Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Sensory histidine kinase DcuS (Staphylococcus aureus) | BDBM50151876 (CHEMBL182783 | GVNACSSLF) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 3.60 | n/a | n/a | n/a | n/a |
University of Nottingham Curated by ChEMBL | Assay Description Effective concentration to antagonise accessory gene regulator C2 of Staphylococcus aureus | J Med Chem 47: 4633-41 (2004) Article DOI: 10.1021/jm0400754 BindingDB Entry DOI: 10.7270/Q2P26XM1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sensory histidine kinase DcuS (Staphylococcus aureus) | BDBM50151880 (CHEMBL426697 | YSTCYFIM) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 13 | n/a | n/a | n/a | n/a |
University of Nottingham Curated by ChEMBL | Assay Description Effective concentration to antagonise accessory gene regulator C4 of Staphylococcus aureus | J Med Chem 47: 4633-41 (2004) Article DOI: 10.1021/jm0400754 BindingDB Entry DOI: 10.7270/Q2P26XM1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sensory histidine kinase DcuS (Staphylococcus aureus) | BDBM50151879 (2-{2-[2-(2-{2-[2-(2-Amino-3-methyl-pentanoylamino)...) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 26 | n/a | n/a | n/a | n/a |
University of Nottingham Curated by ChEMBL | Assay Description Effective concentration to antagonise accessory gene regulator C3 of Staphylococcus aureus | J Med Chem 47: 4633-41 (2004) Article DOI: 10.1021/jm0400754 BindingDB Entry DOI: 10.7270/Q2P26XM1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sensory histidine kinase DcuS (Staphylococcus aureus) | BDBM50151882 (CHEMBL425533 | [15-(2-{2-[2-Amino-3-(4-hydroxy-phe...) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.10E+4 | n/a | n/a | n/a | n/a |
University of Nottingham Curated by ChEMBL | Assay Description Effective concentration to antagonise accessory gene regulator C1 of Staphylococcus aureus; range = 9-11 uM | J Med Chem 47: 4633-41 (2004) Article DOI: 10.1021/jm0400754 BindingDB Entry DOI: 10.7270/Q2P26XM1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sensory histidine kinase DcuS (Staphylococcus aureus) | BDBM50151874 (CHEMBL362838 | Tyr-Ser-Thr-cyclo(Cys-Ala-Phe-Ile-M...) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 21 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Nottingham Curated by ChEMBL | Assay Description Concentration required to inhibit quorum sensor of Staphylococcus aureus | J Med Chem 47: 4633-41 (2004) Article DOI: 10.1021/jm0400754 BindingDB Entry DOI: 10.7270/Q2P26XM1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sensory histidine kinase DcuS (Staphylococcus aureus) | BDBM50151875 (CHEMBL369309 | N-(3-Benzyl-9,12-bis-hydroxymethyl-...) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 4.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Nottingham Curated by ChEMBL | Assay Description Concentration required to inhibit quorum sensor of Staphylococcus aureus | J Med Chem 47: 4633-41 (2004) Article DOI: 10.1021/jm0400754 BindingDB Entry DOI: 10.7270/Q2P26XM1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sensory histidine kinase DcuS (Staphylococcus aureus) | BDBM50151871 (2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]...) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 10 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Nottingham Curated by ChEMBL | Assay Description Concentration required to inhibit quorum sensor of Staphylococcus aureus | J Med Chem 47: 4633-41 (2004) Article DOI: 10.1021/jm0400754 BindingDB Entry DOI: 10.7270/Q2P26XM1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sensory histidine kinase DcuS (Staphylococcus aureus) | BDBM50151874 (CHEMBL362838 | Tyr-Ser-Thr-cyclo(Cys-Ala-Phe-Ile-M...) