The following articles (labelled with PubMed ID or TBD) are for your review
| PMID | Data | Article Title | Organization |
|---|
| 27390066 |
99 |
Discovery of potent and selective inhibitors of human aminopeptidases ERAP1 and ERAP2 by screening libraries of phosphorus-containing amino acid and dipeptide analogues. |
Wroclaw University of Technology |
| 27100031 |
85 |
A structural insight into the P1S1 binding mode of diaminoethylphosphonic and phosphinic acids, selective inhibitors of alanine aminopeptidases. |
Wroclaw University of Technology |
| 27039251 |
66 |
Design, synthesis and anti-HIV-1 evaluation of hydrazide-based peptidomimetics as selective gelatinase inhibitors. |
Shandong University |
| 26629857 |
44 |
Novel leucine ureido derivatives as aminopeptidase N inhibitors. Design, synthesis and activity evaluation. |
Fudan University |
| 26386821 |
15 |
Synthesis of chiral ND-322, ND-364 and ND-364 derivatives as selective inhibitors of human gelatinase. |
Shandong University |
| 25982416 |
43 |
Exploring S1 plasticity and probing S1' subsite of mammalian aminopeptidase N/CD13 with highly potent and selective aminobenzosuberone inhibitors. |
Universit£ |
| 25192493 |
57 |
Structure-guided, single-point modifications in the phosphinic dipeptide structure yield highly potent and selective inhibitors of neutral aminopeptidases. |
University of Athens |
| 24755524 |
60 |
Design, synthesis and preliminary evaluation ofa-sulfonyl¿-(glycinyl-amino)proline peptidomimetics as matrix metalloproteinase inhibitors. |
Shandong University |
| 24055078 |
14 |
Synthesis of amino-hydroxy-benzocycloheptenones as potent, selective, non-peptidic dinuclear zinc metalloaminopeptidase inhibitors. |
Universit£ |
| 23860593 |
17 |
Novelß-dicarbonyl derivatives as inhibitors of aminopeptidase N (APN). |
Shandong University |
| 23528299 |
4 |
Discovery of a synthetic Aminopeptidase N inhibitor LB-4b as a potential anticancer agent. |
Shandong University |
| 23510562 |
30 |
Novel indoline-2,3-dione derivatives as inhibitors of aminopeptidase N (APN). |
Shandong University |
| 23428964 |
9 |
Selective aminopeptidase-N (CD13) inhibitors with relevance to cancer chemotherapy. |
Universit£ |
| 23453219 |
29 |
Novel leucine ureido derivatives as inhibitors of aminopeptidase N (APN). |
Shandong University |
| 24900417 |
59 |
Development of Synthetic Aminopeptidase N/CD13 Inhibitors to Overcome Cancer Metastasis and Angiogenesis. |
TBA |
| 23176597 |
14 |
Structure-activity relationships and blood distribution of antiplasmodial aminopeptidase-1 inhibitors. |
University of Lille |
| 22796349 |
34 |
Rapid and efficient synthesis of a novel series of substituted aminobenzosuberone derivatives as potent, selective, non-peptidic neutral aminopeptidase inhibitors. |
Universit£ |
| 22901392 |
27 |
A novel aminopeptidase N inhibitor developed by virtual screening approach. |
Shandong Academy of Sciences |
| 22607877 |
38 |
Design, synthesis and biological evaluation of novel amino acid ureido derivatives as aminopeptidase N/CD13 inhibitors. |
Shandong University |
| 19339187 |
49 |
Novel aminopeptidase N inhibitors derived from antineoplaston AS2-5 (Part II). |
Shandong University |
| 19329328 |
42 |
Novel aminopeptidase N inhibitors derived from antineoplaston AS2-5 (Part I). |
Shandong University |
| 12801228 |
18 |
The most potent organophosphorus inhibitors of leucine aminopeptidase. Structure-based design, chemistry, and activity. |
Wroclaw University of Technology |
| 10753476 |
84 |
Phosphinic derivatives as new dual enkephalin-degrading enzyme inhibitors: synthesis, biological properties, and antinociceptive activities. |
University of Paris |
| 10602705 |
82 |
Investigation of subsite preferences in aminopeptidase A (EC 3.4.11.7) led to the design of the first highly potent and selective inhibitors of this enzyme. |
University of Paris |
| 1348542 |
23 |
Potent and systemically active aminopeptidase N inhibitors designed from active-site investigation. |
University of Paris |
| 1347791 |
35 |
Analgesic dipeptide derivatives. 7. 3,7-Diamino-2-hydroxyheptanoic acid (DAHHA) containing dipeptide analogues of the analgesic compound H-Lys-Trp(Nps)-OMe. |
