Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Motilin receptor (Homo sapiens (Human)) | BDBM50214268 ((5R,8R,11S)-8-(propan-2-yl)-11-(pyrrolidin-1-ylmet...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 4.60 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Tranzyme Pharma Inc. Curated by ChEMBL | Assay Description Displacement of [125I]-motilin from human motilin receptor expressed in CHO cells | Bioorg Med Chem Lett 17: 4187-90 (2007) Article DOI: 10.1016/j.bmcl.2007.05.043 BindingDB Entry DOI: 10.7270/Q2GF0T62 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Motilin receptor (Homo sapiens (Human)) | BDBM50214264 (1-{[(5R,8R,11S)-6,9,12-trioxo-8-(propan-2-yl)-5-{[...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 6 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Tranzyme Pharma Inc. Curated by ChEMBL | Assay Description Displacement of [125I]-motilin from human motilin receptor expressed in CHO cells | Bioorg Med Chem Lett 17: 4187-90 (2007) Article DOI: 10.1016/j.bmcl.2007.05.043 BindingDB Entry DOI: 10.7270/Q2GF0T62 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Motilin receptor (Homo sapiens (Human)) | BDBM50214270 (1-{[(5R,8R,11S)-5-[(4-chlorophenyl)methyl]-6,9,12-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 6 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Tranzyme Pharma Inc. Curated by ChEMBL | Assay Description Displacement of [125I]-motilin from human motilin receptor expressed in CHO cells | Bioorg Med Chem Lett 17: 4187-90 (2007) Article DOI: 10.1016/j.bmcl.2007.05.043 BindingDB Entry DOI: 10.7270/Q2GF0T62 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Motilin receptor (Homo sapiens (Human)) | BDBM50214266 ((5R,8R,11S)-11-[(methylamino)methyl]-8-(propan-2-y...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 6 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Tranzyme Pharma Inc. Curated by ChEMBL | Assay Description Displacement of [125I]-motilin from human motilin receptor expressed in CHO cells | Bioorg Med Chem Lett 17: 4187-90 (2007) Article DOI: 10.1016/j.bmcl.2007.05.043 BindingDB Entry DOI: 10.7270/Q2GF0T62 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Motilin receptor (Homo sapiens (Human)) | BDBM50214272 ((5R,8R,11S)-11-(aminomethyl)-8-(propan-2-yl)-5-{[3...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 15 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Tranzyme Pharma Inc. Curated by ChEMBL | Assay Description Displacement of [125I]-motilin from human motilin receptor expressed in CHO cells | Bioorg Med Chem Lett 17: 4187-90 (2007) Article DOI: 10.1016/j.bmcl.2007.05.043 BindingDB Entry DOI: 10.7270/Q2GF0T62 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Motilin receptor (Homo sapiens (Human)) | BDBM50214250 ((5R,8R,11S)-5-[(4-chlorophenyl)methyl]-11-[(dimeth...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 16 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Tranzyme Pharma Inc. Curated by ChEMBL | Assay Description Displacement of [125I]-motilin from human motilin receptor expressed in CHO cells | Bioorg Med Chem Lett 17: 4187-90 (2007) Article DOI: 10.1016/j.bmcl.2007.05.043 BindingDB Entry DOI: 10.7270/Q2GF0T62 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Motilin receptor (Homo sapiens (Human)) | BDBM50214255 ((5R,8R,11S)-11-[(5-methyl-1H-1,2,3-triazol-1-yl)me...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 17 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Tranzyme Pharma Inc. Curated by ChEMBL | Assay Description Displacement of [125I]-motilin from human motilin receptor expressed in CHO cells | Bioorg Med Chem Lett 17: 4187-90 (2007) Article DOI: 10.1016/j.bmcl.2007.05.043 BindingDB Entry DOI: 10.7270/Q2GF0T62 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Motilin receptor (Homo sapiens (Human)) | BDBM50214260 ((5R,8R,11S)-5-[(3-chlorophenyl)methyl]-8-(propan-2...