Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Neuronal acetylcholine receptor subunit alpha-4 (Rattus norvegicus (Rat)) | BDBM50216315 ((1R,4R)-2-(6-chloro-3-pyridinyl)-2,5-diazabicyclo[...) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.0180 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Università di Sassari Curated by ChEMBL | Assay Description Displacement of [3H]cytosine form alpha4beta2 nAChR in rat striatum | Bioorg Med Chem Lett 18: 6147-50 (2008) Article DOI: 10.1016/j.bmcl.2008.10.002 BindingDB Entry DOI: 10.7270/Q29G5MPJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuronal acetylcholine receptor subunit alpha-4 (Rattus norvegicus (Rat)) | BDBM50275878 (3-(6-chloropyridin-3-yl)-3,6-diazabicyclo[3.1.1]he...) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.0230 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Università di Sassari Curated by ChEMBL | Assay Description Displacement of [3H]epibatidine form alpha4beta2 nAChR in rat cortex | Bioorg Med Chem Lett 18: 6147-50 (2008) Article DOI: 10.1016/j.bmcl.2008.10.002 BindingDB Entry DOI: 10.7270/Q29G5MPJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuronal acetylcholine receptor subunit alpha-4 (Rattus norvegicus (Rat)) | BDBM50275880 (3-(6-bromopyridin-3-yl)-3,6-diazabicyclo[3.1.1]hep...) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | 0.0390 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Università di Sassari Curated by ChEMBL | Assay Description Displacement of [3H]epibatidine form alpha4beta2 nAChR in rat cortex | Bioorg Med Chem Lett 18: 6147-50 (2008) Article DOI: 10.1016/j.bmcl.2008.10.002 BindingDB Entry DOI: 10.7270/Q29G5MPJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 2 (MOUSE) | BDBM50200169 (6-methyl-1-(2',4'-dichlorophenyl)-N-piperidin-1-yl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | Article PubMed | 0.0400 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Sassari Curated by ChEMBL | Assay Description Displacement of [3H]CP-55940 from CD1 mouse spleen CB2 receptor | J Med Chem 49: 7502-12 (2006) Article DOI: 10.1021/jm060920d BindingDB Entry DOI: 10.7270/Q2057GRN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuronal acetylcholine receptor subunit alpha-4 (Rattus norvegicus (Rat)) | BDBM50275879 (3-(pyridin-3-yl)-3,6-diazabicyclo[3.1.1]heptane | ...) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.0560 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Università di Sassari Curated by ChEMBL | Assay Description Displacement of [3H]epibatidine form alpha4beta2 nAChR in rat cortex | Bioorg Med Chem Lett 18: 6147-50 (2008) Article DOI: 10.1016/j.bmcl.2008.10.002 BindingDB Entry DOI: 10.7270/Q29G5MPJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuronal acetylcholine receptor subunit alpha-4 (Rattus norvegicus (Rat)) | BDBM50275932 (3-(6-chloropyridazin-3-yl)-3,6-diazabicyclo[3.1.1]...) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.168 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Università di Sassari Curated by ChEMBL | Assay Description Displacement of [3H]epibatidine form alpha4beta2 nAChR in rat cortex | Bioorg Med Chem Lett 18: 6147-50 (2008) Article DOI: 10.1016/j.bmcl.2008.10.002 BindingDB Entry DOI: 10.7270/Q29G5MPJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 2 (MOUSE) | BDBM50180022 (5-(4-chloro-3-methyl-phenyl)-1-(4-methyl-benzyl)-1...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 0.280 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Sassari Curated by ChEMBL | Assay Description Displacement of [3H]CP-55940 from CD1 mouse spleen CB2 receptor | J Med Chem 49: 7502-12 (2006) Article DOI: 10.1021/jm060920d BindingDB Entry DOI: 10.7270/Q2057GRN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 2 (MOUSE) | BDBM50176977 (1,4-dihydroindeno[1,2-c]-pyrazole | 6-chloro-1-(2'...