Search and Browse
Download
Enter Data
| Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Bromodomain-containing protein 4 [44-164] (Homo sapiens (Human)) | BDBM425130 (4-[3-[methoxy-[6-(trifluoromethyl)- 3-pyridyl]meth...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet  | PC cid PC sid UniChem | US Patent | n/a | n/a | <1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Plexxikon Inc. US Patent | Assay Description Binding of compounds of formula (I) with bromodomain 2, 3 4 was assessed using Alphascreen binding assay. The inhibition of the interaction between b... | US Patent US10519177 (2019) BindingDB Entry DOI: 10.7270/Q2154KDK | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Bromodomain-containing protein 4 [44-164] (Homo sapiens (Human)) | BDBM425138 (US10519177, Compound P-0020) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Plexxikon Inc. US Patent | Assay Description Binding of compounds of formula (I) with bromodomain 2, 3 4 was assessed using Alphascreen binding assay. The inhibition of the interaction between b... | US Patent US10519177 (2019) BindingDB Entry DOI: 10.7270/Q2154KDK | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Bromodomain-containing protein 4 [44-164] (Homo sapiens (Human)) | BDBM425163 (US10519177, Compound P-0043 | [5-(3,5-dimethylisox...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Plexxikon Inc. US Patent | Assay Description Binding of compounds of formula (I) with bromodomain 2, 3 4 was assessed using Alphascreen binding assay. The inhibition of the interaction between b... | US Patent US10519177 (2019) BindingDB Entry DOI: 10.7270/Q2154KDK | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Bromodomain-containing protein 4 [44-164] (Homo sapiens (Human)) | BDBM425167 (4-[3-[[2-(difluoro- methoxy)phenyl]methyl]- 1H-pyr...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Plexxikon Inc. US Patent | Assay Description Binding of compounds of formula (I) with bromodomain 2, 3 4 was assessed using Alphascreen binding assay. The inhibition of the interaction between b... | US Patent US10519177 (2019) BindingDB Entry DOI: 10.7270/Q2154KDK | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Bromodomain-containing protein 4 [1-477] (Homo sapiens (Human)) | BDBM425729 (4-[3-iodo-1-[(6-methoxy-2- pyridyl)methyl]pyrrolo[...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Plexxikon Inc. US Patent | US Patent US10519177 (2019) BindingDB Entry DOI: 10.7270/Q2154KDK | ||||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Bromodomain-containing protein 4 [1-477] (Homo sapiens (Human)) | BDBM425734 (4-[6-(3,5-dimethylisoxazol-4-yl)-1- [(2- methoxyph...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Plexxikon Inc. US Patent | US Patent US10519177 (2019) BindingDB Entry DOI: 10.7270/Q2154KDK | ||||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Bromodomain-containing protein 4 [1-477] (Homo sapiens (Human)) | BDBM425738 (4-[6-(3,5-dimethylisoxazol-4-yl)-1- [(1S)-1-(2- py...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Plexxikon Inc. US Patent | US Patent US10519177 (2019) BindingDB Entry DOI: 10.7270/Q2154KDK | ||||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Bromodomain-containing protein 4 [1-477] (Homo sapiens (Human)) | BDBM425742 (US10519177, Compound P-0942 | methyl 1-[4-[6-(3,5-...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Plexxikon Inc. US Patent | US Patent US10519177 (2019) BindingDB Entry DOI: 10.7270/Q2154KDK | ||||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Bromodomain-containing protein 4 [1-477] (Homo sapiens (Human)) | BDBM425743 (1-[4-[6-(3,5-dimethylisoxazol-4- yl)-1-[(4-methylt...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Plexxikon Inc. US Patent | US Patent US10519177 (2019) BindingDB Entry DOI: 10.7270/Q2154KDK | ||||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Bromodomain-containing protein 4 [1-477] (Homo sapiens (Human)) | BDBM425748 (US10519177, Compound P-0948 | methyl 4-[6-(3,5-dim...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Plexxikon Inc. US Patent | US Patent US10519177 (2019) BindingDB Entry DOI: 10.7270/Q2154KDK | ||||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Bromodomain-containing protein 4 [1-477] (Homo sapiens (Human)) | BDBM425752 (US10519177, Compound P-0952 | methyl 1-[4-[6-(3,5-...