Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
KiSS-1 receptor (Homo sapiens (Human)) | BDBM50045514 (CHEMBL3315315) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.0260 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Takeda Pharmaceutical Company Ltd. Curated by ChEMBL | Assay Description Displacement of radioligand from human KISS1R transfected in CHO cells | J Med Chem 57: 6105-15 (2014) Article DOI: 10.1021/jm5005489 BindingDB Entry DOI: 10.7270/Q2SF2XSG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
KiSS-1 receptor (Homo sapiens (Human)) | BDBM50045510 (CHEMBL3314227) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | 0.0270 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Takeda Pharmaceutical Company Ltd. Curated by ChEMBL | Assay Description Displacement of radioligand from human KISS1R transfected in CHO cells | J Med Chem 57: 6105-15 (2014) Article DOI: 10.1021/jm5005489 BindingDB Entry DOI: 10.7270/Q2SF2XSG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
KiSS-1 receptor (Homo sapiens (Human)) | BDBM50045500 (CHEMBL3314217) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | 0.0280 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Takeda Pharmaceutical Company Ltd. Curated by ChEMBL | Assay Description Displacement of radioligand from human KISS1R transfected in CHO cells | J Med Chem 57: 6105-15 (2014) Article DOI: 10.1021/jm5005489 BindingDB Entry DOI: 10.7270/Q2SF2XSG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
KiSS-1 receptor (Homo sapiens (Human)) | BDBM50045509 (CHEMBL3314226) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | 0.0340 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Takeda Pharmaceutical Company Ltd. Curated by ChEMBL | Assay Description Displacement of radioligand from human KISS1R transfected in CHO cells | J Med Chem 57: 6105-15 (2014) Article DOI: 10.1021/jm5005489 BindingDB Entry DOI: 10.7270/Q2SF2XSG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
KiSS-1 receptor (Homo sapiens (Human)) | BDBM50045513 (Kisspeptin-10) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem Patents Similars | Article PubMed | 0.0350 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Takeda Pharmaceutical Company Ltd. Curated by ChEMBL | Assay Description Displacement of radioligand from human KISS1R transfected in CHO cells | J Med Chem 57: 6105-15 (2014) Article DOI: 10.1021/jm5005489 BindingDB Entry DOI: 10.7270/Q2SF2XSG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
KiSS-1 receptor (Homo sapiens (Human)) | BDBM50045499 (CHEMBL3314216) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Patents Similars | Article PubMed | 0.0360 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Takeda Pharmaceutical Company Ltd. Curated by ChEMBL | Assay Description Displacement of radioligand from human KISS1R transfected in CHO cells | J Med Chem 57: 6105-15 (2014) Article DOI: 10.1021/jm5005489 BindingDB Entry DOI: 10.7270/Q2SF2XSG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
KiSS-1 receptor (Homo sapiens (Human)) | BDBM50045507 (CHEMBL3314224) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE KEGG PC cid PC sid UniChem Similars | Article PubMed | 0.0360 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Takeda Pharmaceutical Company Ltd. Curated by ChEMBL | Assay Description Displacement of radioligand from human KISS1R transfected in CHO cells | J Med Chem 57: 6105-15 (2014) Article DOI: 10.1021/jm5005489 BindingDB Entry DOI: 10.7270/Q2SF2XSG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
KiSS-1 receptor (Homo sapiens (Human)) | BDBM50045498 (CHEMBL3314215) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Patents Similars | Article PubMed | 0.0370 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Takeda Pharmaceutical Company Ltd. Curated by ChEMBL | Assay Description Displacement of radioligand from human KISS1R transfected in CHO cells | J Med Chem 57: 6105-15 (2014) Article DOI: 10.1021/jm5005489 BindingDB Entry DOI: 10.7270/Q2SF2XSG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
KiSS-1 receptor (Homo sapiens (Human)) | BDBM50045512 (CHEMBL3314229) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | 0.0380 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Takeda Pharmaceutical Company Ltd. Curated by ChEMBL | Assay Description Displacement of radioligand from human KISS1R transfected in CHO cells | J Med Chem 57: 6105-15 (2014) Article DOI: 10.1021/jm5005489 BindingDB Entry DOI: 10.7270/Q2SF2XSG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
