BindingDB PrimarySearch

Found 63 hits with Last Name = 'natale' and Initial = 'nr'
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Voltage-dependent L-type calcium channel subunit alpha-1C (RAT)	BDBM50079458 (2,6-Dimethyl-4-[3-methyl-5-(2-naphthalen-1-yl-ethy...) Show SMILES Show InChI	PDB UniProtKB/SwissProt GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	2.20	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
State University of New York Curated by ChEMBL					Assay Description Displacement of [3H](+)-PN200-110 binding from calcium channels of rat cardiac membranes.				J Med Chem 42: 3087-93 (1999) Article DOI: 10.1021/jm980439q BindingDB Entry DOI: 10.7270/Q20C4TZD
State University of New York Curated by ChEMBL					More data for this Ligand-Target Pair
Voltage-dependent L-type calcium channel subunit alpha-1C (Homo sapiens (Human))	BDBM50079458 (2,6-Dimethyl-4-[3-methyl-5-(2-naphthalen-1-yl-ethy...) Show SMILES Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	4.10	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
State University of New York Curated by ChEMBL					Assay Description Displacement of [3H](+)-PN200-110 binding to calcium channels in guinea pig cardiac membranes.				J Med Chem 42: 3087-93 (1999) Article DOI: 10.1021/jm980439q BindingDB Entry DOI: 10.7270/Q20C4TZD
State University of New York Curated by ChEMBL					More data for this Ligand-Target Pair
Voltage-dependent L-type calcium channel subunit alpha-1C (RAT)	BDBM50079463 (4-{5-[2-(3-Bromo-phenyl)-ethyl]-3-phenyl-isoxazol-...) Show SMILES Show InChI	PDB UniProtKB/SwissProt GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	5.60	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
State University of New York Curated by ChEMBL					Assay Description Displacement of [3H](+)-PN200-110 binding from calcium channels of rat cardiac membranes.				J Med Chem 42: 3087-93 (1999) Article DOI: 10.1021/jm980439q BindingDB Entry DOI: 10.7270/Q20C4TZD
State University of New York Curated by ChEMBL					More data for this Ligand-Target Pair
Voltage-dependent L-type calcium channel subunit alpha-1C (Homo sapiens (Human))	BDBM50079463 (4-{5-[2-(3-Bromo-phenyl)-ethyl]-3-phenyl-isoxazol-...) Show SMILES Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	6.90	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
State University of New York Curated by ChEMBL					Assay Description Displacement of [3H](+)-PN200-110 binding to calcium channels in guinea pig cardiac membranes.				J Med Chem 42: 3087-93 (1999) Article DOI: 10.1021/jm980439q BindingDB Entry DOI: 10.7270/Q20C4TZD
State University of New York Curated by ChEMBL					More data for this Ligand-Target Pair
Voltage-dependent L-type calcium channel subunit alpha-1C (RAT)	BDBM50079459 (4-[5-(2-Biphenyl-4-yl-ethyl)-3-methyl-isoxazol-4-y...) Show SMILES Show InChI	PDB UniProtKB/SwissProt GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	8.70	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
State University of New York Curated by ChEMBL					Assay Description Displacement of [3H](+)-PN200-110 binding from calcium channels of rat cardiac membranes.				J Med Chem 42: 3087-93 (1999) Article DOI: 10.1021/jm980439q BindingDB Entry DOI: 10.7270/Q20C4TZD
State University of New York Curated by ChEMBL					More data for this Ligand-Target Pair
Voltage-dependent L-type calcium channel subunit alpha-1C (RAT)	BDBM50079464 (2,6-Dimethyl-4-[3-methyl-5-(2-naphthalen-2-yl-ethy...) Show SMILES Show InChI	PDB UniProtKB/SwissProt GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	11	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
State University of New York Curated by ChEMBL					Assay Description Displacement of [3H](+)-PN200-110 binding from calcium channels of rat cardiac membranes.				J Med Chem 42: 3087-93 (1999) Article DOI: 10.1021/jm980439q BindingDB Entry DOI: 10.7270/Q20C4TZD