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.340 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Sassari Curated by ChEMBL | Assay Description Displacement of [3H]CP-55940 from CD1 mouse spleen CB2 receptor | J Med Chem 49: 7502-12 (2006) Article DOI: 10.1021/jm060920d BindingDB Entry DOI: 10.7270/Q2057GRN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuronal acetylcholine receptor subunit alpha-4 (Rattus norvegicus (Rat)) | BDBM50275933 (3-(6-chloropyridin-3-yl)-6-methyl-3,6-diazabicyclo...) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.430 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Università di Sassari Curated by ChEMBL | Assay Description Displacement of [3H]epibatidine form alpha4beta2 nAChR in rat cortex | Bioorg Med Chem Lett 18: 6147-50 (2008) Article DOI: 10.1016/j.bmcl.2008.10.002 BindingDB Entry DOI: 10.7270/Q29G5MPJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 2 (MOUSE) | BDBM50072775 (2-((1R,2R,5R)-5-hydroxy-2-(3-hydroxypropyl)cyclohe...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid PDB UniChem Patents Similars | Article PubMed | 1.10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Sassari Curated by ChEMBL | Assay Description Displacement of [3H]CP-55940 from CD1 mouse spleen CB2 receptor | J Med Chem 49: 7502-12 (2006) Article DOI: 10.1021/jm060920d BindingDB Entry DOI: 10.7270/Q2057GRN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuronal acetylcholine receptor subunit alpha-4 (Rattus norvegicus (Rat)) | BDBM50275931 (3-(4-nitrophenyl)-3,6-diazabicyclo[3.1.1]heptane |...) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.20 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Università di Sassari Curated by ChEMBL | Assay Description Displacement of [3H]epibatidine form alpha4beta2 nAChR in rat cortex | Bioorg Med Chem Lett 18: 6147-50 (2008) Article DOI: 10.1016/j.bmcl.2008.10.002 BindingDB Entry DOI: 10.7270/Q29G5MPJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuronal acetylcholine receptor subunit alpha-7 (Rattus norvegicus (Rat)) | BDBM50275879 (3-(pyridin-3-yl)-3,6-diazabicyclo[3.1.1]heptane | ...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.36 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Università di Sassari Curated by ChEMBL | Assay Description Displacement of [3H]alpha-bungarotoxin form alpha7 nAChR in rat cortex | Bioorg Med Chem Lett 18: 6147-50 (2008) Article DOI: 10.1016/j.bmcl.2008.10.002 BindingDB Entry DOI: 10.7270/Q29G5MPJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 1 (Mus musculus (Mouse)) | BDBM50072775 (2-((1R,2R,5R)-5-hydroxy-2-(3-hydroxypropyl)cyclohe...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid PDB UniChem Patents Similars | PDB Article PubMed | 1.5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Sassari Curated by ChEMBL | Assay Description Displacement of [3H]CP-55940 from CD1 mouse brain CB1 receptor | J Med Chem 49: 7502-12 (2006) Article DOI: 10.1021/jm060920d BindingDB Entry DOI: 10.7270/Q2057GRN | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Neuronal acetylcholine receptor subunit alpha-7 (Rattus norvegicus (Rat)) | BDBM50275878 (3-(6-chloropyridin-3-yl)-3,6-diazabicyclo[3.1.1]he...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 4.10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Università di Sassari Curated by ChEMBL | Assay Description Displacement of [3H]alpha-bungarotoxin form alpha7 nAChR in rat cortex | Bioorg Med Chem Lett 18: 6147-50 (2008) Article DOI: 10.1016/j.bmcl.2008.10.002 BindingDB Entry DOI: 10.7270/Q29G5MPJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 2 (MOUSE) | BDBM50200166 (1-(2',4'-dichlorophenyl)-6-methyl-N-cyclohexylamin...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | 7.60 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Sassari Curated by ChEMBL | Assay Description Displacement of [3H]CP-55940 from CD1 mouse spleen CB2 receptor | J Med Chem 49: 7502-12 (2006) Article DOI: 10.1021/jm060920d BindingDB Entry DOI: 10.7270/Q2057GRN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuronal acetylcholine receptor subunit alpha-7 (Rattus norvegicus (Rat)) | BDBM50275933 (3-(6-chloropyridin-3-yl)-6-methyl-3,6-diazabicyclo...