58 articles for thisTarget

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The following articles (labelled with PubMed ID or TBD) are for your review

PMID	Data	Article Title	Organization
27100031	85	A structural insight into the P1S1 binding mode of diaminoethylphosphonic and phosphinic acids, selective inhibitors of alanine aminopeptidases.	Wroclaw University of Technology
26629857	44	Novel leucine ureido derivatives as aminopeptidase N inhibitors. Design, synthesis and activity evaluation.	Fudan University
26463133	22	Influence of polar side chains modifications on the dual enkephalinase inhibitory activity and conformation of human opiorphin, a pain perception related peptide.	Institute of Advanced Chemistry of Catalonia (Iqac-Csic)
26241877	7	Modulation of disulfide dual ENKephalinase inhibitors (DENKIs) activity by a transient N-protection for pain alleviation by oral route.	Pharmaleads
25982416	43	Exploring S1 plasticity and probing S1' subsite of mammalian aminopeptidase N/CD13 with highly potent and selective aminobenzosuberone inhibitors.	Universit£
25192493	57	Structure-guided, single-point modifications in the phosphinic dipeptide structure yield highly potent and selective inhibitors of neutral aminopeptidases.	University of Athens
24927250	18	New orally active dual enkephalinase inhibitors (DENKIs) for central and peripheral pain treatment.	Pharmaleads
23860593	17	Novelß-dicarbonyl derivatives as inhibitors of aminopeptidase N (APN).	Shandong University
23664876	1	Solid phase synthesis and biological evaluation of probestin as an angiogenesis inhibitor.	The University of Oklahoma Health Sciences Center
23528299	4	Discovery of a synthetic Aminopeptidase N inhibitor LB-4b as a potential anticancer agent.	Shandong University
23510562	30	Novel indoline-2,3-dione derivatives as inhibitors of aminopeptidase N (APN).	Shandong University
23428964	9	Selective aminopeptidase-N (CD13) inhibitors with relevance to cancer chemotherapy.	Universit£
23453219	29	Novel leucine ureido derivatives as inhibitors of aminopeptidase N (APN).	Shandong University
19757839	26	The replacement of His(4) in angiotensin IV by conformationally constrained residues provides highly potent and selective analogues.	Vrije Universiteit Brussel
24900417	59	Development of Synthetic Aminopeptidase N/CD13 Inhibitors to Overcome Cancer Metastasis and Angiogenesis.	TBA
22796349	34	Rapid and efficient synthesis of a novel series of substituted aminobenzosuberone derivatives as potent, selective, non-peptidic neutral aminopeptidase inhibitors.	Universit£
21780776	40	Remarkable potential of thea-aminophosphonate/phosphinate structural motif in medicinal chemistry.	Wroclaw University of Technology
22607877	38	Design, synthesis and biological evaluation of novel amino acid ureido derivatives as aminopeptidase N/CD13 inhibitors.	Shandong University
24900367	16	Proposed Bioactive Conformations of Opiorphin, an Endogenous Dual APN/NEP Inhibitor.	TBA
22224710	44	Structure-activity relationship study of opiorphin, a human dual ectopeptidase inhibitor with antinociceptive properties.	Institute of Advanced Chemistry of Catalonia (Iqac-Csic)
19822427	21	Inhibitors of bacterial N-succinyl-L,L-diaminopimelic acid desuccinylase (DapE) and demonstration of in vitro antimicrobial activity.	Loyola University
17331715	19	Synthesis, biological evaluation and structural determination of beta-aminoacyl-containing cyclic hydrazine derivatives as dipeptidyl peptidase IV (DPP-IV) inhibitors.	Korea Research Institute of Chemical Technology
15582436	7	N-hydroxy-2-(naphthalene-2-ylsulfanyl)-acetamide, a novel hydroxamic acid-based inhibitor of aminopeptidase N and its anti-angiogenic activity.	Sejong University
11585456	8	Long lasting antinociceptive properties of enkephalin degrading enzyme (NEP and APN) inhibitor prodrugs.	University of Paris