State University of New York Curated by ChEMBL					More data for this Ligand-Target Pair
Voltage-dependent L-type calcium channel subunit alpha-1C (Homo sapiens (Human))	BDBM50013025 (2,6-Dimethyl-4-(5-methyl-3-phenyl-isoxazol-4-yl)-1...) Show SMILES Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	14	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
State University of New York Curated by ChEMBL					Assay Description Inhibition of [3H]-PN-200110 binding to Calcium channel in guinea pig heart membrane				J Med Chem 33: 2255-9 (1990) BindingDB Entry DOI: 10.7270/Q2KS6QHH
State University of New York Curated by ChEMBL					More data for this Ligand-Target Pair
Voltage-dependent L-type calcium channel subunit alpha-1C (Homo sapiens (Human))	BDBM50079459 (4-[5-(2-Biphenyl-4-yl-ethyl)-3-methyl-isoxazol-4-y...) Show SMILES Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	18	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
State University of New York Curated by ChEMBL					Assay Description Displacement of [3H](+)-PN200-110 binding to calcium channels in guinea pig cardiac membranes.				J Med Chem 42: 3087-93 (1999) Article DOI: 10.1021/jm980439q BindingDB Entry DOI: 10.7270/Q20C4TZD
State University of New York Curated by ChEMBL					More data for this Ligand-Target Pair
Voltage-dependent L-type calcium channel subunit alpha-1C (Homo sapiens (Human))	BDBM50079464 (2,6-Dimethyl-4-[3-methyl-5-(2-naphthalen-2-yl-ethy...) Show SMILES Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	20	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
State University of New York Curated by ChEMBL					Assay Description Displacement of [3H](+)-PN200-110 binding to calcium channels in guinea pig cardiac membranes.				J Med Chem 42: 3087-93 (1999) Article DOI: 10.1021/jm980439q BindingDB Entry DOI: 10.7270/Q20C4TZD
State University of New York Curated by ChEMBL					More data for this Ligand-Target Pair
Voltage-dependent L-type calcium channel subunit alpha-1C/alpha-1D/alpha-1F/alpha-1S (Homo sapiens (Human))	BDBM50013025 (2,6-Dimethyl-4-(5-methyl-3-phenyl-isoxazol-4-yl)-1...) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia antibodypedia antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	22	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
State University of New York Curated by ChEMBL					Assay Description Inhibition of [3H]-PN-200110 binding to Calcium channel in guinea pig heart membrane.				J Med Chem 33: 2255-9 (1990) BindingDB Entry DOI: 10.7270/Q2KS6QHH
State University of New York Curated by ChEMBL					More data for this Ligand-Target Pair
Voltage-dependent L-type calcium channel subunit alpha-1C (Homo sapiens (Human))	BDBM50079462 (2,6-Dimethyl-4-(3-methyl-5-phenethyl-isoxazol-4-yl...) Show SMILES Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	23	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
State University of New York Curated by ChEMBL					Assay Description Displacement of [3H](+)-PN200-110 binding to calcium channels in guinea pig cardiac membranes.				J Med Chem 42: 3087-93 (1999) Article DOI: 10.1021/jm980439q BindingDB Entry DOI: 10.7270/Q20C4TZD
State University of New York Curated by ChEMBL					More data for this Ligand-Target Pair
Voltage-dependent L-type calcium channel subunit alpha-1C (RAT)	BDBM50079462 (2,6-Dimethyl-4-(3-methyl-5-phenethyl-isoxazol-4-yl...) Show SMILES Show InChI	PDB UniProtKB/SwissProt GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	25	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
State University of New York Curated by ChEMBL					Assay Description Displacement of [3H](+)-PN200-110 binding from calcium channels of rat cardiac membranes.				J Med Chem 42: 3087-93 (1999) Article DOI: 10.1021/jm980439q BindingDB Entry DOI: 10.7270/Q20C4TZD
State University of New York Curated by ChEMBL					More data for this Ligand-Target Pair