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 20 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Università di Sassari Curated by ChEMBL | Assay Description Displacement of [3H]alpha-bungarotoxin form alpha7 nAChR in rat cortex | Bioorg Med Chem Lett 18: 6147-50 (2008) Article DOI: 10.1016/j.bmcl.2008.10.002 BindingDB Entry DOI: 10.7270/Q29G5MPJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuronal acetylcholine receptor subunit alpha-7 (Rattus norvegicus (Rat)) | BDBM50275932 (3-(6-chloropyridazin-3-yl)-3,6-diazabicyclo[3.1.1]...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 25 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Università di Sassari Curated by ChEMBL | Assay Description Displacement of [3H]alpha-bungarotoxin form alpha7 nAChR in rat cortex | Bioorg Med Chem Lett 18: 6147-50 (2008) Article DOI: 10.1016/j.bmcl.2008.10.002 BindingDB Entry DOI: 10.7270/Q29G5MPJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 2 (MOUSE) | BDBM50200177 (7-chloro-1-(2',4'-dichlorophenyl)-6-methyl-N-cyclo...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 25 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Sassari Curated by ChEMBL | Assay Description Displacement of [3H]CP-55940 from CD1 mouse spleen CB2 receptor | J Med Chem 49: 7502-12 (2006) Article DOI: 10.1021/jm060920d BindingDB Entry DOI: 10.7270/Q2057GRN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 2 (MOUSE) | BDBM50200163 (1-(2',4'-dichlorophenyl)-6-methyl-N-phenyl-1,4-dih...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 33 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Sassari Curated by ChEMBL | Assay Description Displacement of [3H]CP-55940 from CD1 mouse spleen CB2 receptor | J Med Chem 49: 7502-12 (2006) Article DOI: 10.1021/jm060920d BindingDB Entry DOI: 10.7270/Q2057GRN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuronal acetylcholine receptor subunit alpha-7 (Rattus norvegicus (Rat)) | BDBM50275880 (3-(6-bromopyridin-3-yl)-3,6-diazabicyclo[3.1.1]hep...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | 50.5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Università di Sassari Curated by ChEMBL | Assay Description Displacement of [3H]alpha-bungarotoxin form alpha7 nAChR in rat cortex | Bioorg Med Chem Lett 18: 6147-50 (2008) Article DOI: 10.1016/j.bmcl.2008.10.002 BindingDB Entry DOI: 10.7270/Q29G5MPJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 2 (MOUSE) | BDBM50200175 (1-(2',4'-dichlorophenyl)-6-methyl-N-p-fluorophenyl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 61 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Sassari Curated by ChEMBL | Assay Description Displacement of [3H]CP-55940 from CD1 mouse spleen CB2 receptor | J Med Chem 49: 7502-12 (2006) Article DOI: 10.1021/jm060920d BindingDB Entry DOI: 10.7270/Q2057GRN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 2 (MOUSE) | BDBM50200172 (1-(2',4'-dichlorophenyl)-6-methyl-N-phenyl-1,4-dih...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 63 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Sassari Curated by ChEMBL | Assay Description Displacement of [3H]CP-55940 from CD1 mouse spleen CB2 receptor | J Med Chem 49: 7502-12 (2006) Article DOI: 10.1021/jm060920d BindingDB Entry DOI: 10.7270/Q2057GRN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 1 (Mus musculus (Mouse)) | BDBM50180022 (5-(4-chloro-3-methyl-phenyl)-1-(4-methyl-benzyl)-1...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 70 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Sassari Curated by ChEMBL | Assay Description Displacement of [3H]CP-55940 from CD1 mouse brain CB1 receptor | J Med Chem 49: 7502-12 (2006) Article DOI: 10.1021/jm060920d BindingDB Entry DOI: 10.7270/Q2057GRN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 2 (MOUSE) | BDBM50200167 (1-(2',4'-dichlorophenyl)-6-methyl-N-p-methylphenyl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 74 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Sassari Curated by ChEMBL | Assay Description Displacement of [3H]CP-55940 from CD1 mouse spleen CB2 receptor | J Med Chem 49: 7502-12 (2006) Article DOI: 10.1021/jm060920d BindingDB Entry DOI: 10.7270/Q2057GRN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 2 (MOUSE) | BDBM50200165 (6-chloro-1-(2',4'-dichlorophenyl)-7-methyl-N-piper...