Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Poly [ADP-ribose] polymerase tankyrase-1 [1091-1325] (Homo sapiens (Human)) | BDBM231074 (US9340549, 98) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.316 | n/a | n/a | n/a | n/a | n/a | 25 |
AMGEN INC. US Patent | Assay Description The tankyrase 1 biochemical activity of the compounds was assayed in the following assay buffer (50 mM MOPS pH7.5, 100 mM NaCl, 2.5 mM MgCl2, 0.01% T... | US Patent US9340549 (2016) BindingDB Entry DOI: 10.7270/Q2SN07VD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Poly [ADP-ribose] polymerase tankyrase-1 [1091-1325] (Homo sapiens (Human)) | BDBM231158 (US9340549, 178) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.375 | n/a | n/a | n/a | n/a | n/a | 25 |
AMGEN INC. US Patent | Assay Description The tankyrase 1 biochemical activity of the compounds was assayed in the following assay buffer (50 mM MOPS pH7.5, 100 mM NaCl, 2.5 mM MgCl2, 0.01% T... | US Patent US9340549 (2016) BindingDB Entry DOI: 10.7270/Q2SN07VD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Poly [ADP-ribose] polymerase tankyrase-1 [1091-1325] (Homo sapiens (Human)) | BDBM231152 (US9340549, 174) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 1.01 | n/a | n/a | n/a | n/a | n/a | 25 |
AMGEN INC. US Patent | Assay Description The tankyrase 1 biochemical activity of the compounds was assayed in the following assay buffer (50 mM MOPS pH7.5, 100 mM NaCl, 2.5 mM MgCl2, 0.01% T... | US Patent US9340549 (2016) BindingDB Entry DOI: 10.7270/Q2SN07VD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Poly [ADP-ribose] polymerase tankyrase-1 [1091-1325] (Homo sapiens (Human)) | BDBM50434155 (CHEMBL2381946 | US9340549, 60) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 1.09 | n/a | n/a | n/a | n/a | n/a | 25 |
AMGEN INC. US Patent | Assay Description The tankyrase 1 biochemical activity of the compounds was assayed in the following assay buffer (50 mM MOPS pH7.5, 100 mM NaCl, 2.5 mM MgCl2, 0.01% T... | US Patent US9340549 (2016) BindingDB Entry DOI: 10.7270/Q2SN07VD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Poly [ADP-ribose] polymerase tankyrase-1 [1091-1325] (Homo sapiens (Human)) | BDBM231030 (US9340549, 47) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 1.12 | n/a | n/a | n/a | n/a | n/a | 25 |
AMGEN INC. US Patent | Assay Description The tankyrase 1 biochemical activity of the compounds was assayed in the following assay buffer (50 mM MOPS pH7.5, 100 mM NaCl, 2.5 mM MgCl2, 0.01% T... | US Patent US9340549 (2016) BindingDB Entry DOI: 10.7270/Q2SN07VD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Poly [ADP-ribose] polymerase tankyrase-1 [1091-1325] (Homo sapiens (Human)) | BDBM50444583 (CHEMBL3099716 | US9340549, 74) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid PDB UniChem Similars | PDB US Patent | n/a | n/a | 1.47 | n/a | n/a | n/a | n/a | n/a | 25 |
AMGEN INC. US Patent | Assay Description The tankyrase 1 biochemical activity of the compounds was assayed in the following assay buffer (50 mM MOPS pH7.5, 100 mM NaCl, 2.5 mM MgCl2, 0.01% T... | US Patent US9340549 (2016) BindingDB Entry DOI: 10.7270/Q2SN07VD | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Poly [ADP-ribose] polymerase tankyrase-1 [1091-1325] (Homo sapiens (Human)) | BDBM231039 (US9340549, 56) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 1.48 | n/a | n/a | n/a | n/a | n/a | 25 |
AMGEN INC. US Patent | Assay Description The tankyrase 1 biochemical activity of the compounds was assayed in the following assay buffer (50 mM MOPS pH7.5, 100 mM NaCl, 2.5 mM MgCl2, 0.01% T... | US Patent US9340549 (2016) BindingDB Entry DOI: 10.7270/Q2SN07VD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Poly [ADP-ribose] polymerase tankyrase-1 [1091-1325] (Homo sapiens (Human)) | BDBM231038 (US9340549, 55) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 2.95 | n/a | n/a | n/a | n/a | n/a | 25 |
