Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Epidermal growth factor receptor (Homo sapiens (Human)) | BDBM50099963 (CHEMBL30432 | N*4*-(1-Benzyl-1H-indazol-5-yl)-N*6*...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 1 | n/a | n/a | n/a | n/a | n/a | n/a |
Research Biomet. Glaxo Wellcome Medicines Research Centre Curated by ChEMBL | Assay Description Inhibition of EGF receptor | Bioorg Med Chem Lett 11: 1401-5 (2001) BindingDB Entry DOI: 10.7270/Q2W37VKB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Receptor tyrosine-protein kinase erbB-2 (Rattus norvegicus) | BDBM50099960 ((1-Benzyl-1H-indazol-5-yl)-(6,7-dimethoxy-quinazol...) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 1 | n/a | n/a | n/a | n/a | n/a | n/a |
Research Biomet. Glaxo Wellcome Medicines Research Centre Curated by ChEMBL | Assay Description Inhibition of rat Receptor protein-tyrosine kinase erbB2 | Bioorg Med Chem Lett 11: 1401-5 (2001) BindingDB Entry DOI: 10.7270/Q2W37VKB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Receptor tyrosine-protein kinase erbB-2 (Rattus norvegicus) | BDBM50099969 ((2-Benzyl-1H-benzoimidazol-5-yl)-(6,7-dimethoxy-qu...) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents | PubMed | n/a | n/a | 10 | n/a | n/a | n/a | n/a | n/a | n/a |
Research Biomet. Glaxo Wellcome Medicines Research Centre Curated by ChEMBL | Assay Description Inhibition of rat Receptor protein-tyrosine kinase erbB2 | Bioorg Med Chem Lett 11: 1401-5 (2001) BindingDB Entry DOI: 10.7270/Q2W37VKB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Receptor tyrosine-protein kinase erbB-2 (Rattus norvegicus) | BDBM50099965 ((1-Benzyl-1H-indazol-5-yl)-quinazolin-4-yl-amine |...) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 10 | n/a | n/a | n/a | n/a | n/a | n/a |
Research Biomet. Glaxo Wellcome Medicines Research Centre Curated by ChEMBL | Assay Description Inhibition of rat Receptor protein-tyrosine kinase erbB2 | Bioorg Med Chem Lett 11: 1401-5 (2001) BindingDB Entry DOI: 10.7270/Q2W37VKB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Receptor tyrosine-protein kinase erbB-4 (Homo sapiens (Human)) | BDBM50099963 (CHEMBL30432 | N*4*-(1-Benzyl-1H-indazol-5-yl)-N*6*...) | PDB MMDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 20 | n/a | n/a | n/a | n/a | n/a | n/a |
Research Biomet. Glaxo Wellcome Medicines Research Centre Curated by ChEMBL | Assay Description Inhibition of erbB4 receptor | Bioorg Med Chem Lett 11: 1401-5 (2001) BindingDB Entry DOI: 10.7270/Q2W37VKB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Receptor tyrosine-protein kinase erbB-2 (Rattus norvegicus) | BDBM50099971 (CHEMBL288557 | N*4*-(1-Benzyl-1H-indol-5-yl)-pyrid...) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 26 | n/a | n/a | n/a | n/a | n/a | n/a |
Research Biomet. Glaxo Wellcome Medicines Research Centre Curated by ChEMBL | Assay Description Inhibition of rat Receptor protein-tyrosine kinase erbB2 | Bioorg Med Chem Lett 11: 1401-5 (2001) BindingDB Entry DOI: 10.7270/Q2W37VKB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Receptor tyrosine-protein kinase erbB-2 (Rattus norvegicus) | BDBM50099966 (CHEMBL281006 | N*4*-(1-Benzyl-1H-indazol-5-yl)-pyr...) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 27 | n/a | n/a | n/a | n/a | n/a | n/a |
Research Biomet. Glaxo Wellcome Medicines Research Centre Curated by ChEMBL | Assay Description Inhibition of rat Receptor protein-tyrosine kinase erbB2 | Bioorg Med Chem Lett 11: 1401-5 (2001) BindingDB Entry DOI: 10.7270/Q2W37VKB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Receptor tyrosine-protein kinase erbB-2 (Rattus norvegicus) | BDBM50099968 (CHEMBL31653 | N*4*-(2-Benzyl-1H-benzoimidazol-5-yl...) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 49 | n/a | n/a | n/a | n/a | n/a | n/a |
