Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50215802 (CHEMBL233559 | methyl 4-(6-(diisopentylcarbamoyl)-...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 0.890 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Institut Henri Beaufour Curated by ChEMBL | Assay Description Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CHOK1 cells | Bioorg Med Chem Lett 17: 4464-70 (2007) Article DOI: 10.1016/j.bmcl.2007.06.010 BindingDB Entry DOI: 10.7270/Q24T6J2X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50215802 (CHEMBL233559 | methyl 4-(6-(diisopentylcarbamoyl)-...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 0.890 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Institut Henri Beaufour Curated by ChEMBL | Assay Description Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CHOK1 cells | Bioorg Med Chem Lett 17: 4464-70 (2007) Article DOI: 10.1016/j.bmcl.2007.06.010 BindingDB Entry DOI: 10.7270/Q24T6J2X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50215807 (CHEMBL392092 | N,N-diisopentyl-2-(4-methoxybenzoyl...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 0.950 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Institut Henri Beaufour Curated by ChEMBL | Assay Description Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CHOK1 cells | Bioorg Med Chem Lett 17: 4464-70 (2007) Article DOI: 10.1016/j.bmcl.2007.06.010 BindingDB Entry DOI: 10.7270/Q24T6J2X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50215807 (CHEMBL392092 | N,N-diisopentyl-2-(4-methoxybenzoyl...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 0.950 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Institut Henri Beaufour Curated by ChEMBL | Assay Description Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CHOK1 cells | Bioorg Med Chem Lett 17: 4464-70 (2007) Article DOI: 10.1016/j.bmcl.2007.06.010 BindingDB Entry DOI: 10.7270/Q24T6J2X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50215841 (2-(4-benzoylphenylamino)-N,N-diisopentyl-3-(3-(pip...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 1.70 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Institut Henri Beaufour Curated by ChEMBL | Assay Description Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CHOK1 cells | Bioorg Med Chem Lett 17: 4464-70 (2007) Article DOI: 10.1016/j.bmcl.2007.06.010 BindingDB Entry DOI: 10.7270/Q24T6J2X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50215841 (2-(4-benzoylphenylamino)-N,N-diisopentyl-3-(3-(pip...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 1.70 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Institut Henri Beaufour Curated by ChEMBL | Assay Description Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CHOK1 cells | Bioorg Med Chem Lett 17: 4464-70 (2007) Article DOI: 10.1016/j.bmcl.2007.06.010 BindingDB Entry DOI: 10.7270/Q24T6J2X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50215816 (2-(4-acetylphenylamino)-N,N-diisopentyl-3-(3-(pipe...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 1.90 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Institut Henri Beaufour Curated by ChEMBL | Assay Description Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CHOK1 cells | Bioorg Med Chem Lett 17: 4464-70 (2007) Article DOI: 10.1016/j.bmcl.2007.06.010 BindingDB Entry DOI: 10.7270/Q24T6J2X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50215816 (2-(4-acetylphenylamino)-N,N-diisopentyl-3-(3-(pipe...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 1.90 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Institut Henri Beaufour Curated by ChEMBL | Assay Description Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CHOK1 cells | Bioorg Med Chem Lett 17: 4464-70 (2007) Article DOI: 10.1016/j.bmcl.2007.06.010 BindingDB Entry DOI: 10.7270/Q24T6J2X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50215844 (CHEMBL232161 | N,N-diisopentyl-2-(4-phenoxyphenyla...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 2 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Institut Henri Beaufour Curated by ChEMBL | Assay Description Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CHOK1 cells | Bioorg Med Chem Lett 17: 4464-70 (2007) Article DOI: 10.1016/j.bmcl.2007.06.010 BindingDB Entry DOI: 10.7270/Q24T6J2X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50215844 (CHEMBL232161 | N,N-diisopentyl-2-(4-phenoxyphenyla...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 2 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Institut Henri Beaufour Curated by ChEMBL | Assay Description Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CHOK1 cells | Bioorg Med Chem Lett 17: 4464-70 (2007) Article DOI: 10.1016/j.bmcl.2007.06.010 BindingDB Entry DOI: 10.7270/Q24T6J2X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50215813 (CHEMBL395226 | N,N-diisopentyl-2-(4-nitrophenylami...