Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Mucosa-associated lymphoid tissue lymphoma translocation protein 1 (Homo sapiens (Human)) | BDBM355969 ((S)-1-(5-chloro-6- (difluoromethoxy) pyridin-3-yl)...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.00100 | n/a | n/a | n/a | n/a | n/a | n/a |
Novartis AG US Patent | Assay Description IC50 values of test compounds were determined with an enzyme activity assay using the C-domain of MALT1 (amino acids 329-824). The readout parameter ... | US Patent US9815842 (2017) BindingDB Entry DOI: 10.7270/Q24F1T0N | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mucosa-associated lymphoid tissue lymphoma translocation protein 1 [329-824] (Homo sapiens (Human)) | BDBM355969 ((S)-1-(5-chloro-6- (difluoromethoxy) pyridin-3-yl)...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.00100 | n/a | n/a | n/a | n/a | n/a | n/a |
Novartis AG US Patent | Assay Description The assay employs a short peptide substrate labeled with the single fluorophore PT14 as a fluorescence lifetime probe sensitive to the cleavage state... | US Patent US10442808 (2019) BindingDB Entry DOI: 10.7270/Q2S75JQ3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mucosa-associated lymphoid tissue lymphoma translocation protein 1 [329-824] (Homo sapiens (Human)) | BDBM355970 ((S)-1-(6-(2H-1,2,3- triazol-2-yl)-5- (trifluoromet...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.00200 | n/a | n/a | n/a | n/a | n/a | n/a |
Novartis AG US Patent | Assay Description The assay employs a short peptide substrate labeled with the single fluorophore PT14 as a fluorescence lifetime probe sensitive to the cleavage state... | US Patent US10442808 (2019) BindingDB Entry DOI: 10.7270/Q2S75JQ3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mucosa-associated lymphoid tissue lymphoma translocation protein 1 (Homo sapiens (Human)) | BDBM355980 (1-(5-chloro-6-(2H- 1,2,3-triazol-2- yl)pyridin-3-y...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.00200 | n/a | n/a | n/a | n/a | n/a | n/a |
Novartis AG US Patent | Assay Description IC50 values of test compounds were determined with an enzyme activity assay using the C-domain of MALT1 (amino acids 329-824). The readout parameter ... | US Patent US9815842 (2017) BindingDB Entry DOI: 10.7270/Q24F1T0N | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mucosa-associated lymphoid tissue lymphoma translocation protein 1 [329-824] (Homo sapiens (Human)) | BDBM355980 (1-(5-chloro-6-(2H- 1,2,3-triazol-2- yl)pyridin-3-y...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.00200 | n/a | n/a | n/a | n/a | n/a | n/a |
Novartis AG US Patent | Assay Description The assay employs a short peptide substrate labeled with the single fluorophore PT14 as a fluorescence lifetime probe sensitive to the cleavage state... | US Patent US10442808 (2019) BindingDB Entry DOI: 10.7270/Q2S75JQ3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mucosa-associated lymphoid tissue lymphoma translocation protein 1 (Homo sapiens (Human)) | BDBM50169049 (CHEMBL3806155 | US10442808, Example 1 | US9815842,...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 0.00200 | n/a | n/a | n/a | n/a | n/a | n/a |
Novartis AG US Patent | Assay Description IC50 values of test compounds were determined with an enzyme activity assay using the C-domain of MALT1 (amino acids 329-824). The readout parameter ... | US Patent US9815842 (2017) BindingDB Entry DOI: 10.7270/Q24F1T0N | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mucosa-associated lymphoid tissue lymphoma translocation protein 1 [329-824] (Homo sapiens (Human)) | BDBM50169049 (CHEMBL3806155 | US10442808, Example 1 | US9815842,...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 0.00200 | n/a | n/a | n/a | n/a | n/a | n/a |
Novartis AG US Patent | Assay Description The assay employs a short peptide substrate labeled with the single fluorophore PT14 as a fluorescence lifetime probe sensitive to the cleavage state... | US Patent US10442808 (2019) BindingDB Entry DOI: 10.7270/Q2S75JQ3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mucosa-associated lymphoid tissue lymphoma translocation protein 1 [329-824] (Homo sapiens (Human)) | BDBM355885 ((S)-1-(5-chloro-6- methoxypyridin-3- yl)-3-(2-chlo...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.00200 | n/a | n/a | n/a | n/a | n/a | n/a |