Voltage-dependent L-type calcium channel subunit alpha-1C (Homo sapiens (Human))	BDBM50013022 (4-(3,5-Dimethyl-isoxazol-4-yl)-2,6-dimethyl-1,4-di...) Show SMILES Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	27	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
State University of New York Curated by ChEMBL					Assay Description Inhibition of [3H]-PN-200110 binding to Calcium channel in guinea pig heart membrane				J Med Chem 33: 2255-9 (1990) BindingDB Entry DOI: 10.7270/Q2KS6QHH
State University of New York Curated by ChEMBL					More data for this Ligand-Target Pair
Voltage-dependent L-type calcium channel subunit alpha-1C (Homo sapiens (Human))	BDBM50013022 (4-(3,5-Dimethyl-isoxazol-4-yl)-2,6-dimethyl-1,4-di...) Show SMILES Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	29	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
State University of New York Curated by ChEMBL					Assay Description Inhibition of [3H]-PN-200110 binding to Calcium channel in guinea pig heart membrane.				J Med Chem 33: 2255-9 (1990) BindingDB Entry DOI: 10.7270/Q2KS6QHH
State University of New York Curated by ChEMBL					More data for this Ligand-Target Pair
Voltage-dependent L-type calcium channel subunit alpha-1C (RAT)	BDBM50079460 (4-{5-[2-(3-Methoxy-phenyl)-ethyl]-3-phenyl-isoxazo...) Show SMILES Show InChI	PDB UniProtKB/SwissProt GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	30	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
State University of New York Curated by ChEMBL					Assay Description Displacement of [3H](+)-PN200-110 binding from calcium channels of rat cardiac membranes.				J Med Chem 42: 3087-93 (1999) Article DOI: 10.1021/jm980439q BindingDB Entry DOI: 10.7270/Q20C4TZD
State University of New York Curated by ChEMBL					More data for this Ligand-Target Pair
Voltage-dependent L-type calcium channel subunit alpha-1C/alpha-1D/alpha-1F/alpha-1S (Homo sapiens (Human))	BDBM50013022 (4-(3,5-Dimethyl-isoxazol-4-yl)-2,6-dimethyl-1,4-di...) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia antibodypedia antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	30	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
State University of New York Curated by ChEMBL					Assay Description Inhibition of [3H]PN-200110 binding to Calcium channel in guinea pig ileum membrane.				J Med Chem 33: 2255-9 (1990) BindingDB Entry DOI: 10.7270/Q2KS6QHH
State University of New York Curated by ChEMBL					More data for this Ligand-Target Pair
Metabotropic glutamate receptor 5 (Homo sapiens (Human))	BDBM50105838 (FENOBAM) Show SMILES CN1CC(=O)N=C1NC(=O)Nc1cccc(Cl)c1 \|c:5\| Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase MCE PC cid PC sid PDB UniChem	PDB Article PubMed	32	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
University of Montana Curated by ChEMBL					Assay Description Displacement of MPEP from mGluR5 (unknown origin) after 3 hrs by liquid scintillation counting method				Bioorg Med Chem 26: 4797-4803 (2018) Article DOI: 10.1016/j.bmc.2018.08.012 BindingDB Entry DOI: 10.7270/Q2Q242TX
University of Montana Curated by ChEMBL					More data for this Ligand-Target Pair				3D Structure (crystal)
Voltage-dependent L-type calcium channel subunit alpha-1C/alpha-1D/alpha-1F/alpha-1S (Homo sapiens (Human))	BDBM50013022 (4-(3,5-Dimethyl-isoxazol-4-yl)-2,6-dimethyl-1,4-di...) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia antibodypedia antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	33	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
State University of New York Curated by ChEMBL					Assay Description Inhibition of [3H]PN-200110 binding to Calcium channel in guinea pig ileum membrane				J Med Chem 33: 2255-9 (1990) BindingDB Entry DOI: 10.7270/Q2KS6QHH
State University of New York Curated by ChEMBL					More data for this Ligand-Target Pair
Metabotropic glutamate receptor 5 (Homo sapiens (Human))	BDBM50105838 (FENOBAM) Show SMILES CN1CC(=O)N=C1NC(=O)Nc1cccc(Cl)c1 \|c:5\| Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase MCE PC cid PC sid PDB UniChem	PDB Article PubMed	33	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
