The following articles (labelled with PubMed ID or TBD) are for your review
| PMID | Data | Article Title | Organization |
|---|
| 27639363 |
141 |
Synthesis and biological evaluation of new 6-hydroxypyridazinone benzisoxazoles: Potential multi-receptor-targeting atypical antipsychotics. |
Huazhong University Of Science And Technology |
| 26483200 |
100 |
Synthesis and pharmacological evaluation of piperidine (piperazine)-substituted benzoxazole derivatives as multi-target antipsychotics. |
Huazhong University Of Science And Technology |
| 24487191 |
6 |
Synthesis and evaluation of new coumarin derivatives as potential atypical antipsychotics. |
Huazhong University Of Science And Technology |
| 23675993 |
13 |
Synthesis and biological investigation of coumarin piperazine (piperidine) derivatives as potential multireceptor atypical antipsychotics. |
Huazhong University Of Science And Technology |
| | 3 |
Optical isomers of the H1 antihistamine terfenadine: synthesis and activity |
TBA |
| 21944853 |
41 |
Mepyramine-JNJ7777120-hybrid compounds show high affinity to hH(1)R, but low affinity to hH(4)R. |
University Of Regensburg |
| 9548813 |
53 |
The selective 5-HT1B receptor inverse agonist 1'-methyl-5-[[2'-methyl-4'-(5-methyl-1,2, 4-oxadiazol-3-yl)biphenyl-4-yl]carbonyl]-2,3,6,7-tetrahydro- spiro[furo[2,3-f]indole-3,4'-piperidine] (SB-224289) potently blocks terminal 5-HT autoreceptor function both in vitro and in vivo. |
Smithkline Beecham Pharmaceuticals |
| 7650688 |
6 |
The histamine H1-receptor antagonist binding site. A stereoselective pharmacophoric model based upon (semi-)rigid H1-antagonists and including a known interaction site on the receptor. |
Vrije Universiteit |
| 20875743 |
90 |
Discovery of {1-[4-(2-{hexahydropyrrolo[3,4-c]pyrrol-2(1H)-yl}-1H-benzimidazol-1-yl)piperidin-1-yl]cyclooctyl}methanol, systemically potent novel non-peptide agonist of nociceptin/orphanin FQ receptor as analgesic for the treatment of neuropathic pain: design, synthesis, and structure-activity rela |
Pfizer |
| 18950149 |
75 |
Acylguanidines as bioisosteres of guanidines: NG-acylated imidazolylpropylguanidines, a new class of histamine H2 receptor agonists. |
University Of Regensburg |
| 18052318 |
30 |
4-acyl-1-(4-aminoalkoxyphenyl)-2-ketopiperazines as a novel class of non-brain-penetrant histamine H3 receptor antagonists. |
Glaxosmithkline |
| 12672253 |
60 |
Novel nonimidazole histamine H3 receptor antagonists: 1-(4-(phenoxymethyl)benzyl)piperidines and related compounds. |
Freie Universit£T Berlin |
| 12190321 |
55 |
Influence of bulky substituents on histamine h(3) receptor agonist/antagonist properties. |
Freie Universit£T Berlin |
| 9703460 |
52 |
Studies on quinazolines and 1,2,4-benzothiadiazine 1,1-dioxides. 8.1, 2 synthesis and pharmacological evaluation of tricyclic fused quinazolines and 1,2,4-benzothiadiazine 1,1-dioxides as potential alpha1-adrenoceptor antagonists. |
National Taiwan University |
| 7562938 |
17 |
New antihistamines: substituted piperazine and piperidine derivatives as novel H1-antagonists. |
Wyeth-Ayerst Research |
| 1353796 |
17 |
Synthesis and antihistaminic activity of some thiazolidin-4-ones. |
Universit£ |
| 1350797 |
21 |
Synthesis and antiallergic activity of 11-(aminoalkylidene)-6,11-dihydrodibenz[b,e]oxepin derivatives. |
Kyowa Hakko Kogyo |
| 1908521 |
106 |
Naphthosultam derivatives: a new class of potent and selective 5-HT2 antagonists. |
Centre De Recherches De Vitry Alfortville Rh£Ne-Poulenc Rorer |
| 2879912 |
55 |