Novartis AG US Patent | Assay Description The assay employs a short peptide substrate labeled with the single fluorophore PT14 as a fluorescence lifetime probe sensitive to the cleavage state... | US Patent US10442808 (2019) BindingDB Entry DOI: 10.7270/Q2S75JQ3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mucosa-associated lymphoid tissue lymphoma translocation protein 1 [329-824] (Homo sapiens (Human)) | BDBM355886 ((S)-1-(5-chloro-6- (2H-1,2,3-triazol-2- yl)pyridin...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | US Patent | n/a | n/a | 0.00200 | n/a | n/a | n/a | n/a | n/a | n/a |
Novartis AG US Patent | Assay Description The assay employs a short peptide substrate labeled with the single fluorophore PT14 as a fluorescence lifetime probe sensitive to the cleavage state... | US Patent US10442808 (2019) BindingDB Entry DOI: 10.7270/Q2S75JQ3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mucosa-associated lymphoid tissue lymphoma translocation protein 1 [329-824] (Homo sapiens (Human)) | BDBM355889 ((S)-methyl 3-chloro- 5-(3-(2-chloro-7-(1- methoxye...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.00200 | n/a | n/a | n/a | n/a | n/a | n/a |
Novartis AG US Patent | Assay Description The assay employs a short peptide substrate labeled with the single fluorophore PT14 as a fluorescence lifetime probe sensitive to the cleavage state... | US Patent US10442808 (2019) BindingDB Entry DOI: 10.7270/Q2S75JQ3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mucosa-associated lymphoid tissue lymphoma translocation protein 1 [329-824] (Homo sapiens (Human)) | BDBM355892 (1-(5-chloro-6-(2H- 1,2,3-triazol-2- yl)pyridin-3-y...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.00200 | n/a | n/a | n/a | n/a | n/a | n/a |
Novartis AG US Patent | Assay Description The assay employs a short peptide substrate labeled with the single fluorophore PT14 as a fluorescence lifetime probe sensitive to the cleavage state... | US Patent US10442808 (2019) BindingDB Entry DOI: 10.7270/Q2S75JQ3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mucosa-associated lymphoid tissue lymphoma translocation protein 1 [329-824] (Homo sapiens (Human)) | BDBM355950 ((S)-1-(5-chloro-6- (2H-1,2,3-triazol-2- yl)pyridin...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.00200 | n/a | n/a | n/a | n/a | n/a | n/a |
Novartis AG US Patent | Assay Description The assay employs a short peptide substrate labeled with the single fluorophore PT14 as a fluorescence lifetime probe sensitive to the cleavage state... | US Patent US10442808 (2019) BindingDB Entry DOI: 10.7270/Q2S75JQ3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mucosa-associated lymphoid tissue lymphoma translocation protein 1 [329-824] (Homo sapiens (Human)) | BDBM355967 (1-(5-chloro-6-(2H- 1,2,3-triazol-2- yl)pyridin-3-y...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.00200 | n/a | n/a | n/a | n/a | n/a | n/a |
Novartis AG US Patent | Assay Description The assay employs a short peptide substrate labeled with the single fluorophore PT14 as a fluorescence lifetime probe sensitive to the cleavage state... | US Patent US10442808 (2019) BindingDB Entry DOI: 10.7270/Q2S75JQ3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mucosa-associated lymphoid tissue lymphoma translocation protein 1 (Homo sapiens (Human)) | BDBM355885 ((S)-1-(5-chloro-6- methoxypyridin-3- yl)-3-(2-chlo...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.00200 | n/a | n/a | n/a | n/a | n/a | n/a |
Novartis AG US Patent | Assay Description IC50 values of test compounds were determined with an enzyme activity assay using the C-domain of MALT1 (amino acids 329-824). The readout parameter ... | US Patent US9815842 (2017) BindingDB Entry DOI: 10.7270/Q24F1T0N | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mucosa-associated lymphoid tissue lymphoma translocation protein 1 (Homo sapiens (Human)) | BDBM355886 ((S)-1-(5-chloro-6- (2H-1,2,3-triazol-2- yl)pyridin...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | US Patent | n/a | n/a | 0.00200 | n/a | n/a | n/a | n/a | n/a | n/a |