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents | Article PubMed | 18 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Tranzyme Pharma Inc. Curated by ChEMBL | Assay Description Displacement of [125I]-motilin from human motilin receptor expressed in CHO cells | Bioorg Med Chem Lett 17: 4187-90 (2007) Article DOI: 10.1016/j.bmcl.2007.05.043 BindingDB Entry DOI: 10.7270/Q2GF0T62 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Motilin receptor (Homo sapiens (Human)) | BDBM50214253 ((5R,8R,11S)-8-(propan-2-yl)-11-[(pyrimidin-2-ylami...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 20 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Tranzyme Pharma Inc. Curated by ChEMBL | Assay Description Displacement of [125I]-motilin from human motilin receptor expressed in CHO cells | Bioorg Med Chem Lett 17: 4187-90 (2007) Article DOI: 10.1016/j.bmcl.2007.05.043 BindingDB Entry DOI: 10.7270/Q2GF0T62 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Motilin receptor (Homo sapiens (Human)) | BDBM50214274 ((5R,8R,11S)-11-[(5-methyl-1H-1,2,3,4-tetrazol-1-yl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents | Article PubMed | 21 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Tranzyme Pharma Inc. Curated by ChEMBL | Assay Description Displacement of [125I]-motilin from human motilin receptor expressed in CHO cells | Bioorg Med Chem Lett 17: 4187-90 (2007) Article DOI: 10.1016/j.bmcl.2007.05.043 BindingDB Entry DOI: 10.7270/Q2GF0T62 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Motilin receptor (Homo sapiens (Human)) | BDBM50214261 ((5R,8R,11S)-11-[(4,5-dimethyl-1H-1,2,3-triazol-1-y...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 23 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Tranzyme Pharma Inc. Curated by ChEMBL | Assay Description Displacement of [125I]-motilin from human motilin receptor expressed in CHO cells | Bioorg Med Chem Lett 17: 4187-90 (2007) Article DOI: 10.1016/j.bmcl.2007.05.043 BindingDB Entry DOI: 10.7270/Q2GF0T62 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Motilin receptor (Homo sapiens (Human)) | BDBM50214251 ((5R,8R,11S)-5-[(3-chlorophenyl)methyl]-11-[(dimeth...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 27 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Tranzyme Pharma Inc. Curated by ChEMBL | Assay Description Displacement of [125I]-motilin from human motilin receptor expressed in CHO cells | Bioorg Med Chem Lett 17: 4187-90 (2007) Article DOI: 10.1016/j.bmcl.2007.05.043 BindingDB Entry DOI: 10.7270/Q2GF0T62 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Motilin receptor (Homo sapiens (Human)) | BDBM50214276 (3-[(5R,8R,11S)-5-[(3-chlorophenyl)methyl]-6,9,12-t...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 27 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Tranzyme Pharma Inc. Curated by ChEMBL | Assay Description Displacement of [125I]-motilin from human motilin receptor expressed in CHO cells | Bioorg Med Chem Lett 17: 4187-90 (2007) Article DOI: 10.1016/j.bmcl.2007.05.043 BindingDB Entry DOI: 10.7270/Q2GF0T62 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Motilin receptor (Homo sapiens (Human)) | BDBM50214262 ((5R,8R,11S)-5-[(4-chlorophenyl)methyl]-11-[(methyl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 31 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Tranzyme Pharma Inc. Curated by ChEMBL | Assay Description Displacement of [125I]-motilin from human motilin receptor expressed in CHO cells | Bioorg Med Chem Lett 17: 4187-90 (2007) Article DOI: 10.1016/j.bmcl.2007.05.043 BindingDB Entry DOI: 10.7270/Q2GF0T62 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Motilin receptor (Homo sapiens (Human)) | BDBM50214267 (1-{2-[(5R,8R,11S)-5-[(3-chlorophenyl)methyl]-6,9,1...