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.300 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Nottingham Curated by ChEMBL | Assay Description Concentration required to inhibit quorum sensor of Staphylococcus aureus | J Med Chem 47: 4633-41 (2004) Article DOI: 10.1021/jm0400754 BindingDB Entry DOI: 10.7270/Q2P26XM1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sensory histidine kinase DcuS (Staphylococcus aureus) | BDBM50151876 (CHEMBL182783 | GVNACSSLF) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 86 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Nottingham Curated by ChEMBL | Assay Description Concentration required to antagonise accessory gene regulator C4 of Staphylococcus aureus | J Med Chem 47: 4633-41 (2004) Article DOI: 10.1021/jm0400754 BindingDB Entry DOI: 10.7270/Q2P26XM1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sensory histidine kinase DcuS (Staphylococcus aureus) | BDBM50151876 (CHEMBL182783 | GVNACSSLF) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.90 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Nottingham Curated by ChEMBL | Assay Description Antagonistic concentration for accessory gene regulator C1 of Staphylococcus aureus | J Med Chem 47: 4633-41 (2004) Article DOI: 10.1021/jm0400754 BindingDB Entry DOI: 10.7270/Q2P26XM1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sensory histidine kinase DcuS (Staphylococcus aureus) | BDBM50151878 (2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]...) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 256 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Nottingham Curated by ChEMBL | Assay Description Concentration required to inhibit quorum sensor of Staphylococcus aureus | J Med Chem 47: 4633-41 (2004) Article DOI: 10.1021/jm0400754 BindingDB Entry DOI: 10.7270/Q2P26XM1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sensory histidine kinase DcuS (Staphylococcus aureus) | BDBM50151881 (CHEMBL362839 | Cyclo(Ac-Cys-Asp-Phe-Ile-Met)) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 8.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Nottingham Curated by ChEMBL | Assay Description Concentration required to inhibit quorum sensor of Staphylococcus aureus | J Med Chem 47: 4633-41 (2004) Article DOI: 10.1021/jm0400754 BindingDB Entry DOI: 10.7270/Q2P26XM1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sensory histidine kinase DcuS (Staphylococcus aureus) | BDBM50151879 (2-{2-[2-(2-{2-[2-(2-Amino-3-methyl-pentanoylamino)...) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 150 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Nottingham Curated by ChEMBL | Assay Description Concentration required to antagonise accessory gene regulator C4 of Staphylococcus aureus | J Med Chem 47: 4633-41 (2004) Article DOI: 10.1021/jm0400754 BindingDB Entry DOI: 10.7270/Q2P26XM1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sensory histidine kinase DcuS (Staphylococcus aureus) | BDBM50151880 (CHEMBL426697 | YSTCYFIM) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 7.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Nottingham Curated by ChEMBL | Assay Description Antagonistic concentration for accessory gene regulator C1 of Staphylococcus aureus | J Med Chem 47: 4633-41 (2004) Article DOI: 10.1021/jm0400754 BindingDB Entry DOI: 10.7270/Q2P26XM1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sensory histidine kinase DcuS (Staphylococcus aureus) | BDBM50151877 (CHEMBL182114 | N-[9-Benzyl-6-sec-butyl-12-methyl-3...) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 5 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Nottingham Curated by ChEMBL | Assay Description Concentration required to inhibit quorum sensor of Staphylococcus aureus | J Med Chem 47: 4633-41 (2004) Article DOI: 10.1021/jm0400754 BindingDB Entry DOI: 10.7270/Q2P26XM1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sensory histidine kinase DcuS (Staphylococcus aureus) | BDBM50151879 (2-{2-[2-(2-{2-[2-(2-Amino-3-methyl-pentanoylamino)...) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 70 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Nottingham Curated by ChEMBL | Assay Description Antagonistic concentration for accessory gene regulator C1 of Staphylococcus aureus | J Med Chem 47: 4633-41 (2004) Article DOI: 10.1021/jm0400754 BindingDB Entry DOI: 10.7270/Q2P26XM1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sensory histidine kinase DcuS (Staphylococcus aureus) | BDBM50151879 (2-{2-[2-(2-{2-[2-(2-Amino-3-methyl-pentanoylamino)...) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 6 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Nottingham Curated by ChEMBL | Assay Description Concentration required to antagonise accessory gene regulator C2 of Staphylococcus aureus | J Med Chem 47: 4633-41 (2004) Article DOI: 10.1021/jm0400754 BindingDB Entry DOI: 10.7270/Q2P26XM1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sensory histidine kinase DcuS (Staphylococcus aureus) | BDBM50151880 (CHEMBL426697 | YSTCYFIM) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Nottingham Curated by ChEMBL | Assay Description Concentration required to antagonise accessory gene regulator C3 of Staphylococcus aureus | J Med Chem 47: 4633-41 (2004) Article DOI: 10.1021/jm0400754 BindingDB Entry DOI: 10.7270/Q2P26XM1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sensory histidine kinase DcuS (Staphylococcus aureus) | BDBM50151878 (2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]...) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 256 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Nottingham Curated by ChEMBL | Assay Description Concentration required to inhibit quorum sensor of Staphylococcus aureus | J Med Chem 47: 4633-41 (2004) Article DOI: 10.1021/jm0400754 BindingDB Entry DOI: 10.7270/Q2P26XM1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sensory histidine kinase DcuS (Staphylococcus aureus) | BDBM50151880 (CHEMBL426697 | YSTCYFIM) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Nottingham Curated by ChEMBL | Assay Description Concentration required to antagonise accessory gene regulator C2 of Staphylococcus aureus | J Med Chem 47: 4633-41 (2004) Article DOI: 10.1021/jm0400754 BindingDB Entry DOI: 10.7270/Q2P26XM1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sensory histidine kinase DcuS (Staphylococcus aureus) | BDBM50151877 (CHEMBL182114 | N-[9-Benzyl-6-sec-butyl-12-methyl-3...) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 5 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Nottingham Curated by ChEMBL | Assay Description Concentration required to inhibit quorum sensor of Staphylococcus aureus | J Med Chem 47: 4633-41 (2004) Article DOI: 10.1021/jm0400754 BindingDB Entry DOI: 10.7270/Q2P26XM1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sensory histidine kinase DcuS (Staphylococcus aureus) | BDBM50151871 (2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]...) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 10 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Nottingham Curated by ChEMBL | Assay Description Concentration required to inhibit quorum sensor of Staphylococcus aureus | J Med Chem 47: 4633-41 (2004) Article DOI: 10.1021/jm0400754 BindingDB Entry DOI: 10.7270/Q2P26XM1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sensory histidine kinase DcuS (Staphylococcus aureus) | BDBM50151883 (CHEMBL276191 | N-[9-Benzyl-6-sec-butyl-12-methyl-3...) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 295 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Nottingham Curated by ChEMBL | Assay Description Concentration required to inhibit quorum sensor of Staphylococcus aureus | J Med Chem 47: 4633-41 (2004) Article DOI: 10.1021/jm0400754 BindingDB Entry DOI: 10.7270/Q2P26XM1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sensory histidine kinase DcuS (Staphylococcus aureus) | BDBM50151874 (CHEMBL362838 | Tyr-Ser-Thr-cyclo(Cys-Ala-Phe-Ile-M...) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 8 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Nottingham Curated by ChEMBL | Assay Description Concentration required to inhibit quorum sensor of Staphylococcus aureus | J Med Chem 47: 4633-41 (2004) Article DOI: 10.1021/jm0400754 BindingDB Entry DOI: 10.7270/Q2P26XM1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sensory histidine kinase DcuS (Staphylococcus aureus) | BDBM50151876 (CHEMBL182783 | GVNACSSLF) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Nottingham Curated by ChEMBL | Assay Description Concentration required to antagonise accessory gene regulator C3 of Staphylococcus aureus | J Med Chem 47: 4633-41 (2004) Article DOI: 10.1021/jm0400754 BindingDB Entry DOI: 10.7270/Q2P26XM1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sensory histidine kinase DcuS (Staphylococcus aureus) | BDBM50151874 (CHEMBL362838 | Tyr-Ser-Thr-cyclo(Cys-Ala-Phe-Ile-M...) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 21 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Nottingham Curated by ChEMBL | Assay Description Concentration required to inhibit quorum sensor of Staphylococcus aureus | J Med Chem 47: 4633-41 (2004) Article DOI: 10.1021/jm0400754 BindingDB Entry DOI: 10.7270/Q2P26XM1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sensory histidine kinase DcuS (Staphylococcus aureus) | BDBM50151883 (CHEMBL276191 | N-[9-Benzyl-6-sec-butyl-12-methyl-3...) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 19 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Nottingham Curated by ChEMBL | Assay Description Concentration required to inhibit quorum sensor of Staphylococcus aureus | J Med Chem 47: 4633-41 (2004) Article DOI: 10.1021/jm0400754 BindingDB Entry DOI: 10.7270/Q2P26XM1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sensory histidine kinase DcuS (Staphylococcus aureus) | BDBM50151872 (2-{2-[4-(4-Benzoyl-phenoxy)-butyrylamino]-3-hydrox...) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 303 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Nottingham Curated by ChEMBL | Assay Description Concentration required to inhibit quorum sensor of Staphylococcus aureus | J Med Chem 47: 4633-41 (2004) Article DOI: 10.1021/jm0400754 BindingDB Entry DOI: 10.7270/Q2P26XM1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sensory histidine kinase DcuS (Staphylococcus aureus) | BDBM50151875 (CHEMBL369309 | N-(3-Benzyl-9,12-bis-hydroxymethyl-...) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 4.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Nottingham Curated by ChEMBL | Assay Description Concentration required to inhibit quorum sensor of Staphylococcus aureus | J Med Chem 47: 4633-41 (2004) Article DOI: 10.1021/jm0400754 BindingDB Entry DOI: 10.7270/Q2P26XM1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sensory histidine kinase DcuS (Staphylococcus aureus) | BDBM50151873 (2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]...) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.80 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Nottingham Curated by ChEMBL | Assay Description Concentration required to inhibit quorum sensor of Staphylococcus aureus | J Med Chem 47: 4633-41 (2004) Article DOI: 10.1021/jm0400754 BindingDB Entry DOI: 10.7270/Q2P26XM1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sensory histidine kinase DcuS (Staphylococcus aureus) | BDBM50406270 (CHEMBL4163103) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.91E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Inhibition of AIP-stimulated quorum sensing system AgrC activation in Staphylococcus aureus RN10829 harboring P3:blaZ fusion assessed as reduction in... | Eur J Med Chem 152: 370-376 (2018) Article DOI: 10.1016/j.ejmech.2018.04.053 BindingDB Entry DOI: 10.7270/Q2JM2D66 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sensory histidine kinase DcuS (Staphylococcus aureus) | BDBM50406354 (CHEMBL4169312) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 622 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Inhibition of AIP-stimulated quorum sensing system AgrC activation in Staphylococcus aureus RN10829 harboring P3:blaZ fusion assessed as reduction in... | Eur J Med Chem 152: 370-376 (2018) Article DOI: 10.1016/j.ejmech.2018.04.053 BindingDB Entry DOI: 10.7270/Q2JM2D66 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sensory histidine kinase DcuS (Staphylococcus aureus) | BDBM50406360 (CHEMBL4167382) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.43E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Inhibition of AIP-stimulated quorum sensing system AgrC activation in Staphylococcus aureus RN10829 harboring P3:blaZ fusion assessed as reduction in... | Eur J Med Chem 152: 370-376 (2018) Article DOI: 10.1016/j.ejmech.2018.04.053 BindingDB Entry DOI: 10.7270/Q2JM2D66 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sensory histidine kinase DcuS (Staphylococcus aureus) | BDBM50406396 (CHEMBL4159129) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 456 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Inhibition of AIP-stimulated quorum sensing system AgrC activation in Staphylococcus aureus RN10829 harboring P3:blaZ fusion assessed as reduction in... | Eur J Med Chem 152: 370-376 (2018) Article DOI: 10.1016/j.ejmech.2018.04.053 BindingDB Entry DOI: 10.7270/Q2JM2D66 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sensory histidine kinase DcuS (Staphylococcus aureus) | BDBM50406397 (CHEMBL4162686) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 