Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
D(2) dopamine receptor (Rattus norvegicus (rat)) | BDBM50001888 ((chloropromazine) [3-(2-Chloro-phenothiazin-10-yl)...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG MMDB PC cid PC sid PDB UniChem Patents Similars | PubMed | 1.20 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Compound was tested for inhibitory activity against the binding of [3H]-spiperone to Dopamine receptor D2 in rat striatal membranes | J Med Chem 30: 1631-5 (1987) BindingDB Entry DOI: 10.7270/Q2FB51ZZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(2) dopamine receptor (Mus musculus (Mouse)) | BDBM50016778 (1-Ethyl-2-[(2-methoxy-5-sulfamoyl-benzoylamino)-me...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | PubMed | 5.20 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Ohio State University Curated by ChEMBL | Assay Description Compound was tested for its ability to displace [3H]- spiperone from D2 binding site in rat striatal membranes | J Med Chem 32: 874-80 (1989) BindingDB Entry DOI: 10.7270/Q23B5Z48 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(2) dopamine receptor (Rattus norvegicus (rat)) | BDBM11638 (CHEMBL26 | Compound 7 | N-[(1-ethylpyrrolidin-2-yl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE PC cid PC sid UniChem Patents Similars | PubMed | 5.5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Ohio State University Curated by ChEMBL | Assay Description Compound was tested for its ability to displace [3H]- spiperone from Dopamine receptor D2 in rat striatal membranes | J Med Chem 32: 874-80 (1989) BindingDB Entry DOI: 10.7270/Q23B5Z48 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(2) dopamine receptor (Rattus norvegicus (rat)) | BDBM50019878 (CHEMBL44394 | [3-(2-Chloro-phenothiazin-10-yl)-pro...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 280 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Compound was tested for inhibitory activity against the binding of [3H]-spiperone toDopamine receptor D2 in rat striatal membranes | J Med Chem 30: 1631-5 (1987) BindingDB Entry DOI: 10.7270/Q2FB51ZZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(2) dopamine receptor (Rattus norvegicus (rat)) | BDBM50019879 (CHEMBL279905 | [3-(2-Chloro-phenothiazin-10-yl)-pr...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | PubMed | 2.15E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Compound was tested for inhibitory activity against the binding of [3H]-spiperone to Dopamine receptor D2 in rat striatal membranes | J Med Chem 30: 1631-5 (1987) BindingDB Entry DOI: 10.7270/Q2FB51ZZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human)) | BDBM50213092 ((1R,2R)-1-(1-naphthalenethoxy)-2-(4-morpholinyl)cy...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Cardiome Pharma Corporation Curated by ChEMBL | Assay Description Inhibition of human potassium channel Kv1.5 by patch-clamp method | J Med Chem 50: 2818-41 (2007) Article DOI: 10.1021/jm0604528 BindingDB Entry DOI: 10.7270/Q29Z95QZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily D member 2 (Rattus norvegicus) | BDBM50121975 ((6-Methoxy-quinolin-4-yl)-(5-vinyl-1-aza-bicyclo[2...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG PC cid PC sid PDB UniChem Patents Similars | Article PubMed | n/a | n/a | 2.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Cardiome Pharma Corporation Curated by ChEMBL | Assay Description Inhibition of rat potassium channel Kv4.2 by patch-clamp method | J Med Chem 50: 2818-41 (2007) Article DOI: 10.1021/jm0604528 BindingDB Entry DOI: 10.7270/Q29Z95QZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily B member 1 (Rattus norvegicus) | BDBM50213094 ((1R,2R)-1-(3,4-dichlorophenethoxy)-2-(4-morpholiny...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Cardiome Pharma Corporation Curated by ChEMBL | Assay Description Inhibition of rat potassium channel Kv2.1 by patch-clamp method | J Med Chem 50: 2818-41 (2007) Article DOI: 10.1021/jm0604528 BindingDB Entry DOI: 10.7270/Q29Z95QZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily B member 1 (Rattus norvegicus) | BDBM50213092 ((1R,2R)-1-(1-naphthalenethoxy)-2-(4-morpholinyl)cy...