Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Cysteinyl leukotriene receptor 1/2 (Homo sapiens (Human)) | BDBM50227363 (CHEMBL299837) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 0.100 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
ICI Pharmaceuticals Group Curated by ChEMBL | Assay Description Inhibition constant for displacement of [3H]LTD4 on guinea pig lung parenchymal membranes. | J Med Chem 33: 1781-90 (1990) BindingDB Entry DOI: 10.7270/Q2862FDP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cysteinyl leukotriene receptor 1/2 (Homo sapiens (Human)) | BDBM50227366 (CHEMBL48927) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 0.200 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
ICI Pharmaceuticals Group Curated by ChEMBL | Assay Description Inhibition constant for displacement of [3H]LTD4 on guinea pig lung parenchymal membranes. | J Med Chem 33: 1781-90 (1990) BindingDB Entry DOI: 10.7270/Q2862FDP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cysteinyl leukotriene receptor 1/2 (Homo sapiens (Human)) | BDBM50227361 (CHEMBL51585) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 0.25 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
ICI Pharmaceuticals Group Curated by ChEMBL | Assay Description Inhibition constant for displacement of [3H]LTD4 on guinea pig lung parenchymal membranes. | J Med Chem 33: 1781-90 (1990) BindingDB Entry DOI: 10.7270/Q2862FDP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cysteinyl leukotriene receptor 1/2 (Homo sapiens (Human)) | BDBM50227364 (CHEMBL299093) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 0.25 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
ICI Pharmaceuticals Group Curated by ChEMBL | Assay Description Inhibition constant for displacement of [3H]LTD4 on guinea pig lung parenchymal membranes. | J Med Chem 33: 1781-90 (1990) BindingDB Entry DOI: 10.7270/Q2862FDP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cysteinyl leukotriene receptor 1 (GUINEA PIG) | BDBM50009073 (4-(5-cyclopentyloxycarbonylamino-1-methyl-1H-indol...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG PC cid PC sid PDB UniChem Patents Similars | PDB PubMed | 0.300 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
ICI Pharmaceuticals Group Curated by ChEMBL | Assay Description Displacement of [3H]-LTD4 on guinea pig lung parenchymal membranes | J Med Chem 33: 1781-90 (1990) BindingDB Entry DOI: 10.7270/Q2862FDP | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Cysteinyl leukotriene receptor 1/2 (Homo sapiens (Human)) | BDBM50227365 (CHEMBL300096) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 0.300 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
ICI Pharmaceuticals Group Curated by ChEMBL | Assay Description Inhibition constant for displacement of [3H]LTD4 on guinea pig lung parenchymal membranes. | J Med Chem 33: 1781-90 (1990) BindingDB Entry DOI: 10.7270/Q2862FDP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-C chemokine receptor type 5 (Homo sapiens (Human)) | BDBM50124943 ((4-{(4-Bromo-phenyl)-[(Z)-ethoxyimino]-methyl}-4'-...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 0.300 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Schering-Plough Research Institute Curated by ChEMBL | Assay Description Inhibition of [125I]RANTES binding to CCR5 receptor. | Bioorg Med Chem Lett 13: 709-12 (2003) BindingDB Entry DOI: 10.7270/Q2VM4CTD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cysteinyl leukotriene receptor 1/2 (Homo sapiens (Human)) | BDBM50227358 (CHEMBL412056) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 0.300 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
ICI Pharmaceuticals Group Curated by ChEMBL | Assay Description Inhibition constant for displacement of [3H]LTD4 on guinea pig lung parenchymal membranes. | J Med Chem 33: 1781-90 (1990) BindingDB Entry DOI: 10.7270/Q2862FDP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cysteinyl leukotriene receptor 1/2 (Homo sapiens (Human)) | BDBM50227356 (CHEMBL49944) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 0.300 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