6.90E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Inhibition of AIP-stimulated quorum sensing system AgrC activation in Staphylococcus aureus RN10829 harboring P3:blaZ fusion assessed as reduction in... | Eur J Med Chem 152: 370-376 (2018) Article DOI: 10.1016/j.ejmech.2018.04.053 BindingDB Entry DOI: 10.7270/Q2JM2D66 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sensory histidine kinase DcuS (Staphylococcus aureus) | BDBM50406399 (CHEMBL4161642) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 738 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Inhibition of AIP-stimulated quorum sensing system AgrC activation in Staphylococcus aureus RN10829 harboring P3:blaZ fusion assessed as reduction in... | Eur J Med Chem 152: 370-376 (2018) Article DOI: 10.1016/j.ejmech.2018.04.053 BindingDB Entry DOI: 10.7270/Q2JM2D66 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sensory histidine kinase DcuS (Staphylococcus aureus) | BDBM50406468 (CHEMBL4169564) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 608 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Inhibition of AIP-stimulated quorum sensing system AgrC activation in Staphylococcus aureus RN10829 harboring P3:blaZ fusion assessed as reduction in... | Eur J Med Chem 152: 370-376 (2018) Article DOI: 10.1016/j.ejmech.2018.04.053 BindingDB Entry DOI: 10.7270/Q2JM2D66 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sensory histidine kinase DcuS (Staphylococcus aureus) | BDBM50406469 (CHEMBL4174843) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 913 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Inhibition of AIP-stimulated quorum sensing system AgrC activation in Staphylococcus aureus RN10829 harboring P3:blaZ fusion assessed as reduction in... | Eur J Med Chem 152: 370-376 (2018) Article DOI: 10.1016/j.ejmech.2018.04.053 BindingDB Entry DOI: 10.7270/Q2JM2D66 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sensory histidine kinase DcuS (Staphylococcus aureus) | BDBM76798 ((E)-1-[2,4-dihydroxy-3-[(2E)-6-hydroxy-3,7-dimethy...) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.39E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Southampton Curated by ChEMBL | Assay Description Inhibition of recombinant Staphylococcus aureus AgrC autophosphorylation expressed in Escherichia coli BL21(DE3) preincubated for 15 mins followed by... | J Med Chem 61: 10473-10487 (2018) Article DOI: 10.1021/acs.jmedchem.8b01012 BindingDB Entry DOI: 10.7270/Q20P12PP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sensory histidine kinase DcuS (Staphylococcus aureus) | BDBM50468034 (CHEMBL4286992) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.40E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Southampton Curated by ChEMBL | Assay Description Inhibition of recombinant Staphylococcus aureus AgrC autophosphorylation expressed in Escherichia coli BL21(DE3) preincubated for 15 mins followed by... | J Med Chem 61: 10473-10487 (2018) Article DOI: 10.1021/acs.jmedchem.8b01012 BindingDB Entry DOI: 10.7270/Q20P12PP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sensory histidine kinase DcuS (Staphylococcus aureus) | BDBM50497017 (CHEMBL3235596) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 2.30E+4 | n/a | n/a | n/a | n/a | n/a |
University of Nottingham Curated by ChEMBL | Assay Description Binding affinity to AgrC in Staphylococcus aureus assessed as disruption of membrane dipole potential by di-8-ANEPPS fluorescence assay | J Med Chem 57: 2813-9 (2014) Article DOI: 10.1021/jm500215s BindingDB Entry DOI: 10.7270/Q2XG9V4C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sensory histidine kinase DcuS (Staphylococcus aureus) | BDBM50497018 (CHEMBL3235589) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 7.20E+4 | n/a | n/a | n/a | n/a | n/a |
University of Nottingham Curated by ChEMBL | Assay Description Binding affinity to AgrC in Staphylococcus aureus assessed as disruption of membrane dipole potential by di-8-ANEPPS fluorescence assay | J Med Chem 57: 2813-9 (2014) Article DOI: 10.1021/jm500215s BindingDB Entry DOI: 10.7270/Q2XG9V4C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sensory histidine kinase DcuS (Staphylococcus aureus) | BDBM50497019 (CHEMBL3235588) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 2.58E+5 | n/a | n/a | n/a | n/a | n/a |