Novartis AG US Patent | Assay Description IC50 values of test compounds were determined with an enzyme activity assay using the C-domain of MALT1 (amino acids 329-824). The readout parameter ... | US Patent US9815842 (2017) BindingDB Entry DOI: 10.7270/Q24F1T0N | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mucosa-associated lymphoid tissue lymphoma translocation protein 1 (Homo sapiens (Human)) | BDBM355889 ((S)-methyl 3-chloro- 5-(3-(2-chloro-7-(1- methoxye...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.00200 | n/a | n/a | n/a | n/a | n/a | n/a |
Novartis AG US Patent | Assay Description IC50 values of test compounds were determined with an enzyme activity assay using the C-domain of MALT1 (amino acids 329-824). The readout parameter ... | US Patent US9815842 (2017) BindingDB Entry DOI: 10.7270/Q24F1T0N | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mucosa-associated lymphoid tissue lymphoma translocation protein 1 (Homo sapiens (Human)) | BDBM355892 (1-(5-chloro-6-(2H- 1,2,3-triazol-2- yl)pyridin-3-y...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.00200 | n/a | n/a | n/a | n/a | n/a | n/a |
Novartis AG US Patent | Assay Description IC50 values of test compounds were determined with an enzyme activity assay using the C-domain of MALT1 (amino acids 329-824). The readout parameter ... | US Patent US9815842 (2017) BindingDB Entry DOI: 10.7270/Q24F1T0N | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mucosa-associated lymphoid tissue lymphoma translocation protein 1 (Homo sapiens (Human)) | BDBM355950 ((S)-1-(5-chloro-6- (2H-1,2,3-triazol-2- yl)pyridin...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.00200 | n/a | n/a | n/a | n/a | n/a | n/a |
Novartis AG US Patent | Assay Description IC50 values of test compounds were determined with an enzyme activity assay using the C-domain of MALT1 (amino acids 329-824). The readout parameter ... | US Patent US9815842 (2017) BindingDB Entry DOI: 10.7270/Q24F1T0N | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mucosa-associated lymphoid tissue lymphoma translocation protein 1 (Homo sapiens (Human)) | BDBM355967 (1-(5-chloro-6-(2H- 1,2,3-triazol-2- yl)pyridin-3-y...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.00200 | n/a | n/a | n/a | n/a | n/a | n/a |
Novartis AG US Patent | Assay Description IC50 values of test compounds were determined with an enzyme activity assay using the C-domain of MALT1 (amino acids 329-824). The readout parameter ... | US Patent US9815842 (2017) BindingDB Entry DOI: 10.7270/Q24F1T0N | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mucosa-associated lymphoid tissue lymphoma translocation protein 1 (Homo sapiens (Human)) | BDBM355970 ((S)-1-(6-(2H-1,2,3- triazol-2-yl)-5- (trifluoromet...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.00200 | n/a | n/a | n/a | n/a | n/a | n/a |
Novartis AG US Patent | Assay Description IC50 values of test compounds were determined with an enzyme activity assay using the C-domain of MALT1 (amino acids 329-824). The readout parameter ... | US Patent US9815842 (2017) BindingDB Entry DOI: 10.7270/Q24F1T0N | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mucosa-associated lymphoid tissue lymphoma translocation protein 1 (Homo sapiens (Human)) | BDBM355971 ((S)-1-(5-chloro-6- (2H-1,2,3-triazol-2- yl)pyridin...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.00200 | n/a | n/a | n/a | n/a | n/a | n/a |
Novartis AG US Patent | Assay Description IC50 values of test compounds were determined with an enzyme activity assay using the C-domain of MALT1 (amino acids 329-824). The readout parameter ... | US Patent US9815842 (2017) BindingDB Entry DOI: 10.7270/Q24F1T0N | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mucosa-associated lymphoid tissue lymphoma translocation protein 1 [329-824] (Homo sapiens (Human)) | BDBM355971 ((S)-1-(5-chloro-6- (2H-1,2,3-triazol-2- yl)pyridin...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.00200 | n/a | n/a | n/a | n/a | n/a | n/a |
