Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Neuropeptide Y receptor type 5 (Homo sapiens (Human)) | BDBM50258001 (CHEMBL492370 | N-(3,4-dichlorophenyl)-1-(methylsul...) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 0.200 | n/a | n/a | n/a | n/a | n/a | n/a |
Tsukuba Research Institute Curated by ChEMBL | Assay Description Displacement of [125I]PYY from human recombinant Y5 receptor expressed in mouse LMtk cells | Bioorg Med Chem Lett 19: 1564-8 (2009) Article DOI: 10.1016/j.bmcl.2009.02.035 BindingDB Entry DOI: 10.7270/Q2TQ61FT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 5 (Homo sapiens (Human)) | BDBM50093652 (2-Methyl-6-pentyl-4-piperidin-1-yl-5H-pyrrolo[3,2-...) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 0.200 | n/a | n/a | n/a | n/a | n/a | n/a |
Amgen, Inc. Curated by ChEMBL | Assay Description Affinity for human neuropeptide Y receptor Y5, binding was evaluated in an in vitro radioligand [125I]-PYY binding assay | J Med Chem 43: 4288-312 (2000) BindingDB Entry DOI: 10.7270/Q2C828J1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 5 (Homo sapiens (Human)) | BDBM50111656 (1-[2-(5-Chloro-2-oxo-benzothiazol-3-yl)-acetyl]-pi...) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 0.230 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co., Ltd. Curated by ChEMBL | Assay Description Tested for the inhibition of [125I]-PYY binding to HEK 293 cells stably expressed with human neuropeptide NPY Y5 receptor | Bioorg Med Chem Lett 12: 1171-5 (2002) BindingDB Entry DOI: 10.7270/Q26M365J | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 5 (Homo sapiens (Human)) | BDBM50093696 (6-(3-Fluoro-phenyl)-2-methyl-4-piperidin-1-yl-5H-p...) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 0.300 | n/a | n/a | n/a | n/a | n/a | n/a |
Amgen, Inc. Curated by ChEMBL | Assay Description Affinity for human neuropeptide Y receptor Y5, binding was evaluated in an in vitro radioligand [125I]-PYY binding assay | J Med Chem 43: 4288-312 (2000) BindingDB Entry DOI: 10.7270/Q2C828J1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 5 (Homo sapiens (Human)) | BDBM50093664 (6-(4-Fluoro-phenyl)-2-methyl-4-piperidin-1-yl-5H-p...) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 0.300 | n/a | n/a | n/a | n/a | n/a | n/a |
Amgen, Inc. Curated by ChEMBL | Assay Description Affinity for human neuropeptide Y receptor Y5, binding was evaluated in an in vitro radioligand [125I]-PYY binding assay | J Med Chem 43: 4288-312 (2000) BindingDB Entry DOI: 10.7270/Q2C828J1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 5 (Homo sapiens (Human)) | BDBM50093646 (6-Benzofuran-2-yl-2-methyl-4-piperidin-1-yl-5H-pyr...) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 0.300 | n/a | n/a | n/a | n/a | n/a | n/a |
Amgen, Inc. Curated by ChEMBL | Assay Description Affinity for human neuropeptide Y receptor Y5, binding was evaluated in an in vitro radioligand [125I]-PYY binding assay | J Med Chem 43: 4288-312 (2000) BindingDB Entry DOI: 10.7270/Q2C828J1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 5 (Homo sapiens (Human)) | BDBM50093691 (4-(3,6-Dihydro-2H-pyridin-1-yl)-2-methyl-6-phenyl-...) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 0.400 | n/a | n/a | n/a | n/a | n/a | n/a |
Amgen, Inc. Curated by ChEMBL | Assay Description Affinity for human neuropeptide Y receptor Y5, binding was evaluated in an in vitro radioligand [125I]-PYY binding assay | J Med Chem 43: 4288-312 (2000) BindingDB Entry DOI: 10.7270/Q2C828J1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 5 (Homo sapiens (Human)) | BDBM50093675 (6-(3,5-Difluoro-phenyl)-2-methyl-4-piperidin-1-yl-...) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 0.400 | n/a | n/a | n/a | n/a | n/a | n/a |