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Cardiome Pharma Corporation Curated by ChEMBL | Assay Description Inhibition of rat potassium channel Kv2.1 by patch-clamp method | J Med Chem 50: 2818-41 (2007) Article DOI: 10.1021/jm0604528 BindingDB Entry DOI: 10.7270/Q29Z95QZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human)) | BDBM50213094 ((1R,2R)-1-(3,4-dichlorophenethoxy)-2-(4-morpholiny...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.60E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Cardiome Pharma Corporation Curated by ChEMBL | Assay Description Inhibition of human potassium channel Kv1.5 by patch-clamp method | J Med Chem 50: 2818-41 (2007) Article DOI: 10.1021/jm0604528 BindingDB Entry DOI: 10.7270/Q29Z95QZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium channel protein type 5 subunit alpha (Homo sapiens (Human)) | BDBM50213092 ((1R,2R)-1-(1-naphthalenethoxy)-2-(4-morpholinyl)cy...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 4.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Cardiome Pharma Corporation Curated by ChEMBL | Assay Description Inhibition of human heart sodium channel Nav1.5 by patch-clamp method | J Med Chem 50: 2818-41 (2007) Article DOI: 10.1021/jm0604528 BindingDB Entry DOI: 10.7270/Q29Z95QZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human)) | BDBM50213093 ((1R,2R)-1-(1-naphthalenethoxy)-2-(3-ketopyrrolidin...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 5.90E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Cardiome Pharma Corporation Curated by ChEMBL | Assay Description Inhibition of human potassium channel Kv1.5 by patch-clamp method | J Med Chem 50: 2818-41 (2007) Article DOI: 10.1021/jm0604528 BindingDB Entry DOI: 10.7270/Q29Z95QZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human)) | BDBM50213093 ((1R,2R)-1-(1-naphthalenethoxy)-2-(3-ketopyrrolidin...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 5.90E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Cardiome Pharma Corporation Curated by ChEMBL | Assay Description Inhibition of human potassium channel Kv1.5 by patch-clamp method | J Med Chem 50: 2818-41 (2007) Article DOI: 10.1021/jm0604528 BindingDB Entry DOI: 10.7270/Q29Z95QZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily B member 1 (Rattus norvegicus) | BDBM50213093 ((1R,2R)-1-(1-naphthalenethoxy)-2-(3-ketopyrrolidin...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 6.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Cardiome Pharma Corporation Curated by ChEMBL | Assay Description Inhibition of rat potassium channel Kv2.1 by patch-clamp method | J Med Chem 50: 2818-41 (2007) Article DOI: 10.1021/jm0604528 BindingDB Entry DOI: 10.7270/Q29Z95QZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily B member 1 (Rattus norvegicus) | BDBM50213093 ((1R,2R)-1-(1-naphthalenethoxy)-2-(3-ketopyrrolidin...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 6.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Cardiome Pharma Corporation Curated by ChEMBL | Assay Description Inhibition of rat potassium channel Kv2.1 by patch-clamp method | J Med Chem 50: 2818-41 (2007) Article DOI: 10.1021/jm0604528 BindingDB Entry DOI: 10.7270/Q29Z95QZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium channel protein type 5 subunit alpha (Homo sapiens (Human)) | BDBM50131434 (CHEMBL652 | FLECAINIDE | N-(piperidin-2-ylmethyl)-...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG PC cid PC sid PDB UniChem Patents Similars | DrugBank Article PubMed | n/a | n/a | 6.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Cardiome Pharma Corporation Curated by ChEMBL | Assay Description Inhibition of human heart sodium channel Nav1.5 by patch-clamp method | J Med Chem 50: 2818-41 (2007) Article DOI: 10.1021/jm0604528 BindingDB Entry DOI: 10.7270/Q29Z95QZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human)) | BDBM50213095 ((1S,2S)-1-(1-Naphthalenethoxy)-2-(3-ketopyrrolidin...