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Plexxikon Inc. US Patent | US Patent US10519177 (2019) BindingDB Entry DOI: 10.7270/Q2154KDK | ||||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Bromodomain-containing protein 4 [1-477] (Homo sapiens (Human)) | BDBM425768 (US10519177, Compound P-0968 | methyl 1-[4-[6-(3,5-...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Plexxikon Inc. US Patent | US Patent US10519177 (2019) BindingDB Entry DOI: 10.7270/Q2154KDK | ||||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Bromodomain-containing protein 4 [44-164] (Homo sapiens (Human)) | BDBM425199 (US10519177, Compound P-0079) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Plexxikon Inc. US Patent | Assay Description Binding of compounds of formula (I) with bromodomain 2, 3 4 was assessed using Alphascreen binding assay. The inhibition of the interaction between b... | US Patent US10519177 (2019) BindingDB Entry DOI: 10.7270/Q2154KDK | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Bromodomain-containing protein 4 [44-164] (Homo sapiens (Human)) | BDBM425220 (US10519177, Compound P-0098) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Plexxikon Inc. US Patent | Assay Description Binding of compounds of formula (I) with bromodomain 2, 3 4 was assessed using Alphascreen binding assay. The inhibition of the interaction between b... | US Patent US10519177 (2019) BindingDB Entry DOI: 10.7270/Q2154KDK | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Bromodomain-containing protein 4 [44-164] (Homo sapiens (Human)) | BDBM425229 (US10519177, Compound P-0108) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Plexxikon Inc. US Patent | Assay Description Binding of compounds of formula (I) with bromodomain 2, 3 4 was assessed using Alphascreen binding assay. The inhibition of the interaction between b... | US Patent US10519177 (2019) BindingDB Entry DOI: 10.7270/Q2154KDK | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Bromodomain-containing protein 4 [44-164] (Homo sapiens (Human)) | BDBM425231 (4-[1-(benzenesulfonyl)-3-(1- methylpyrazol-4-yl)py...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Plexxikon Inc. US Patent | Assay Description Binding of compounds of formula (I) with bromodomain 2, 3 4 was assessed using Alphascreen binding assay. The inhibition of the interaction between b... | US Patent US10519177 (2019) BindingDB Entry DOI: 10.7270/Q2154KDK | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Bromodomain-containing protein 4 [44-164] (Homo sapiens (Human)) | BDBM425242 (4-[1-(2-fluorophenyl) sulfonyl-3-(1-methyl- pyrazo...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Plexxikon Inc. US Patent | Assay Description Binding of compounds of formula (I) with bromodomain 2, 3 4 was assessed using Alphascreen binding assay. The inhibition of the interaction between b... | US Patent US10519177 (2019) BindingDB Entry DOI: 10.7270/Q2154KDK | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Bromodomain-containing protein 4 [44-164] (Homo sapiens (Human)) | BDBM425254 (4-[1-cyclopentylsulfonyl- 3-[1-(difluoromethyl) py...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Plexxikon Inc. US Patent | Assay Description Binding of compounds of formula (I) with bromodomain 2, 3 4 was assessed using Alphascreen binding assay. The inhibition of the interaction between b... | US Patent US10519177 (2019) BindingDB Entry DOI: 10.7270/Q2154KDK | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Bromodomain-containing protein 4 [44-164] (Homo sapiens (Human)) | BDBM425284 (4-[1-(benzenesulfonyl)-3- (1H-pyrazol-4-yl)pyrrolo...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Plexxikon Inc. US Patent | Assay Description Binding of compounds of formula (I) with bromodomain 2, 3 4 was assessed using Alphascreen binding assay. The inhibition of the interaction between b... | US Patent US10519177 (2019) BindingDB Entry DOI: 10.7270/Q2154KDK | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Bromodomain-containing protein 4 [44-164] (Homo sapiens (Human)) | BDBM425293 (4-[1-[(2-fluorophenyl)methyl]-3-(1- methylpyrazol-...