University of Montana Curated by ChEMBL					Assay Description Displacement of MPEP from mGluR5 (unknown origin) after 3 hrs by liquid scintillation counting method				Bioorg Med Chem 26: 4797-4803 (2018) Article DOI: 10.1016/j.bmc.2018.08.012 BindingDB Entry DOI: 10.7270/Q2Q242TX
University of Montana Curated by ChEMBL					More data for this Ligand-Target Pair				3D Structure (crystal)
Voltage-dependent L-type calcium channel subunit alpha-1C (Homo sapiens (Human))	BDBM50079460 (4-{5-[2-(3-Methoxy-phenyl)-ethyl]-3-phenyl-isoxazo...) Show SMILES Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	40	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
State University of New York Curated by ChEMBL					Assay Description Displacement of [3H](+)-PN200-110 binding to calcium channels in guinea pig cardiac membranes.				J Med Chem 42: 3087-93 (1999) Article DOI: 10.1021/jm980439q BindingDB Entry DOI: 10.7270/Q20C4TZD
State University of New York Curated by ChEMBL					More data for this Ligand-Target Pair
Voltage-dependent L-type calcium channel subunit alpha-1C (RAT)	BDBM50079465 (4-[5-(2-Biphenyl-2-yl-ethyl)-3-methyl-isoxazol-4-y...) Show SMILES Show InChI	PDB UniProtKB/SwissProt GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	46	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
State University of New York Curated by ChEMBL					Assay Description Displacement of [3H](+)-PN200-110 binding from calcium channels of rat cardiac membranes.				J Med Chem 42: 3087-93 (1999) Article DOI: 10.1021/jm980439q BindingDB Entry DOI: 10.7270/Q20C4TZD
State University of New York Curated by ChEMBL					More data for this Ligand-Target Pair
Voltage-dependent L-type calcium channel subunit alpha-1C (Homo sapiens (Human))	BDBM50013021 (4-(5-Ethyl-3-methyl-isoxazol-4-yl)-2,6-dimethyl-1,...) Show SMILES Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	52	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
State University of New York Curated by ChEMBL					Assay Description Inhibition of [3H]-PN-200110 binding to Calcium channel in guinea pig heart membrane				J Med Chem 33: 2255-9 (1990) BindingDB Entry DOI: 10.7270/Q2KS6QHH
State University of New York Curated by ChEMBL					More data for this Ligand-Target Pair
Voltage-dependent L-type calcium channel subunit alpha-1C (RAT)	BDBM50079461 (2,6-Dimethyl-4-(5-phenethyl-3-phenyl-isoxazol-4-yl...) Show SMILES Show InChI	PDB UniProtKB/SwissProt GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	55	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
State University of New York Curated by ChEMBL					Assay Description Displacement of [3H](+)-PN200-110 binding from calcium channels of rat cardiac membranes.				J Med Chem 42: 3087-93 (1999) Article DOI: 10.1021/jm980439q BindingDB Entry DOI: 10.7270/Q20C4TZD
State University of New York Curated by ChEMBL					More data for this Ligand-Target Pair
Voltage-dependent L-type calcium channel subunit alpha-1C/alpha-1D/alpha-1F/alpha-1S (Homo sapiens (Human))	BDBM50013021 (4-(5-Ethyl-3-methyl-isoxazol-4-yl)-2,6-dimethyl-1,...) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia antibodypedia antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	63	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
State University of New York Curated by ChEMBL					Assay Description Inhibition of [3H]PN-200110 binding to Calcium channel in guinea pig ileum membrane				J Med Chem 33: 2255-9 (1990) BindingDB Entry DOI: 10.7270/Q2KS6QHH
State University of New York Curated by ChEMBL					More data for this Ligand-Target Pair
Voltage-dependent L-type calcium channel subunit alpha-1C (Homo sapiens (Human))	BDBM50079461 (2,6-Dimethyl-4-(5-phenethyl-3-phenyl-isoxazol-4-yl...) Show SMILES Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	73	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
