Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Steroid hormone receptor ERR2 (Homo sapiens (Human)) | BDBM50233271 (CHEMBL4071073) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 10 | n/a | n/a | n/a | n/a | n/a | n/a |
The Beckman Research Institute Curated by ChEMBL | Assay Description Inverse agonist activity at GAL4-DNA binding domain-fused human ERRbeta ligand binding domain expressed in African green monkey CV1 cells assessed as... | Bioorg Med Chem 25: 1585-1599 (2017) Article DOI: 10.1016/j.bmc.2017.01.019 BindingDB Entry DOI: 10.7270/Q2DF6TFV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen-related receptor gamma (Homo sapiens (Human)) | BDBM50233271 (CHEMBL4071073) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 10 | n/a | n/a | n/a | n/a | n/a | n/a |
The Beckman Research Institute Curated by ChEMBL | Assay Description Inverse agonist activity at GAL4-DNA binding domain-fused mouse ERRgamma ligand binding domain expressed in African green monkey CV1 cells assessed a... | Bioorg Med Chem 25: 1585-1599 (2017) Article DOI: 10.1016/j.bmc.2017.01.019 BindingDB Entry DOI: 10.7270/Q2DF6TFV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Steroid hormone receptor ERR2 (Homo sapiens (Human)) | BDBM50233269 (CHEMBL4100590) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 50 | n/a | n/a | n/a | n/a | n/a | n/a |
The Beckman Research Institute Curated by ChEMBL | Assay Description Inverse agonist activity at GAL4-DNA binding domain-fused human ERRbeta ligand binding domain expressed in African green monkey CV1 cells assessed as... | Bioorg Med Chem 25: 1585-1599 (2017) Article DOI: 10.1016/j.bmc.2017.01.019 BindingDB Entry DOI: 10.7270/Q2DF6TFV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Steroid hormone receptor ERR2 (Homo sapiens (Human)) | BDBM50233266 (CHEMBL4092854) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 210 | n/a | n/a | n/a | n/a | n/a | n/a |
The Beckman Research Institute Curated by ChEMBL | Assay Description Inverse agonist activity at GAL4-DNA binding domain-fused human ERRbeta ligand binding domain expressed in African green monkey CV1 cells assessed as... | Bioorg Med Chem 25: 1585-1599 (2017) Article DOI: 10.1016/j.bmc.2017.01.019 BindingDB Entry DOI: 10.7270/Q2DF6TFV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen-related receptor gamma (Homo sapiens (Human)) | BDBM50233266 (CHEMBL4092854) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 290 | n/a | n/a | n/a | n/a | n/a | n/a |
The Beckman Research Institute Curated by ChEMBL | Assay Description Inverse agonist activity at GAL4-DNA binding domain-fused mouse ERRgamma ligand binding domain expressed in African green monkey CV1 cells assessed a... | Bioorg Med Chem 25: 1585-1599 (2017) Article DOI: 10.1016/j.bmc.2017.01.019 BindingDB Entry DOI: 10.7270/Q2DF6TFV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Steroid hormone receptor ERR2 (Homo sapiens (Human)) | BDBM50233264 (CHEMBL4085105) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 300 | n/a | n/a | n/a | n/a | n/a | n/a |
The Beckman Research Institute Curated by ChEMBL | Assay Description Inverse agonist activity at GAL4-DNA binding domain-fused human ERRbeta ligand binding domain expressed in African green monkey CV1 cells assessed as... | Bioorg Med Chem 25: 1585-1599 (2017) Article DOI: 10.1016/j.bmc.2017.01.019 BindingDB Entry DOI: 10.7270/Q2DF6TFV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen-related receptor gamma (Homo sapiens (Human)) | BDBM50233272 (CHEMBL4064246) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 300 | n/a | n/a | n/a | n/a | n/a | n/a |
The Beckman Research Institute Curated by ChEMBL | Assay Description Inverse agonist activity at GAL4-DNA binding domain-fused mouse ERRgamma ligand binding domain expressed in African green monkey CV1 cells assessed a... | Bioorg Med Chem 25: 1585-1599 (2017) Article DOI: 10.1016/j.bmc.2017.01.019 BindingDB Entry DOI: 10.7270/Q2DF6TFV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen-related receptor gamma (Homo sapiens (Human)) | BDBM50233273 (CHEMBL4064664) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 350 | n/a | n/a | n/a | n/a | n/a | n/a |
The Beckman Research Institute Curated by ChEMBL | Assay Description Inverse agonist activity at GAL4-DNA binding domain-fused mouse ERRgamma ligand binding domain expressed in African green monkey CV1 cells assessed a... | Bioorg Med Chem 25: 1585-1599 (2017) Article DOI: 10.1016/j.bmc.2017.01.019 BindingDB Entry DOI: 10.7270/Q2DF6TFV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Steroid hormone receptor ERR2 (Homo sapiens (Human)) | BDBM50233267 (CHEMBL4084142) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 350 | n/a | n/a | n/a | n/a | n/a | n/a |