University of Nottingham Curated by ChEMBL | Assay Description Binding affinity to AgrC in Staphylococcus aureus assessed as disruption of membrane dipole potential by di-8-ANEPPS fluorescence assay | J Med Chem 57: 2813-9 (2014) Article DOI: 10.1021/jm500215s BindingDB Entry DOI: 10.7270/Q2XG9V4C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sensory histidine kinase DcuS (Staphylococcus aureus) | BDBM50497020 (CHEMBL3235590) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 4.00E+3 | n/a | n/a | n/a | n/a | n/a |
University of Nottingham Curated by ChEMBL | Assay Description Binding affinity to AgrC in Staphylococcus aureus assessed as disruption of membrane dipole potential by di-8-ANEPPS fluorescence assay | J Med Chem 57: 2813-9 (2014) Article DOI: 10.1021/jm500215s BindingDB Entry DOI: 10.7270/Q2XG9V4C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sensory histidine kinase DcuS (Staphylococcus aureus) | BDBM50497021 (CHEMBL3235597) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 2.00E+3 | n/a | n/a | n/a | n/a | n/a |
University of Nottingham Curated by ChEMBL | Assay Description Binding affinity to AgrC in Staphylococcus aureus assessed as disruption of membrane dipole potential by di-8-ANEPPS fluorescence assay | J Med Chem 57: 2813-9 (2014) Article DOI: 10.1021/jm500215s BindingDB Entry DOI: 10.7270/Q2XG9V4C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sensory histidine kinase DcuS (Staphylococcus aureus) | BDBM50497022 (CHEMBL1213657) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 2.22E+5 | n/a | n/a | n/a | n/a | n/a |
University of Nottingham Curated by ChEMBL | Assay Description Binding affinity to AgrC in Staphylococcus aureus assessed as disruption of membrane dipole potential by di-8-ANEPPS fluorescence assay | J Med Chem 57: 2813-9 (2014) Article DOI: 10.1021/jm500215s BindingDB Entry DOI: 10.7270/Q2XG9V4C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sensory histidine kinase DcuS (Staphylococcus aureus) | BDBM50020375 (CHEMBL3289785) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 2.90 | n/a | n/a | n/a | n/a | n/a | n/a |
Veterans Affairs Eastern Colorado Health Care System Curated by ChEMBL | Assay Description Inhibition of AgrC in mid-exponential phase Staphylococcus aureus RN6390B assessed as beta-lactamase activity incubated for 80 mins by spectrophotome... | J Med Chem 63: 2705-2730 (2020) Article DOI: 10.1021/acs.jmedchem.9b00798 BindingDB Entry DOI: 10.7270/Q2CF9TJ1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sensory histidine kinase DcuS (Staphylococcus aureus) | BDBM50526859 (CHEMBL4518791) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 7.90 | n/a | n/a | n/a | n/a | n/a | n/a |
Veterans Affairs Eastern Colorado Health Care System Curated by ChEMBL | Assay Description Inhibition of AgrC in mid-exponential phase Staphylococcus aureus RN6390B assessed as beta-lactamase activity incubated for 80 mins by spectrophotome... | J Med Chem 63: 2705-2730 (2020) Article DOI: 10.1021/acs.jmedchem.9b00798 BindingDB Entry DOI: 10.7270/Q2CF9TJ1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sensory histidine kinase DcuS (Staphylococcus aureus) | BDBM50526860 (CHEMBL4554516) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | <1 | n/a | n/a | n/a | n/a | n/a | n/a |
Veterans Affairs Eastern Colorado Health Care System Curated by ChEMBL | Assay Description Inhibition of AgrC in mid-exponential phase Staphylococcus aureus RN6390B assessed as beta-lactamase activity incubated for 80 mins by spectrophotome... | J Med Chem 63: 2705-2730 (2020) Article DOI: 10.1021/acs.jmedchem.9b00798 BindingDB Entry DOI: 10.7270/Q2CF9TJ1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sensory histidine kinase DcuS (Staphylococcus aureus) | BDBM50526861 (CHEMBL2337554) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.10 | n/a | n/a | n/a | n/a | n/a | n/a |
Veterans Affairs Eastern Colorado Health Care System Curated by ChEMBL | Assay Description Inhibition of AgrC in mid-exponential phase Staphylococcus aureus RN8463 assessed as beta-lactamase activity incubated for 80 mins by spectrophotomet... | J Med Chem 63: 2705-2730 (2020) Article DOI: 10.1021/acs.jmedchem.9b00798 BindingDB Entry DOI: 10.7270/Q2CF9TJ1 | |||||||||||
More data for this Ligand-Target Pair |
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