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Plexxikon Inc. US Patent | Assay Description Binding of compounds of formula (I) with bromodomain 2, 3 4 was assessed using Alphascreen binding assay. The inhibition of the interaction between b... | US Patent US10519177 (2019) BindingDB Entry DOI: 10.7270/Q2154KDK | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Bromodomain-containing protein 4 [44-164] (Homo sapiens (Human)) | BDBM425317 (3-cyclopentyl-3-[6-(3,5- dimethylisoxazol-4- yl)py...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Plexxikon Inc. US Patent | Assay Description Binding of compounds of formula (I) with bromodomain 2, 3 4 was assessed using Alphascreen binding assay. The inhibition of the interaction between b... | US Patent US10519177 (2019) BindingDB Entry DOI: 10.7270/Q2154KDK | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Bromodomain-containing protein 4 [44-164] (Homo sapiens (Human)) | BDBM425318 (US10519177, Compound P-0197) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Plexxikon Inc. US Patent | Assay Description Binding of compounds of formula (I) with bromodomain 2, 3 4 was assessed using Alphascreen binding assay. The inhibition of the interaction between b... | US Patent US10519177 (2019) BindingDB Entry DOI: 10.7270/Q2154KDK | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Bromodomain-containing protein 4 [44-164] (Homo sapiens (Human)) | BDBM425329 (US10519177, Compound P-0208) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Plexxikon Inc. US Patent | Assay Description Binding of compounds of formula (I) with bromodomain 2, 3 4 was assessed using Alphascreen binding assay. The inhibition of the interaction between b... | US Patent US10519177 (2019) BindingDB Entry DOI: 10.7270/Q2154KDK | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Bromodomain-containing protein 4 [44-164] (Homo sapiens (Human)) | BDBM425341 (4-[3-(1-cyclopropylpyrazol- 4-yl)-1-[dideuterio-(4...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Plexxikon Inc. US Patent | Assay Description Binding of compounds of formula (I) with bromodomain 2, 3 4 was assessed using Alphascreen binding assay. The inhibition of the interaction between b... | US Patent US10519177 (2019) BindingDB Entry DOI: 10.7270/Q2154KDK | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Bromodomain-containing protein 4 [44-164] (Homo sapiens (Human)) | BDBM425342 (4-[1-[dideuterio-(4,4- difluorocyclohexyl)methyl]-...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Plexxikon Inc. US Patent | Assay Description Binding of compounds of formula (I) with bromodomain 2, 3 4 was assessed using Alphascreen binding assay. The inhibition of the interaction between b... | US Patent US10519177 (2019) BindingDB Entry DOI: 10.7270/Q2154KDK | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Bromodomain-containing protein 4 [1-477] (Homo sapiens (Human)) | BDBM425347 (3-cyclopentyl-3-[3-[1- (difluoromethyl)pyrazol-4-y...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Plexxikon Inc. US Patent | US Patent US10519177 (2019) BindingDB Entry DOI: 10.7270/Q2154KDK | ||||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Bromodomain-containing protein 4 [44-164] (Homo sapiens (Human)) | BDBM425362 (3,5-dimethyl-4-[1-(1-phenylethyl)-3- (3-pyridyl)py...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Plexxikon Inc. US Patent | Assay Description Binding of compounds of formula (I) with bromodomain 2, 3 4 was assessed using Alphascreen binding assay. The inhibition of the interaction between b... | US Patent US10519177 (2019) BindingDB Entry DOI: 10.7270/Q2154KDK | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Bromodomain-containing protein 4 [1-477] (Homo sapiens (Human)) | BDBM425362 (3,5-dimethyl-4-[1-(1-phenylethyl)-3- (3-pyridyl)py...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Plexxikon Inc. US Patent | US Patent US10519177 (2019) BindingDB Entry DOI: 10.7270/Q2154KDK | ||||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Bromodomain-containing protein 4 [44-164] (Homo sapiens (Human)) | BDBM425367 (3,5-dimethyl-4-[3-(6-methyl-3- pyridyl)-1-(1-pheny...