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 33 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Tranzyme Pharma Inc. Curated by ChEMBL | Assay Description Displacement of [125I]-motilin from human motilin receptor expressed in CHO cells | Bioorg Med Chem Lett 17: 4187-90 (2007) Article DOI: 10.1016/j.bmcl.2007.05.043 BindingDB Entry DOI: 10.7270/Q2GF0T62 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Motilin receptor (Homo sapiens (Human)) | BDBM50214273 ((5R,8R,11S)-5-[(3-chlorophenyl)methyl]-8-(propan-2...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents | Article PubMed | 41 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Tranzyme Pharma Inc. Curated by ChEMBL | Assay Description Displacement of [125I]-motilin from human motilin receptor expressed in CHO cells | Bioorg Med Chem Lett 17: 4187-90 (2007) Article DOI: 10.1016/j.bmcl.2007.05.043 BindingDB Entry DOI: 10.7270/Q2GF0T62 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Motilin receptor (Homo sapiens (Human)) | BDBM50214257 ((5R,8R,11S)-5-[(3-chlorophenyl)methyl]-11-[(4,5-di...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 51 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Tranzyme Pharma Inc. Curated by ChEMBL | Assay Description Displacement of [125I]-motilin from human motilin receptor expressed in CHO cells | Bioorg Med Chem Lett 17: 4187-90 (2007) Article DOI: 10.1016/j.bmcl.2007.05.043 BindingDB Entry DOI: 10.7270/Q2GF0T62 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Motilin receptor (Homo sapiens (Human)) | BDBM50214269 (1-{[(5R,8R,11S)-5-[(3-chlorophenyl)methyl]-6,9,12-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 57 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Tranzyme Pharma Inc. Curated by ChEMBL | Assay Description Displacement of [125I]-motilin from human motilin receptor expressed in CHO cells | Bioorg Med Chem Lett 17: 4187-90 (2007) Article DOI: 10.1016/j.bmcl.2007.05.043 BindingDB Entry DOI: 10.7270/Q2GF0T62 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Motilin receptor (Homo sapiens (Human)) | BDBM50214275 ((5R,8R,11S)-11-(aminomethyl)-5-[(4-chlorophenyl)me...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 60 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Tranzyme Pharma Inc. Curated by ChEMBL | Assay Description Displacement of [125I]-motilin from human motilin receptor expressed in CHO cells | Bioorg Med Chem Lett 17: 4187-90 (2007) Article DOI: 10.1016/j.bmcl.2007.05.043 BindingDB Entry DOI: 10.7270/Q2GF0T62 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Motilin receptor (Homo sapiens (Human)) | BDBM50214254 ((5R,8R,11S)-5-[(3-chlorophenyl)methyl]-11-(1H-imid...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents | Article PubMed | 62 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Tranzyme Pharma Inc. Curated by ChEMBL | Assay Description Displacement of [125I]-motilin from human motilin receptor expressed in CHO cells | Bioorg Med Chem Lett 17: 4187-90 (2007) Article DOI: 10.1016/j.bmcl.2007.05.043 BindingDB Entry DOI: 10.7270/Q2GF0T62 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Motilin receptor (Homo sapiens (Human)) | BDBM50214278 ((5R,8R,11S)-11-(aminomethyl)-5-[(3-chlorophenyl)me...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 64 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Tranzyme Pharma Inc. Curated by ChEMBL | Assay Description Displacement of [125I]-motilin from human motilin receptor expressed in CHO cells | Bioorg Med Chem Lett 17: 4187-90 (2007) Article DOI: 10.1016/j.bmcl.2007.05.043 BindingDB Entry DOI: 10.7270/Q2GF0T62 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Motilin receptor (Homo sapiens (Human)) | BDBM50214279 ((5R,8R,11S)-5-[(3-chlorophenyl)methyl]-8-(propan-2...