Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Sterol O-acyltransferase 1 (Homo sapiens (Human)) | BDBM182852 (US9149492, Compound 1D) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 3.20 | n/a | n/a | n/a | n/a | n/a | n/a |
Trustees of Dartmouth College US Patent | Assay Description Methods for assessing the selectively of ACAT1 inhibitors are known in the art and can be based upon any conventional assay including, but not limite... | US Patent US9149492 (2015) BindingDB Entry DOI: 10.7270/Q2N015BF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Homo sapiens (Human)) | BDBM182851 (US9149492, Compound 1C) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 3.60 | n/a | n/a | n/a | n/a | n/a | n/a |
Trustees of Dartmouth College US Patent | Assay Description Methods for assessing the selectively of ACAT1 inhibitors are known in the art and can be based upon any conventional assay including, but not limite... | US Patent US9149492 (2015) BindingDB Entry DOI: 10.7270/Q2N015BF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Homo sapiens (Human)) | BDBM182849 (US9149492, Compound 1A) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 4.20 | n/a | n/a | n/a | n/a | n/a | n/a |
Trustees of Dartmouth College US Patent | Assay Description Methods for assessing the selectively of ACAT1 inhibitors are known in the art and can be based upon any conventional assay including, but not limite... | US Patent US9149492 (2015) BindingDB Entry DOI: 10.7270/Q2N015BF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Homo sapiens (Human)) | BDBM182850 (US9149492, Compound 1B) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 10.3 | n/a | n/a | n/a | n/a | n/a | n/a |
Trustees of Dartmouth College US Patent | Assay Description Methods for assessing the selectively of ACAT1 inhibitors are known in the art and can be based upon any conventional assay including, but not limite... | US Patent US9149492 (2015) BindingDB Entry DOI: 10.7270/Q2N015BF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Homo sapiens (Human)) | BDBM182848 (US9149492, Eflucimibe (F12511)) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | MCE PC cid PC sid UniChem | US Patent | n/a | n/a | 39 | n/a | n/a | n/a | n/a | n/a | n/a |
Trustees of Dartmouth College US Patent | Assay Description Methods for assessing the selectively of ACAT1 inhibitors are known in the art and can be based upon any conventional assay including, but not limite... | US Patent US9149492 (2015) BindingDB Entry DOI: 10.7270/Q2N015BF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 2 (Homo sapiens (Human)) | BDBM182848 (US9149492, Eflucimibe (F12511)) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | MCE PC cid PC sid UniChem | US Patent | n/a | n/a | 110 | n/a | n/a | n/a | n/a | n/a | n/a |
Trustees of Dartmouth College US Patent | Assay Description Methods for assessing the selectively of ACAT1 inhibitors are known in the art and can be based upon any conventional assay including, but not limite... | US Patent US9149492 (2015) BindingDB Entry DOI: 10.7270/Q2N015BF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 2 (Homo sapiens (Human)) | BDBM182849 (US9149492, Compound 1A) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 275 | n/a | n/a | n/a | n/a | n/a | n/a |
Trustees of Dartmouth College US Patent | Assay Description Methods for assessing the selectively of ACAT1 inhibitors are known in the art and can be based upon any conventional assay including, but not limite... | US Patent US9149492 (2015) BindingDB Entry DOI: 10.7270/Q2N015BF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Homo sapiens (Human)) | BDBM182847 (US9149492, K-604) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | US Patent | n/a | n/a | 450 | n/a | n/a | n/a | n/a | n/a | n/a |
Trustees of Dartmouth College US Patent | Assay Description Methods for assessing the selectively of ACAT1 inhibitors are known in the art and can be based upon any conventional assay including, but not limite... | US Patent US9149492 (2015) BindingDB Entry DOI: 10.7270/Q2N015BF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 2 (Homo sapiens (Human)) | BDBM182851 (US9149492, Compound 1C) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 530 | n/a | n/a | n/a | n/a | n/a | n/a |
Trustees of Dartmouth College US Patent | Assay Description Methods for assessing the selectively of ACAT1 inhibitors are known in the art and can be based upon any conventional assay including, but not limite... | US Patent US9149492 (2015) BindingDB Entry DOI: 10.7270/Q2N015BF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Homo sapiens (Human)) | BDBM50360304 (CHEMBL516093 | US9149492, Beauveriolide I) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 600 | n/a | n/a | n/a | n/a | n/a | n/a |
Trustees of Dartmouth College US Patent | Assay Description Methods for assessing the selectively of ACAT1 inhibitors are known in the art and can be based upon any conventional assay including, but not limite... | US Patent US9149492 (2015) BindingDB Entry DOI: 10.7270/Q2N015BF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 2 (Homo sapiens (Human)) | BDBM182852 (US9149492, Compound 1D) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 600 | n/a | n/a | n/a | n/a | n/a | n/a |
Trustees of Dartmouth College US Patent | Assay Description Methods for assessing the selectively of ACAT1 inhibitors are known in the art and can be based upon any conventional assay including, but not limite... | US Patent US9149492 (2015) BindingDB Entry DOI: 10.7270/Q2N015BF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Homo sapiens (Human)) | BDBM50360305 (CHEMBL409855 | US9149492, Beauveriolide III) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 900 | n/a | n/a | n/a | n/a | n/a | n/a |