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Plexxikon Inc. US Patent | Assay Description Binding of compounds of formula (I) with bromodomain 2, 3 4 was assessed using Alphascreen binding assay. The inhibition of the interaction between b... | US Patent US10519177 (2019) BindingDB Entry DOI: 10.7270/Q2154KDK | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Bromodomain-containing protein 4 [1-477] (Homo sapiens (Human)) | BDBM425372 (5-[6-(3,5-dimethylisoxazol-4-yl)-1-(1- phenylethyl...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Plexxikon Inc. US Patent | US Patent US10519177 (2019) BindingDB Entry DOI: 10.7270/Q2154KDK | ||||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Bromodomain-containing protein 4 [44-164] (Homo sapiens (Human)) | BDBM425383 (2-[6-(3,5-dimethylisoxazol-4-yl)-1-(1- phenylethyl...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Plexxikon Inc. US Patent | Assay Description Binding of compounds of formula (I) with bromodomain 2, 3 4 was assessed using Alphascreen binding assay. The inhibition of the interaction between b... | US Patent US10519177 (2019) BindingDB Entry DOI: 10.7270/Q2154KDK | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Bromodomain-containing protein 4 [1-477] (Homo sapiens (Human)) | BDBM425392 (4-[1-[(4,4-difluorocyclohexyl)methyl]- 3-(1-isobut...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Plexxikon Inc. US Patent | US Patent US10519177 (2019) BindingDB Entry DOI: 10.7270/Q2154KDK | ||||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Bromodomain-containing protein 4 [1-477] (Homo sapiens (Human)) | BDBM425393 (3-[4-[1-[(4,4- difluorocyclohexyl)methyl]-6-(3,5- ...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Plexxikon Inc. US Patent | US Patent US10519177 (2019) BindingDB Entry DOI: 10.7270/Q2154KDK | ||||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Bromodomain-containing protein 4 [44-164] (Homo sapiens (Human)) | BDBM425351 (4-[1-[dideuterio-(3,3- difluorocyclobutyl)methyl]-...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Plexxikon Inc. US Patent | Assay Description Binding of compounds of formula (I) with bromodomain 2, 3 4 was assessed using Alphascreen binding assay. The inhibition of the interaction between b... | US Patent US10519177 (2019) BindingDB Entry DOI: 10.7270/Q2154KDK | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Bromodomain-containing protein 4 [1-477] (Homo sapiens (Human)) | BDBM425351 (4-[1-[dideuterio-(3,3- difluorocyclobutyl)methyl]-...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Plexxikon Inc. US Patent | US Patent US10519177 (2019) BindingDB Entry DOI: 10.7270/Q2154KDK | ||||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Bromodomain-containing protein 4 [1-477] (Homo sapiens (Human)) | BDBM425352 (4-[1-[dideuterio-(3,3- difluorocyclobutyl)methyl]-...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Plexxikon Inc. US Patent | US Patent US10519177 (2019) BindingDB Entry DOI: 10.7270/Q2154KDK | ||||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Bromodomain-containing protein 4 [44-164] (Homo sapiens (Human)) | BDBM425402 (3-[3-chloro-6-(3,5-dimethylisoxazol-4- yl)pyrrolo[...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Plexxikon Inc. US Patent | Assay Description Binding of compounds of formula (I) with bromodomain 2, 3 4 was assessed using Alphascreen binding assay. The inhibition of the interaction between b... | US Patent US10519177 (2019) BindingDB Entry DOI: 10.7270/Q2154KDK | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Bromodomain-containing protein 4 [1-477] (Homo sapiens (Human)) | BDBM425402 (3-[3-chloro-6-(3,5-dimethylisoxazol-4- yl)pyrrolo[...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Plexxikon Inc. US Patent | US Patent US10519177 (2019) BindingDB Entry DOI: 10.7270/Q2154KDK | ||||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Bromodomain-containing protein 4 [44-164] (Homo sapiens (Human)) | BDBM425406 (1-[(4,4-difluorocyclohexyl)methyl]-6- (3,5-dimethy...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Plexxikon Inc. US Patent | Assay Description Binding of compounds of formula (I) with bromodomain 2, 3 4 was assessed using Alphascreen binding assay. The inhibition of the interaction between b... | US Patent US10519177 (2019) BindingDB Entry DOI: 10.7270/Q2154KDK | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Bromodomain-containing protein 4 [1-477] (Homo sapiens (Human)) | BDBM425779 (N-[4-[6-(3,5-dimethylisoxazol-4- yl)-1-[(1S)-1-(2-...