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 87 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Tranzyme Pharma Inc. Curated by ChEMBL | Assay Description Displacement of [125I]-motilin from human motilin receptor expressed in CHO cells | Bioorg Med Chem Lett 17: 4187-90 (2007) Article DOI: 10.1016/j.bmcl.2007.05.043 BindingDB Entry DOI: 10.7270/Q2GF0T62 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Motilin receptor (Homo sapiens (Human)) | BDBM50214263 (1-{[(5R,8R,11S)-5-[(3-chlorophenyl)methyl]-6,9,12-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 100 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Tranzyme Pharma Inc. Curated by ChEMBL | Assay Description Displacement of [125I]-motilin from human motilin receptor expressed in CHO cells | Bioorg Med Chem Lett 17: 4187-90 (2007) Article DOI: 10.1016/j.bmcl.2007.05.043 BindingDB Entry DOI: 10.7270/Q2GF0T62 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Motilin receptor (Homo sapiens (Human)) | BDBM50214256 ((5R,8R,11S)-5-[(3-fluorophenyl)methyl]-8-(propan-2...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | 116 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Tranzyme Pharma Inc. Curated by ChEMBL | Assay Description Displacement of [125I]-motilin from human motilin receptor expressed in CHO cells | Bioorg Med Chem Lett 17: 4187-90 (2007) Article DOI: 10.1016/j.bmcl.2007.05.043 BindingDB Entry DOI: 10.7270/Q2GF0T62 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Motilin receptor (Homo sapiens (Human)) | BDBM50199365 ((E)-(9R,12R,15S)-9-(4-hydroxy-benzyl)-12-isopropyl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 137 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Tranzyme Pharma Inc. Curated by ChEMBL | Assay Description Displacement of [125I]-motilin from human motilin receptor expressed in CHO cells | Bioorg Med Chem Lett 17: 4187-90 (2007) Article DOI: 10.1016/j.bmcl.2007.05.043 BindingDB Entry DOI: 10.7270/Q2GF0T62 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Motilin receptor (Homo sapiens (Human)) | BDBM50214258 ((5R,8R,11S)-11-(aminomethyl)-5-[(4-hydroxyphenyl)m...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 171 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Tranzyme Pharma Inc. Curated by ChEMBL | Assay Description Displacement of [125I]-motilin from human motilin receptor expressed in CHO cells | Bioorg Med Chem Lett 17: 4187-90 (2007) Article DOI: 10.1016/j.bmcl.2007.05.043 BindingDB Entry DOI: 10.7270/Q2GF0T62 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Motilin receptor (Homo sapiens (Human)) | BDBM50214265 ((5R,8R,11S)-11-(2-aminoethyl)-5-[(4-hydroxyphenyl)...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 342 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Tranzyme Pharma Inc. Curated by ChEMBL | Assay Description Displacement of [125I]-motilin from human motilin receptor expressed in CHO cells | Bioorg Med Chem Lett 17: 4187-90 (2007) Article DOI: 10.1016/j.bmcl.2007.05.043 BindingDB Entry DOI: 10.7270/Q2GF0T62 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Motilin receptor (Homo sapiens (Human)) | BDBM50214259 ((5R,8R,11S)-5-[(4-hydroxyphenyl)methyl]-8-(propan-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 376 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Tranzyme Pharma Inc. Curated by ChEMBL | Assay Description Displacement of [125I]-motilin from human motilin receptor expressed in CHO cells | Bioorg Med Chem Lett 17: 4187-90 (2007) Article DOI: 10.1016/j.bmcl.2007.05.043 BindingDB Entry DOI: 10.7270/Q2GF0T62 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Motilin receptor (Homo sapiens (Human)) | BDBM50214271 (CHEMBL232359 | {[(5R,8R,11S)-5-[(4-chlorophenyl)me...