Amgen, Inc. Curated by ChEMBL | Assay Description Affinity for human neuropeptide Y receptor Y5, binding was evaluated in an in vitro radioligand [125I]-PYY binding assay | J Med Chem 43: 4288-312 (2000) BindingDB Entry DOI: 10.7270/Q2C828J1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 5 (Homo sapiens (Human)) | BDBM50073048 (2-[4-(2-Oxo-2,3-dihydro-benzoimidazol-1-yl)-piperi...) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents | Article PubMed | n/a | n/a | 0.470 | n/a | n/a | n/a | n/a | n/a | n/a |
The R. W. Johnson Pharmaceutical Research Institute Curated by ChEMBL | Assay Description The compound was tested for the binding affinity against Neuropeptide Y receptor type 5 in rat | J Med Chem 42: 181-201 (1999) Article DOI: 10.1021/jm980521l BindingDB Entry DOI: 10.7270/Q2T43S8P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 5 (Homo sapiens (Human)) | BDBM50073048 (2-[4-(2-Oxo-2,3-dihydro-benzoimidazol-1-yl)-piperi...) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents | PubMed | n/a | n/a | 0.470 | n/a | n/a | n/a | n/a | n/a | n/a |
The R. W. Johnson Pharmaceutical Research Institute Curated by ChEMBL | Assay Description Binding affinity of the compound against human Neuropeptide Y receptor type 5 in HEK 293 cell line by using [125I]-PYY as radioligand | Bioorg Med Chem Lett 11: 2283-6 (2001) BindingDB Entry DOI: 10.7270/Q2NZ86WB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 5 (Homo sapiens (Human)) | BDBM50093647 (2-Methyl-6-(5-methyl-furan-2-yl)-4-piperidin-1-yl-...) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 0.5 | n/a | n/a | n/a | n/a | n/a | n/a |
Amgen, Inc. Curated by ChEMBL | Assay Description Affinity for human neuropeptide Y receptor Y5, binding was evaluated in an in vitro radioligand [125I]-PYY binding assay | J Med Chem 43: 4288-312 (2000) BindingDB Entry DOI: 10.7270/Q2C828J1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 5 (Homo sapiens (Human)) | BDBM50093697 (2-Methyl-4-piperidin-1-yl-6-p-tolyl-5H-pyrrolo[3,2...) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 0.5 | n/a | n/a | n/a | n/a | n/a | n/a |
Amgen, Inc. Curated by ChEMBL | Assay Description Affinity for human neuropeptide Y receptor Y5, binding was evaluated in an in vitro radioligand [125I]-PYY binding assay | J Med Chem 43: 4288-312 (2000) BindingDB Entry DOI: 10.7270/Q2C828J1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 5 (Homo sapiens (Human)) | BDBM50101571 (1-Methyl-1-(1-methyl-2-pyridin-4-yl-ethyl)-3-(4-ph...) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 0.5 | n/a | n/a | n/a | n/a | n/a | n/a |
Amgen Inc. Curated by ChEMBL | Assay Description Inhibitory activity tested against Human Neuropeptide Y5 Receptor. | J Med Chem 44: 2344-56 (2001) BindingDB Entry DOI: 10.7270/Q2DV1J56 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 5 (Homo sapiens (Human)) | BDBM50110571 (CHEMBL167991 | FR-230481 | Naphthalene-1-sulfonic ...) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 0.540 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co., Ltd. Curated by ChEMBL | Assay Description Inhibition of 125 I-PYY binding to human Neuropeptide Y receptor type 5 | Bioorg Med Chem Lett 12: 799-802 (2002) BindingDB Entry DOI: 10.7270/Q2M044R7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 5 (Homo sapiens (Human)) | BDBM50258232 (1-(Methylsulfonyl)-N-(5-phenylpyrimidin-2-yl)-1,2-...) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.570 | n/a | n/a | n/a | n/a | n/a | n/a |