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Plexxikon Inc. US Patent | US Patent US10519177 (2019) BindingDB Entry DOI: 10.7270/Q2154KDK | ||||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Bromodomain-containing protein 4 [1-477] (Homo sapiens (Human)) | BDBM425644 (1-[4-[6-(3,5-dimethylisoxazol-4-yl)-1- [(1S)-1-(2-...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Plexxikon Inc. US Patent | US Patent US10519177 (2019) BindingDB Entry DOI: 10.7270/Q2154KDK | ||||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Bromodomain-containing protein 4 [1-477] (Homo sapiens (Human)) | BDBM425784 (N-[4-[6-(3,5-dimethylisoxazol-4- yl)-1-[(1S)-1-(2-...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Plexxikon Inc. US Patent | US Patent US10519177 (2019) BindingDB Entry DOI: 10.7270/Q2154KDK | ||||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Bromodomain-containing protein 4 [1-477] (Homo sapiens (Human)) | BDBM425796 (2-[4-[1-[cyclopentyl(2- pyridyl)methyl]-6-(3,5- di...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | KEGG PC cid PC sid UniChem | US Patent | n/a | n/a | <1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Plexxikon Inc. US Patent | US Patent US10519177 (2019) BindingDB Entry DOI: 10.7270/Q2154KDK | ||||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Bromodomain-containing protein 4 [1-477] (Homo sapiens (Human)) | BDBM425811 (US10519177, Compound P-1011 | methyl 4-[1-[cyclobu...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Plexxikon Inc. US Patent | US Patent US10519177 (2019) BindingDB Entry DOI: 10.7270/Q2154KDK | ||||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Bromodomain-containing protein 4 [44-164] (Homo sapiens (Human)) | BDBM425412 (4-[1-benzyl-3-[1-(2,2,2- trifluoroethyl)pyrazol-4-...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Plexxikon Inc. US Patent | Assay Description Binding of compounds of formula (I) with bromodomain 2, 3 4 was assessed using Alphascreen binding assay. The inhibition of the interaction between b... | US Patent US10519177 (2019) BindingDB Entry DOI: 10.7270/Q2154KDK | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Bromodomain-containing protein 4 [1-477] (Homo sapiens (Human)) | BDBM425412 (4-[1-benzyl-3-[1-(2,2,2- trifluoroethyl)pyrazol-4-...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Plexxikon Inc. US Patent | US Patent US10519177 (2019) BindingDB Entry DOI: 10.7270/Q2154KDK | ||||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Bromodomain-containing protein 4 [44-164] (Homo sapiens (Human)) | BDBM425416 (3,5-dimethyl-4-(1-[(1,4,4- trifluorocyclohexyl)met...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Plexxikon Inc. US Patent | Assay Description Binding of compounds of formula (I) with bromodomain 2, 3 4 was assessed using Alphascreen binding assay. The inhibition of the interaction between b... | US Patent US10519177 (2019) BindingDB Entry DOI: 10.7270/Q2154KDK | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Bromodomain-containing protein 4 [44-164] (Homo sapiens (Human)) | BDBM425419 (4-[1-[(4,4-difluorocyclohexyl)methyl]- 6-(3,5-dime...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Plexxikon Inc. US Patent | Assay Description Binding of compounds of formula (I) with bromodomain 2, 3 4 was assessed using Alphascreen binding assay. The inhibition of the interaction between b... | US Patent US10519177 (2019) BindingDB Entry DOI: 10.7270/Q2154KDK | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Bromodomain-containing protein 4 [1-477] (Homo sapiens (Human)) | BDBM425419 (4-[1-[(4,4-difluorocyclohexyl)methyl]- 6-(3,5-dime...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Plexxikon Inc. US Patent | US Patent US10519177 (2019) BindingDB Entry DOI: 10.7270/Q2154KDK | ||||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Bromodomain-containing protein 4 [1-477] (Homo sapiens (Human)) | BDBM425420 (3,5-dimethyl-4-[3-(1-methylpyrazol-4- yl)-1-(pyrim...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Plexxikon Inc. US Patent | US Patent US10519177 (2019) BindingDB Entry DOI: 10.7270/Q2154KDK | ||||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Displayed 1 to 50 (of 802 total ) | Next | Last >> |