The Beckman Research Institute Curated by ChEMBL | Assay Description Inverse agonist activity at GAL4-DNA binding domain-fused human ERRbeta ligand binding domain expressed in African green monkey CV1 cells assessed as... | Bioorg Med Chem 25: 1585-1599 (2017) Article DOI: 10.1016/j.bmc.2017.01.019 BindingDB Entry DOI: 10.7270/Q2DF6TFV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Steroid hormone receptor ERR2 (Homo sapiens (Human)) | BDBM50233273 (CHEMBL4064664) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 550 | n/a | n/a | n/a | n/a | n/a | n/a |
The Beckman Research Institute Curated by ChEMBL | Assay Description Inverse agonist activity at GAL4-DNA binding domain-fused human ERRbeta ligand binding domain expressed in African green monkey CV1 cells assessed as... | Bioorg Med Chem 25: 1585-1599 (2017) Article DOI: 10.1016/j.bmc.2017.01.019 BindingDB Entry DOI: 10.7270/Q2DF6TFV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Steroid hormone receptor ERR2 (Homo sapiens (Human)) | BDBM50233265 (CHEMBL4065193) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 600 | n/a | n/a | n/a | n/a | n/a | n/a |
The Beckman Research Institute Curated by ChEMBL | Assay Description Inverse agonist activity at GAL4-DNA binding domain-fused human ERRbeta ligand binding domain expressed in African green monkey CV1 cells assessed as... | Bioorg Med Chem 25: 1585-1599 (2017) Article DOI: 10.1016/j.bmc.2017.01.019 BindingDB Entry DOI: 10.7270/Q2DF6TFV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen-related receptor gamma (Homo sapiens (Human)) | BDBM20608 (4-Hydroxytamoxifen | 4-Hydroxytamoxifen (9) | 4-[(...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE KEGG MMDB PC cid PC sid PDB UniChem Patents Similars | MMDB PDB Article PubMed | n/a | n/a | 600 | n/a | n/a | n/a | n/a | n/a | n/a |
The Beckman Research Institute Curated by ChEMBL | Assay Description Inverse agonist activity at GAL4-DNA binding domain-fused mouse ERRgamma ligand binding domain expressed in African green monkey CV1 cells assessed a... | Bioorg Med Chem 25: 1585-1599 (2017) Article DOI: 10.1016/j.bmc.2017.01.019 BindingDB Entry DOI: 10.7270/Q2DF6TFV | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Steroid hormone receptor ERR2 (Homo sapiens (Human)) | BDBM20608 (4-Hydroxytamoxifen | 4-Hydroxytamoxifen (9) | 4-[(...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE KEGG MMDB PC cid PC sid PDB UniChem Patents Similars | Article PubMed | n/a | n/a | 650 | n/a | n/a | n/a | n/a | n/a | n/a |
The Beckman Research Institute Curated by ChEMBL | Assay Description Inverse agonist activity at GAL4-DNA binding domain-fused human ERRbeta ligand binding domain expressed in African green monkey CV1 cells assessed as... | Bioorg Med Chem 25: 1585-1599 (2017) Article DOI: 10.1016/j.bmc.2017.01.019 BindingDB Entry DOI: 10.7270/Q2DF6TFV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Steroid hormone receptor ERR2 (Homo sapiens (Human)) | BDBM50233268 (CHEMBL4073790) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 750 | n/a | n/a | n/a | n/a | n/a | n/a |
The Beckman Research Institute Curated by ChEMBL | Assay Description Inverse agonist activity at GAL4-DNA binding domain-fused human ERRbeta ligand binding domain expressed in African green monkey CV1 cells assessed as... | Bioorg Med Chem 25: 1585-1599 (2017) Article DOI: 10.1016/j.bmc.2017.01.019 BindingDB Entry DOI: 10.7270/Q2DF6TFV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen-related receptor gamma (Homo sapiens (Human)) | BDBM50233268 (CHEMBL4073790) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
The Beckman Research Institute Curated by ChEMBL | Assay Description Inverse agonist activity at GAL4-DNA binding domain-fused mouse ERRgamma ligand binding domain expressed in African green monkey CV1 cells assessed a... | Bioorg Med Chem 25: 1585-1599 (2017) Article DOI: 10.1016/j.bmc.2017.01.019 BindingDB Entry DOI: 10.7270/Q2DF6TFV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Steroid hormone receptor ERR2 (Homo sapiens (Human)) | BDBM50233272 (CHEMBL4064246) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
The Beckman Research Institute Curated by ChEMBL | Assay Description Inverse agonist activity at GAL4-DNA binding domain-fused human ERRbeta ligand binding domain expressed in African green monkey CV1 cells assessed as... | Bioorg Med Chem 25: 1585-1599 (2017) Article DOI: 10.1016/j.bmc.2017.01.019 BindingDB Entry DOI: 10.7270/Q2DF6TFV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Steroid hormone receptor ERR2 (Homo sapiens (Human)) | BDBM50233270 (CHEMBL4091901) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.25E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