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 85 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Sassari Curated by ChEMBL | Assay Description Displacement of [3H]CP-55940 from CD1 mouse spleen CB2 receptor | J Med Chem 49: 7502-12 (2006) Article DOI: 10.1021/jm060920d BindingDB Entry DOI: 10.7270/Q2057GRN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 2 (MOUSE) | BDBM50200171 (1-(2',4'-dichlorophenyl)-6-methyl-N-p-methoxypheny...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 114 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Sassari Curated by ChEMBL | Assay Description Displacement of [3H]CP-55940 from CD1 mouse spleen CB2 receptor | J Med Chem 49: 7502-12 (2006) Article DOI: 10.1021/jm060920d BindingDB Entry DOI: 10.7270/Q2057GRN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 2 (MOUSE) | BDBM50200162 (1-(2',4'-dichlorophenyl)-6-methyl-N-p-chlorophenyl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 177 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Sassari Curated by ChEMBL | Assay Description Displacement of [3H]CP-55940 from CD1 mouse spleen CB2 receptor | J Med Chem 49: 7502-12 (2006) Article DOI: 10.1021/jm060920d BindingDB Entry DOI: 10.7270/Q2057GRN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 2 (MOUSE) | BDBM50200168 (7-chloro-1-(2',4'-dichlorophenyl)-6-methyl-N-piper...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 200 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Sassari Curated by ChEMBL | Assay Description Displacement of [3H]CP-55940 from CD1 mouse spleen CB2 receptor | J Med Chem 49: 7502-12 (2006) Article DOI: 10.1021/jm060920d BindingDB Entry DOI: 10.7270/Q2057GRN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 1 (Mus musculus (Mouse)) | BDBM50200169 (6-methyl-1-(2',4'-dichlorophenyl)-N-piperidin-1-yl...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | Article PubMed | 363 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Sassari Curated by ChEMBL | Assay Description Displacement of [3H]CP-55940 from CD1 mouse brain CB1 receptor | J Med Chem 49: 7502-12 (2006) Article DOI: 10.1021/jm060920d BindingDB Entry DOI: 10.7270/Q2057GRN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 1 (Mus musculus (Mouse)) | BDBM50200177 (7-chloro-1-(2',4'-dichlorophenyl)-6-methyl-N-cyclo...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 833 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Sassari Curated by ChEMBL | Assay Description Displacement of [3H]CP-55940 from CD1 mouse brain CB1 receptor | J Med Chem 49: 7502-12 (2006) Article DOI: 10.1021/jm060920d BindingDB Entry DOI: 10.7270/Q2057GRN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 1 (Mus musculus (Mouse)) | BDBM50200166 (1-(2',4'-dichlorophenyl)-6-methyl-N-cyclohexylamin...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | 900 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Sassari Curated by ChEMBL | Assay Description Displacement of [3H]CP-55940 from CD1 mouse brain CB1 receptor | J Med Chem 49: 7502-12 (2006) Article DOI: 10.1021/jm060920d BindingDB Entry DOI: 10.7270/Q2057GRN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 1 (Mus musculus (Mouse)) | BDBM50200168 (7-chloro-1-(2',4'-dichlorophenyl)-6-methyl-N-piper...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 916 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Sassari Curated by ChEMBL | Assay Description Displacement of [3H]CP-55940 from CD1 mouse brain CB1 receptor | J Med Chem 49: 7502-12 (2006) Article DOI: 10.1021/jm060920d BindingDB Entry DOI: 10.7270/Q2057GRN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 1 (Mus musculus (Mouse)) | BDBM50200165 (6-chloro-1-(2',4'-dichlorophenyl)-7-methyl-N-piper...