Novartis AG US Patent | Assay Description The assay employs a short peptide substrate labeled with the single fluorophore PT14 as a fluorescence lifetime probe sensitive to the cleavage state... | US Patent US10442808 (2019) BindingDB Entry DOI: 10.7270/Q2S75JQ3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mucosa-associated lymphoid tissue lymphoma translocation protein 1 [329-824] (Homo sapiens (Human)) | BDBM355973 ((S)-1-(5-chloro-6- (difluoromethoxy)py- ridin-3-yl...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.00300 | n/a | n/a | n/a | n/a | n/a | n/a |
Novartis AG US Patent | Assay Description The assay employs a short peptide substrate labeled with the single fluorophore PT14 as a fluorescence lifetime probe sensitive to the cleavage state... | US Patent US10442808 (2019) BindingDB Entry DOI: 10.7270/Q2S75JQ3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mucosa-associated lymphoid tissue lymphoma translocation protein 1 (Homo sapiens (Human)) | BDBM355978 (1-(5-chloro-6-(2H- 1,2,3-triazol-2- yl)pyridin-3-y...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.00300 | n/a | n/a | n/a | n/a | n/a | n/a |
Novartis AG US Patent | Assay Description IC50 values of test compounds were determined with an enzyme activity assay using the C-domain of MALT1 (amino acids 329-824). The readout parameter ... | US Patent US9815842 (2017) BindingDB Entry DOI: 10.7270/Q24F1T0N | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mucosa-associated lymphoid tissue lymphoma translocation protein 1 [329-824] (Homo sapiens (Human)) | BDBM355987 ((R)-1-(6-(2H-1,2,3- triazol-2-yl)-5- (trifluoromet...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.00300 | n/a | n/a | n/a | n/a | n/a | n/a |
Novartis AG US Patent | Assay Description The assay employs a short peptide substrate labeled with the single fluorophore PT14 as a fluorescence lifetime probe sensitive to the cleavage state... | US Patent US10442808 (2019) BindingDB Entry DOI: 10.7270/Q2S75JQ3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mucosa-associated lymphoid tissue lymphoma translocation protein 1 (Homo sapiens (Human)) | BDBM355896 (1-(3-chloro-4-(2H- 1,2,3-triazol-2- yl)phenyl)-3-(...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.00300 | n/a | n/a | n/a | n/a | n/a | n/a |
Novartis AG US Patent | Assay Description IC50 values of test compounds were determined with an enzyme activity assay using the C-domain of MALT1 (amino acids 329-824). The readout parameter ... | US Patent US9815842 (2017) BindingDB Entry DOI: 10.7270/Q24F1T0N | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mucosa-associated lymphoid tissue lymphoma translocation protein 1 (Homo sapiens (Human)) | BDBM355987 ((R)-1-(6-(2H-1,2,3- triazol-2-yl)-5- (trifluoromet...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.00300 | n/a | n/a | n/a | n/a | n/a | n/a |
Novartis AG US Patent | Assay Description IC50 values of test compounds were determined with an enzyme activity assay using the C-domain of MALT1 (amino acids 329-824). The readout parameter ... | US Patent US9815842 (2017) BindingDB Entry DOI: 10.7270/Q24F1T0N | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mucosa-associated lymphoid tissue lymphoma translocation protein 1 [329-824] (Homo sapiens (Human)) | BDBM355890 (1-(5-chloro-6-(2H- 1,2,3-triazol-2- yl)pyridin-3-y...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.00300 | n/a | n/a | n/a | n/a | n/a | n/a |
Novartis AG US Patent | Assay Description The assay employs a short peptide substrate labeled with the single fluorophore PT14 as a fluorescence lifetime probe sensitive to the cleavage state... | US Patent US10442808 (2019) BindingDB Entry DOI: 10.7270/Q2S75JQ3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mucosa-associated lymphoid tissue lymphoma translocation protein 1 [329-824] (Homo sapiens (Human)) | BDBM355894 (1-(5-chloro-6- methoxypyridin-3- yl)-3-(2-chloro-7...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.00300 | n/a | n/a | n/a | n/a | n/a | n/a |