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 2.10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Institut Henri Beaufour Curated by ChEMBL | Assay Description Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CHOK1 cells | Bioorg Med Chem Lett 17: 4464-70 (2007) Article DOI: 10.1016/j.bmcl.2007.06.010 BindingDB Entry DOI: 10.7270/Q24T6J2X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50215813 (CHEMBL395226 | N,N-diisopentyl-2-(4-nitrophenylami...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 2.10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Institut Henri Beaufour Curated by ChEMBL | Assay Description Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CHOK1 cells | Bioorg Med Chem Lett 17: 4464-70 (2007) Article DOI: 10.1016/j.bmcl.2007.06.010 BindingDB Entry DOI: 10.7270/Q24T6J2X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50215836 (CHEMBL233757 | N,N-diisopentyl-3-(3-(piperidin-1-y...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 2.70 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Institut Henri Beaufour Curated by ChEMBL | Assay Description Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CHOK1 cells | Bioorg Med Chem Lett 17: 4464-70 (2007) Article DOI: 10.1016/j.bmcl.2007.06.010 BindingDB Entry DOI: 10.7270/Q24T6J2X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50215836 (CHEMBL233757 | N,N-diisopentyl-3-(3-(piperidin-1-y...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 2.70 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Institut Henri Beaufour Curated by ChEMBL | Assay Description Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CHOK1 cells | Bioorg Med Chem Lett 17: 4464-70 (2007) Article DOI: 10.1016/j.bmcl.2007.06.010 BindingDB Entry DOI: 10.7270/Q24T6J2X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50215820 (2-(benzo[b]thiophen-2-yl)-N,N-diisopentyl-3-(3-(pi...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents | Article PubMed | 3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Institut Henri Beaufour Curated by ChEMBL | Assay Description Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CHOK1 cells | Bioorg Med Chem Lett 17: 4464-70 (2007) Article DOI: 10.1016/j.bmcl.2007.06.010 BindingDB Entry DOI: 10.7270/Q24T6J2X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50215820 (2-(benzo[b]thiophen-2-yl)-N,N-diisopentyl-3-(3-(pi...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents | Article PubMed | 3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Institut Henri Beaufour Curated by ChEMBL | Assay Description Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CHOK1 cells | Bioorg Med Chem Lett 17: 4464-70 (2007) Article DOI: 10.1016/j.bmcl.2007.06.010 BindingDB Entry DOI: 10.7270/Q24T6J2X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50215801 (CHEMBL391664 | N,N-diisopentyl-2-(1-methyl-1H-indo...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 3.20 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Institut Henri Beaufour Curated by ChEMBL | Assay Description Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CHOK1 cells | Bioorg Med Chem Lett 17: 4464-70 (2007) Article DOI: 10.1016/j.bmcl.2007.06.010 BindingDB Entry DOI: 10.7270/Q24T6J2X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50215801 (CHEMBL391664 | N,N-diisopentyl-2-(1-methyl-1H-indo...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 3.20 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Institut Henri Beaufour Curated by ChEMBL | Assay Description Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CHOK1 cells | Bioorg Med Chem Lett 17: 4464-70 (2007) Article DOI: 10.1016/j.bmcl.2007.06.010 BindingDB Entry DOI: 10.7270/Q24T6J2X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50215828 (CHEMBL233758 | N,N-diisopentyl-2-(4-(methylcarbamo...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 3.30 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Institut Henri Beaufour Curated by ChEMBL | Assay Description Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CHOK1 cells | Bioorg Med Chem Lett 17: 4464-70 (2007) Article DOI: 10.1016/j.bmcl.2007.06.010 BindingDB Entry DOI: 10.7270/Q24T6J2X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50215828 (CHEMBL233758 | N,N-diisopentyl-2-(4-(methylcarbamo...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 3.30 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Institut Henri Beaufour Curated by ChEMBL | Assay Description Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CHOK1 cells | Bioorg Med Chem Lett 17: 4464-70 (2007) Article DOI: 10.1016/j.bmcl.2007.06.010 BindingDB Entry DOI: 10.7270/Q24T6J2X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50215812 (2-(4-acetamidophenylamino)-N,N-diisopentyl-3-(3-(p...