ICI Pharmaceuticals Group Curated by ChEMBL | Assay Description Inhibition constant for displacement of [3H]LTD4 on guinea pig lung parenchymal membranes. | J Med Chem 33: 1781-90 (1990) BindingDB Entry DOI: 10.7270/Q2862FDP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cysteinyl leukotriene receptor 1/2 (Homo sapiens (Human)) | BDBM50227355 (CHEMBL296821) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 0.300 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
ICI Pharmaceuticals Group Curated by ChEMBL | Assay Description Inhibition constant for displacement of [3H]LTD4 on guinea pig lung parenchymal membranes. | J Med Chem 33: 1781-90 (1990) BindingDB Entry DOI: 10.7270/Q2862FDP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cysteinyl leukotriene receptor 1/2 (Homo sapiens (Human)) | BDBM50227642 (CHEMBL50562) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 0.300 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
ICI Pharmaceuticals Group Curated by ChEMBL | Assay Description Inhibition constant for displacement of [3H]LTD4 on guinea pig lung parenchymal membranes. | J Med Chem 33: 1781-90 (1990) BindingDB Entry DOI: 10.7270/Q2862FDP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cysteinyl leukotriene receptor 1/2 (Homo sapiens (Human)) | BDBM50227640 (CHEMBL297952) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | 0.300 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
ICI Pharmaceuticals Group Curated by ChEMBL | Assay Description Inhibition constant for displacement of [3H]LTD4 on guinea pig lung parenchymal membranes. | J Med Chem 33: 1781-90 (1990) BindingDB Entry DOI: 10.7270/Q2862FDP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cysteinyl leukotriene receptor 1 (GUINEA PIG) | BDBM50015528 (CHEMBL50370 | N-[3-(4-Benzenesulfonylaminocarbonyl...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | 0.300 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
ICI Pharmaceuticals Group Curated by ChEMBL | Assay Description Displacement of [3H]-LTD4 on guinea pig lung parenchymal membranes | J Med Chem 33: 1781-90 (1990) BindingDB Entry DOI: 10.7270/Q2862FDP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-C chemokine receptor type 5 (Homo sapiens (Human)) | BDBM50124953 ((4-{(4-Bromo-phenyl)-[(Z)-ethoxyimino]-methyl}-4'-...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 0.400 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Schering-Plough Research Institute Curated by ChEMBL | Assay Description Inhibition of [125I]RANTES binding to CCR5 receptor. | Bioorg Med Chem Lett 13: 709-12 (2003) BindingDB Entry DOI: 10.7270/Q2VM4CTD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cysteinyl leukotriene receptor 1/2 (Homo sapiens (Human)) | BDBM50227390 (CHEMBL301616) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | PubMed | 0.5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
ICI Pharmaceuticals Group Curated by ChEMBL | Assay Description Inhibition constant for displacement of [3H]LTD4 on guinea pig lung parenchymal membranes. | J Med Chem 33: 1781-90 (1990) BindingDB Entry DOI: 10.7270/Q2862FDP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cysteinyl leukotriene receptor 1 (GUINEA PIG) | BDBM50015523 (CHEMBL52492 | N-{4-[5-(3-Cyclopentyl-ureido)-1-pro...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 0.5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
ICI Pharmaceuticals Group Curated by ChEMBL | Assay Description Displacement of [3H]-LTD4 on guinea pig lung parenchymal membranes | J Med Chem 33: 1781-90 (1990) BindingDB Entry DOI: 10.7270/Q2862FDP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cysteinyl leukotriene receptor 1 (GUINEA PIG) | BDBM50000819 (2-Cyclopentyl-N-{3-[2-methoxy-4-(toluene-2-sulfony...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | 0.5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
ICI Pharmaceuticals Group Curated by ChEMBL | Assay Description Displacement of [3H]-LTD4 on guinea pig lung parenchymal membranes | J Med Chem 33: 1781-90 (1990) BindingDB Entry DOI: 10.7270/Q2862FDP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cysteinyl leukotriene receptor 1/2 (Homo sapiens (Human)) | BDBM50227389 (CHEMBL51580) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 0.700 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