Research Biomet. Glaxo Wellcome Medicines Research Centre Curated by ChEMBL | Assay Description Inhibition of rat Receptor protein-tyrosine kinase erbB2 | Bioorg Med Chem Lett 11: 1401-5 (2001) BindingDB Entry DOI: 10.7270/Q2W37VKB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Receptor tyrosine-protein kinase erbB-2 (Rattus norvegicus) | BDBM50099970 ((1-Benzyl-1H-indol-5-yl)-(6,7-dimethoxy-quinazolin...) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents | PubMed | n/a | n/a | 49 | n/a | n/a | n/a | n/a | n/a | n/a |
Research Biomet. Glaxo Wellcome Medicines Research Centre Curated by ChEMBL | Assay Description Inhibition of rat Receptor protein-tyrosine kinase erbB2 | Bioorg Med Chem Lett 11: 1401-5 (2001) BindingDB Entry DOI: 10.7270/Q2W37VKB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Receptor tyrosine-protein kinase erbB-2 (Homo sapiens (Human)) | BDBM50099963 (CHEMBL30432 | N*4*-(1-Benzyl-1H-indazol-5-yl)-N*6*...) | PDB MMDB UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 70 | n/a | n/a | n/a | n/a | n/a | n/a |
Research Biomet. Glaxo Wellcome Medicines Research Centre Curated by ChEMBL | Assay Description Inhibition of erbB2 overexpressing BT 474 cell proliferation | Bioorg Med Chem Lett 11: 1401-5 (2001) BindingDB Entry DOI: 10.7270/Q2W37VKB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Receptor tyrosine-protein kinase erbB-2 (Rattus norvegicus) | BDBM50099967 ((1-Benzyl-1H-indol-5-yl)-quinazolin-4-yl-amine | C...) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 90 | n/a | n/a | n/a | n/a | n/a | n/a |
Research Biomet. Glaxo Wellcome Medicines Research Centre Curated by ChEMBL | Assay Description Inhibition of rat Receptor protein-tyrosine kinase erbB2 | Bioorg Med Chem Lett 11: 1401-5 (2001) BindingDB Entry DOI: 10.7270/Q2W37VKB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Receptor tyrosine-protein kinase erbB-2 (Homo sapiens (Human)) | BDBM50099966 (CHEMBL281006 | N*4*-(1-Benzyl-1H-indazol-5-yl)-pyr...) | PDB MMDB UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 97 | n/a | n/a | n/a | n/a | n/a | n/a |
Research Biomet. Glaxo Wellcome Medicines Research Centre Curated by ChEMBL | Assay Description Inhibition of c-erbB-2 overexpressing HB4a cell proliferation | Bioorg Med Chem Lett 11: 1401-5 (2001) BindingDB Entry DOI: 10.7270/Q2W37VKB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Receptor tyrosine-protein kinase erbB-2 (Homo sapiens (Human)) | BDBM50099963 (CHEMBL30432 | N*4*-(1-Benzyl-1H-indazol-5-yl)-N*6*...) | PDB MMDB UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 97 | n/a | n/a | n/a | n/a | n/a | n/a |
Research Biomet. Glaxo Wellcome Medicines Research Centre Curated by ChEMBL | Assay Description Inhibition of erbB2 overexpressing HB4a.e5.2 cell proliferation | Bioorg Med Chem Lett 11: 1401-5 (2001) BindingDB Entry DOI: 10.7270/Q2W37VKB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Epidermal growth factor receptor (Homo sapiens (Human)) | BDBM50099963 (CHEMBL30432 | N*4*-(1-Benzyl-1H-indazol-5-yl)-N*6*...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 210 | n/a | n/a | n/a | n/a | n/a | n/a |