Synthesis of 2-(4-substituted-1-piperazinyl)benzimidazoles as H1-antihistaminic agents. |
TBA |
| 21498080 |
45 |
N-Alkenyl and cycloalkyl carbamates as dual acting histamine H3 and H4 receptor ligands. |
Jagiellonian University Medical College |
| 20812727 |
157 |
Synthesis, structure-affinity relationships, and radiolabeling of selective high-affinity 5-HT4 receptor ligands as prospective imaging probes for positron emission tomography. |
National Institute Of Mental Health |
| 19072656 |
110 |
Discovery of a new class of potential multifunctional atypical antipsychotic agents targeting dopamine D3 and serotonin 5-HT1A and 5-HT2A receptors: design, synthesis, and effects on behavior. |
University Of Siena |
| 16246552 |
57 |
Novel histamine H3 receptor antagonists based on the 4-[(1H-imidazol-4-yl)methyl]piperidine scaffold. |
The Schering Plough Research Institute |
| 15686934 |
20 |
Synthesis and structure-activity relationships of piperidinylpyrrolopyridine derivatives as potent and selective H1 antagonists. |
RhôNe-Poulenc Rorer |
| 15566302 |
101 |
Synthesis and structure-activity relationships of novel histamine H1 antagonists: indolylpiperidinyl benzoic acid derivatives. |
RhôNe-Poulenc Rorer |
| 15115409 |
72 |
4-(omega-(alkyloxy)alkyl)-1H-imidazole derivatives as histamine H(3) receptor antagonists/agonists. |
Freie UniversitäT Berlin |
| 11855993 |
91 |
Development of a new class of nonimidazole histamine H(3) receptor ligands with combined inhibitory histamine N-methyltransferase activity. |
Freie UniversitäT Berlin |
| 10966752 |
60 |
New histamine H(3)-receptor ligands of the proxifan series: imoproxifan and other selective antagonists with high oral in vivo potency. |
Freie UniversitäT Berlin |
| 10866399 |
10 |
Conformationally-restricted ligands for the histamine H1 receptor. |
University Of Bath |
| 10841797 |
110 |
Design, synthesis, and structure-activity relationships of phthalimide-phenylpiperazines: a novel series of potent and selective alpha(1)(a)-adrenergic receptor antagonists. |
The R. W. Johnson Pharmaceutical Research Institute |
| 9873505 |
50 |
Novel H3 receptor antagonists. Sulfonamide homologs of histamine. |
Schering-Plough Research Institute |
| 9871662 |
15 |
Trans-4-methyl-3-imidazoyl pyrrolidine as a potent, highly selective histamine H3 receptor agonist in vivo. |
Schering-Plough Research Institute |
| 8676353 |
140 |
Novel carbamates as potent histamine H3 receptor antagonists with high in vitro and oral in vivo activity. |
Freie UniversitäT Berlin |
| 8093908 |
15 |
Dibenz[b,e]oxepin derivatives: novel antiallergic agents possessing thromboxane A2 and histamine H1 dual antagonizing activity. 1. |
Kyowa Hakko Kogyo |
| 7752184 |
12 |
A novel pyrrolidine analog of histamine as a potent, highly selective histamine H3 receptor agonist. |
Schering-Plough Research Institute |
| 7608912 |
6 |
(Piperidinylalkoxy)chromones: novel antihistamines with additional antagonistic activity against leukotriene D4. |
Vrije Universiteit |
| 2562852 |
6 |
Synthesis and antiallergy activity of 4-(diarylhydroxymethyl)-1-[3-(aryloxy)propyl]piperidines and structurally related compounds. |
A.H. Robins |
| 1673158 |
9 |
Optical isomers of rocastine and close analogues: synthesis and H1 antihistaminic activity of its enantiomers and their structural relationship to the classical antihistamines. |
A.H. Robins |
| 26214585 |
23 |
Virtual Screening for UDP-Galactopyranose Mutase Ligands Identifies a New Class of Antimycobacterial Agents. |
University Of Wisconsin-Madison |
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