KiSS-1 receptor (Homo sapiens (Human)) | BDBM50045506 (CHEMBL3314223) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | 0.0390 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Takeda Pharmaceutical Company Ltd. Curated by ChEMBL | Assay Description Displacement of radioligand from human KISS1R transfected in CHO cells | J Med Chem 57: 6105-15 (2014) Article DOI: 10.1021/jm5005489 BindingDB Entry DOI: 10.7270/Q2SF2XSG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
KiSS-1 receptor (Homo sapiens (Human)) | BDBM50045517 (CHEMBL3314209) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | 0.0520 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Takeda Pharmaceutical Company Ltd. Curated by ChEMBL | Assay Description Displacement of radioligand from human KISS1R transfected in CHO cells | J Med Chem 57: 6105-15 (2014) Article DOI: 10.1021/jm5005489 BindingDB Entry DOI: 10.7270/Q2SF2XSG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
KiSS-1 receptor (Rattus norvegicus) | BDBM50045507 (CHEMBL3314224) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE KEGG PC cid PC sid UniChem Similars | Article PubMed | 0.0690 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Takeda Pharmaceutical Company Ltd. Curated by ChEMBL | Assay Description Displacement of radioligand from rat KISS1R transfected in CHO cells | J Med Chem 57: 6105-15 (2014) Article DOI: 10.1021/jm5005489 BindingDB Entry DOI: 10.7270/Q2SF2XSG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
KiSS-1 receptor (Homo sapiens (Human)) | BDBM50045515 (CHEMBL3314207) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Patents Similars | Article PubMed | 0.0740 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Takeda Pharmaceutical Company Ltd. Curated by ChEMBL | Assay Description Displacement of radioligand from human KISS1R transfected in CHO cells | J Med Chem 57: 6105-15 (2014) Article DOI: 10.1021/jm5005489 BindingDB Entry DOI: 10.7270/Q2SF2XSG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
KiSS-1 receptor (Rattus norvegicus) | BDBM50045498 (CHEMBL3314215) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Patents Similars | Article PubMed | 0.0770 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Takeda Pharmaceutical Company Ltd. Curated by ChEMBL | Assay Description Displacement of radioligand from rat KISS1R transfected in CHO cells | J Med Chem 57: 6105-15 (2014) Article DOI: 10.1021/jm5005489 BindingDB Entry DOI: 10.7270/Q2SF2XSG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
KiSS-1 receptor (Homo sapiens (Human)) | BDBM50045516 (CHEMBL3314208) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Patents Similars | Article PubMed | 0.0860 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Takeda Pharmaceutical Company Ltd. Curated by ChEMBL | Assay Description Displacement of radioligand from human KISS1R transfected in CHO cells | J Med Chem 57: 6105-15 (2014) Article DOI: 10.1021/jm5005489 BindingDB Entry DOI: 10.7270/Q2SF2XSG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
KiSS-1 receptor (Rattus norvegicus) | BDBM50045512 (CHEMBL3314229) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | 0.0870 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Takeda Pharmaceutical Company Ltd. Curated by ChEMBL | Assay Description Displacement of radioligand from rat KISS1R transfected in CHO cells | J Med Chem 57: 6105-15 (2014) Article DOI: 10.1021/jm5005489 BindingDB Entry DOI: 10.7270/Q2SF2XSG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
KiSS-1 receptor (Rattus norvegicus) | BDBM50045509 (CHEMBL3314226) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | 0.0870 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Takeda Pharmaceutical Company Ltd. Curated by ChEMBL | Assay Description Displacement of radioligand from rat KISS1R transfected in CHO cells | J Med Chem 57: 6105-15 (2014) Article DOI: 10.1021/jm5005489 BindingDB Entry DOI: 10.7270/Q2SF2XSG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