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 543 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Tranzyme Pharma Inc. Curated by ChEMBL | Assay Description Displacement of [125I]-motilin from human motilin receptor expressed in CHO cells | Bioorg Med Chem Lett 17: 4187-90 (2007) Article DOI: 10.1016/j.bmcl.2007.05.043 BindingDB Entry DOI: 10.7270/Q2GF0T62 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Motilin receptor (Homo sapiens (Human)) | BDBM50199378 ((9R,12R,15S)-15-(4-amino-butyl)-9-(4-hydroxy-benzy...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 664 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Tranzyme Pharma Inc. Curated by ChEMBL | Assay Description Displacement of [125I]-motilin from human motilin receptor expressed in CHO cells | Bioorg Med Chem Lett 17: 4187-90 (2007) Article DOI: 10.1016/j.bmcl.2007.05.043 BindingDB Entry DOI: 10.7270/Q2GF0T62 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Motilin receptor (Homo sapiens (Human)) | BDBM50214252 ((5R,8R,11S)-11-(3-aminopropyl)-5-[(4-hydroxyphenyl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 889 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Tranzyme Pharma Inc. Curated by ChEMBL | Assay Description Displacement of [125I]-motilin from human motilin receptor expressed in CHO cells | Bioorg Med Chem Lett 17: 4187-90 (2007) Article DOI: 10.1016/j.bmcl.2007.05.043 BindingDB Entry DOI: 10.7270/Q2GF0T62 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Motilin receptor (Homo sapiens (Human)) | BDBM50214277 (CHEMBL232551 | N-{[(5R,8R,11S)-5-[(4-hydroxyphenyl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.95E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Tranzyme Pharma Inc. Curated by ChEMBL | Assay Description Displacement of [125I]-motilin from human motilin receptor expressed in CHO cells | Bioorg Med Chem Lett 17: 4187-90 (2007) Article DOI: 10.1016/j.bmcl.2007.05.043 BindingDB Entry DOI: 10.7270/Q2GF0T62 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Motilin receptor (Homo sapiens (Human)) | BDBM50199382 ((9R,12R,15S)-9-(4-hydroxy-benzyl)-12-isopropyl-10,...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2.55E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Tranzyme Pharma Inc. Curated by ChEMBL | Assay Description Displacement of [125I]-motilin from human motilin receptor expressed in CHO cells | Bioorg Med Chem Lett 17: 4187-90 (2007) Article DOI: 10.1016/j.bmcl.2007.05.043 BindingDB Entry DOI: 10.7270/Q2GF0T62 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Motilin receptor (Homo sapiens (Human)) | BDBM50214268 ((5R,8R,11S)-8-(propan-2-yl)-11-(pyrrolidin-1-ylmet...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 2 | n/a | n/a | n/a | n/a | n/a | n/a |
Tranzyme Pharma Inc. Curated by ChEMBL | Assay Description Antagonist activity against human motilin receptor in aequoscreen cells assessed as inhibition of motilin induced calcium release by aequorin assay | Bioorg Med Chem Lett 17: 4187-90 (2007) Article DOI: 10.1016/j.bmcl.2007.05.043 BindingDB Entry DOI: 10.7270/Q2GF0T62 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Motilin receptor (Homo sapiens (Human)) | BDBM50214266 ((5R,8R,11S)-11-[(methylamino)methyl]-8-(propan-2-y...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 3 | n/a | n/a | n/a | n/a | n/a | n/a |