State University of New York Curated by ChEMBL					Assay Description Displacement of [3H](+)-PN200-110 binding to calcium channels in guinea pig cardiac membranes.				J Med Chem 42: 3087-93 (1999) Article DOI: 10.1021/jm980439q BindingDB Entry DOI: 10.7270/Q20C4TZD
State University of New York Curated by ChEMBL					More data for this Ligand-Target Pair
Voltage-dependent L-type calcium channel subunit alpha-1C/alpha-1D/alpha-1F/alpha-1S (Homo sapiens (Human))	BDBM50013026 (2,6-Dimethyl-4-(5-pentyl-3-phenyl-isoxazol-4-yl)-1...) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia antibodypedia antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	78	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
State University of New York Curated by ChEMBL					Assay Description Inhibition of [3H]PN-200110 binding to Calcium channel in guinea pig ileum membrane				J Med Chem 33: 2255-9 (1990) BindingDB Entry DOI: 10.7270/Q2KS6QHH
State University of New York Curated by ChEMBL					More data for this Ligand-Target Pair
Voltage-dependent L-type calcium channel subunit alpha-1C (Homo sapiens (Human))	BDBM50013026 (2,6-Dimethyl-4-(5-pentyl-3-phenyl-isoxazol-4-yl)-1...) Show SMILES Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	79	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
State University of New York Curated by ChEMBL					Assay Description Inhibition of [3H]-PN-200110 binding to Calcium channel in guinea pig heart membrane				J Med Chem 33: 2255-9 (1990) BindingDB Entry DOI: 10.7270/Q2KS6QHH
State University of New York Curated by ChEMBL					More data for this Ligand-Target Pair
Voltage-dependent L-type calcium channel subunit alpha-1C (Homo sapiens (Human))	BDBM50079465 (4-[5-(2-Biphenyl-2-yl-ethyl)-3-methyl-isoxazol-4-y...) Show SMILES Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	91	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
State University of New York Curated by ChEMBL					Assay Description Displacement of [3H](+)-PN200-110 binding to calcium channels in guinea pig cardiac membranes.				J Med Chem 42: 3087-93 (1999) Article DOI: 10.1021/jm980439q BindingDB Entry DOI: 10.7270/Q20C4TZD
State University of New York Curated by ChEMBL					More data for this Ligand-Target Pair
Voltage-dependent L-type calcium channel subunit alpha-1C (Homo sapiens (Human))	BDBM50013024 (4-(3,5-Dimethyl-isoxazol-4-yl)-2,6-dimethyl-1,4-di...) Show SMILES Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	122	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
State University of New York Curated by ChEMBL					Assay Description Inhibition of [3H]-PN-200110 binding to Calcium channel in guinea pig heart membrane				J Med Chem 33: 2255-9 (1990) BindingDB Entry DOI: 10.7270/Q2KS6QHH
State University of New York Curated by ChEMBL					More data for this Ligand-Target Pair
Voltage-dependent L-type calcium channel subunit alpha-1C/alpha-1D/alpha-1F/alpha-1S (Homo sapiens (Human))	BDBM50013024 (4-(3,5-Dimethyl-isoxazol-4-yl)-2,6-dimethyl-1,4-di...) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia antibodypedia antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	173	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
State University of New York Curated by ChEMBL					Assay Description Inhibition of [3H]PN-200110 binding to Calcium channel in guinea pig ileum membrane				J Med Chem 33: 2255-9 (1990) BindingDB Entry DOI: 10.7270/Q2KS6QHH
State University of New York Curated by ChEMBL					More data for this Ligand-Target Pair
Voltage-dependent L-type calcium channel subunit alpha-1C/alpha-1D/alpha-1F/alpha-1S (Homo sapiens (Human))	BDBM50013023 (4-(5-Isopropyl-3-phenyl-isoxazol-4-yl)-2,6-dimethy...) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia antibodypedia antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	254	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