AMGEN INC. US Patent | Assay Description The tankyrase 1 biochemical activity of the compounds was assayed in the following assay buffer (50 mM MOPS pH7.5, 100 mM NaCl, 2.5 mM MgCl2, 0.01% T... | US Patent US9340549 (2016) BindingDB Entry DOI: 10.7270/Q2SN07VD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Poly [ADP-ribose] polymerase tankyrase-1 [1091-1325] (Homo sapiens (Human)) | BDBM231070 (US9340549, 93) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 3 | n/a | n/a | n/a | n/a | n/a | 25 |
AMGEN INC. US Patent | Assay Description The tankyrase 1 biochemical activity of the compounds was assayed in the following assay buffer (50 mM MOPS pH7.5, 100 mM NaCl, 2.5 mM MgCl2, 0.01% T... | US Patent US9340549 (2016) BindingDB Entry DOI: 10.7270/Q2SN07VD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Poly [ADP-ribose] polymerase tankyrase-1 [1091-1325] (Homo sapiens (Human)) | BDBM231005 (US9340549, 23) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 3.04 | n/a | n/a | n/a | n/a | n/a | 25 |
AMGEN INC. US Patent | Assay Description The tankyrase 1 biochemical activity of the compounds was assayed in the following assay buffer (50 mM MOPS pH7.5, 100 mM NaCl, 2.5 mM MgCl2, 0.01% T... | US Patent US9340549 (2016) BindingDB Entry DOI: 10.7270/Q2SN07VD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Poly [ADP-ribose] polymerase tankyrase-1 [1091-1325] (Homo sapiens (Human)) | BDBM231042 (US9340549, 61) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 3.42 | n/a | n/a | n/a | n/a | n/a | 25 |
AMGEN INC. US Patent | Assay Description The tankyrase 1 biochemical activity of the compounds was assayed in the following assay buffer (50 mM MOPS pH7.5, 100 mM NaCl, 2.5 mM MgCl2, 0.01% T... | US Patent US9340549 (2016) BindingDB Entry DOI: 10.7270/Q2SN07VD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Poly [ADP-ribose] polymerase tankyrase-1 [1091-1325] (Homo sapiens (Human)) | BDBM50434156 (CHEMBL2381945 | US9340549, 103) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 3.48 | n/a | n/a | n/a | n/a | n/a | 25 |
AMGEN INC. US Patent | Assay Description The tankyrase 1 biochemical activity of the compounds was assayed in the following assay buffer (50 mM MOPS pH7.5, 100 mM NaCl, 2.5 mM MgCl2, 0.01% T... | US Patent US9340549 (2016) BindingDB Entry DOI: 10.7270/Q2SN07VD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Poly [ADP-ribose] polymerase tankyrase-1 [1091-1325] (Homo sapiens (Human)) | BDBM231034 (US9340549, 51) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 3.56 | n/a | n/a | n/a | n/a | n/a | 25 |
AMGEN INC. US Patent | Assay Description The tankyrase 1 biochemical activity of the compounds was assayed in the following assay buffer (50 mM MOPS pH7.5, 100 mM NaCl, 2.5 mM MgCl2, 0.01% T... | US Patent US9340549 (2016) BindingDB Entry DOI: 10.7270/Q2SN07VD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Poly [ADP-ribose] polymerase tankyrase-1 [1091-1325] (Homo sapiens (Human)) | BDBM50434158 (CHEMBL2381936 | US9340549, 59) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | US Patent | n/a | n/a | 3.86 | n/a | n/a | n/a | n/a | n/a | 25 |
AMGEN INC. US Patent | Assay Description The tankyrase 1 biochemical activity of the compounds was assayed in the following assay buffer (50 mM MOPS pH7.5, 100 mM NaCl, 2.5 mM MgCl2, 0.01% T... | US Patent US9340549 (2016) BindingDB Entry DOI: 10.7270/Q2SN07VD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Poly [ADP-ribose] polymerase tankyrase-1 [1091-1325] (Homo sapiens (Human)) | BDBM231163 (US9340549, 183) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 3.94 | n/a | n/a | n/a | n/a | n/a | 25 |