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 7.70E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Cardiome Pharma Corporation Curated by ChEMBL | Assay Description Inhibition of human potassium channel Kv1.5 by patch-clamp method | J Med Chem 50: 2818-41 (2007) Article DOI: 10.1021/jm0604528 BindingDB Entry DOI: 10.7270/Q29Z95QZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily B member 1 (Rattus norvegicus) | BDBM50213095 ((1S,2S)-1-(1-Naphthalenethoxy)-2-(3-ketopyrrolidin...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 8.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Cardiome Pharma Corporation Curated by ChEMBL | Assay Description Inhibition of rat potassium channel Kv2.1 by patch-clamp method | J Med Chem 50: 2818-41 (2007) Article DOI: 10.1021/jm0604528 BindingDB Entry DOI: 10.7270/Q29Z95QZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily D member 2 (Rattus norvegicus) | BDBM50213095 ((1S,2S)-1-(1-Naphthalenethoxy)-2-(3-ketopyrrolidin...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 9.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Cardiome Pharma Corporation Curated by ChEMBL | Assay Description Inhibition of rat potassium channel Kv4.2 by patch-clamp method | J Med Chem 50: 2818-41 (2007) Article DOI: 10.1021/jm0604528 BindingDB Entry DOI: 10.7270/Q29Z95QZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily D member 2 (Rattus norvegicus) | BDBM50131434 (CHEMBL652 | FLECAINIDE | N-(piperidin-2-ylmethyl)-...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG PC cid PC sid PDB UniChem Patents Similars | Article PubMed | n/a | n/a | 1.01E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Cardiome Pharma Corporation Curated by ChEMBL | Assay Description Inhibition of rat potassium channel Kv4.2 by patch-clamp method | J Med Chem 50: 2818-41 (2007) Article DOI: 10.1021/jm0604528 BindingDB Entry DOI: 10.7270/Q29Z95QZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium channel protein type 5 subunit alpha (Homo sapiens (Human)) | BDBM50213093 ((1R,2R)-1-(1-naphthalenethoxy)-2-(3-ketopyrrolidin...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.10E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Cardiome Pharma Corporation Curated by ChEMBL | Assay Description Inhibition of human heart sodium channel Nav1.5 by patch-clamp method | J Med Chem 50: 2818-41 (2007) Article DOI: 10.1021/jm0604528 BindingDB Entry DOI: 10.7270/Q29Z95QZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily D member 2 (Rattus norvegicus) | BDBM50213093 ((1R,2R)-1-(1-naphthalenethoxy)-2-(3-ketopyrrolidin...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.10E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Cardiome Pharma Corporation Curated by ChEMBL | Assay Description Inhibition of rat potassium channel Kv4.2 by patch-clamp method | J Med Chem 50: 2818-41 (2007) Article DOI: 10.1021/jm0604528 BindingDB Entry DOI: 10.7270/Q29Z95QZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily D member 2 (Rattus norvegicus) | BDBM50213093 ((1R,2R)-1-(1-naphthalenethoxy)-2-(3-ketopyrrolidin...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.10E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Cardiome Pharma Corporation Curated by ChEMBL | Assay Description Inhibition of rat potassium channel Kv4.2 by patch-clamp method | J Med Chem 50: 2818-41 (2007) Article DOI: 10.1021/jm0604528 BindingDB Entry DOI: 10.7270/Q29Z95QZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium channel protein type 5 subunit alpha (Homo sapiens (Human)) | BDBM50213093 ((1R,2R)-1-(1-naphthalenethoxy)-2-(3-ketopyrrolidin...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.10E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Cardiome Pharma Corporation Curated by ChEMBL | Assay Description Inhibition of human heart sodium channel Nav1.5 by patch-clamp method | J Med Chem 50: 2818-41 (2007) Article DOI: 10.1021/jm0604528 BindingDB Entry DOI: 10.7270/Q29Z95QZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily D member 2 (Rattus norvegicus) | BDBM50213094 ((1R,2R)-1-(3,4-dichlorophenethoxy)-2-(4-morpholiny...