State University of New York Curated by ChEMBL					Assay Description Inhibition of [3H]PN-200110 binding to Calcium channel in guinea pig ileum membrane				J Med Chem 33: 2255-9 (1990) BindingDB Entry DOI: 10.7270/Q2KS6QHH
State University of New York Curated by ChEMBL					More data for this Ligand-Target Pair
Voltage-dependent L-type calcium channel subunit alpha-1C (Homo sapiens (Human))	BDBM50013023 (4-(5-Isopropyl-3-phenyl-isoxazol-4-yl)-2,6-dimethy...) Show SMILES Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	417	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
State University of New York Curated by ChEMBL					Assay Description Inhibition of [3H]-PN-200110 binding to Calcium channel in guinea pig heart membrane				J Med Chem 33: 2255-9 (1990) BindingDB Entry DOI: 10.7270/Q2KS6QHH
State University of New York Curated by ChEMBL					More data for this Ligand-Target Pair
Metabotropic glutamate receptor 5 (Homo sapiens (Human))	BDBM50450061 (CHEMBL4166199) Show SMILES Cc1ccc(cc1)-n1nc(C)c2conc2c1=O Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	1.88E+3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
University of Montana Curated by ChEMBL					Assay Description Displacement of MPEP from mGluR5 (unknown origin) after 3 hrs by liquid scintillation counting method				Bioorg Med Chem 26: 4797-4803 (2018) Article DOI: 10.1016/j.bmc.2018.08.012 BindingDB Entry DOI: 10.7270/Q2Q242TX
University of Montana Curated by ChEMBL					More data for this Ligand-Target Pair
Metabotropic glutamate receptor 5 (Homo sapiens (Human))	BDBM50450078 (CHEMBL4167825) Show SMILES Cc1nn(-c2cc(Cl)cc(Cl)c2)c(=O)c2nocc12 Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	3.08E+3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
University of Montana Curated by ChEMBL					Assay Description Displacement of MPEP from mGluR5 (unknown origin) after 3 hrs by liquid scintillation counting method				Bioorg Med Chem 26: 4797-4803 (2018) Article DOI: 10.1016/j.bmc.2018.08.012 BindingDB Entry DOI: 10.7270/Q2Q242TX
University of Montana Curated by ChEMBL					More data for this Ligand-Target Pair
Metabotropic glutamate receptor 5 (Homo sapiens (Human))	BDBM50450074 (CHEMBL4171187) Show SMILES COc1ccc(cc1)-n1nc(C)c2conc2c1=O Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	>1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
University of Montana Curated by ChEMBL					Assay Description Displacement of MPEP from mGluR5 (unknown origin) after 3 hrs by liquid scintillation counting method				Bioorg Med Chem 26: 4797-4803 (2018) Article DOI: 10.1016/j.bmc.2018.08.012 BindingDB Entry DOI: 10.7270/Q2Q242TX
University of Montana Curated by ChEMBL					More data for this Ligand-Target Pair
Metabotropic glutamate receptor 5 (Homo sapiens (Human))	BDBM50450059 (CHEMBL4160584) Show SMILES Cc1nn(-c2ccc(F)cc2)c(=O)c2nocc12 Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	>1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
University of Montana Curated by ChEMBL					Assay Description Displacement of MPEP from mGluR5 (unknown origin) after 3 hrs by liquid scintillation counting method				Bioorg Med Chem 26: 4797-4803 (2018) Article DOI: 10.1016/j.bmc.2018.08.012 BindingDB Entry DOI: 10.7270/Q2Q242TX
University of Montana Curated by ChEMBL					More data for this Ligand-Target Pair
Metabotropic glutamate receptor 5 (Homo sapiens (Human))	BDBM50450076 (CHEMBL4163974) Show SMILES Cc1nn(-c2ccc(F)cc2F)c(=O)c2nocc12 Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	>1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
University of Montana Curated by ChEMBL					Assay Description Displacement of MPEP from mGluR5 (unknown origin) after 3 hrs by liquid scintillation counting method				Bioorg Med Chem 26: 4797-4803 (2018) Article DOI: 10.1016/j.bmc.2018.08.012 BindingDB Entry DOI: 10.7270/Q2Q242TX
University of Montana Curated by ChEMBL					More data for this Ligand-Target Pair