Research Biomet. Glaxo Wellcome Medicines Research Centre Curated by ChEMBL | Assay Description Inhibition of EGF receptor overexpressing HN5 cell proliferation | Bioorg Med Chem Lett 11: 1401-5 (2001) BindingDB Entry DOI: 10.7270/Q2W37VKB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Receptor tyrosine-protein kinase erbB-2 (Rattus norvegicus) | BDBM50099961 ((2-Benzyl-2H-indazol-5-yl)-(6,7-dimethoxy-quinazol...) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 290 | n/a | n/a | n/a | n/a | n/a | n/a |
Research Biomet. Glaxo Wellcome Medicines Research Centre Curated by ChEMBL | Assay Description Inhibition of rat Receptor protein-tyrosine kinase erbB2 | Bioorg Med Chem Lett 11: 1401-5 (2001) BindingDB Entry DOI: 10.7270/Q2W37VKB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Receptor tyrosine-protein kinase erbB-2 (Homo sapiens (Human)) | BDBM50099960 ((1-Benzyl-1H-indazol-5-yl)-(6,7-dimethoxy-quinazol...) | PDB MMDB UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 290 | n/a | n/a | n/a | n/a | n/a | n/a |
Research Biomet. Glaxo Wellcome Medicines Research Centre Curated by ChEMBL | Assay Description Inhibition of c-erbB-2 overexpressing HB4a cell proliferation | Bioorg Med Chem Lett 11: 1401-5 (2001) BindingDB Entry DOI: 10.7270/Q2W37VKB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Receptor tyrosine-protein kinase erbB-2 (Homo sapiens (Human)) | BDBM50099970 ((1-Benzyl-1H-indol-5-yl)-(6,7-dimethoxy-quinazolin...) | PDB MMDB UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents | PubMed | n/a | n/a | 350 | n/a | n/a | n/a | n/a | n/a | n/a |
Research Biomet. Glaxo Wellcome Medicines Research Centre Curated by ChEMBL | Assay Description Inhibition of c-erbB-2 overexpressing HB4a cell proliferation | Bioorg Med Chem Lett 11: 1401-5 (2001) BindingDB Entry DOI: 10.7270/Q2W37VKB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Receptor tyrosine-protein kinase erbB-2 (Rattus norvegicus) | BDBM50099963 (CHEMBL30432 | N*4*-(1-Benzyl-1H-indazol-5-yl)-N*6*...) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 390 | n/a | n/a | n/a | n/a | n/a | n/a |
Research Biomet. Glaxo Wellcome Medicines Research Centre Curated by ChEMBL | Assay Description Inhibition of erbB2 overexpressing Calu3 cell proliferation | Bioorg Med Chem Lett 11: 1401-5 (2001) BindingDB Entry DOI: 10.7270/Q2W37VKB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Receptor tyrosine-protein kinase erbB-2 (Rattus norvegicus) | BDBM50099963 (CHEMBL30432 | N*4*-(1-Benzyl-1H-indazol-5-yl)-N*6*...) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 390 | n/a | n/a | n/a | n/a | n/a | n/a |
Research Biomet. Glaxo Wellcome Medicines Research Centre Curated by ChEMBL | Assay Description Inhibition of erbB2 overexpressing Calu3 cell proliferation | Bioorg Med Chem Lett 11: 1401-5 (2001) BindingDB Entry DOI: 10.7270/Q2W37VKB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Receptor tyrosine-protein kinase erbB-2 (Rattus norvegicus) | BDBM50099959 ((2-Benzyl-1H-benzoimidazol-5-yl)-quinazolin-4-yl-a...) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 560 | n/a | n/a | n/a | n/a | n/a | n/a |
Research Biomet. Glaxo Wellcome Medicines Research Centre Curated by ChEMBL | Assay Description Inhibition of rat Receptor protein-tyrosine kinase erbB2 | Bioorg Med Chem Lett 11: 1401-5 (2001) BindingDB Entry DOI: 10.7270/Q2W37VKB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Receptor tyrosine-protein kinase erbB-2 (Homo sapiens (Human)) | BDBM50099969 ((2-Benzyl-1H-benzoimidazol-5-yl)-(6,7-dimethoxy-qu...) | PDB MMDB UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents | PubMed | n/a | n/a | 1.