Novartis AG US Patent | Assay Description The assay employs a short peptide substrate labeled with the single fluorophore PT14 as a fluorescence lifetime probe sensitive to the cleavage state... | US Patent US10442808 (2019) BindingDB Entry DOI: 10.7270/Q2S75JQ3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mucosa-associated lymphoid tissue lymphoma translocation protein 1 [329-824] (Homo sapiens (Human)) | BDBM355895 (1-(2-chloro-7- isopropylpyrazolo[1, 5-a]pyrimidin-...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.00300 | n/a | n/a | n/a | n/a | n/a | n/a |
Novartis AG US Patent | Assay Description The assay employs a short peptide substrate labeled with the single fluorophore PT14 as a fluorescence lifetime probe sensitive to the cleavage state... | US Patent US10442808 (2019) BindingDB Entry DOI: 10.7270/Q2S75JQ3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mucosa-associated lymphoid tissue lymphoma translocation protein 1 [329-824] (Homo sapiens (Human)) | BDBM355896 (1-(3-chloro-4-(2H- 1,2,3-triazol-2- yl)phenyl)-3-(...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.00300 | n/a | n/a | n/a | n/a | n/a | n/a |
Novartis AG US Patent | Assay Description The assay employs a short peptide substrate labeled with the single fluorophore PT14 as a fluorescence lifetime probe sensitive to the cleavage state... | US Patent US10442808 (2019) BindingDB Entry DOI: 10.7270/Q2S75JQ3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mucosa-associated lymphoid tissue lymphoma translocation protein 1 [329-824] (Homo sapiens (Human)) | BDBM355897 (1-(5-chloro-6-(2H- 1,2,3-triazol-2- yl)pyridin-3-y...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.00300 | n/a | n/a | n/a | n/a | n/a | n/a |
Novartis AG US Patent | Assay Description The assay employs a short peptide substrate labeled with the single fluorophore PT14 as a fluorescence lifetime probe sensitive to the cleavage state... | US Patent US10442808 (2019) BindingDB Entry DOI: 10.7270/Q2S75JQ3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mucosa-associated lymphoid tissue lymphoma translocation protein 1 [329-824] (Homo sapiens (Human)) | BDBM355906 (1-(2-chloro-7- isopropylpyrazolo[1, 5-a]pyrimidin-...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.00300 | n/a | n/a | n/a | n/a | n/a | n/a |
Novartis AG US Patent | Assay Description The assay employs a short peptide substrate labeled with the single fluorophore PT14 as a fluorescence lifetime probe sensitive to the cleavage state... | US Patent US10442808 (2019) BindingDB Entry DOI: 10.7270/Q2S75JQ3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mucosa-associated lymphoid tissue lymphoma translocation protein 1 [329-824] (Homo sapiens (Human)) | BDBM355911 (1-(7-(sec-butyl)-2- chloropyrazolo[1,5- a]pyrimidi...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.00300 | n/a | n/a | n/a | n/a | n/a | n/a |
Novartis AG US Patent | Assay Description The assay employs a short peptide substrate labeled with the single fluorophore PT14 as a fluorescence lifetime probe sensitive to the cleavage state... | US Patent US10442808 (2019) BindingDB Entry DOI: 10.7270/Q2S75JQ3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mucosa-associated lymphoid tissue lymphoma translocation protein 1 [329-824] (Homo sapiens (Human)) | BDBM355915 ((S)-1-(5-chloro-6- (2H-1,2,3-triazol-2- yl)pyridin...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.00300 | n/a | n/a | n/a | n/a | n/a | n/a |
Novartis AG US Patent | Assay Description The assay employs a short peptide substrate labeled with the single fluorophore PT14 as a fluorescence lifetime probe sensitive to the cleavage state... | US Patent US10442808 (2019) BindingDB Entry DOI: 10.7270/Q2S75JQ3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mucosa-associated lymphoid tissue lymphoma translocation protein 1 [329-824] (Homo sapiens (Human)) | BDBM355921 ((R)-1-(5-chloro-6- (2H-1,2,3-triazol-2- yl)pyridin...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.00300 | n/a | n/a | n/a | n/a | n/a | n/a |