Metabotropic glutamate receptor 5 (Homo sapiens (Human))	BDBM50450077 (CHEMBL4164391) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	>1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
University of Montana Curated by ChEMBL					Assay Description Displacement of MPEP from mGluR5 (unknown origin) after 3 hrs by liquid scintillation counting method				Bioorg Med Chem 26: 4797-4803 (2018) Article DOI: 10.1016/j.bmc.2018.08.012 BindingDB Entry DOI: 10.7270/Q2Q242TX
University of Montana Curated by ChEMBL					More data for this Ligand-Target Pair
Metabotropic glutamate receptor 5 (Homo sapiens (Human))	BDBM50450075 (CHEMBL4174628) Show SMILES Cc1nn(-c2ccccc2)c(=O)c2nocc12 Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	>1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
University of Montana Curated by ChEMBL					Assay Description Displacement of MPEP from mGluR5 (unknown origin) after 3 hrs by liquid scintillation counting method				Bioorg Med Chem 26: 4797-4803 (2018) Article DOI: 10.1016/j.bmc.2018.08.012 BindingDB Entry DOI: 10.7270/Q2Q242TX
University of Montana Curated by ChEMBL					More data for this Ligand-Target Pair
Metabotropic glutamate receptor 5 (Homo sapiens (Human))	BDBM50450060 (CHEMBL4172276) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	>1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
University of Montana Curated by ChEMBL					Assay Description Displacement of MPEP from mGluR5 (unknown origin) after 3 hrs by liquid scintillation counting method				Bioorg Med Chem 26: 4797-4803 (2018) Article DOI: 10.1016/j.bmc.2018.08.012 BindingDB Entry DOI: 10.7270/Q2Q242TX
University of Montana Curated by ChEMBL					More data for this Ligand-Target Pair
Cystine/glutamate transporter (Homo sapiens (Human))	BDBM50378670 (CHEMBL600474) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	5.20E+4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
The University of Montana Curated by ChEMBL					Assay Description Competitive inhibition of [3H]L-glutamate uptake at amino acid transport system xc- in human SNB19 cells by liquid scintillation counting				Bioorg Med Chem 18: 202-13 (2010) Article DOI: 10.1016/j.bmc.2009.11.001 BindingDB Entry DOI: 10.7270/Q23J3DX8
The University of Montana Curated by ChEMBL					More data for this Ligand-Target Pair
Cystine/glutamate transporter (Homo sapiens (Human))	BDBM50109609 ((2R)-2-amino-3-mercaptopropanoic acid \| (2R)-2-ami...) Show SMILES N[C@@H](CS)C(O)=O \|r\| Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	Purchase CHEMBL DrugBank MCE KEGG MMDB PC cid PC sid UniChem Patents Similars	Article PubMed	5.90E+4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
The University of Montana Curated by ChEMBL					Assay Description Competitive inhibition of [3H]L-glutamate uptake at amino acid transport system xc- in human SNB19 cells by liquid scintillation counting				Bioorg Med Chem 18: 202-13 (2010) Article DOI: 10.1016/j.bmc.2009.11.001 BindingDB Entry DOI: 10.7270/Q23J3DX8
The University of Montana Curated by ChEMBL					More data for this Ligand-Target Pair
Cystine/glutamate transporter (Homo sapiens (Human))	BDBM50378666 (CHEMBL601837) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	6.00E+4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
The University of Montana Curated by ChEMBL					Assay Description Competitive inhibition of [3H]L-glutamate uptake at amino acid transport system xc- in human SNB19 cells by liquid scintillation counting				Bioorg Med Chem 18: 202-13 (2010) Article DOI: 10.1016/j.bmc.2009.11.001 BindingDB Entry DOI: 10.7270/Q23J3DX8
The University of Montana Curated by ChEMBL					More data for this Ligand-Target Pair
Cystine/glutamate transporter (Homo sapiens (Human))	BDBM50378667 (CHEMBL604574) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem	Article PubMed	6.40E+4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