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Research Biomet. Glaxo Wellcome Medicines Research Centre Curated by ChEMBL | Assay Description Inhibition of c-erbB-2 overexpressing HB4a cell proliferation | Bioorg Med Chem Lett 11: 1401-5 (2001) BindingDB Entry DOI: 10.7270/Q2W37VKB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Receptor tyrosine-protein kinase erbB-2 (Homo sapiens (Human)) | BDBM50099967 ((1-Benzyl-1H-indol-5-yl)-quinazolin-4-yl-amine | C...) | PDB MMDB UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 1.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Research Biomet. Glaxo Wellcome Medicines Research Centre Curated by ChEMBL | Assay Description Inhibition of c-erbB-2 overexpressing HB4a cell proliferation | Bioorg Med Chem Lett 11: 1401-5 (2001) BindingDB Entry DOI: 10.7270/Q2W37VKB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Receptor tyrosine-protein kinase erbB-2 (Homo sapiens (Human)) | BDBM50099959 ((2-Benzyl-1H-benzoimidazol-5-yl)-quinazolin-4-yl-a...) | PDB MMDB UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 1.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Research Biomet. Glaxo Wellcome Medicines Research Centre Curated by ChEMBL | Assay Description Inhibition of c-erbB-2 overexpressing HB4a cell proliferation | Bioorg Med Chem Lett 11: 1401-5 (2001) BindingDB Entry DOI: 10.7270/Q2W37VKB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Receptor tyrosine-protein kinase erbB-2 (Homo sapiens (Human)) | BDBM50099968 (CHEMBL31653 | N*4*-(2-Benzyl-1H-benzoimidazol-5-yl...) | PDB MMDB UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 1.86E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Research Biomet. Glaxo Wellcome Medicines Research Centre Curated by ChEMBL | Assay Description Inhibition of c-erbB-2 overexpressing HB4a cell proliferation | Bioorg Med Chem Lett 11: 1401-5 (2001) BindingDB Entry DOI: 10.7270/Q2W37VKB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Receptor tyrosine-protein kinase erbB-2 (Homo sapiens (Human)) | BDBM50099961 ((2-Benzyl-2H-indazol-5-yl)-(6,7-dimethoxy-quinazol...) | PDB MMDB UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 3.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Research Biomet. Glaxo Wellcome Medicines Research Centre Curated by ChEMBL | Assay Description Inhibition of c-erbB-2 overexpressing HB4a cell proliferation | Bioorg Med Chem Lett 11: 1401-5 (2001) BindingDB Entry DOI: 10.7270/Q2W37VKB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Receptor tyrosine-protein kinase erbB-2 (Rattus norvegicus) | BDBM50099962 ((3-Benzyl-3H-benzoimidazol-5-yl)-quinazolin-4-yl-a...) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 4.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Research Biomet. Glaxo Wellcome Medicines Research Centre Curated by ChEMBL | Assay Description Inhibition of rat Receptor protein-tyrosine kinase erbB2 | Bioorg Med Chem Lett 11: 1401-5 (2001) BindingDB Entry DOI: 10.7270/Q2W37VKB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Receptor tyrosine-protein kinase erbB-2 (Rattus norvegicus) | BDBM50099964 ((1-Benzyl-1H-benzoimidazol-5-yl)-quinazolin-4-yl-a...) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 6.60E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Research Biomet. Glaxo Wellcome Medicines Research Centre Curated by ChEMBL | Assay Description Inhibition of rat Receptor protein-tyrosine kinase erbB2 | Bioorg Med Chem Lett 11: 1401-5 (2001) BindingDB Entry DOI: 10.7270/Q2W37VKB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-dependent kinase 1 (Homo sapiens (Human)) | BDBM50099963 (CHEMBL30432 | N*4*-(1-Benzyl-1H-indazol-5-yl)-N*6*...