Novartis AG US Patent | Assay Description The assay employs a short peptide substrate labeled with the single fluorophore PT14 as a fluorescence lifetime probe sensitive to the cleavage state... | US Patent US10442808 (2019) BindingDB Entry DOI: 10.7270/Q2S75JQ3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mucosa-associated lymphoid tissue lymphoma translocation protein 1 [329-824] (Homo sapiens (Human)) | BDBM355925 (1-(5-chloro-6-(2H- 1,2,3-triazol-2- yl)pyridin-3-y...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.00300 | n/a | n/a | n/a | n/a | n/a | n/a |
Novartis AG US Patent | Assay Description The assay employs a short peptide substrate labeled with the single fluorophore PT14 as a fluorescence lifetime probe sensitive to the cleavage state... | US Patent US10442808 (2019) BindingDB Entry DOI: 10.7270/Q2S75JQ3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mucosa-associated lymphoid tissue lymphoma translocation protein 1 [329-824] (Homo sapiens (Human)) | BDBM355948 (1-(5-chloro-6-(2H- 1,2,3-triazol-2- yl)pyridin-3-y...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.00300 | n/a | n/a | n/a | n/a | n/a | n/a |
Novartis AG US Patent | Assay Description The assay employs a short peptide substrate labeled with the single fluorophore PT14 as a fluorescence lifetime probe sensitive to the cleavage state... | US Patent US10442808 (2019) BindingDB Entry DOI: 10.7270/Q2S75JQ3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mucosa-associated lymphoid tissue lymphoma translocation protein 1 [329-824] (Homo sapiens (Human)) | BDBM355965 ((S)-1-(2-chloro-7-(1- methoxyethyl)pyrazo- lo[1,5-...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.00300 | n/a | n/a | n/a | n/a | n/a | n/a |
Novartis AG US Patent | Assay Description The assay employs a short peptide substrate labeled with the single fluorophore PT14 as a fluorescence lifetime probe sensitive to the cleavage state... | US Patent US10442808 (2019) BindingDB Entry DOI: 10.7270/Q2S75JQ3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mucosa-associated lymphoid tissue lymphoma translocation protein 1 (Homo sapiens (Human)) | BDBM355911 (1-(7-(sec-butyl)-2- chloropyrazolo[1,5- a]pyrimidi...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.00300 | n/a | n/a | n/a | n/a | n/a | n/a |
Novartis AG US Patent | Assay Description IC50 values of test compounds were determined with an enzyme activity assay using the C-domain of MALT1 (amino acids 329-824). The readout parameter ... | US Patent US9815842 (2017) BindingDB Entry DOI: 10.7270/Q24F1T0N | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mucosa-associated lymphoid tissue lymphoma translocation protein 1 (Homo sapiens (Human)) | BDBM355890 (1-(5-chloro-6-(2H- 1,2,3-triazol-2- yl)pyridin-3-y...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.00300 | n/a | n/a | n/a | n/a | n/a | n/a |
Novartis AG US Patent | Assay Description IC50 values of test compounds were determined with an enzyme activity assay using the C-domain of MALT1 (amino acids 329-824). The readout parameter ... | US Patent US9815842 (2017) BindingDB Entry DOI: 10.7270/Q24F1T0N | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mucosa-associated lymphoid tissue lymphoma translocation protein 1 (Homo sapiens (Human)) | BDBM355894 (1-(5-chloro-6- methoxypyridin-3- yl)-3-(2-chloro-7...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.00300 | n/a | n/a | n/a | n/a | n/a | n/a |
Novartis AG US Patent | Assay Description IC50 values of test compounds were determined with an enzyme activity assay using the C-domain of MALT1 (amino acids 329-824). The readout parameter ... | US Patent US9815842 (2017) BindingDB Entry DOI: 10.7270/Q24F1T0N | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mucosa-associated lymphoid tissue lymphoma translocation protein 1 (Homo sapiens (Human)) | BDBM355895 (1-(2-chloro-7- isopropylpyrazolo[1, 5-a]pyrimidin-...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.00300 | n/a | n/a | n/a | n/a | n/a | n/a |