ICI Pharmaceuticals Group Curated by ChEMBL | Assay Description Inhibition constant for displacement of [3H]LTD4 on guinea pig lung parenchymal membranes. | J Med Chem 33: 1781-90 (1990) BindingDB Entry DOI: 10.7270/Q2862FDP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-C chemokine receptor type 5 (Homo sapiens (Human)) | BDBM50124957 ((4-{(4-Bromo-phenyl)-[(Z)-ethoxyimino]-methyl}-4'-...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 0.700 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Schering-Plough Research Institute Curated by ChEMBL | Assay Description Inhibition of [125I]RANTES binding to CCR5 receptor. | Bioorg Med Chem Lett 13: 709-12 (2003) BindingDB Entry DOI: 10.7270/Q2VM4CTD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cysteinyl leukotriene receptor 1 (GUINEA PIG) | BDBM50015551 (CHEMBL301498 | N-{4-[5-(3-Cyclopentyl-ureido)-1-me...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 0.800 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
ICI Pharmaceuticals Group Curated by ChEMBL | Assay Description Displacement of [3H]-LTD4 on guinea pig lung parenchymal membranes | J Med Chem 33: 1781-90 (1990) BindingDB Entry DOI: 10.7270/Q2862FDP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cysteinyl leukotriene receptor 1/2 (Homo sapiens (Human)) | BDBM50227367 (CHEMBL48435) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 0.800 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
ICI Pharmaceuticals Group Curated by ChEMBL | Assay Description Inhibition constant for displacement of [3H]LTD4 on guinea pig lung parenchymal membranes. | J Med Chem 33: 1781-90 (1990) BindingDB Entry DOI: 10.7270/Q2862FDP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cysteinyl leukotriene receptor 1 (GUINEA PIG) | BDBM50015517 (2-Cyclopentyl-N-{3-[2-methoxy-4-(toluene-2-sulfony...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | 1 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
ICI Pharmaceuticals Group Curated by ChEMBL | Assay Description Displacement of [3H]-LTD4 on guinea pig lung parenchymal membranes | J Med Chem 33: 1781-90 (1990) BindingDB Entry DOI: 10.7270/Q2862FDP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-C chemokine receptor type 5 (Homo sapiens (Human)) | BDBM50104942 ((4-Fluoro-naphthalen-1-yl)-{4-[4-(4-methoxy-benzen...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents | PubMed | 1 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Schering-Plough Research Institute Curated by ChEMBL | Assay Description Inhibition of RANTES binding to C-C chemokine receptor type 5 | J Med Chem 44: 3339-42 (2001) BindingDB Entry DOI: 10.7270/Q27M0771 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-C chemokine receptor type 5 (Homo sapiens (Human)) | BDBM50104933 (CHEMBL105821 | {4-[(4-Bromo-phenyl)-ethoxyimino-me...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 1.10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Schering-Plough Research Institute Curated by ChEMBL | Assay Description Inhibition of RANTES binding to C-C chemokine receptor type 5 | J Med Chem 44: 3339-42 (2001) BindingDB Entry DOI: 10.7270/Q27M0771 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-C chemokine receptor type 5 (Mus musculus) | BDBM50104933 (CHEMBL105821 | {4-[(4-Bromo-phenyl)-ethoxyimino-me...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 1.10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Schering-Plough Research Institute Curated by ChEMBL | Assay Description Inhibition of RANTES binding to Chemokine receptor type 5 receptor from NIH 3T3 cells | J Med Chem 45: 3143-60 (2002) BindingDB Entry DOI: 10.7270/Q2HD7TZJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-C chemokine receptor type 5 (Mus musculus) | BDBM50104940 (CHEMBL323172 | {4-[(4-Bromo-phenyl)-methoxyimino-m...