KiSS-1 receptor (Rattus norvegicus) | BDBM50045513 (Kisspeptin-10) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem Patents Similars | Article PubMed | 0.0880 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Takeda Pharmaceutical Company Ltd. Curated by ChEMBL | Assay Description Displacement of radioligand from rat KISS1R transfected in CHO cells | J Med Chem 57: 6105-15 (2014) Article DOI: 10.1021/jm5005489 BindingDB Entry DOI: 10.7270/Q2SF2XSG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
KiSS-1 receptor (Homo sapiens (Human)) | BDBM50045511 (CHEMBL3314228) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | 0.0890 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Takeda Pharmaceutical Company Ltd. Curated by ChEMBL | Assay Description Displacement of radioligand from human KISS1R transfected in CHO cells | J Med Chem 57: 6105-15 (2014) Article DOI: 10.1021/jm5005489 BindingDB Entry DOI: 10.7270/Q2SF2XSG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
KiSS-1 receptor (Homo sapiens (Human)) | BDBM50045518 (CHEMBL3314213) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | 0.0960 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Takeda Pharmaceutical Company Ltd. Curated by ChEMBL | Assay Description Displacement of radioligand from human KISS1R transfected in CHO cells | J Med Chem 57: 6105-15 (2014) Article DOI: 10.1021/jm5005489 BindingDB Entry DOI: 10.7270/Q2SF2XSG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
KiSS-1 receptor (Homo sapiens (Human)) | BDBM50442961 (CHEMBL3086284) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.110 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Takeda Pharmaceutical Company Ltd. Curated by ChEMBL | Assay Description Displacement of radioligand from human KISS1R transfected in CHO cells | J Med Chem 57: 6105-15 (2014) Article DOI: 10.1021/jm5005489 BindingDB Entry DOI: 10.7270/Q2SF2XSG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
KiSS-1 receptor (Rattus norvegicus) | BDBM50045508 (CHEMBL3314225) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Patents Similars | Article PubMed | 0.110 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Takeda Pharmaceutical Company Ltd. Curated by ChEMBL | Assay Description Displacement of radioligand from rat KISS1R transfected in CHO cells | J Med Chem 57: 6105-15 (2014) Article DOI: 10.1021/jm5005489 BindingDB Entry DOI: 10.7270/Q2SF2XSG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
KiSS-1 receptor (Homo sapiens (Human)) | BDBM50045505 (CHEMBL3314222) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | 0.120 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Takeda Pharmaceutical Company Ltd. Curated by ChEMBL | Assay Description Displacement of radioligand from human KISS1R transfected in CHO cells | J Med Chem 57: 6105-15 (2014) Article DOI: 10.1021/jm5005489 BindingDB Entry DOI: 10.7270/Q2SF2XSG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
KiSS-1 receptor (Rattus norvegicus) | BDBM50045515 (CHEMBL3314207) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Patents Similars | Article PubMed | 0.130 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Takeda Pharmaceutical Company Ltd. Curated by ChEMBL | Assay Description Displacement of radioligand from rat KISS1R transfected in CHO cells | J Med Chem 57: 6105-15 (2014) Article DOI: 10.1021/jm5005489 BindingDB Entry DOI: 10.7270/Q2SF2XSG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
KiSS-1 receptor (Rattus norvegicus) | BDBM50442961 (CHEMBL3086284) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.140 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Takeda Pharmaceutical Company Ltd. Curated by ChEMBL | Assay Description Displacement of radioligand from rat KISS1R transfected in CHO cells | J Med Chem 57: 6105-15 (2014) Article DOI: 10.1021/jm5005489 BindingDB Entry DOI: 10.7270/Q2SF2XSG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
KiSS-1 receptor (Rattus norvegicus) | BDBM50045511 (CHEMBL3314228) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | 0.170 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Takeda Pharmaceutical Company Ltd. Curated by ChEMBL | Assay Description Displacement of radioligand from rat KISS1R transfected in CHO cells | J Med Chem 57: 6105-15 (2014) Article DOI: 10.1021/jm5005489 BindingDB Entry DOI: 10.7270/Q2SF2XSG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