AMGEN INC. US Patent | Assay Description The tankyrase 1 biochemical activity of the compounds was assayed in the following assay buffer (50 mM MOPS pH7.5, 100 mM NaCl, 2.5 mM MgCl2, 0.01% T... | US Patent US9340549 (2016) BindingDB Entry DOI: 10.7270/Q2SN07VD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Poly [ADP-ribose] polymerase tankyrase-1 [1091-1325] (Homo sapiens (Human)) | BDBM231060 (US9340549, 83) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 4.07 | n/a | n/a | n/a | n/a | n/a | 25 |
AMGEN INC. US Patent | Assay Description The tankyrase 1 biochemical activity of the compounds was assayed in the following assay buffer (50 mM MOPS pH7.5, 100 mM NaCl, 2.5 mM MgCl2, 0.01% T... | US Patent US9340549 (2016) BindingDB Entry DOI: 10.7270/Q2SN07VD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Poly [ADP-ribose] polymerase tankyrase-1 [1091-1325] (Homo sapiens (Human)) | BDBM231007 (US9340549, 25) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 4.56 | n/a | n/a | n/a | n/a | n/a | 25 |
AMGEN INC. US Patent | Assay Description The tankyrase 1 biochemical activity of the compounds was assayed in the following assay buffer (50 mM MOPS pH7.5, 100 mM NaCl, 2.5 mM MgCl2, 0.01% T... | US Patent US9340549 (2016) BindingDB Entry DOI: 10.7270/Q2SN07VD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Poly [ADP-ribose] polymerase tankyrase-2 [946-1162] (Homo sapiens (Human)) | BDBM231008 (US9340549, 26 | US9340549, 27) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 4.78 | n/a | n/a | n/a | n/a | n/a | 25 |
AMGEN INC. US Patent | Assay Description The tankyrase 1 biochemical activity of the compounds was assayed in the following assay buffer (50 mM MOPS pH7.5, 100 mM NaCl, 2.5 mM MgCl2, 0.01% T... | US Patent US9340549 (2016) BindingDB Entry DOI: 10.7270/Q2SN07VD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Poly [ADP-ribose] polymerase tankyrase-1 [1091-1325] (Homo sapiens (Human)) | BDBM231069 (US9340549, 92) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 4.90 | n/a | n/a | n/a | n/a | n/a | 25 |
AMGEN INC. US Patent | Assay Description The tankyrase 1 biochemical activity of the compounds was assayed in the following assay buffer (50 mM MOPS pH7.5, 100 mM NaCl, 2.5 mM MgCl2, 0.01% T... | US Patent US9340549 (2016) BindingDB Entry DOI: 10.7270/Q2SN07VD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Poly [ADP-ribose] polymerase tankyrase-2 [946-1162] (Homo sapiens (Human)) | BDBM231012 (US9340549, 29) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 4.98 | n/a | n/a | n/a | n/a | n/a | 25 |
AMGEN INC. US Patent | Assay Description The tankyrase 1 biochemical activity of the compounds was assayed in the following assay buffer (50 mM MOPS pH7.5, 100 mM NaCl, 2.5 mM MgCl2, 0.01% T... | US Patent US9340549 (2016) BindingDB Entry DOI: 10.7270/Q2SN07VD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Poly [ADP-ribose] polymerase tankyrase-1 [1091-1325] (Homo sapiens (Human)) | BDBM231033 (US9340549, 50) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 5.11 | n/a | n/a | n/a | n/a | n/a | 25 |
AMGEN INC. US Patent | Assay Description The tankyrase 1 biochemical activity of the compounds was assayed in the following assay buffer (50 mM MOPS pH7.5, 100 mM NaCl, 2.5 mM MgCl2, 0.01% T... | US Patent US9340549 (2016) BindingDB Entry DOI: 10.7270/Q2SN07VD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Poly [ADP-ribose] polymerase tankyrase-1 [1091-1325] (Homo sapiens (Human)) | BDBM231111 (US9340549, 136) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 5.17 | n/a | n/a | n/a | n/a | n/a | 25 |