7909847	33	Investigation of the active site of aminopeptidase A using a series of new thiol-containing inhibitors.	University of Paris
12873488	11	Design, synthesis and antimalarial activity of novel, quinoline-based, zinc metallo-aminopeptidase inhibitors.	Universit£
10098663	81	Nonpeptide small-molecular inhibitors of dipeptidyl peptidase IV: N-phenylphthalimide analogs.	University of Tokyo
	40	Pseudopeptide inhibitors of aminopeptidases containing the [CH(CN)NH] surrogate as a transition-state MIMIC	TBA
21911297	40	Design, synthesis and biological evaluation of novel 1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid derivatives as aminopeptidase N/CD13 inhibitors.	Shandong University
21802307	64	Novel aminopeptidase N (APN/CD13) inhibitors derived from chloramphenicol amine.	Shandong University
21476495	31	Potent macrocyclic inhibitors of insulin-regulated aminopeptidase (IRAP) by olefin ring-closing metathesis.	Uppsala University
21306895	46	Discovery ofß-aminoacyl containing thiazolidine derivatives as potent and selective dipeptidyl peptidase IV inhibitors.	Korea Research Institute of Chemical Technology
21292493	23	Amino-benzosuberone: a novel warhead for selective inhibition of human aminopeptidase-N/CD13.	Merck Sharpe and Dohme
21047126	51	Disulfide cyclized tripeptide analogues of angiotensin IV as potent and selective inhibitors of insulin-regulated aminopeptidase (IRAP).	Uppsala University
20129718	32	Novel cyclic-imide peptidomimetics as aminopeptidase N inhibitors. Structure-based design, chemistry and activity evaluation. II.	Shandong University
20347318	49	New aromatic monoesters of alpha-aminoaralkylphosphonic acids as inhibitors of aminopeptidase N/CD13.	Wroclaw University of Technology
18718763	50	Synthesis of new sulfonyl pyrrolidine derivatives as matrix metalloproteinase inhibitors.	Shandong University
18556208	48	Ligands to the (IRAP)/AT4 receptor encompassing a 4-hydroxydiphenylmethane scaffold replacing Tyr2.	Uppsala University
18440232	38	Design, synthesis and evaluation of novel sulfonyl pyrrolidine derivatives as matrix metalloproteinase inhibitors.	Shandong University
18362041	59	Design, synthesis and preliminary evaluation of novel pyrrolidine derivatives as matrix metalloproteinase inhibitors.	Shandong University
17270439	23	Novel hydroxamic acid-related phosphinates: inhibition of neutral aminopeptidase N (APN).	Wroclaw University of Technology
31251594	57	Novel Human Aminopeptidase N Inhibitors: Discovery and Optimization of Subsite Binding Interactions.	Monash University
10090787	25	Structure-activity relationship of diaryl phosphonate esters as potent irreversible dipeptidyl peptidase IV inhibitors.	University of Antwerp (Uia)
30537832	7	Hydroxamic Acid Inhibitors Provide Cross-Species Inhibition of Plasmodium M1 and M17 Aminopeptidases.	Monash University
30737134	52	Leucine ureido derivatives as aminopeptidase N inhibitors using click chemistry. Part II.	Shandong University
22707871	12	Kinetic studies of novel inhibitors of endomorphin degrading enzymes.	TBA
18386881	38	Beta-homo-amino acid scan of angiotensin IV.	Vrije Universiteit Brussel
9464355	59	Novel potent nonpeptide aminopeptidase N inhibitors with a cyclic imide skeleton.	University of Tokyo
29630364	63	Design of Aminopeptidase N Inhibitors as Anti-cancer Agents.	Jadavpur University
29202398	17	Synthesis and biological characterization of ubenimex-fluorouracil conjugates for anti-cancer therapy.	Shandong University
28803047	20	Puromycin based inhibitors of aminopeptidases for the potential treatment of hematologic malignancies.	University of Minnesota
29859750	56	Novel leucine ureido derivatives as aminopeptidase N inhibitors using click chemistry.	Shandong University
1738140	26	alpha-Keto amide inhibitors of aminopeptidases.	University of Wisconsin-Madison
28442252	62	Approaches towards the development of chimeric DPP4/ACE inhibitors for treating metabolic syndrome.	Ranbaxy Laboratories