KiSS-1 receptor (Homo sapiens (Human)) | BDBM50045501 (CHEMBL3314218) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | 0.200 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Takeda Pharmaceutical Company Ltd. Curated by ChEMBL | Assay Description Displacement of radioligand from human KISS1R transfected in CHO cells | J Med Chem 57: 6105-15 (2014) Article DOI: 10.1021/jm5005489 BindingDB Entry DOI: 10.7270/Q2SF2XSG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
KiSS-1 receptor (Rattus norvegicus) | BDBM50045505 (CHEMBL3314222) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | 0.830 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Takeda Pharmaceutical Company Ltd. Curated by ChEMBL | Assay Description Displacement of radioligand from rat KISS1R transfected in CHO cells | J Med Chem 57: 6105-15 (2014) Article DOI: 10.1021/jm5005489 BindingDB Entry DOI: 10.7270/Q2SF2XSG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
KiSS-1 receptor (Rattus norvegicus) | BDBM50045501 (CHEMBL3314218) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | 3.60 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Takeda Pharmaceutical Company Ltd. Curated by ChEMBL | Assay Description Displacement of radioligand from rat KISS1R transfected in CHO cells | J Med Chem 57: 6105-15 (2014) Article DOI: 10.1021/jm5005489 BindingDB Entry DOI: 10.7270/Q2SF2XSG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gonadotropin-releasing hormone receptor (Homo sapiens (Human)) | BDBM50122654 (1-(4-(1-(2,6-difluorobenzyl)-5-((benzyl(methyl)ami...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 0.0600 | n/a | n/a | n/a | n/a | n/a | n/a |
Takeda Pharmaceutical Company, Ltd. Curated by ChEMBL | Assay Description Antagonist activity at human GnRH receptor expressed in CHO cells assessed as inhibition of GnRH-induced arachadonic acid release using [5,6,8,9,11,1... | J Med Chem 54: 4998-5012 (2011) Article DOI: 10.1021/jm200216q BindingDB Entry DOI: 10.7270/Q22N52MK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gonadotropin-releasing hormone receptor (Homo sapiens (Human)) | BDBM50347985 (CHEMBL1800156) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.0700 | n/a | n/a | n/a | n/a | n/a | n/a |
Takeda Pharmaceutical Company, Ltd. Curated by ChEMBL | Assay Description Antagonist activity at human GnRH receptor expressed in CHO cells assessed as inhibition of GnRH-induced arachadonic acid release using [5,6,8,9,11,1... | J Med Chem 54: 4998-5012 (2011) Article DOI: 10.1021/jm200216q BindingDB Entry DOI: 10.7270/Q22N52MK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gonadotropin-releasing hormone receptor (Homo sapiens (Human)) | BDBM50347996 (CHEMBL1800663) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 0.0700 | n/a | n/a | n/a | n/a | n/a | n/a |
Takeda Pharmaceutical Company, Ltd. Curated by ChEMBL | Assay Description Displacement of [125I]leuprorelin from recombinant human GnRH receptor expressed in CHO cells after 60 mins by X-ray counter | J Med Chem 54: 4998-5012 (2011) Article DOI: 10.1021/jm200216q BindingDB Entry DOI: 10.7270/Q22N52MK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gonadotropin-releasing hormone receptor (Homo sapiens (Human)) | BDBM50347996 (CHEMBL1800663) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 0.0700 | n/a | n/a | n/a | n/a | n/a | n/a |
Takeda Pharmaceutical Company, Ltd. Curated by ChEMBL | Assay Description Antagonist activity at human GnRH receptor expressed in CHO cells assessed as inhibition of GnRH-induced arachadonic acid release using [5,6,8,9,11,1... | J Med Chem 54: 4998-5012 (2011) Article DOI: 10.1021/jm200216q BindingDB Entry DOI: 10.7270/Q22N52MK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gonadotropin-releasing hormone receptor (Homo sapiens (Human)) | BDBM50347986 (CHEMBL1800155) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 0.0700 | n/a | n/a | n/a | n/a | n/a | n/a |
Takeda Pharmaceutical Company, Ltd. Curated by ChEMBL | Assay Description Displacement of [125I]leuprorelin from recombinant human GnRH receptor expressed in CHO cells after 60 mins by X-ray counter | J Med Chem 54: 4998-5012 (2011) Article DOI: 10.1021/jm200216q BindingDB Entry DOI: 10.7270/Q22N52MK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gonadotropin-releasing hormone receptor (Homo sapiens (Human)) | BDBM50347989 (CHEMBL1800668) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 0.0800 | n/a | n/a | n/a | n/a | n/a | n/a |