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 3.70 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Institut Henri Beaufour Curated by ChEMBL | Assay Description Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CHOK1 cells | Bioorg Med Chem Lett 17: 4464-70 (2007) Article DOI: 10.1016/j.bmcl.2007.06.010 BindingDB Entry DOI: 10.7270/Q24T6J2X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50215812 (2-(4-acetamidophenylamino)-N,N-diisopentyl-3-(3-(p...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 3.70 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Institut Henri Beaufour Curated by ChEMBL | Assay Description Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CHOK1 cells | Bioorg Med Chem Lett 17: 4464-70 (2007) Article DOI: 10.1016/j.bmcl.2007.06.010 BindingDB Entry DOI: 10.7270/Q24T6J2X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50215800 (2-(4-acetylbenzyl)-N,N-diisopentyl-3-(3-(piperidin...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 3.90 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Institut Henri Beaufour Curated by ChEMBL | Assay Description Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CHOK1 cells | Bioorg Med Chem Lett 17: 4464-70 (2007) Article DOI: 10.1016/j.bmcl.2007.06.010 BindingDB Entry DOI: 10.7270/Q24T6J2X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50215800 (2-(4-acetylbenzyl)-N,N-diisopentyl-3-(3-(piperidin...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 3.90 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Institut Henri Beaufour Curated by ChEMBL | Assay Description Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CHOK1 cells | Bioorg Med Chem Lett 17: 4464-70 (2007) Article DOI: 10.1016/j.bmcl.2007.06.010 BindingDB Entry DOI: 10.7270/Q24T6J2X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50215823 (CHEMBL232584 | N,N-diisopentyl-3-(3-(piperidin-1-y...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 4.20 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Institut Henri Beaufour Curated by ChEMBL | Assay Description Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CHOK1 cells | Bioorg Med Chem Lett 17: 4464-70 (2007) Article DOI: 10.1016/j.bmcl.2007.06.010 BindingDB Entry DOI: 10.7270/Q24T6J2X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50215823 (CHEMBL232584 | N,N-diisopentyl-3-(3-(piperidin-1-y...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 4.20 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Institut Henri Beaufour Curated by ChEMBL | Assay Description Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CHOK1 cells | Bioorg Med Chem Lett 17: 4464-70 (2007) Article DOI: 10.1016/j.bmcl.2007.06.010 BindingDB Entry DOI: 10.7270/Q24T6J2X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50215846 (2-(3-acetylphenylamino)-N,N-diisopentyl-3-(3-(pipe...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 4.5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Institut Henri Beaufour Curated by ChEMBL | Assay Description Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CHOK1 cells | Bioorg Med Chem Lett 17: 4464-70 (2007) Article DOI: 10.1016/j.bmcl.2007.06.010 BindingDB Entry DOI: 10.7270/Q24T6J2X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50215846 (2-(3-acetylphenylamino)-N,N-diisopentyl-3-(3-(pipe...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 4.5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Institut Henri Beaufour Curated by ChEMBL | Assay Description Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CHOK1 cells | Bioorg Med Chem Lett 17: 4464-70 (2007) Article DOI: 10.1016/j.bmcl.2007.06.010 BindingDB Entry DOI: 10.7270/Q24T6J2X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50215805 (2-(4-acetylphenylamino)-N,N-diisopentyl-3-(3-(pyrr...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 4.90 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Institut Henri Beaufour Curated by ChEMBL | Assay Description Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CHOK1 cells | Bioorg Med Chem Lett 17: 4464-70 (2007) Article DOI: 10.1016/j.bmcl.2007.06.010 BindingDB Entry DOI: 10.7270/Q24T6J2X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50215805 (2-(4-acetylphenylamino)-N,N-diisopentyl-3-(3-(pyrr...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 4.90 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Institut Henri Beaufour Curated by ChEMBL | Assay Description Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CHOK1 cells | Bioorg Med Chem Lett 17: 4464-70 (2007) Article DOI: 10.1016/j.bmcl.2007.06.010 BindingDB Entry DOI: 10.7270/Q24T6J2X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50215815 (CHEMBL429943 | N,N-diisopentyl-2-(4-methoxyphenyla...