Tranzyme Pharma Inc. Curated by ChEMBL | Assay Description Antagonist activity against human motilin receptor in aequoscreen cells assessed as inhibition of motilin induced calcium release by aequorin assay | Bioorg Med Chem Lett 17: 4187-90 (2007) Article DOI: 10.1016/j.bmcl.2007.05.043 BindingDB Entry DOI: 10.7270/Q2GF0T62 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Motilin receptor (Homo sapiens (Human)) | BDBM50214272 ((5R,8R,11S)-11-(aminomethyl)-8-(propan-2-yl)-5-{[3...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 8 | n/a | n/a | n/a | n/a | n/a | n/a |
Tranzyme Pharma Inc. Curated by ChEMBL | Assay Description Antagonist activity against human motilin receptor in aequoscreen cells assessed as inhibition of motilin induced calcium release by aequorin assay | Bioorg Med Chem Lett 17: 4187-90 (2007) Article DOI: 10.1016/j.bmcl.2007.05.043 BindingDB Entry DOI: 10.7270/Q2GF0T62 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Motilin receptor (Homo sapiens (Human)) | BDBM50214264 (1-{[(5R,8R,11S)-6,9,12-trioxo-8-(propan-2-yl)-5-{[...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 28 | n/a | n/a | n/a | n/a | n/a | n/a |
Tranzyme Pharma Inc. Curated by ChEMBL | Assay Description Antagonist activity against human motilin receptor in aequoscreen cells assessed as inhibition of motilin induced calcium release by aequorin assay | Bioorg Med Chem Lett 17: 4187-90 (2007) Article DOI: 10.1016/j.bmcl.2007.05.043 BindingDB Entry DOI: 10.7270/Q2GF0T62 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Motilin receptor (Homo sapiens (Human)) | BDBM50214262 ((5R,8R,11S)-5-[(4-chlorophenyl)methyl]-11-[(methyl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 33 | n/a | n/a | n/a | n/a | n/a | n/a |
Tranzyme Pharma Inc. Curated by ChEMBL | Assay Description Antagonist activity against human motilin receptor in aequoscreen cells assessed as inhibition of motilin induced calcium release by aequorin assay | Bioorg Med Chem Lett 17: 4187-90 (2007) Article DOI: 10.1016/j.bmcl.2007.05.043 BindingDB Entry DOI: 10.7270/Q2GF0T62 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Motilin receptor (Homo sapiens (Human)) | BDBM50214260 ((5R,8R,11S)-5-[(3-chlorophenyl)methyl]-8-(propan-2...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents | Article PubMed | n/a | n/a | 56 | n/a | n/a | n/a | n/a | n/a | n/a |
Tranzyme Pharma Inc. Curated by ChEMBL | Assay Description Antagonist activity against human motilin receptor in aequoscreen cells assessed as inhibition of motilin induced calcium release by aequorin assay | Bioorg Med Chem Lett 17: 4187-90 (2007) Article DOI: 10.1016/j.bmcl.2007.05.043 BindingDB Entry DOI: 10.7270/Q2GF0T62 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Motilin receptor (Homo sapiens (Human)) | BDBM50199365 ((E)-(9R,12R,15S)-9-(4-hydroxy-benzyl)-12-isopropyl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 74 | n/a | n/a | n/a | n/a | n/a | n/a |
Tranzyme Pharma Inc. Curated by ChEMBL | Assay Description Antagonist activity against human motilin receptor in aequoscreen cells assessed as inhibition of motilin induced calcium release by aequorin assay | Bioorg Med Chem Lett 17: 4187-90 (2007) Article DOI: 10.1016/j.bmcl.2007.05.043 BindingDB Entry DOI: 10.7270/Q2GF0T62 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Motilin receptor (Homo sapiens (Human)) | BDBM50214251 ((5R,8R,11S)-5-[(3-chlorophenyl)methyl]-11-[(dimeth...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 95 | n/a | n/a | n/a | n/a | n/a | n/a |
Tranzyme Pharma Inc. Curated by ChEMBL | Assay Description Antagonist activity against human motilin receptor in aequoscreen cells assessed as inhibition of motilin induced calcium release by aequorin assay | Bioorg Med Chem Lett 17: 4187-90 (2007) Article DOI: 10.1016/j.bmcl.2007.05.043 BindingDB Entry DOI: 10.7270/Q2GF0T62 | |||||||||||
More data for this Ligand-Target Pair |