Tsukuba Research Institute Curated by ChEMBL | Assay Description Displacement of [125I]PYY from human recombinant Y5 receptor expressed in mouse LMtk cells | Bioorg Med Chem Lett 19: 1564-8 (2009) Article DOI: 10.1016/j.bmcl.2009.02.035 BindingDB Entry DOI: 10.7270/Q2TQ61FT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 5 (Homo sapiens (Human)) | BDBM50258232 (1-(Methylsulfonyl)-N-(5-phenylpyrimidin-2-yl)-1,2-...) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.570 | n/a | n/a | n/a | n/a | n/a | n/a |
Tsukuba Research Institute Curated by ChEMBL | Assay Description Binding affinity to human neuropeptide Y5 receptor | Bioorg Med Chem 17: 5015-26 (2009) Article DOI: 10.1016/j.bmc.2009.05.064 BindingDB Entry DOI: 10.7270/Q2KK9BT2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 5 (Homo sapiens (Human)) | BDBM50111644 (1-[2-(5-Chloro-2-oxo-benzothiazol-3-yl)-acetyl]-pi...) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 0.590 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co., Ltd. Curated by ChEMBL | Assay Description Inhibitory concentration of total specific binding of [125I]- -PYY to HEK 293 cells transfected with the Human NPY-Y5 cDNA (compound prepared by para... | Bioorg Med Chem Lett 12: 1171-5 (2002) BindingDB Entry DOI: 10.7270/Q26M365J | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 5 (Homo sapiens (Human)) | BDBM50111645 (1-[2-(5-Chloro-2-oxo-benzothiazol-3-yl)-acetyl]-pi...) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 0.590 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co., Ltd. Curated by ChEMBL | Assay Description Inhibitory concentration of total specific binding of [125I]- -PYY to HEK 293 cells transfected with Human NPY-Y5 cDNA (compound prepared by manual s... | Bioorg Med Chem Lett 12: 1171-5 (2002) BindingDB Entry DOI: 10.7270/Q26M365J | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 5 (Homo sapiens (Human)) | BDBM50354066 (CHEMBL1836324) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 0.600 | n/a | n/a | n/a | n/a | n/a | n/a |
Lundbeck Research USA, Inc. Curated by ChEMBL | Assay Description Antagonist activity at human NPY5 receptor assessed as calcium mobilization by FLIPR assay | Bioorg Med Chem Lett 21: 5436-41 (2011) Article DOI: 10.1016/j.bmcl.2011.06.124 BindingDB Entry DOI: 10.7270/Q2RN387K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 5 (Homo sapiens (Human)) | BDBM50089055 (CHEMBL273811 | N*2*-(4-Ethanesulfonylmethyl-phenyl...) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 0.600 | n/a | n/a | n/a | n/a | n/a | n/a |
Novartis Pharma AG Curated by ChEMBL | Assay Description Antagonistic activity against neuropeptide Y receptor type 5 subtype stably expressed in LM(tk-)cells | Bioorg Med Chem Lett 10: 1175-9 (2000) BindingDB Entry DOI: 10.7270/Q2KH0MJP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 5 (Homo sapiens (Human)) | BDBM50301643 (CHEMBL570633 | trans-3'-oxo-N-(5-phenylpyrimidin-2...) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.640 | n/a | n/a | n/a | n/a | n/a | n/a |
Tsukuba Research Institute Curated by ChEMBL | Assay Description Displacement of [125I]PYY from human recombinant NPY Y5 receptor expressed in mouse LMtk cells | Bioorg Med Chem Lett 19: 5436-9 (2009) Article DOI: 10.1016/j.bmcl.2009.07.103 BindingDB Entry DOI: 10.7270/Q27D2V6Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 5 (Homo sapiens (Human)) | BDBM50298636 (1-(Methylsulfonyl)-N-[4-(phenylcarbonyl)phenyl]-1,...) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 0.680 | n/a | n/a | n/a | n/a | n/a | n/a |