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Institut Henri Beaufour Curated by ChEMBL | Assay Description Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CHOK1 cells | Bioorg Med Chem Lett 17: 4464-70 (2007) Article DOI: 10.1016/j.bmcl.2007.06.010 BindingDB Entry DOI: 10.7270/Q24T6J2X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50215815 (CHEMBL429943 | N,N-diisopentyl-2-(4-methoxyphenyla...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Institut Henri Beaufour Curated by ChEMBL | Assay Description Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CHOK1 cells | Bioorg Med Chem Lett 17: 4464-70 (2007) Article DOI: 10.1016/j.bmcl.2007.06.010 BindingDB Entry DOI: 10.7270/Q24T6J2X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50215839 (2-(biphenyl-4-ylamino)-3-(3-piperidin-1-yl-propyl)...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 5.20 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Institut Henri Beaufour Curated by ChEMBL | Assay Description Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CHOK1 cells | Bioorg Med Chem Lett 17: 4464-70 (2007) Article DOI: 10.1016/j.bmcl.2007.06.010 BindingDB Entry DOI: 10.7270/Q24T6J2X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50215839 (2-(biphenyl-4-ylamino)-3-(3-piperidin-1-yl-propyl)...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 5.20 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Institut Henri Beaufour Curated by ChEMBL | Assay Description Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CHOK1 cells | Bioorg Med Chem Lett 17: 4464-70 (2007) Article DOI: 10.1016/j.bmcl.2007.06.010 BindingDB Entry DOI: 10.7270/Q24T6J2X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50215831 (2-(4-acetylbenzylamino)-N,N-diisopentyl-3-(3-(pipe...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 5.80 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Institut Henri Beaufour Curated by ChEMBL | Assay Description Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CHOK1 cells | Bioorg Med Chem Lett 17: 4464-70 (2007) Article DOI: 10.1016/j.bmcl.2007.06.010 BindingDB Entry DOI: 10.7270/Q24T6J2X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50215831 (2-(4-acetylbenzylamino)-N,N-diisopentyl-3-(3-(pipe...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 5.80 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Institut Henri Beaufour Curated by ChEMBL | Assay Description Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CHOK1 cells | Bioorg Med Chem Lett 17: 4464-70 (2007) Article DOI: 10.1016/j.bmcl.2007.06.010 BindingDB Entry DOI: 10.7270/Q24T6J2X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50215835 (2-(4-carbamoylphenylamino)-N,N-diisopentyl-3-(3-(p...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 6.5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Institut Henri Beaufour Curated by ChEMBL | Assay Description Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CHOK1 cells | Bioorg Med Chem Lett 17: 4464-70 (2007) Article DOI: 10.1016/j.bmcl.2007.06.010 BindingDB Entry DOI: 10.7270/Q24T6J2X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50215835 (2-(4-carbamoylphenylamino)-N,N-diisopentyl-3-(3-(p...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 6.5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Institut Henri Beaufour Curated by ChEMBL | Assay Description Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CHOK1 cells | Bioorg Med Chem Lett 17: 4464-70 (2007) Article DOI: 10.1016/j.bmcl.2007.06.010 BindingDB Entry DOI: 10.7270/Q24T6J2X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50215804 (2-(1H-indol-3-yl)-N,N-diisopentyl-3-(3-(piperidin-...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 7.10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Institut Henri Beaufour Curated by ChEMBL | Assay Description Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CHOK1 cells | Bioorg Med Chem Lett 17: 4464-70 (2007) Article DOI: 10.1016/j.bmcl.2007.06.010 BindingDB Entry DOI: 10.7270/Q24T6J2X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50215804 (2-(1H-indol-3-yl)-N,N-diisopentyl-3-(3-(piperidin-...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 7.10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Institut Henri Beaufour Curated by ChEMBL | Assay Description Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CHOK1 cells | Bioorg Med Chem Lett 17: 4464-70 (2007) Article DOI: 10.1016/j.bmcl.2007.06.010 BindingDB Entry DOI: 10.7270/Q24T6J2X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50215845 (CHEMBL430165 | N,N-diisopentyl-2-(phenylamino)-3-(...