AMGEN INC. US Patent | Assay Description The tankyrase 1 biochemical activity of the compounds was assayed in the following assay buffer (50 mM MOPS pH7.5, 100 mM NaCl, 2.5 mM MgCl2, 0.01% T... | US Patent US9340549 (2016) BindingDB Entry DOI: 10.7270/Q2SN07VD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Poly [ADP-ribose] polymerase tankyrase-1 [1091-1325] (Homo sapiens (Human)) | BDBM231131 (US9340549, 156) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 5.18 | n/a | n/a | n/a | n/a | n/a | 25 |
AMGEN INC. US Patent | Assay Description The tankyrase 1 biochemical activity of the compounds was assayed in the following assay buffer (50 mM MOPS pH7.5, 100 mM NaCl, 2.5 mM MgCl2, 0.01% T... | US Patent US9340549 (2016) BindingDB Entry DOI: 10.7270/Q2SN07VD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Poly [ADP-ribose] polymerase tankyrase-1 [1091-1325] (Homo sapiens (Human)) | BDBM231012 (US9340549, 29) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 5.33 | n/a | n/a | n/a | n/a | n/a | 25 |
AMGEN INC. US Patent | Assay Description The tankyrase 1 biochemical activity of the compounds was assayed in the following assay buffer (50 mM MOPS pH7.5, 100 mM NaCl, 2.5 mM MgCl2, 0.01% T... | US Patent US9340549 (2016) BindingDB Entry DOI: 10.7270/Q2SN07VD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Poly [ADP-ribose] polymerase tankyrase-2 [946-1162] (Homo sapiens (Human)) | BDBM231007 (US9340549, 25) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 5.46 | n/a | n/a | n/a | n/a | n/a | 25 |
AMGEN INC. US Patent | Assay Description The tankyrase 1 biochemical activity of the compounds was assayed in the following assay buffer (50 mM MOPS pH7.5, 100 mM NaCl, 2.5 mM MgCl2, 0.01% T... | US Patent US9340549 (2016) BindingDB Entry DOI: 10.7270/Q2SN07VD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Poly [ADP-ribose] polymerase tankyrase-1 [1091-1325] (Homo sapiens (Human)) | BDBM231036 (US9340549, 53) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 6.52 | n/a | n/a | n/a | n/a | n/a | 25 |
AMGEN INC. US Patent | Assay Description The tankyrase 1 biochemical activity of the compounds was assayed in the following assay buffer (50 mM MOPS pH7.5, 100 mM NaCl, 2.5 mM MgCl2, 0.01% T... | US Patent US9340549 (2016) BindingDB Entry DOI: 10.7270/Q2SN07VD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Poly [ADP-ribose] polymerase tankyrase-1 [1091-1325] (Homo sapiens (Human)) | BDBM231164 (US9340549, 87) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 6.91 | n/a | n/a | n/a | n/a | n/a | 25 |
AMGEN INC. US Patent | Assay Description The tankyrase 1 biochemical activity of the compounds was assayed in the following assay buffer (50 mM MOPS pH7.5, 100 mM NaCl, 2.5 mM MgCl2, 0.01% T... | US Patent US9340549 (2016) BindingDB Entry DOI: 10.7270/Q2SN07VD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Poly [ADP-ribose] polymerase tankyrase-1 [1091-1325] (Homo sapiens (Human)) | BDBM50444584 (CHEMBL3099718 | US9340549, 95) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 6.98 | n/a | n/a | n/a | n/a | n/a | 25 |
AMGEN INC. US Patent | Assay Description The tankyrase 1 biochemical activity of the compounds was assayed in the following assay buffer (50 mM MOPS pH7.5, 100 mM NaCl, 2.5 mM MgCl2, 0.01% T... | US Patent US9340549 (2016) BindingDB Entry DOI: 10.7270/Q2SN07VD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Poly [ADP-ribose] polymerase tankyrase-1 [1091-1325] (Homo sapiens (Human)) | BDBM231037 (US9340549, 54) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 7.42 | n/a | n/a | n/a | n/a | n/a | 25 |