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Sassari Curated by ChEMBL | Assay Description Displacement of [3H]CP-55940 from CD1 mouse brain CB1 receptor | J Med Chem 49: 7502-12 (2006) Article DOI: 10.1021/jm060920d BindingDB Entry DOI: 10.7270/Q2057GRN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 1 (Mus musculus (Mouse)) | BDBM50176977 (1,4-dihydroindeno[1,2-c]-pyrazole | 6-chloro-1-(2'...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2.05E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Sassari Curated by ChEMBL | Assay Description Displacement of [3H]CP-55940 from CD1 mouse brain CB1 receptor | J Med Chem 49: 7502-12 (2006) Article DOI: 10.1021/jm060920d BindingDB Entry DOI: 10.7270/Q2057GRN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 2 (MOUSE) | BDBM50200160 (1-(2',4'-dichlorphenyl)-6-methyl-N-p-nitrophenyl-1...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2.12E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Sassari Curated by ChEMBL | Assay Description Displacement of [3H]CP-55940 from CD1 mouse spleen CB2 receptor | J Med Chem 49: 7502-12 (2006) Article DOI: 10.1021/jm060920d BindingDB Entry DOI: 10.7270/Q2057GRN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 1 (Mus musculus (Mouse)) | BDBM50200172 (1-(2',4'-dichlorophenyl)-6-methyl-N-phenyl-1,4-dih...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2.28E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Sassari Curated by ChEMBL | Assay Description Displacement of [3H]CP-55940 from CD1 mouse brain CB1 receptor | J Med Chem 49: 7502-12 (2006) Article DOI: 10.1021/jm060920d BindingDB Entry DOI: 10.7270/Q2057GRN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 1 (Mus musculus (Mouse)) | BDBM50200163 (1-(2',4'-dichlorophenyl)-6-methyl-N-phenyl-1,4-dih...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2.41E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Sassari Curated by ChEMBL | Assay Description Displacement of [3H]CP-55940 from CD1 mouse brain CB1 receptor | J Med Chem 49: 7502-12 (2006) Article DOI: 10.1021/jm060920d BindingDB Entry DOI: 10.7270/Q2057GRN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 1 (Mus musculus (Mouse)) | BDBM50200161 (1-(2',4'-dichlorophenyl)-6-methyl-N-o,p-dichloroph...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2.63E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Sassari Curated by ChEMBL | Assay Description Displacement of [3H]CP-55940 from CD1 mouse brain CB1 receptor | J Med Chem 49: 7502-12 (2006) Article DOI: 10.1021/jm060920d BindingDB Entry DOI: 10.7270/Q2057GRN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 2 (MOUSE) | BDBM50200164 (1-(2',4'-dichlorophenyl)-6-methyl-N-p-methoxypheny...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 3.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Sassari Curated by ChEMBL | Assay Description Displacement of [3H]CP-55940 from CD1 mouse spleen CB2 receptor | J Med Chem 49: 7502-12 (2006) Article DOI: 10.1021/jm060920d BindingDB Entry DOI: 10.7270/Q2057GRN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 1 (Mus musculus (Mouse)) | BDBM50200160 (1-(2',4'-dichlorphenyl)-6-methyl-N-p-nitrophenyl-1...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 4.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Sassari Curated by ChEMBL | Assay Description Displacement of [3H]CP-55940 from CD1 mouse brain CB1 receptor | J Med Chem 49: 7502-12 (2006) Article DOI: 10.1021/jm060920d BindingDB Entry DOI: 10.7270/Q2057GRN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 2 (MOUSE) | BDBM50200161 (1-(2',4'-dichlorophenyl)-6-methyl-N-o,p-dichloroph...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | >5.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Sassari Curated by ChEMBL | Assay Description Displacement of [3H]CP-55940 from CD1 mouse spleen CB2 receptor | J Med Chem 49: 7502-12 (2006) Article DOI: 10.1021/jm060920d BindingDB Entry DOI: 10.7270/Q2057GRN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 1 (Mus musculus (Mouse)) | BDBM50200167 (1-(2',4'-dichlorophenyl)-6-methyl-N-p-methylphenyl...