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | >8.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Research Biomet. Glaxo Wellcome Medicines Research Centre Curated by ChEMBL | Assay Description Inhibition of Cyclin-dependent kinase 1 | Bioorg Med Chem Lett 11: 1401-5 (2001) BindingDB Entry DOI: 10.7270/Q2W37VKB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-dependent kinase 2 (Homo sapiens (Human)) | BDBM50099963 (CHEMBL30432 | N*4*-(1-Benzyl-1H-indazol-5-yl)-N*6*...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | >8.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Research Biomet. Glaxo Wellcome Medicines Research Centre Curated by ChEMBL | Assay Description Inhibition of Cyclin-dependent kinase 2 | Bioorg Med Chem Lett 11: 1401-5 (2001) BindingDB Entry DOI: 10.7270/Q2W37VKB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dual specificity mitogen-activated protein kinase kinase 1/2 (Homo sapiens (Human)) | BDBM50099963 (CHEMBL30432 | N*4*-(1-Benzyl-1H-indazol-5-yl)-N*6*...) | PDB KEGG UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 9.70E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Research Biomet. Glaxo Wellcome Medicines Research Centre Curated by ChEMBL | Assay Description Inhibition of erbB2 overexpressing BT 474 cell proliferation | Bioorg Med Chem Lett 11: 1401-5 (2001) BindingDB Entry DOI: 10.7270/Q2W37VKB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Receptor tyrosine-protein kinase erbB-2 (Homo sapiens (Human)) | BDBM50099962 ((3-Benzyl-3H-benzoimidazol-5-yl)-quinazolin-4-yl-a...) | PDB MMDB UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 2.10E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Research Biomet. Glaxo Wellcome Medicines Research Centre Curated by ChEMBL | Assay Description Inhibition of c-erbB-2 overexpressing HB4a cell proliferation | Bioorg Med Chem Lett 11: 1401-5 (2001) BindingDB Entry DOI: 10.7270/Q2W37VKB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Receptor tyrosine-protein kinase erbB-2 (Homo sapiens (Human)) | BDBM50099964 ((1-Benzyl-1H-benzoimidazol-5-yl)-quinazolin-4-yl-a...) | PDB MMDB UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 2.70E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Research Biomet. Glaxo Wellcome Medicines Research Centre Curated by ChEMBL | Assay Description Inhibition of c-erbB-2 overexpressing HB4a cell proliferation | Bioorg Med Chem Lett 11: 1401-5 (2001) BindingDB Entry DOI: 10.7270/Q2W37VKB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
RAF proto-oncogene serine/threonine-protein kinase (Homo sapiens (Human)) | BDBM50099963 (CHEMBL30432 | N*4*-(1-Benzyl-1H-indazol-5-yl)-N*6*...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 4.90E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Research Biomet. Glaxo Wellcome Medicines Research Centre Curated by ChEMBL | Assay Description Inhibition of Raf kinase | Bioorg Med Chem Lett 11: 1401-5 (2001) BindingDB Entry DOI: 10.7270/Q2W37VKB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proto-oncogene tyrosine-protein kinase Src (Homo sapiens (Human)) | BDBM50099963 (CHEMBL30432 | N*4*-(1-Benzyl-1H-indazol-5-yl)-N*6*...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | >5.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Research Biomet. Glaxo Wellcome Medicines Research Centre Curated by ChEMBL | Assay Description Inhibition of Src kinase | Bioorg Med Chem Lett 11: 1401-5 (2001) BindingDB Entry DOI: 10.7270/Q2W37VKB | |||||||||||
More data for this Ligand-Target Pair |