AMGEN INC. US Patent | Assay Description The tankyrase 1 biochemical activity of the compounds was assayed in the following assay buffer (50 mM MOPS pH7.5, 100 mM NaCl, 2.5 mM MgCl2, 0.01% T... | US Patent US9340549 (2016) BindingDB Entry DOI: 10.7270/Q2SN07VD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Poly [ADP-ribose] polymerase tankyrase-1 [1091-1325] (Homo sapiens (Human)) | BDBM231041 (US9340549, 58) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 7.46 | n/a | n/a | n/a | n/a | n/a | 25 |
AMGEN INC. US Patent | Assay Description The tankyrase 1 biochemical activity of the compounds was assayed in the following assay buffer (50 mM MOPS pH7.5, 100 mM NaCl, 2.5 mM MgCl2, 0.01% T... | US Patent US9340549 (2016) BindingDB Entry DOI: 10.7270/Q2SN07VD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Poly [ADP-ribose] polymerase tankyrase-1 [1091-1325] (Homo sapiens (Human)) | BDBM231043 (US9340549, 62) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 7.63 | n/a | n/a | n/a | n/a | n/a | 25 |
AMGEN INC. US Patent | Assay Description The tankyrase 1 biochemical activity of the compounds was assayed in the following assay buffer (50 mM MOPS pH7.5, 100 mM NaCl, 2.5 mM MgCl2, 0.01% T... | US Patent US9340549 (2016) BindingDB Entry DOI: 10.7270/Q2SN07VD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Poly [ADP-ribose] polymerase tankyrase-1 [1091-1325] (Homo sapiens (Human)) | BDBM50444583 (CHEMBL3099716 | US9340549, 74) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid PDB UniChem Similars | PDB US Patent | n/a | n/a | 8.30 | n/a | n/a | n/a | n/a | n/a | 25 |
AMGEN INC. US Patent | Assay Description The tankyrase 1 biochemical activity of the compounds was assayed in the following assay buffer (50 mM MOPS pH7.5, 100 mM NaCl, 2.5 mM MgCl2, 0.01% T... | US Patent US9340549 (2016) BindingDB Entry DOI: 10.7270/Q2SN07VD | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Poly [ADP-ribose] polymerase tankyrase-1 [1091-1325] (Homo sapiens (Human)) | BDBM231068 (US9340549, 91) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 9.01 | n/a | n/a | n/a | n/a | n/a | 25 |
AMGEN INC. US Patent | Assay Description The tankyrase 1 biochemical activity of the compounds was assayed in the following assay buffer (50 mM MOPS pH7.5, 100 mM NaCl, 2.5 mM MgCl2, 0.01% T... | US Patent US9340549 (2016) BindingDB Entry DOI: 10.7270/Q2SN07VD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Poly [ADP-ribose] polymerase tankyrase-1 [1091-1325] (Homo sapiens (Human)) | BDBM231121 (US9340549, 146) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 9.18 | n/a | n/a | n/a | n/a | n/a | 25 |
AMGEN INC. US Patent | Assay Description The tankyrase 1 biochemical activity of the compounds was assayed in the following assay buffer (50 mM MOPS pH7.5, 100 mM NaCl, 2.5 mM MgCl2, 0.01% T... | US Patent US9340549 (2016) BindingDB Entry DOI: 10.7270/Q2SN07VD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Poly [ADP-ribose] polymerase tankyrase-1 [1091-1325] (Homo sapiens (Human)) | BDBM231150 (US9340549, 173) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 9.26 | n/a | n/a | n/a | n/a | n/a | 25 |
AMGEN INC. US Patent | Assay Description The tankyrase 1 biochemical activity of the compounds was assayed in the following assay buffer (50 mM MOPS pH7.5, 100 mM NaCl, 2.5 mM MgCl2, 0.01% T... | US Patent US9340549 (2016) BindingDB Entry DOI: 10.7270/Q2SN07VD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Poly [ADP-ribose] polymerase tankyrase-1 [1091-1325] (Homo sapiens (Human)) | BDBM231008 (US9340549, 26 | US9340549, 27) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 10.3 | n/a | n/a | n/a | n/a | n/a | 25 |