Tsukuba Research Institute Curated by ChEMBL | Assay Description Binding affinity to human neuropeptide Y5 receptor | Bioorg Med Chem 17: 5015-26 (2009) Article DOI: 10.1016/j.bmc.2009.05.064 BindingDB Entry DOI: 10.7270/Q2KK9BT2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 5 (Homo sapiens (Human)) | BDBM50268739 (CHEMBL524085 | N-(3-(4-chlorophenyl)isoxazol-5-yl)...) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.690 | n/a | n/a | n/a | n/a | n/a | n/a |
Tsukuba Research Institute Curated by ChEMBL | Assay Description Displacement of [125I]PYY from human recombinant NPY Y5 receptor expressed in mouse LMtk- cells | Bioorg Med Chem Lett 19: 3511-6 (2009) Article DOI: 10.1016/j.bmcl.2009.05.013 BindingDB Entry DOI: 10.7270/Q21C1WS5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 5 (Homo sapiens (Human)) | BDBM50111645 (1-[2-(5-Chloro-2-oxo-benzothiazol-3-yl)-acetyl]-pi...) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 0.700 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co., Ltd. Curated by ChEMBL | Assay Description Inhibitory concentration of total specific binding of [125I]- -PYY to HEK 293 cells transfected with the Human NPY-Y5 cDNA (compound prepared by para... | Bioorg Med Chem Lett 12: 1171-5 (2002) BindingDB Entry DOI: 10.7270/Q26M365J | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 5 (Homo sapiens (Human)) | BDBM50110562 (5-Chloro-3-(2-{4-[(3-methoxy-6,7,8,9-tetrahydro-5H...) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 0.700 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co., Ltd. Curated by ChEMBL | Assay Description Inhibition of 125 I-PYY binding to human Neuropeptide Y receptor type 5 | Bioorg Med Chem Lett 12: 799-802 (2002) BindingDB Entry DOI: 10.7270/Q2M044R7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 5 (Homo sapiens (Human)) | BDBM50093673 (2-Methyl-4-piperidin-1-yl-6-(4-trifluoromethyl-phe...) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 0.700 | n/a | n/a | n/a | n/a | n/a | n/a |
Amgen, Inc. Curated by ChEMBL | Assay Description Affinity for human neuropeptide Y receptor Y5, binding was evaluated in an in vitro radioligand [125I]-PYY binding assay | J Med Chem 43: 4288-312 (2000) BindingDB Entry DOI: 10.7270/Q2C828J1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 5 (Homo sapiens (Human)) | BDBM50093678 (2-Methyl-6-phenyl-4-pyrrolidin-1-yl-5H-pyrrolo[3,2...) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 0.700 | n/a | n/a | n/a | n/a | n/a | n/a |
Amgen, Inc. Curated by ChEMBL | Assay Description Affinity for human neuropeptide Y receptor Y5, binding was evaluated in an in vitro radioligand [125I]-PYY binding assay | J Med Chem 43: 4288-312 (2000) BindingDB Entry DOI: 10.7270/Q2C828J1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 5 (Homo sapiens (Human)) | BDBM50111646 (1-[2-(5-Chloro-2-oxo-benzothiazol-3-yl)-acetyl]-pi...) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 0.710 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co., Ltd. Curated by ChEMBL | Assay Description Inhibitory concentration of total specific binding of [125I]- -PYY to HEK 293 cells transfected with the Human NPY-Y5 cDNA (compound prepared by para... | Bioorg Med Chem Lett 12: 1171-5 (2002) BindingDB Entry DOI: 10.7270/Q26M365J | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 5 (Homo sapiens (Human)) | BDBM141344 (US8916594, I-017) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 0.810 | n/a | n/a | n/a | n/a | 7.4 | 25 |