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.10E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Cardiome Pharma Corporation Curated by ChEMBL | Assay Description Inhibition of rat potassium channel Kv4.2 by patch-clamp method | J Med Chem 50: 2818-41 (2007) Article DOI: 10.1021/jm0604528 BindingDB Entry DOI: 10.7270/Q29Z95QZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium channel protein type 5 subunit alpha (Homo sapiens (Human)) | BDBM50213095 ((1S,2S)-1-(1-Naphthalenethoxy)-2-(3-ketopyrrolidin...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.30E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Cardiome Pharma Corporation Curated by ChEMBL | Assay Description Inhibition of human heart sodium channel Nav1.5 by patch-clamp method | J Med Chem 50: 2818-41 (2007) Article DOI: 10.1021/jm0604528 BindingDB Entry DOI: 10.7270/Q29Z95QZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium channel protein type 5 subunit alpha (Homo sapiens (Human)) | BDBM50213094 ((1R,2R)-1-(3,4-dichlorophenethoxy)-2-(4-morpholiny...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.50E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Cardiome Pharma Corporation Curated by ChEMBL | Assay Description Inhibition of human heart sodium channel Nav1.5 by patch-clamp method | J Med Chem 50: 2818-41 (2007) Article DOI: 10.1021/jm0604528 BindingDB Entry DOI: 10.7270/Q29Z95QZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily D member 2 (Rattus norvegicus) | BDBM50213092 ((1R,2R)-1-(1-naphthalenethoxy)-2-(4-morpholinyl)cy...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.70E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Cardiome Pharma Corporation Curated by ChEMBL | Assay Description Inhibition of rat potassium channel Kv4.2 by patch-clamp method | J Med Chem 50: 2818-41 (2007) Article DOI: 10.1021/jm0604528 BindingDB Entry DOI: 10.7270/Q29Z95QZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human)) | BDBM50131434 (CHEMBL652 | FLECAINIDE | N-(piperidin-2-ylmethyl)-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG PC cid PC sid PDB UniChem Patents Similars | Article PubMed | n/a | n/a | 5.10E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Cardiome Pharma Corporation Curated by ChEMBL | Assay Description Inhibition of human potassium channel Kv1.5 by patch-clamp method | J Med Chem 50: 2818-41 (2007) Article DOI: 10.1021/jm0604528 BindingDB Entry DOI: 10.7270/Q29Z95QZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium channel protein type 5 subunit alpha (Homo sapiens (Human)) | BDBM50017662 (2-(Diethylamino)-2',6'-acetoxylidide | 2-(Diethyla...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG MMDB PC cid PC sid PDB UniChem Patents Similars | DrugBank Article PubMed | n/a | n/a | 1.08E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Cardiome Pharma Corporation Curated by ChEMBL | Assay Description Inhibition of human heart sodium channel Nav1.5 by patch-clamp method | J Med Chem 50: 2818-41 (2007) Article DOI: 10.1021/jm0604528 BindingDB Entry DOI: 10.7270/Q29Z95QZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily D member 2 (Rattus norvegicus) | BDBM50017662 (2-(Diethylamino)-2',6'-acetoxylidide | 2-(Diethyla...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG MMDB PC cid PC sid PDB UniChem Patents Similars | Article PubMed | n/a | n/a | 1.21E+6 | n/a | n/a | n/a | n/a | n/a | n/a |
Cardiome Pharma Corporation Curated by ChEMBL | Assay Description Inhibition of rat potassium channel Kv4.2 by patch-clamp method | J Med Chem 50: 2818-41 (2007) Article DOI: 10.1021/jm0604528 BindingDB Entry DOI: 10.7270/Q29Z95QZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human)) | BDBM50017662 (2-(Diethylamino)-2',6'-acetoxylidide | 2-(Diethyla...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG MMDB PC cid PC sid PDB UniChem Patents Similars | Article PubMed | n/a | n/a | 2.19E+6 | n/a | n/a | n/a | n/a | n/a | n/a |
Cardiome Pharma Corporation Curated by ChEMBL | Assay Description Inhibition of human potassium channel Kv1.5 by patch-clamp method | J Med Chem 50: 2818-41 (2007) Article DOI: 10.1021/jm0604528 BindingDB Entry DOI: 10.7270/Q29Z95QZ | |||||||||||
More data for this Ligand-Target Pair |