AMGEN INC. US Patent | Assay Description The tankyrase 1 biochemical activity of the compounds was assayed in the following assay buffer (50 mM MOPS pH7.5, 100 mM NaCl, 2.5 mM MgCl2, 0.01% T... | US Patent US9340549 (2016) BindingDB Entry DOI: 10.7270/Q2SN07VD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Poly [ADP-ribose] polymerase tankyrase-1 [1091-1325] (Homo sapiens (Human)) | BDBM231013 (US9340549, 30) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 10.7 | n/a | n/a | n/a | n/a | n/a | 25 |
AMGEN INC. US Patent | Assay Description The tankyrase 1 biochemical activity of the compounds was assayed in the following assay buffer (50 mM MOPS pH7.5, 100 mM NaCl, 2.5 mM MgCl2, 0.01% T... | US Patent US9340549 (2016) BindingDB Entry DOI: 10.7270/Q2SN07VD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Poly [ADP-ribose] polymerase tankyrase-2 [946-1162] (Homo sapiens (Human)) | BDBM231015 (US9340549, 32) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 10.9 | n/a | n/a | n/a | n/a | n/a | 25 |
AMGEN INC. US Patent | Assay Description The tankyrase 1 biochemical activity of the compounds was assayed in the following assay buffer (50 mM MOPS pH7.5, 100 mM NaCl, 2.5 mM MgCl2, 0.01% T... | US Patent US9340549 (2016) BindingDB Entry DOI: 10.7270/Q2SN07VD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Poly [ADP-ribose] polymerase tankyrase-2 [946-1162] (Homo sapiens (Human)) | BDBM230983 (US9340549, 1) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 11 | n/a | n/a | n/a | n/a | n/a | 25 |
AMGEN INC. US Patent | Assay Description The tankyrase 1 biochemical activity of the compounds was assayed in the following assay buffer (50 mM MOPS pH7.5, 100 mM NaCl, 2.5 mM MgCl2, 0.01% T... | US Patent US9340549 (2016) BindingDB Entry DOI: 10.7270/Q2SN07VD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Poly [ADP-ribose] polymerase tankyrase-1 [1091-1325] (Homo sapiens (Human)) | BDBM231058 (US9340549, 81) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 11.4 | n/a | n/a | n/a | n/a | n/a | 25 |
AMGEN INC. US Patent | Assay Description The tankyrase 1 biochemical activity of the compounds was assayed in the following assay buffer (50 mM MOPS pH7.5, 100 mM NaCl, 2.5 mM MgCl2, 0.01% T... | US Patent US9340549 (2016) BindingDB Entry DOI: 10.7270/Q2SN07VD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Poly [ADP-ribose] polymerase tankyrase-1 [1091-1325] (Homo sapiens (Human)) | BDBM231123 (US9340549, 148) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 11.4 | n/a | n/a | n/a | n/a | n/a | 25 |
AMGEN INC. US Patent | Assay Description The tankyrase 1 biochemical activity of the compounds was assayed in the following assay buffer (50 mM MOPS pH7.5, 100 mM NaCl, 2.5 mM MgCl2, 0.01% T... | US Patent US9340549 (2016) BindingDB Entry DOI: 10.7270/Q2SN07VD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Poly [ADP-ribose] polymerase tankyrase-1 [1091-1325] (Homo sapiens (Human)) | BDBM231114 (US9340549, 139) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 11.5 | n/a | n/a | n/a | n/a | n/a | 25 |
AMGEN INC. US Patent | Assay Description The tankyrase 1 biochemical activity of the compounds was assayed in the following assay buffer (50 mM MOPS pH7.5, 100 mM NaCl, 2.5 mM MgCl2, 0.01% T... | US Patent US9340549 (2016) BindingDB Entry DOI: 10.7270/Q2SN07VD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Poly [ADP-ribose] polymerase tankyrase-1 [1091-1325] (Homo sapiens (Human)) | BDBM231020 (US9340549, 37) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 11.8 | n/a | n/a | n/a | n/a | n/a | 25 |