Shionogi & Co., Ltd. US Patent | Assay Description cDNA sequence encoding a human NPY Y5 receptor (WO96/16542) was cloned in a vector (pME18S, Takebe et al. Mol. Cell. Biol. 8, 466-472). The obtained ... | US Patent US8916594 (2014) BindingDB Entry DOI: 10.7270/Q21G0K0S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 5 (Homo sapiens (Human)) | BDBM50258191 (1-(Methylsulfonyl)-N-(6-phenylpyridin-3-yl)-1,2-di...) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 0.820 | n/a | n/a | n/a | n/a | n/a | n/a |
Tsukuba Research Institute Curated by ChEMBL | Assay Description Displacement of [125I]PYY from human recombinant Y5 receptor expressed in mouse LMtk cells | Bioorg Med Chem Lett 19: 1564-8 (2009) Article DOI: 10.1016/j.bmcl.2009.02.035 BindingDB Entry DOI: 10.7270/Q2TQ61FT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 5 (Homo sapiens (Human)) | BDBM50258191 (1-(Methylsulfonyl)-N-(6-phenylpyridin-3-yl)-1,2-di...) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 0.820 | n/a | n/a | n/a | n/a | n/a | n/a |
Tsukuba Research Institute Curated by ChEMBL | Assay Description Binding affinity to human neuropeptide Y5 receptor | Bioorg Med Chem 17: 5015-26 (2009) Article DOI: 10.1016/j.bmc.2009.05.064 BindingDB Entry DOI: 10.7270/Q2KK9BT2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 5 (Homo sapiens (Human)) | BDBM50268737 (CHEMBL526084 | N-(3-(2-chlorophenyl)isoxazol-5-yl)...) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.830 | n/a | n/a | n/a | n/a | n/a | n/a |
Tsukuba Research Institute Curated by ChEMBL | Assay Description Displacement of [125I]PYY from human recombinant NPY Y5 receptor expressed in mouse LMtk- cells | Bioorg Med Chem Lett 19: 3511-6 (2009) Article DOI: 10.1016/j.bmcl.2009.05.013 BindingDB Entry DOI: 10.7270/Q21C1WS5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 5 (Homo sapiens (Human)) | BDBM50268700 (3-oxo-N-(3-phenylisoxazol-5-yl)-3H-spiro[isobenzof...) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.840 | n/a | n/a | n/a | n/a | n/a | n/a |
Tsukuba Research Institute Curated by ChEMBL | Assay Description Displacement of [125I]PYY from human recombinant NPY Y5 receptor expressed in mouse LMtk- cells | Bioorg Med Chem Lett 19: 3511-6 (2009) Article DOI: 10.1016/j.bmcl.2009.05.013 BindingDB Entry DOI: 10.7270/Q21C1WS5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 5 (Homo sapiens (Human)) | BDBM50268651 (3-oxo-N-(5-(3-(trifluoromethyl)phenyl)pyrimidin-2-...) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.850 | n/a | n/a | n/a | n/a | n/a | n/a |
Tsukuba Research Institute Curated by ChEMBL | Assay Description Displacement of [125I]PYY from human recombinant NPY Y5 receptor expressed in mouse LMtk- cells | Bioorg Med Chem Lett 19: 3511-6 (2009) Article DOI: 10.1016/j.bmcl.2009.05.013 BindingDB Entry DOI: 10.7270/Q21C1WS5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 5 (Homo sapiens (Human)) | BDBM50258053 (CHEMBL492568 | N-(biphenyl-4-yl)-1-(methylsulfonyl...) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 0.850 | n/a | n/a | n/a | n/a | n/a | n/a |
Tsukuba Research Institute Curated by ChEMBL | Assay Description Displacement of [125I]PYY from human recombinant Y5 receptor expressed in mouse LMtk cells | Bioorg Med Chem Lett 19: 1564-8 (2009) Article DOI: 10.1016/j.bmcl.2009.02.035 BindingDB Entry DOI: 10.7270/Q2TQ61FT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 5 (Homo sapiens (Human)) | BDBM50111647 (1-[2-(5-Chloro-2-oxo-benzothiazol-3-yl)-acetyl]-pi...) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 0.850 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co., Ltd. Curated by ChEMBL | Assay Description Inhibitory concentration of total specific binding of [125I]- -PYY to HEK 293 cells transfected with the Human NPY-Y5 cDNA (compound prepared by para... | Bioorg Med Chem Lett 12: 1171-5 (2002) BindingDB Entry DOI: 10.7270/Q26M365J | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 5 (Homo sapiens (Human)) | BDBM50258194 (1-(Methylsulfonyl)-N-(2-phenylpyrimidin-5-yl)-1,2-...) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 0.860 | n/a | n/a | n/a | n/a | n/a | n/a |