Trustees of Dartmouth College US Patent | Assay Description Methods for assessing the selectively of ACAT1 inhibitors are known in the art and can be based upon any conventional assay including, but not limite... | US Patent US9149492 (2015) BindingDB Entry DOI: 10.7270/Q2N015BF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 2 (Homo sapiens (Human)) | BDBM182850 (US9149492, Compound 1B) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 1.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Trustees of Dartmouth College US Patent | Assay Description Methods for assessing the selectively of ACAT1 inhibitors are known in the art and can be based upon any conventional assay including, but not limite... | US Patent US9149492 (2015) BindingDB Entry DOI: 10.7270/Q2N015BF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 2 (Homo sapiens (Human)) | BDBM50360304 (CHEMBL516093 | US9149492, Beauveriolide I) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 2.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Trustees of Dartmouth College US Patent | Assay Description Methods for assessing the selectively of ACAT1 inhibitors are known in the art and can be based upon any conventional assay including, but not limite... | US Patent US9149492 (2015) BindingDB Entry DOI: 10.7270/Q2N015BF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 2 (Homo sapiens (Human)) | BDBM50360305 (CHEMBL409855 | US9149492, Beauveriolide III) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | US Patent | n/a | n/a | >2.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Trustees of Dartmouth College US Patent | Assay Description Methods for assessing the selectively of ACAT1 inhibitors are known in the art and can be based upon any conventional assay including, but not limite... | US Patent US9149492 (2015) BindingDB Entry DOI: 10.7270/Q2N015BF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Homo sapiens (Human)) | BDBM182854 (US9149492, 14) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 2.30E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Trustees of Dartmouth College US Patent | Assay Description Methods for assessing the selectively of ACAT1 inhibitors are known in the art and can be based upon any conventional assay including, but not limite... | US Patent US9149492 (2015) BindingDB Entry DOI: 10.7270/Q2N015BF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Homo sapiens (Human)) | BDBM182853 (US9149492, 13) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 2.40E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Trustees of Dartmouth College US Patent | Assay Description Methods for assessing the selectively of ACAT1 inhibitors are known in the art and can be based upon any conventional assay including, but not limite... | US Patent US9149492 (2015) BindingDB Entry DOI: 10.7270/Q2N015BF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Homo sapiens (Human)) | BDBM182855 (US9149492, 16) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 3.90E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Trustees of Dartmouth College US Patent | Assay Description Methods for assessing the selectively of ACAT1 inhibitors are known in the art and can be based upon any conventional assay including, but not limite... | US Patent US9149492 (2015) BindingDB Entry DOI: 10.7270/Q2N015BF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 2 (Homo sapiens (Human)) | BDBM182853 (US9149492, 13) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 5.30E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Trustees of Dartmouth College US Patent | Assay Description Methods for assessing the selectively of ACAT1 inhibitors are known in the art and can be based upon any conventional assay including, but not limite... | US Patent US9149492 (2015) BindingDB Entry DOI: 10.7270/Q2N015BF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Homo sapiens (Human)) | BDBM50371698 (CHEMBL408322 | US9149492, 1) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 6.10E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Trustees of Dartmouth College US Patent | Assay Description Methods for assessing the selectively of ACAT1 inhibitors are known in the art and can be based upon any conventional assay including, but not limite... | US Patent US9149492 (2015) BindingDB Entry DOI: 10.7270/Q2N015BF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Homo sapiens (Human)) | BDBM50371699 (CHEMBL270041 | US9149492, 2) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 6.50E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Trustees of Dartmouth College US Patent | Assay Description Methods for assessing the selectively of ACAT1 inhibitors are known in the art and can be based upon any conventional assay including, but not limite... | US Patent US9149492 (2015) BindingDB Entry DOI: 10.7270/Q2N015BF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 2 (Homo sapiens (Human)) | BDBM182854 (US9149492, 14) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 7.50E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Trustees of Dartmouth College US Patent | Assay Description Methods for assessing the selectively of ACAT1 inhibitors are known in the art and can be based upon any conventional assay including, but not limite... | US Patent US9149492 (2015) BindingDB Entry DOI: 10.7270/Q2N015BF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 2 (Homo sapiens (Human)) | BDBM182855 (US9149492, 16) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 9.70E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Trustees of Dartmouth College US Patent | Assay Description Methods for assessing the selectively of ACAT1 inhibitors are known in the art and can be based upon any conventional assay including, but not limite... | US Patent US9149492 (2015) BindingDB Entry DOI: 10.7270/Q2N015BF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 2 (Homo sapiens (Human)) | BDBM182847 (US9149492, K-604) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | US Patent | n/a | n/a | 1.03E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Trustees of Dartmouth College US Patent | Assay Description Methods for assessing the selectively of ACAT1 inhibitors are known in the art and can be based upon any conventional assay including, but not limite... | US Patent US9149492 (2015) BindingDB Entry DOI: 10.7270/Q2N015BF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 2 (Homo sapiens (Human)) | BDBM50371698 (CHEMBL408322 | US9149492, 1) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 2.30E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Trustees of Dartmouth College US Patent | Assay Description Methods for assessing the selectively of ACAT1 inhibitors are known in the art and can be based upon any conventional assay including, but not limite... | US Patent US9149492 (2015) BindingDB Entry DOI: 10.7270/Q2N015BF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 2 (Homo sapiens (Human)) | BDBM50371699 (CHEMBL270041 | US9149492, 2) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 4.14E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Trustees of Dartmouth College US Patent | Assay Description Methods for assessing the selectively of ACAT1 inhibitors are known in the art and can be based upon any conventional assay including, but not limite... | US Patent US9149492 (2015) BindingDB Entry DOI: 10.7270/Q2N015BF | |||||||||||
More data for this Ligand-Target Pair |