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | >5.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Sassari Curated by ChEMBL | Assay Description Displacement of [3H]CP-55940 from CD1 mouse brain CB1 receptor | J Med Chem 49: 7502-12 (2006) Article DOI: 10.1021/jm060920d BindingDB Entry DOI: 10.7270/Q2057GRN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 1 (Mus musculus (Mouse)) | BDBM50200175 (1-(2',4'-dichlorophenyl)-6-methyl-N-p-fluorophenyl...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | >5.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Sassari Curated by ChEMBL | Assay Description Displacement of [3H]CP-55940 from CD1 mouse brain CB1 receptor | J Med Chem 49: 7502-12 (2006) Article DOI: 10.1021/jm060920d BindingDB Entry DOI: 10.7270/Q2057GRN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 2 (MOUSE) | BDBM50200173 (1-(2',4'-dichlorphenyl)-6-methyl-N-p-chlorophenyl-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | >5.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Sassari Curated by ChEMBL | Assay Description Displacement of [3H]CP-55940 from CD1 mouse spleen CB2 receptor | J Med Chem 49: 7502-12 (2006) Article DOI: 10.1021/jm060920d BindingDB Entry DOI: 10.7270/Q2057GRN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 2 (MOUSE) | BDBM50200174 (1-(2',4'-dichlorophenyl)-6-methyl-N-p-trifluoromet...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | >5.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Sassari Curated by ChEMBL | Assay Description Displacement of [3H]CP-55940 from CD1 mouse spleen CB2 receptor | J Med Chem 49: 7502-12 (2006) Article DOI: 10.1021/jm060920d BindingDB Entry DOI: 10.7270/Q2057GRN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 1 (Mus musculus (Mouse)) | BDBM50200164 (1-(2',4'-dichlorophenyl)-6-methyl-N-p-methoxypheny...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | >5.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Sassari Curated by ChEMBL | Assay Description Displacement of [3H]CP-55940 from CD1 mouse brain CB1 receptor | J Med Chem 49: 7502-12 (2006) Article DOI: 10.1021/jm060920d BindingDB Entry DOI: 10.7270/Q2057GRN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 1 (Mus musculus (Mouse)) | BDBM50200178 (1-(2',4'-dichlorophenyl)-6-methyl-N-m,p-dichloroph...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Sassari Curated by ChEMBL | Assay Description Displacement of [3H]CP-55940 from CD1 mouse brain CB1 receptor | J Med Chem 49: 7502-12 (2006) Article DOI: 10.1021/jm060920d BindingDB Entry DOI: 10.7270/Q2057GRN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 2 (MOUSE) | BDBM50200178 (1-(2',4'-dichlorophenyl)-6-methyl-N-m,p-dichloroph...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Sassari Curated by ChEMBL | Assay Description Displacement of [3H]CP-55940 from CD1 mouse spleen CB2 receptor | J Med Chem 49: 7502-12 (2006) Article DOI: 10.1021/jm060920d BindingDB Entry DOI: 10.7270/Q2057GRN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 1 (Mus musculus (Mouse)) | BDBM50200173 (1-(2',4'-dichlorphenyl)-6-methyl-N-p-chlorophenyl-...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Sassari Curated by ChEMBL | Assay Description Displacement of [3H]CP-55940 from CD1 mouse brain CB1 receptor | J Med Chem 49: 7502-12 (2006) Article DOI: 10.1021/jm060920d BindingDB Entry DOI: 10.7270/Q2057GRN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 1 (Mus musculus (Mouse)) | BDBM50200174 (1-(2',4'-dichlorophenyl)-6-methyl-N-p-trifluoromet...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Sassari Curated by ChEMBL | Assay Description Displacement of [3H]CP-55940 from CD1 mouse brain CB1 receptor | J Med Chem 49: 7502-12 (2006) Article DOI: 10.1021/jm060920d BindingDB Entry DOI: 10.7270/Q2057GRN | |||||||||||
More data for this Ligand-Target Pair |
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