Tsukuba Research Institute Curated by ChEMBL | Assay Description Displacement of [125I]PYY from human recombinant Y5 receptor expressed in mouse LMtk cells | Bioorg Med Chem Lett 19: 1564-8 (2009) Article DOI: 10.1016/j.bmcl.2009.02.035 BindingDB Entry DOI: 10.7270/Q2TQ61FT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 5 (Homo sapiens (Human)) | BDBM141349 (US8916594, I-029) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 0.860 | n/a | n/a | n/a | n/a | 7.4 | 25 |
Shionogi & Co., Ltd. US Patent | Assay Description cDNA sequence encoding a human NPY Y5 receptor (WO96/16542) was cloned in a vector (pME18S, Takebe et al. Mol. Cell. Biol. 8, 466-472). The obtained ... | US Patent US8916594 (2014) BindingDB Entry DOI: 10.7270/Q21G0K0S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 5 (Homo sapiens (Human)) | BDBM50258194 (1-(Methylsulfonyl)-N-(2-phenylpyrimidin-5-yl)-1,2-...) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 0.860 | n/a | n/a | n/a | n/a | n/a | n/a |
Tsukuba Research Institute Curated by ChEMBL | Assay Description Binding affinity to human neuropeptide Y5 receptor | Bioorg Med Chem 17: 5015-26 (2009) Article DOI: 10.1016/j.bmc.2009.05.064 BindingDB Entry DOI: 10.7270/Q2KK9BT2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 5 (Homo sapiens (Human)) | BDBM50111641 (1-[2-(5-Chloro-2-oxo-benzothiazol-3-yl)-acetyl]-pi...) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 0.890 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co., Ltd. Curated by ChEMBL | Assay Description Inhibitory concentration of total specific binding of [125I]- -PYY to HEK 293 cells transfected with Human NPY-Y5 cDNA (compound prepared by manual s... | Bioorg Med Chem Lett 12: 1171-5 (2002) BindingDB Entry DOI: 10.7270/Q26M365J | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 5 (Homo sapiens (Human)) | BDBM50304315 (CHEMBL593465 | trans-3-Oxo-N-(2-phenyl-2H-1,2,3-tr...) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 0.890 | n/a | n/a | n/a | n/a | n/a | n/a |
Tsukuba Research Institute Curated by ChEMBL | Assay Description Displacement of [125I]PYY from human recombinant Y5 receptor | Bioorg Med Chem 17: 6971-82 (2009) Article DOI: 10.1016/j.bmc.2009.08.019 BindingDB Entry DOI: 10.7270/Q2P26Z62 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 5 (Homo sapiens (Human)) | BDBM50354070 (CHEMBL1836319) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 0.900 | n/a | n/a | n/a | n/a | n/a | n/a |
Lundbeck Research USA, Inc. Curated by ChEMBL | Assay Description Antagonist activity at human NPY5 receptor assessed as calcium mobilization by FLIPR assay | Bioorg Med Chem Lett 21: 5436-41 (2011) Article DOI: 10.1016/j.bmcl.2011.06.124 BindingDB Entry DOI: 10.7270/Q2RN387K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 5 (Homo sapiens (Human)) | BDBM50089048 (CHEMBL18163 | N,N-Dimethyl-C-[4-(4-phenylamino-qui...) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 0.900 | n/a | n/a | n/a | n/a | n/a | n/a |