Takeda Pharmaceutical Company, Ltd. Curated by ChEMBL | Assay Description Antagonist activity at human GnRH receptor expressed in CHO cells assessed as inhibition of GnRH-induced arachadonic acid release using [5,6,8,9,11,1... | J Med Chem 54: 4998-5012 (2011) Article DOI: 10.1021/jm200216q BindingDB Entry DOI: 10.7270/Q22N52MK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gonadotropin-releasing hormone receptor (Homo sapiens (Human)) | BDBM50347982 (CHEMBL1800159) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 0.0800 | n/a | n/a | n/a | n/a | n/a | n/a |
Takeda Pharmaceutical Company, Ltd. Curated by ChEMBL | Assay Description Displacement of [125I]leuprorelin from recombinant human GnRH receptor expressed in CHO cells after 60 mins by X-ray counter | J Med Chem 54: 4998-5012 (2011) Article DOI: 10.1021/jm200216q BindingDB Entry DOI: 10.7270/Q22N52MK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gonadotropin-releasing hormone receptor (Homo sapiens (Human)) | BDBM50347984 (CHEMBL1800157) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 0.0800 | n/a | n/a | n/a | n/a | n/a | n/a |
Takeda Pharmaceutical Company, Ltd. Curated by ChEMBL | Assay Description Displacement of [125I]leuprorelin from recombinant human GnRH receptor expressed in CHO cells after 60 mins by X-ray counter | J Med Chem 54: 4998-5012 (2011) Article DOI: 10.1021/jm200216q BindingDB Entry DOI: 10.7270/Q22N52MK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gonadotropin-releasing hormone receptor (Homo sapiens (Human)) | BDBM50347997 (CHEMBL1800661) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 0.0800 | n/a | n/a | n/a | n/a | n/a | n/a |
Takeda Pharmaceutical Company, Ltd. Curated by ChEMBL | Assay Description Antagonist activity at human GnRH receptor expressed in CHO cells assessed as inhibition of GnRH-induced arachadonic acid release using [5,6,8,9,11,1... | J Med Chem 54: 4998-5012 (2011) Article DOI: 10.1021/jm200216q BindingDB Entry DOI: 10.7270/Q22N52MK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gonadotropin-releasing hormone receptor (Homo sapiens (Human)) | BDBM50347997 (CHEMBL1800661) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 0.0900 | n/a | n/a | n/a | n/a | n/a | n/a |
Takeda Pharmaceutical Company, Ltd. Curated by ChEMBL | Assay Description Displacement of [125I]leuprorelin from recombinant human GnRH receptor expressed in CHO cells after 60 mins by X-ray counter | J Med Chem 54: 4998-5012 (2011) Article DOI: 10.1021/jm200216q BindingDB Entry DOI: 10.7270/Q22N52MK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gonadotropin-releasing hormone receptor (Homo sapiens (Human)) | BDBM50347994 (CHEMBL1800666) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 0.0900 | n/a | n/a | n/a | n/a | n/a | n/a |
Takeda Pharmaceutical Company, Ltd. Curated by ChEMBL | Assay Description Displacement of [125I]leuprorelin from recombinant human GnRH receptor expressed in CHO cells after 60 mins by X-ray counter | J Med Chem 54: 4998-5012 (2011) Article DOI: 10.1021/jm200216q BindingDB Entry DOI: 10.7270/Q22N52MK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gonadotropin-releasing hormone receptor (Homo sapiens (Human)) | BDBM50347987 (CHEMBL1800153) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 0.100 | n/a | n/a | n/a | n/a | n/a | n/a |
Takeda Pharmaceutical Company, Ltd. Curated by ChEMBL | Assay Description Displacement of [125I]leuprorelin from recombinant human GnRH receptor expressed in CHO cells after 60 mins by X-ray counter | J Med Chem 54: 4998-5012 (2011) Article DOI: 10.1021/jm200216q BindingDB Entry DOI: 10.7270/Q22N52MK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gonadotropin-releasing hormone receptor (Homo sapiens (Human)) | BDBM50347989 (CHEMBL1800668) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 0.100 | n/a | n/a | n/a | n/a | n/a | n/a |
Takeda Pharmaceutical Company, Ltd. Curated by ChEMBL | Assay Description Displacement of [125I]leuprorelin from recombinant human GnRH receptor expressed in CHO cells after 60 mins by X-ray counter | J Med Chem 54: 4998-5012 (2011) Article DOI: 10.1021/jm200216q BindingDB Entry DOI: 10.7270/Q22N52MK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gonadotropin-releasing hormone receptor (Homo sapiens (Human)) | BDBM50347995 (CHEMBL1800664) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 0.100 | n/a | n/a | n/a | n/a | n/a | n/a |