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 1.10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Schering-Plough Research Institute Curated by ChEMBL | Assay Description Inhibition of RANTES binding to Chemokine receptor type 5 receptor from NIH 3T3 cells | J Med Chem 45: 3143-60 (2002) BindingDB Entry DOI: 10.7270/Q2HD7TZJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-C chemokine receptor type 5 (Homo sapiens (Human)) | BDBM50104940 (CHEMBL323172 | {4-[(4-Bromo-phenyl)-methoxyimino-m...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 1.10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Schering-Plough Research Institute Curated by ChEMBL | Assay Description Inhibition of RANTES binding to C-C chemokine receptor type 5 | J Med Chem 44: 3339-42 (2001) BindingDB Entry DOI: 10.7270/Q27M0771 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-C chemokine receptor type 5 (Homo sapiens (Human)) | BDBM50124946 ((4-{(4-Bromo-phenyl)-[(Z)-ethoxyimino]-methyl}-4'-...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 1.20 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Schering-Plough Research Institute Curated by ChEMBL | Assay Description Inhibition of [125I]RANTES binding to CCR5 receptor. | Bioorg Med Chem Lett 13: 709-12 (2003) BindingDB Entry DOI: 10.7270/Q2VM4CTD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-C chemokine receptor type 5 (Homo sapiens (Human)) | BDBM50124956 ((4-{(4-Bromo-phenyl)-[(E)-ethoxyimino]-methyl}-4'-...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 1.30 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Schering-Plough Research Institute Curated by ChEMBL | Assay Description Inhibition of [125I]RANTES binding to CCR5 receptor. | Bioorg Med Chem Lett 13: 709-12 (2003) BindingDB Entry DOI: 10.7270/Q2VM4CTD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Muscarinic acetylcholine receptor M2 (Homo sapiens (Human)) | BDBM50104942 ((4-Fluoro-naphthalen-1-yl)-{4-[4-(4-methoxy-benzen...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents | PubMed | 1.30 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Schering-Plough Research Institute Curated by ChEMBL | Assay Description Inhibitory activity against Muscarinic acetylcholine receptor M2 | J Med Chem 45: 3143-60 (2002) BindingDB Entry DOI: 10.7270/Q2HD7TZJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cysteinyl leukotriene receptor 1 (GUINEA PIG) | BDBM50015540 (CHEMBL431348 | N-{4-[5-(3-Cyclopentyl-ureido)-1-me...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | 1.40 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
ICI Pharmaceuticals Group Curated by ChEMBL | Assay Description Displacement of [3H]-LTD4 on guinea pig lung parenchymal membranes | J Med Chem 33: 1781-90 (1990) BindingDB Entry DOI: 10.7270/Q2862FDP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cysteinyl leukotriene receptor 1/2 (Homo sapiens (Human)) | BDBM50227638 (CHEMBL49566) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | 1.40 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
ICI Pharmaceuticals Group Curated by ChEMBL | Assay Description Inhibition constant for displacement of [3H]LTD4 on guinea pig lung parenchymal membranes. | J Med Chem 33: 1781-90 (1990) BindingDB Entry DOI: 10.7270/Q2862FDP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanin-concentrating hormone receptor 1 (Homo sapiens (Human)) | BDBM50170625 (3-(3-Chloro-4-fluoro-phenyl)-1-(3'-cyano-biphenyl-...) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 1.60 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Schering-Plough Research Institute Curated by ChEMBL | Assay Description Inhibition of human melanin concentrating hormone receptor 1 | J Med Chem 48: 4746-9 (2005) Article DOI: 10.1021/jm0503852 BindingDB Entry DOI: 10.7270/Q2P55N26 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanin-concentrating hormone receptor 1 (Homo sapiens (Human)) | BDBM50184944 (CHEMBL382668 | N-[trans-5-(3-cyanophenyl)bicyclo[3...) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 1.60 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Schering-Plough Research Institute Curated by ChEMBL | Assay Description Displacement of [125I]MCH from human MCHR1 expressed in CHO cell | J Med Chem 49: 2294-310 (2006) Article DOI: 10.1021/jm050886n BindingDB Entry DOI: 10.7270/Q2HQ3ZGH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanin-concentrating hormone receptor 1 (Homo sapiens (Human)) | BDBM50164243 ((R)-1-(3'-cyanobiphenyl-4-yl)-3-(4-fluoro-3-(trifl...) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 1.80 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Schering-Plough Research Institute Curated by ChEMBL | Assay Description Inhibition of human melanin concentrating hormone receptor 1 | J Med Chem 48: 4746-9 (2005) Article DOI: 10.1021/jm0503852 BindingDB Entry DOI: 10.7270/Q2P55N26 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanin-concentrating hormone receptor 1 (Homo sapiens (Human)) | BDBM50184925 (CHEMBL380509 | N-[trans-5-(4-fluorophenyl)bicyclo[...) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.80 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Schering-Plough Research Institute Curated by ChEMBL | Assay Description Displacement of [125I]MCH from human MCHR1 expressed in CHO cell | J Med Chem 49: 2294-310 (2006) Article DOI: 10.1021/jm050886n BindingDB Entry DOI: 10.7270/Q2HQ3ZGH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-C chemokine receptor type 5 (Homo sapiens (Human)) | BDBM50115528 ((Z)-(4-((4-bromophenyl)(ethoxyimino)methyl)-4'-met...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 1.80 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Schering-Plough Research Institute Curated by ChEMBL | Assay Description Inhibition of RANTES binding to C-C chemokine receptor type 5 | J Med Chem 44: 3339-42 (2001) BindingDB Entry DOI: 10.7270/Q27M0771 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanin-concentrating hormone receptor 1 (Homo sapiens (Human)) | BDBM50170614 (1-(3'-Cyano-biphenyl-4-yl)-1-(1-cyclopentyl-piperi...) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 1.90 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Schering-Plough Research Institute Curated by ChEMBL | Assay Description Inhibition of human melanin concentrating hormone receptor 1 | J Med Chem 48: 4746-9 (2005) Article DOI: 10.1021/jm0503852 BindingDB Entry DOI: 10.7270/Q2P55N26 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-C chemokine receptor type 5 (Homo sapiens (Human)) | BDBM50124958 ((4-{(4-Bromo-phenyl)-[(E)-propoxyimino]-methyl}-4'...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 2 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Schering-Plough Research Institute Curated by ChEMBL | Assay Description Inhibition of [125I]RANTES binding to CCR5 receptor. | Bioorg Med Chem Lett 13: 709-12 (2003) BindingDB Entry DOI: 10.7270/Q2VM4CTD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-C chemokine receptor type 5 (Mus musculus) | BDBM50115512 (CHEMBL324671 | {4-[(4-Bromo-phenyl)-methoxyimino-m...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | 2 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Schering-Plough Research Institute Curated by ChEMBL | Assay Description Inhibition of RANTES binding to Chemokine receptor type 5 receptor from NIH 3T3 cells | J Med Chem 45: 3143-60 (2002) BindingDB Entry DOI: 10.7270/Q2HD7TZJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-C chemokine receptor type 5 (Mus musculus) | BDBM50115528 ((Z)-(4-((4-bromophenyl)(ethoxyimino)methyl)-4'-met...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 2 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Schering-Plough Research Institute Curated by ChEMBL | Assay Description Inhibition of RANTES binding to Chemokine receptor type 5 receptor from NIH 3T3 cells | J Med Chem 45: 3143-60 (2002) BindingDB Entry DOI: 10.7270/Q2HD7TZJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-C chemokine receptor type 5 (Homo sapiens (Human)) | BDBM50104930 ((Z)-{4-[(4-Bromo-phenyl)-methoxyimino-methyl]-[1,4...