lett 16: 3449-53 (2006) Article DOI: 10.1016/j.bmcl.2006.04.002 BindingDB Entry DOI: 10.7270/Q2ST7PFS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50186126 (CHEMBL379051 | N-((R)-3-(4-chlorophenyl)-1-(4-(2,6...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 18 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Lilly Research Laboratories Curated by ChEMBL | Assay Description Inhibition of [125]I-NDP-alpha-MSH binding to human MC4R transfected in HEK293 cells | Bioorg Med Chem Lett 16: 3449-53 (2006) Article DOI: 10.1016/j.bmcl.2006.04.002 BindingDB Entry DOI: 10.7270/Q2ST7PFS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50177561 ((R)-N-((R)-3-(4-chlorophenyl)-1-(4-(2-(diethylamin...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 20 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Lilly Research Laboratories Curated by ChEMBL | Assay Description Inhibition of [125]I-NDP-alpha-MSH binding to human MC4R transfected in HEK293 cells | Bioorg Med Chem Lett 16: 3449-53 (2006) Article DOI: 10.1016/j.bmcl.2006.04.002 BindingDB Entry DOI: 10.7270/Q2ST7PFS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50174055 (CHEMBL198379 | Diethyl-[2-(2-fluoro-phenyl)-2-(4-m...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 20 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Lilly Research Laboratories Curated by ChEMBL | Assay Description Inhibition of [125I]-NDP MSH binding to human Melanocortin 4 receptor | Bioorg Med Chem Lett 15: 4973-8 (2005) Article DOI: 10.1016/j.bmcl.2005.08.018 BindingDB Entry DOI: 10.7270/Q2HT2NWT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50139046 (1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic acid ...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 24 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Lilly Research Laboratories Curated by ChEMBL | Assay Description Agonistic potency towards human melanocortin 4 receptor, determined by 50% maximum cAMP release | J Med Chem 47: 744-55 (2004) Article DOI: 10.1021/jm0304109 BindingDB Entry DOI: 10.7270/Q2DJ5F21 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50186134 (CHEMBL209559 | N-((R)-3-(4-chlorophenyl)-1-(4-(1-c...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 26 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Lilly Research Laboratories Curated by ChEMBL | Assay Description Inhibition of [125]I-NDP-alpha-MSH binding to human MC4R transfected in HEK293 cells | Bioorg Med Chem Lett 16: 3449-53 (2006) Article DOI: 10.1016/j.bmcl.2006.04.002 BindingDB Entry DOI: 10.7270/Q2ST7PFS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50139032 (1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic acid ...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 27 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Lilly Research Laboratories Curated by ChEMBL | Assay Description Agonistic potency towards human melanocortin 4 receptor, determined by 50% maximum cAMP release | J Med Chem 47: 744-55 (2004) Article DOI: 10.1021/jm0304109 BindingDB Entry DOI: 10.7270/Q2DJ5F21 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50186869 (CHEMBL375388 | N-{(R)-1-(4-chloro-benzyl)-2-[4-(4-...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 27 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Lilly Research Laboratories Curated by ChEMBL | Assay Description Displacement of [125I]NDP-alpha-MSH from human MC4 receptor transfected in HEK293 cells | Bioorg Med Chem Lett 16: 3843-6 (2006) Article DOI: 10.1016/j.bmcl.2006.04.016 BindingDB Entry DOI: 10.7270/Q2SQ900D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50186861 (CHEMBL213940 | N-{(R)-1-(4-chloro-benzyl)-2-[4-(4-...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 31 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Lilly Research Laboratories Curated by ChEMBL | Assay Description Displacement of [125I]NDP-alpha-MSH from human MC4 receptor transfected in HEK293 cells | Bioorg Med Chem Lett 16: 3843-6 (2006) Article DOI: 10.1016/j.bmcl.2006.04.016 BindingDB Entry DOI: 10.7270/Q2SQ900D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50139027 ((R)-1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic a...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 34 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Lilly Research Laboratories Curated by ChEMBL | Assay Description Agonistic potency towards human melanocortin 4 receptor, determined by 50% maximum cAMP release | J Med Chem 47: 744-55 (2004) Article DOI: 10.1021/jm0304109 BindingDB Entry DOI: 10.7270/Q2DJ5F21 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50186130 (CHEMBL211078 | N-((R)-3-(4-chlorophenyl)-1-(4-(dic...