The University of Montana Curated by ChEMBL					Assay Description Competitive inhibition of [3H]L-glutamate uptake at amino acid transport system xc- in human SNB19 cells by liquid scintillation counting				Bioorg Med Chem 18: 202-13 (2010) Article DOI: 10.1016/j.bmc.2009.11.001 BindingDB Entry DOI: 10.7270/Q23J3DX8
The University of Montana Curated by ChEMBL					More data for this Ligand-Target Pair
Cystine/glutamate transporter (Homo sapiens (Human))	BDBM50378668 (CHEMBL606915) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	1.13E+5	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
The University of Montana Curated by ChEMBL					Assay Description Competitive inhibition of [3H]L-glutamate uptake at amino acid transport system xc- in human SNB19 cells by liquid scintillation counting				Bioorg Med Chem 18: 202-13 (2010) Article DOI: 10.1016/j.bmc.2009.11.001 BindingDB Entry DOI: 10.7270/Q23J3DX8
The University of Montana Curated by ChEMBL					More data for this Ligand-Target Pair
Cystine/glutamate transporter (Homo sapiens (Human))	BDBM50378669 (CHEMBL591770) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	1.17E+5	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
The University of Montana Curated by ChEMBL					Assay Description Competitive inhibition of [3H]L-glutamate uptake at amino acid transport system xc- in human SNB19 cells by liquid scintillation counting				Bioorg Med Chem 18: 202-13 (2010) Article DOI: 10.1016/j.bmc.2009.11.001 BindingDB Entry DOI: 10.7270/Q23J3DX8
The University of Montana Curated by ChEMBL					More data for this Ligand-Target Pair
Cystine/glutamate transporter (Homo sapiens (Human))	BDBM50378665 (CHEMBL590556) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	1.47E+5	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
The University of Montana Curated by ChEMBL					Assay Description Competitive inhibition of [3H]L-glutamate uptake at amino acid transport system xc- in human SNB19 cells by liquid scintillation counting				Bioorg Med Chem 18: 202-13 (2010) Article DOI: 10.1016/j.bmc.2009.11.001 BindingDB Entry DOI: 10.7270/Q23J3DX8
The University of Montana Curated by ChEMBL					More data for this Ligand-Target Pair
ATP-dependent translocase ABCB1 (Homo sapiens (Human))	BDBM50242247 (CHEMBL4074268) Show SMILES Show InChI	PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	510	n/a	n/a	n/a	n/a	n/a	n/a
University of Montana Curated by ChEMBL					Assay Description Inhibition of MDR-1 in human Caco-2 cells after 30 mins by calcein-AM dye based fluorescence assay				Bioorg Med Chem 25: 3223-3234 (2017) Article DOI: 10.1016/j.bmc.2017.04.008 BindingDB Entry DOI: 10.7270/Q2348NS4
University of Montana Curated by ChEMBL					More data for this Ligand-Target Pair
ATP-dependent translocase ABCB1 (Homo sapiens (Human))	BDBM50242253 (CHEMBL4092304) Show SMILES Show InChI	PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	1.30E+3	n/a	n/a	n/a	n/a	n/a	n/a
University of Montana Curated by ChEMBL					Assay Description Inhibition of MDR-1 in human Caco-2 cells after 30 mins by calcein-AM dye based fluorescence assay				Bioorg Med Chem 25: 3223-3234 (2017) Article DOI: 10.1016/j.bmc.2017.04.008 BindingDB Entry DOI: 10.7270/Q2348NS4
University of Montana Curated by ChEMBL					More data for this Ligand-Target Pair
ATP-dependent translocase ABCB1 (Homo sapiens (Human))	BDBM50242254 (CHEMBL4104354) Show SMILES Show InChI	PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	1.39E+3	n/a	n/a	n/a	n/a	n/a	n/a
University of Montana Curated by ChEMBL					Assay Description Inhibition of MDR-1 in human Caco-2 cells after 30 mins by calcein-AM dye based fluorescence assay				Bioorg Med Chem 25: 3223-3234 (2017) Article DOI: 10.1016/j.bmc.2017.04.008 BindingDB Entry DOI: 10.7270/Q2348NS4
University of Montana Curated by ChEMBL					More data for this Ligand-Target Pair

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