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 2 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Schering-Plough Research Institute Curated by ChEMBL | Assay Description Inhibition of RANTES binding to C-C chemokine receptor type 5 | J Med Chem 44: 3339-42 (2001) BindingDB Entry DOI: 10.7270/Q27M0771 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanin-concentrating hormone receptor 1 (Homo sapiens (Human)) | BDBM50184935 (3-(3-chloro-4-fluorophenyl)-1-(3-(4-methylpiperazi...) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Schering-Plough Research Institute Curated by ChEMBL | Assay Description Binding affinity to MCHR1 | Bioorg Med Chem Lett 16: 4262-5 (2006) Article DOI: 10.1016/j.bmcl.2006.05.069 BindingDB Entry DOI: 10.7270/Q2BC3Z5G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanin-concentrating hormone receptor 1 (Homo sapiens (Human)) | BDBM50184935 (3-(3-chloro-4-fluorophenyl)-1-(3-(4-methylpiperazi...) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Schering-Plough Research Institute Curated by ChEMBL | Assay Description Displacement of [125I]MCH from human MCHR1 expressed in CHO cell | J Med Chem 49: 2294-310 (2006) Article DOI: 10.1021/jm050886n BindingDB Entry DOI: 10.7270/Q2HQ3ZGH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-C chemokine receptor type 5 (Homo sapiens (Human)) | BDBM50145685 ((4,6-Dimethyl-pyrimidin-5-yl)-(4-{(S)-4-[(R)-2-met...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | PubMed | 2.10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Schering-Plough Research Institute Curated by ChEMBL | Assay Description Inhibition of [125I]RANTES binding to CCR5 receptor. | Bioorg Med Chem Lett 13: 709-12 (2003) BindingDB Entry DOI: 10.7270/Q2VM4CTD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-C chemokine receptor type 5 (Homo sapiens (Human)) | BDBM50104931 ((4-{(4-Bromo-phenyl)-[(E)-ethoxyimino]-methyl}-4''...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | 2.10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Schering-Plough Research Institute Curated by ChEMBL | Assay Description Inhibition of RANTES binding to C-C chemokine receptor type 5 | J Med Chem 44: 3339-42 (2001) BindingDB Entry DOI: 10.7270/Q27M0771 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-C chemokine receptor type 5 (Mus musculus) | BDBM50104931 ((4-{(4-Bromo-phenyl)-[(E)-ethoxyimino]-methyl}-4''...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | 2.10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Schering-Plough Research Institute Curated by ChEMBL | Assay Description Inhibition of RANTES binding to Chemokine receptor type 5 receptor from NIH 3T3 cells | J Med Chem 45: 3143-60 (2002) BindingDB Entry DOI: 10.7270/Q2HD7TZJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-C chemokine receptor type 5 (Homo sapiens (Human)) | BDBM50124951 ((4-{(4-Bromo-phenyl)-[(E)-ethoxyimino]-methyl}-4'-...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 2.10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Schering-Plough Research Institute Curated by ChEMBL | Assay Description Inhibition of [125I]RANTES binding to CCR5 receptor. | Bioorg Med Chem Lett 13: 709-12 (2003) BindingDB Entry DOI: 10.7270/Q2VM4CTD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanin-concentrating hormone receptor 1 (Homo sapiens (Human)) | BDBM50184928 (CHEMBL382140 | N-[trans-5-(3-cyanophenyl)bicyclo[3...) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 2.20 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Schering-Plough Research Institute Curated by ChEMBL | Assay Description Displacement of [125I]MCH from human MCHR1 expressed in CHO cell | J Med Chem 49: 2294-310 (2006) Article DOI: 10.1021/jm050886n BindingDB Entry DOI: 10.7270/Q2HQ3ZGH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-C chemokine receptor type 5 (Homo sapiens (Human)) | BDBM50124948 ((4-{(4-Bromo-phenyl)-[(Z)-ethoxyimino]-methyl}-4'-...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | 2.20 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Schering-Plough Research Institute Curated by ChEMBL | Assay Description Inhibition of [125I]RANTES binding to CCR5 receptor. | Bioorg Med Chem Lett 13: 709-12 (2003) BindingDB Entry DOI: 10.7270/Q2VM4CTD | |||||||||||
More data for this Ligand-Target Pair |
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