Novartis Pharma AG Curated by ChEMBL | Assay Description Antagonistic activity against neuropeptide Y receptor type 5 subtype stably expressed in LM(tk-)cells | Bioorg Med Chem Lett 10: 1175-9 (2000) BindingDB Entry DOI: 10.7270/Q2KH0MJP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 5 (Homo sapiens (Human)) | BDBM50101533 (1-[2-(4-Chloro-phenyl)-1-methyl-ethyl]-1-methyl-3-...) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 0.900 | n/a | n/a | n/a | n/a | n/a | n/a |
Amgen Inc. Curated by ChEMBL | Assay Description Inhibitory activity tested against Human Neuropeptide Y5 Receptor. | J Med Chem 44: 2344-56 (2001) BindingDB Entry DOI: 10.7270/Q2DV1J56 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 5 (Homo sapiens (Human)) | BDBM50268534 (CHEMBL521545 | N-(5-(3-chlorophenyl)pyrimidin-2-yl...) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.910 | n/a | n/a | n/a | n/a | n/a | n/a |
Tsukuba Research Institute Curated by ChEMBL | Assay Description Displacement of [125I]PYY from human recombinant NPY Y5 receptor expressed in mouse LMtk- cells | Bioorg Med Chem Lett 19: 3511-6 (2009) Article DOI: 10.1016/j.bmcl.2009.05.013 BindingDB Entry DOI: 10.7270/Q21C1WS5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 5 (Homo sapiens (Human)) | BDBM50304301 (CHEMBL595790 | trans-N-[1-(3-Fluorophenyl)-1H-pyra...) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.920 | n/a | n/a | n/a | n/a | n/a | n/a |
Tsukuba Research Institute Curated by ChEMBL | Assay Description Displacement of [125I]PYY from human recombinant Y5 receptor | Bioorg Med Chem 17: 6971-82 (2009) Article DOI: 10.1016/j.bmc.2009.08.019 BindingDB Entry DOI: 10.7270/Q2P26Z62 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 5 (Homo sapiens (Human)) | BDBM50258151 (1-(Methylsulfonyl)-N-(5-phenylpyridin-2-yl)-1,2-di...) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 0.960 | n/a | n/a | n/a | n/a | n/a | n/a |
Tsukuba Research Institute Curated by ChEMBL | Assay Description Binding affinity to human neuropeptide Y5 receptor | Bioorg Med Chem 17: 5015-26 (2009) Article DOI: 10.1016/j.bmc.2009.05.064 BindingDB Entry DOI: 10.7270/Q2KK9BT2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 5 (Homo sapiens (Human)) | BDBM50258151 (1-(Methylsulfonyl)-N-(5-phenylpyridin-2-yl)-1,2-di...) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 0.960 | n/a | n/a | n/a | n/a | n/a | n/a |
Tsukuba Research Institute Curated by ChEMBL | Assay Description Displacement of [125I]PYY from human recombinant Y5 receptor expressed in mouse LMtk cells | Bioorg Med Chem Lett 19: 1564-8 (2009) Article DOI: 10.1016/j.bmcl.2009.02.035 BindingDB Entry DOI: 10.7270/Q2TQ61FT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 5 (Homo sapiens (Human)) | BDBM50258193 (1-(Methylsulfonyl)-N-(5-phenylpyrazin-2-yl)-1,2-di...) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 0.970 | n/a | n/a | n/a | n/a | n/a | n/a |
Tsukuba Research Institute Curated by ChEMBL | Assay Description Displacement of [125I]PYY from human recombinant Y5 receptor expressed in mouse LMtk cells | Bioorg Med Chem Lett 19: 1564-8 (2009) Article DOI: 10.1016/j.bmcl.2009.02.035 BindingDB Entry DOI: 10.7270/Q2TQ61FT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 5 (Homo sapiens (Human)) | BDBM50258193 (1-(Methylsulfonyl)-N-(5-phenylpyrazin-2-yl)-1,2-di...) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 0.970 | n/a | n/a | n/a | n/a | n/a | n/a |
Tsukuba Research Institute Curated by ChEMBL | Assay Description Binding affinity to human neuropeptide Y5 receptor | Bioorg Med Chem 17: 5015-26 (2009) Article DOI: 10.1016/j.bmc.2009.05.064 BindingDB Entry DOI: 10.7270/Q2KK9BT2 | |||||||||||
More data for this Ligand-Target Pair |
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