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 7.20 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Institut Henri Beaufour Curated by ChEMBL | Assay Description Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CHOK1 cells | Bioorg Med Chem Lett 17: 4464-70 (2007) Article DOI: 10.1016/j.bmcl.2007.06.010 BindingDB Entry DOI: 10.7270/Q24T6J2X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50215845 (CHEMBL430165 | N,N-diisopentyl-2-(phenylamino)-3-(...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 7.20 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Institut Henri Beaufour Curated by ChEMBL | Assay Description Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CHOK1 cells | Bioorg Med Chem Lett 17: 4464-70 (2007) Article DOI: 10.1016/j.bmcl.2007.06.010 BindingDB Entry DOI: 10.7270/Q24T6J2X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50215829 (2-(4-bromophenylamino)-N,N-diisopentyl-3-(3-(piper...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 7.60 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Institut Henri Beaufour Curated by ChEMBL | Assay Description Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CHOK1 cells | Bioorg Med Chem Lett 17: 4464-70 (2007) Article DOI: 10.1016/j.bmcl.2007.06.010 BindingDB Entry DOI: 10.7270/Q24T6J2X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50215829 (2-(4-bromophenylamino)-N,N-diisopentyl-3-(3-(piper...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 7.60 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Institut Henri Beaufour Curated by ChEMBL | Assay Description Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CHOK1 cells | Bioorg Med Chem Lett 17: 4464-70 (2007) Article DOI: 10.1016/j.bmcl.2007.06.010 BindingDB Entry DOI: 10.7270/Q24T6J2X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50215833 (2-(4-acetylphenylamino)-3-(3-(diethylamino)propyl)...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 7.90 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Institut Henri Beaufour Curated by ChEMBL | Assay Description Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CHOK1 cells | Bioorg Med Chem Lett 17: 4464-70 (2007) Article DOI: 10.1016/j.bmcl.2007.06.010 BindingDB Entry DOI: 10.7270/Q24T6J2X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50215833 (2-(4-acetylphenylamino)-3-(3-(diethylamino)propyl)...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 7.90 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Institut Henri Beaufour Curated by ChEMBL | Assay Description Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CHOK1 cells | Bioorg Med Chem Lett 17: 4464-70 (2007) Article DOI: 10.1016/j.bmcl.2007.06.010 BindingDB Entry DOI: 10.7270/Q24T6J2X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50215852 (2-(4-fluorophenylamino)-N,N-diisopentyl-3-(3-(pipe...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 8.30 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Institut Henri Beaufour Curated by ChEMBL | Assay Description Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CHOK1 cells | Bioorg Med Chem Lett 17: 4464-70 (2007) Article DOI: 10.1016/j.bmcl.2007.06.010 BindingDB Entry DOI: 10.7270/Q24T6J2X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50215852 (2-(4-fluorophenylamino)-N,N-diisopentyl-3-(3-(pipe...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 8.30 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Institut Henri Beaufour Curated by ChEMBL | Assay Description Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CHOK1 cells | Bioorg Med Chem Lett 17: 4464-70 (2007) Article DOI: 10.1016/j.bmcl.2007.06.010 BindingDB Entry DOI: 10.7270/Q24T6J2X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50215811 (2-(4-chlorophenylamino)-N,N-diisopentyl-3-(3-(pipe...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 8.70 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Institut Henri Beaufour Curated by ChEMBL | Assay Description Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CHOK1 cells | Bioorg Med Chem Lett 17: 4464-70 (2007) Article DOI: 10.1016/j.bmcl.2007.06.010 BindingDB Entry DOI: 10.7270/Q24T6J2X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50215811 (2-(4-chlorophenylamino)-N,N-diisopentyl-3-(3-(pipe...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 8.70 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Institut Henri Beaufour Curated by ChEMBL | Assay Description Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CHOK1 cells | Bioorg Med Chem Lett 17: 4464-70 (2007) Article DOI: 10.1016/j.bmcl.2007.06.010 BindingDB Entry DOI: 10.7270/Q24T6J2X | |||||||||||
More data for this Ligand-Target Pair |
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