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 35 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Lilly Research Laboratories Curated by ChEMBL | Assay Description Inhibition of [125]I-NDP-alpha-MSH binding to human MC4R transfected in HEK293 cells | Bioorg Med Chem Lett 16: 3449-53 (2006) Article DOI: 10.1016/j.bmcl.2006.04.002 BindingDB Entry DOI: 10.7270/Q2ST7PFS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50139043 (1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic acid ...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 35 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Lilly Research Laboratories Curated by ChEMBL | Assay Description Binding affinity towards human melanocortin 4 receptor using [125I]NDP-alpha-MSH as a radioligand in HEK293 cells | J Med Chem 47: 744-55 (2004) Article DOI: 10.1021/jm0304109 BindingDB Entry DOI: 10.7270/Q2DJ5F21 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50186864 (CHEMBL373735 | N-[(R)-2-[4-(1-acetyl-4-isobutyl-pi...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 38 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Lilly Research Laboratories Curated by ChEMBL | Assay Description Displacement of [125I]NDP-alpha-MSH from human MC4 receptor transfected in HEK293 cells | Bioorg Med Chem Lett 16: 3843-6 (2006) Article DOI: 10.1016/j.bmcl.2006.04.016 BindingDB Entry DOI: 10.7270/Q2SQ900D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50174050 (CHEMBL365184 | Diethyl-[2-(4-methyl-piperazin-1-yl...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | 40 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Lilly Research Laboratories Curated by ChEMBL | Assay Description Inhibition of [125I]-NDP MSH binding to human Melanocortin 4 receptor | Bioorg Med Chem Lett 15: 4973-8 (2005) Article DOI: 10.1016/j.bmcl.2005.08.018 BindingDB Entry DOI: 10.7270/Q2HT2NWT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50174062 (CHEMBL371896 | Diethyl-[2-(4-methyl-piperazin-1-yl...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 40 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Lilly Research Laboratories Curated by ChEMBL | Assay Description Inhibition of [125I]-NDP MSH binding to human Melanocortin 4 receptor | Bioorg Med Chem Lett 15: 4973-8 (2005) Article DOI: 10.1016/j.bmcl.2005.08.018 BindingDB Entry DOI: 10.7270/Q2HT2NWT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50177561 ((R)-N-((R)-3-(4-chlorophenyl)-1-(4-(2-(diethylamin...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 41 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Lilly Research Laboratories Curated by ChEMBL | Assay Description Displacement of [125I]NDP-alpha-MSH from cloned human MC4R expressed in HEK293 cells | Bioorg Med Chem Lett 16: 2341-6 (2006) Article DOI: 10.1016/j.bmcl.2005.10.103 BindingDB Entry DOI: 10.7270/Q2NS0TF6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50186871 (CHEMBL211032 | N-{(R)-1-(4-chloro-benzyl)-2-[4-(4-...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 42 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Lilly Research Laboratories Curated by ChEMBL | Assay Description Displacement of [125I]NDP-alpha-MSH from human MC4 receptor transfected in HEK293 cells | Bioorg Med Chem Lett 16: 3843-6 (2006) Article DOI: 10.1016/j.bmcl.2006.04.016 BindingDB Entry DOI: 10.7270/Q2SQ900D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50186867 (CHEMBL378415 | N-[(R)-2-[4-(4-benzyl-1-methyl-pipe...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 44 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Lilly Research Laboratories Curated by ChEMBL | Assay Description Displacement of [125I]NDP-alpha-MSH from human MC4 receptor transfected in HEK293 cells | Bioorg Med Chem Lett 16: 3843-6 (2006) Article DOI: 10.1016/j.bmcl.2006.04.016 BindingDB Entry DOI: 10.7270/Q2SQ900D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50186875 (CHEMBL375389 | N-{(R)-1-(4-chloro-benzyl)-2-[4-(1-...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 47 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Lilly Research Laboratories Curated by ChEMBL | Assay Description Displacement of [125I]NDP-alpha-MSH from human MC4 receptor transfected in HEK293 cells | Bioorg Med Chem Lett 16: 3843-6 (2006) Article DOI: 10.1016/j.bmcl.2006.04.016 BindingDB Entry DOI: 10.7270/Q2SQ900D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50174045 (CHEMBL373042 | Diethyl-[(R)-2-(4-methyl-piperazin-...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 50 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Lilly Research Laboratories Curated by ChEMBL | Assay Description Inhibition of [125I]-NDP MSH binding to human Melanocortin 4 receptor | Bioorg Med Chem Lett 15: 4973-8 (2005) Article DOI: 10.1016/j.bmcl.2005.08.018 BindingDB Entry DOI: 10.7270/Q2HT2NWT | |||||||||||
More data for this Ligand-Target Pair |
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