Novartis AG US Patent | Assay Description IC50 values of test compounds were determined with an enzyme activity assay using the C-domain of MALT1 (amino acids 329-824). The readout parameter ... | US Patent US9815842 (2017) BindingDB Entry DOI: 10.7270/Q24F1T0N | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mucosa-associated lymphoid tissue lymphoma translocation protein 1 (Homo sapiens (Human)) | BDBM355897 (1-(5-chloro-6-(2H- 1,2,3-triazol-2- yl)pyridin-3-y...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.00300 | n/a | n/a | n/a | n/a | n/a | n/a |
Novartis AG US Patent | Assay Description IC50 values of test compounds were determined with an enzyme activity assay using the C-domain of MALT1 (amino acids 329-824). The readout parameter ... | US Patent US9815842 (2017) BindingDB Entry DOI: 10.7270/Q24F1T0N | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mucosa-associated lymphoid tissue lymphoma translocation protein 1 (Homo sapiens (Human)) | BDBM355906 (1-(2-chloro-7- isopropylpyrazolo[1, 5-a]pyrimidin-...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.00300 | n/a | n/a | n/a | n/a | n/a | n/a |
Novartis AG US Patent | Assay Description IC50 values of test compounds were determined with an enzyme activity assay using the C-domain of MALT1 (amino acids 329-824). The readout parameter ... | US Patent US9815842 (2017) BindingDB Entry DOI: 10.7270/Q24F1T0N | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mucosa-associated lymphoid tissue lymphoma translocation protein 1 (Homo sapiens (Human)) | BDBM355915 ((S)-1-(5-chloro-6- (2H-1,2,3-triazol-2- yl)pyridin...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.00300 | n/a | n/a | n/a | n/a | n/a | n/a |
Novartis AG US Patent | Assay Description IC50 values of test compounds were determined with an enzyme activity assay using the C-domain of MALT1 (amino acids 329-824). The readout parameter ... | US Patent US9815842 (2017) BindingDB Entry DOI: 10.7270/Q24F1T0N | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mucosa-associated lymphoid tissue lymphoma translocation protein 1 (Homo sapiens (Human)) | BDBM355921 ((R)-1-(5-chloro-6- (2H-1,2,3-triazol-2- yl)pyridin...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.00300 | n/a | n/a | n/a | n/a | n/a | n/a |
Novartis AG US Patent | Assay Description IC50 values of test compounds were determined with an enzyme activity assay using the C-domain of MALT1 (amino acids 329-824). The readout parameter ... | US Patent US9815842 (2017) BindingDB Entry DOI: 10.7270/Q24F1T0N | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mucosa-associated lymphoid tissue lymphoma translocation protein 1 (Homo sapiens (Human)) | BDBM355925 (1-(5-chloro-6-(2H- 1,2,3-triazol-2- yl)pyridin-3-y...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.00300 | n/a | n/a | n/a | n/a | n/a | n/a |
Novartis AG US Patent | Assay Description IC50 values of test compounds were determined with an enzyme activity assay using the C-domain of MALT1 (amino acids 329-824). The readout parameter ... | US Patent US9815842 (2017) BindingDB Entry DOI: 10.7270/Q24F1T0N | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mucosa-associated lymphoid tissue lymphoma translocation protein 1 (Homo sapiens (Human)) | BDBM355948 (1-(5-chloro-6-(2H- 1,2,3-triazol-2- yl)pyridin-3-y...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.00300 | n/a | n/a | n/a | n/a | n/a | n/a |
Novartis AG US Patent | Assay Description IC50 values of test compounds were determined with an enzyme activity assay using the C-domain of MALT1 (amino acids 329-824). The readout parameter ... | US Patent US9815842 (2017) BindingDB Entry DOI: 10.7270/Q24F1T0N | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mucosa-associated lymphoid tissue lymphoma translocation protein 1 (Homo sapiens (Human)) | BDBM355965 ((S)-1-(2-chloro-7-(1- methoxyethyl)pyrazo- lo[1,5-...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.00300 | n/a | n/a | n/a | n/a | n/a | n/a |
Novartis AG US Patent | Assay Description IC50 values of test compounds were determined with an enzyme activity assay using the C-domain of MALT1 (amino acids 329-824). The readout parameter ... | US Patent US9815842 (2017) BindingDB Entry DOI: 10.7270/Q24F1T0N | |||||||||||
More data for this Ligand-Target Pair |
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