AMGEN INC. US Patent | Assay Description The tankyrase 1 biochemical activity of the compounds was assayed in the following assay buffer (50 mM MOPS pH7.5, 100 mM NaCl, 2.5 mM MgCl2, 0.01% T... | US Patent US9340549 (2016) BindingDB Entry DOI: 10.7270/Q2SN07VD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Poly [ADP-ribose] polymerase tankyrase-1 [1091-1325] (Homo sapiens (Human)) | BDBM231018 (US9340549, 35) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 11.8 | n/a | n/a | n/a | n/a | n/a | 25 |
AMGEN INC. US Patent | Assay Description The tankyrase 1 biochemical activity of the compounds was assayed in the following assay buffer (50 mM MOPS pH7.5, 100 mM NaCl, 2.5 mM MgCl2, 0.01% T... | US Patent US9340549 (2016) BindingDB Entry DOI: 10.7270/Q2SN07VD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Poly [ADP-ribose] polymerase tankyrase-1 [1091-1325] (Homo sapiens (Human)) | BDBM231065 (US9340549, 88) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 11.8 | n/a | n/a | n/a | n/a | n/a | 25 |
AMGEN INC. US Patent | Assay Description The tankyrase 1 biochemical activity of the compounds was assayed in the following assay buffer (50 mM MOPS pH7.5, 100 mM NaCl, 2.5 mM MgCl2, 0.01% T... | US Patent US9340549 (2016) BindingDB Entry DOI: 10.7270/Q2SN07VD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Poly [ADP-ribose] polymerase tankyrase-1 [1091-1325] (Homo sapiens (Human)) | BDBM231120 (US9340549, 145) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 13.7 | n/a | n/a | n/a | n/a | n/a | 25 |
AMGEN INC. US Patent | Assay Description The tankyrase 1 biochemical activity of the compounds was assayed in the following assay buffer (50 mM MOPS pH7.5, 100 mM NaCl, 2.5 mM MgCl2, 0.01% T... | US Patent US9340549 (2016) BindingDB Entry DOI: 10.7270/Q2SN07VD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Poly [ADP-ribose] polymerase tankyrase-1 [1091-1325] (Homo sapiens (Human)) | BDBM231075 (US9340549, 99) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 14.3 | n/a | n/a | n/a | n/a | n/a | 25 |
AMGEN INC. US Patent | Assay Description The tankyrase 1 biochemical activity of the compounds was assayed in the following assay buffer (50 mM MOPS pH7.5, 100 mM NaCl, 2.5 mM MgCl2, 0.01% T... | US Patent US9340549 (2016) BindingDB Entry DOI: 10.7270/Q2SN07VD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Poly [ADP-ribose] polymerase tankyrase-1 [1091-1325] (Homo sapiens (Human)) | BDBM231106 (US9340549, 131) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 16 | n/a | n/a | n/a | n/a | n/a | 25 |
AMGEN INC. US Patent | Assay Description The tankyrase 1 biochemical activity of the compounds was assayed in the following assay buffer (50 mM MOPS pH7.5, 100 mM NaCl, 2.5 mM MgCl2, 0.01% T... | US Patent US9340549 (2016) BindingDB Entry DOI: 10.7270/Q2SN07VD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Poly [ADP-ribose] polymerase tankyrase-1 [1091-1325] (Homo sapiens (Human)) | BDBM231077 (US9340549, 101) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 16.2 | n/a | n/a | n/a | n/a | n/a | 25 |
AMGEN INC. US Patent | Assay Description The tankyrase 1 biochemical activity of the compounds was assayed in the following assay buffer (50 mM MOPS pH7.5, 100 mM NaCl, 2.5 mM MgCl2, 0.01% T... | US Patent US9340549 (2016) BindingDB Entry DOI: 10.7270/Q2SN07VD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Poly [ADP-ribose] polymerase tankyrase-1 [1091-1325] (Homo sapiens (Human)) | BDBM231015 (US9340549, 32) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 16.8 | n/a | n/a | n/a | n/a | n/a | 25 |
AMGEN INC. US Patent | Assay Description The tankyrase 1 biochemical activity of the compounds was assayed in the following assay buffer (50 mM MOPS pH7.5, 100 mM NaCl, 2.5 mM MgCl2, 0.01% T... | US Patent US9340549 (2016) BindingDB Entry DOI: 10.7270/Q2SN07VD | |||||||||||
More data for this Ligand-Target Pair |
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