Takeda Pharmaceutical Company, Ltd. Curated by ChEMBL | Assay Description Displacement of [125I]leuprorelin from recombinant human GnRH receptor expressed in CHO cells after 60 mins by X-ray counter | J Med Chem 54: 4998-5012 (2011) Article DOI: 10.1021/jm200216q BindingDB Entry DOI: 10.7270/Q22N52MK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gonadotropin-releasing hormone receptor (Homo sapiens (Human)) | BDBM50122654 (1-(4-(1-(2,6-difluorobenzyl)-5-((benzyl(methyl)ami...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 0.100 | n/a | n/a | n/a | n/a | n/a | n/a |
Takeda Pharmaceutical Company, Ltd. Curated by ChEMBL | Assay Description Displacement of [125I]leuprorelin from recombinant human GnRH receptor expressed in CHO cells after 60 mins by X-ray counter | J Med Chem 54: 4998-5012 (2011) Article DOI: 10.1021/jm200216q BindingDB Entry DOI: 10.7270/Q22N52MK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gonadotropin-releasing hormone receptor (Homo sapiens (Human)) | BDBM230879 (US9346822, 41) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.100 | n/a | n/a | n/a | n/a | n/a | n/a |
Takeda Pharmaceutical Company Limited US Patent | Assay Description The monkey and human membrane fractions prepared were diluted with the assay buffer to yield a 200 g/ml dilution, each of which was then dispensed at... | US Patent US9346822 (2016) BindingDB Entry DOI: 10.7270/Q2251H2F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gonadotropin-releasing hormone receptor (Homo sapiens (Human)) | BDBM50347983 (CHEMBL1800158) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 0.120 | n/a | n/a | n/a | n/a | n/a | n/a |
Takeda Pharmaceutical Company, Ltd. Curated by ChEMBL | Assay Description Displacement of [125I]leuprorelin from recombinant human GnRH receptor expressed in CHO cells after 60 mins by X-ray counter | J Med Chem 54: 4998-5012 (2011) Article DOI: 10.1021/jm200216q BindingDB Entry DOI: 10.7270/Q22N52MK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gonadotropin-releasing hormone receptor (Homo sapiens (Human)) | BDBM50347986 (CHEMBL1800155) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 0.170 | n/a | n/a | n/a | n/a | n/a | n/a |
Takeda Pharmaceutical Company, Ltd. Curated by ChEMBL | Assay Description Antagonist activity at human GnRH receptor expressed in CHO cells assessed as inhibition of GnRH-induced arachadonic acid release using [5,6,8,9,11,1... | J Med Chem 54: 4998-5012 (2011) Article DOI: 10.1021/jm200216q BindingDB Entry DOI: 10.7270/Q22N52MK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gonadotropin-releasing hormone receptor (Homo sapiens (Human)) | BDBM50347987 (CHEMBL1800153) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 0.180 | n/a | n/a | n/a | n/a | n/a | n/a |
Takeda Pharmaceutical Company, Ltd. Curated by ChEMBL | Assay Description Antagonist activity at human GnRH receptor expressed in CHO cells assessed as inhibition of GnRH-induced arachadonic acid release using [5,6,8,9,11,1... | J Med Chem 54: 4998-5012 (2011) Article DOI: 10.1021/jm200216q BindingDB Entry DOI: 10.7270/Q22N52MK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gonadotropin-releasing hormone receptor (Homo sapiens (Human)) | BDBM50348001 (CHEMBL1800662) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 0.200 | n/a | n/a | n/a | n/a | n/a | n/a |
Takeda Pharmaceutical Company, Ltd. Curated by ChEMBL | Assay Description Displacement of [125I]leuprorelin from recombinant human GnRH receptor expressed in CHO cells after 60 mins by X-ray counter | J Med Chem 54: 4998-5012 (2011) Article DOI: 10.1021/jm200216q BindingDB Entry DOI: 10.7270/Q22N52MK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gonadotropin-releasing hormone receptor (Homo sapiens (Human)) | BDBM50347988 (CHEMBL1800152 | US9346822, 40) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | US Patent | n/a | n/a | 0.200 | n/a | n/a | n/a | n/a | n/a | n/a |
Takeda Pharmaceutical Company Limited US Patent | Assay Description The monkey and human membrane fractions prepared were diluted with the assay buffer to yield a 200 g/ml dilution, each of which was then dispensed at... | US Patent US9346822 (2016) BindingDB Entry DOI: 10.7270/Q2251H2F | |||||||||||
More data for this Ligand-Target Pair |
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