The Beckman Research Institute Curated by ChEMBL | Assay Description Inverse agonist activity at GAL4-DNA binding domain-fused human ERRbeta ligand binding domain expressed in African green monkey CV1 cells assessed as... | Bioorg Med Chem 25: 1585-1599 (2017) Article DOI: 10.1016/j.bmc.2017.01.019 BindingDB Entry DOI: 10.7270/Q2DF6TFV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen-related receptor gamma (Homo sapiens (Human)) | BDBM50233270 (CHEMBL4091901) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
The Beckman Research Institute Curated by ChEMBL | Assay Description Inverse agonist activity at GAL4-DNA binding domain-fused mouse ERRgamma ligand binding domain expressed in African green monkey CV1 cells assessed a... | Bioorg Med Chem 25: 1585-1599 (2017) Article DOI: 10.1016/j.bmc.2017.01.019 BindingDB Entry DOI: 10.7270/Q2DF6TFV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen-related receptor gamma (Homo sapiens (Human)) | BDBM22435 (4-[(1Z)-1-{4-[2-(dimethylamino)ethoxy]phenyl}-5-hy...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase MCE MMDB PC cid PC sid PDB UniChem Similars | MMDB PDB Article PubMed | n/a | n/a | 2.70E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
The Beckman Research Institute Curated by ChEMBL | Assay Description Inverse agonist activity at GAL4-DNA binding domain-fused mouse ERRgamma ligand binding domain expressed in African green monkey CV1 cells assessed a... | Bioorg Med Chem 25: 1585-1599 (2017) Article DOI: 10.1016/j.bmc.2017.01.019 BindingDB Entry DOI: 10.7270/Q2DF6TFV | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Estrogen-related receptor gamma (Homo sapiens (Human)) | BDBM50233269 (CHEMBL4100590) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.78E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
The Beckman Research Institute Curated by ChEMBL | Assay Description Inverse agonist activity at GAL4-DNA binding domain-fused mouse ERRgamma ligand binding domain expressed in African green monkey CV1 cells assessed a... | Bioorg Med Chem 25: 1585-1599 (2017) Article DOI: 10.1016/j.bmc.2017.01.019 BindingDB Entry DOI: 10.7270/Q2DF6TFV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Steroid hormone receptor ERR2 (Homo sapiens (Human)) | BDBM22435 (4-[(1Z)-1-{4-[2-(dimethylamino)ethoxy]phenyl}-5-hy...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase MCE MMDB PC cid PC sid PDB UniChem Similars | Article PubMed | n/a | n/a | 3.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
The Beckman Research Institute Curated by ChEMBL | Assay Description Inverse agonist activity at GAL4-DNA binding domain-fused human ERRbeta ligand binding domain expressed in African green monkey CV1 cells assessed as... | Bioorg Med Chem 25: 1585-1599 (2017) Article DOI: 10.1016/j.bmc.2017.01.019 BindingDB Entry DOI: 10.7270/Q2DF6TFV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen-related receptor gamma (Homo sapiens (Human)) | BDBM50233267 (CHEMBL4084142) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
The Beckman Research Institute Curated by ChEMBL | Assay Description Inverse agonist activity at GAL4-DNA binding domain-fused mouse ERRgamma ligand binding domain expressed in African green monkey CV1 cells assessed a... | Bioorg Med Chem 25: 1585-1599 (2017) Article DOI: 10.1016/j.bmc.2017.01.019 BindingDB Entry DOI: 10.7270/Q2DF6TFV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen-related receptor gamma (Homo sapiens (Human)) | BDBM50233264 (CHEMBL4085105) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 5.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
The Beckman Research Institute Curated by ChEMBL | Assay Description Inverse agonist activity at GAL4-DNA binding domain-fused mouse ERRgamma ligand binding domain expressed in African green monkey CV1 cells assessed a... | Bioorg Med Chem 25: 1585-1599 (2017) Article DOI: 10.1016/j.bmc.2017.01.019 BindingDB Entry DOI: 10.7270/Q2DF6TFV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen-related receptor gamma (Homo sapiens (Human)) | BDBM50233265 (CHEMBL4065193) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 6.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
The Beckman Research Institute Curated by ChEMBL | Assay Description Inverse agonist activity at GAL4-DNA binding domain-fused mouse ERRgamma ligand binding domain expressed in African green monkey CV1 cells assessed a... | Bioorg Med Chem 25: 1585-1599 (2017) Article DOI: 10.1016/j.bmc.2017.01.019 BindingDB Entry DOI: 10.7270/Q2DF6TFV | |||||||||||
More data for this Ligand-Target Pair |