Instituto De Qu£Mica M£Dica |
| 3184126 |
46 |
Synthesis of sulfur-containing analogues of bestatin. Inhibition of aminopeptidases by alpha-thiolbestatin analogues. |
University of Wisconsin |
| 3897541 |
27 |
New bidentates as full inhibitors of enkephalin-degrading enzymes: synthesis and analgesic properties. |
TBA |
| 6142952 |
42 |
Inhibition of aminopeptidases by amastatin and bestatin derivatives. Effect of inhibitor structure on slow-binding processes. |
TBA |
| 10386926 |
32 |
Design of the first highly potent and selective aminopeptidase N (EC 3.4.11.2) inhibitor. |
University of Paris |
| 22206607 |
9 |
Novel potent 2,5-pyrrolidinedione peptidomimetics as aminopeptidase N inhibitors. Design, synthesis and activity evaluation. |
Central South University |
| 21911297 |
40 |
Design, synthesis and biological evaluation of novel 1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid derivatives as aminopeptidase N/CD13 inhibitors. |
Shandong University |
| 21843945 |
36 |
A novel amino-benzosuberone derivative is a picomolar inhibitor of mammalian aminopeptidase N/CD13. |
Universit£ |
| 21802307 |
64 |
Novel aminopeptidase N (APN/CD13) inhibitors derived from chloramphenicol amine. |
Shandong University |
| 18458130 |
8 |
Chemical target validation studies of aminopeptidase in malaria parasites using alpha-aminoalkylphosphonate and phosphonopeptide inhibitors. |
Trinity College |
| 21194957 |
27 |
Design, synthesis and biological evaluation of novel L-lysine ureido derivatives as aminopeptidase N inhibitors. |
Shandong University |
| 20637634 |
48 |
Novel aminopeptidase N (APN/CD13) inhibitors derived from 3-phenylalanyl-N'-substituted-2,6-piperidinedione. |
Shandong University |
| 20347318 |
49 |
New aromatic monoesters of alpha-aminoaralkylphosphonic acids as inhibitors of aminopeptidase N/CD13. |
Wroclaw University of Technology |
| 19969464 |
56 |
Design, synthesis and primary activity assay of bi- or tri-peptide analogues with the scaffold l-arginine as amino-peptidase N/CD13 inhibitors. |
Shandong University |
| 19782572 |
62 |
Design, synthesis, and preliminary studies of the activity of novel derivatives of N-cinnamoyl-L-aspartic acid as inhibitors of aminopeptidase N/CD13. |
Shandong University |
| 19683842 |
27 |
Novel cyclic-imide peptidomimetics as aminopeptidase N inhibitors. Design, chemistry and activity evaluation. Part I. |
Shandong University |
| 19454370 |
52 |
Design, synthesis and primary activity evaluation of L-arginine derivatives as amino-peptidase N/CD13 inhibitors. |
Shandong University |
| 19423354 |
26 |
Design and synthesis of novel chloramphenicol amine derivatives as potent aminopeptidase N (APN/CD13) inhibitors. |
Shandong University |
| 19299146 |
33 |
Design, synthesis and SAR studies of tripeptide analogs with the scaffold 3-phenylpropane-1,2-diamine as aminopeptidase N/CD13 inhibitors. |
Shandong University |
| 18996018 |
42 |
Novel 3-phenylpropane-1,2-diamine derivates as inhibitors of aminopeptidase N (APN). |
Shandong University |
| 18571419 |
24 |
Novel aminopeptidase N inhibitors derived from 1,3,4-thiadiazole scaffold. |
Shandong University |
| 18524593 |
12 |
First synthesis of alpha-aminoalkyl-(N-substituted)thiocarbamoyl-phosphinates: inhibitors of aminopeptidase N (APN/CD13) with the new zinc-binding group. |
Wroclaw University of Technology |
| 17433673 |
44 |
Novel 3-galloylamido-N'-substituted-2,6-piperidinedione-N-acetamide peptidomimetics as metalloproteinase inhibitors. |
Shandong University |
| 17326615 |
49 |
Novel selective inhibitors of the zinc plasmodial aminopeptidase PfA-M1 as potential antimalarial agents. |
University of Lille |
| 17070058 |
15 |
A library of novel hydroxamic acids targeting the metallo-protease family: design, parallel synthesis and screening. |
University of Lille 2 |
| 12930151 |
1 |
Synthesis and biological evaluation of novel flavone-8-acetic acid derivatives as reversible inhibitors of aminopeptidase N/CD13. |
Institut Curie |
| 30737134 |
52 |
Leucine ureido derivatives as aminopeptidase N inhibitors using click chemistry. Part II. |
Shandong University |
| 30846252 |
23 |
Recent developments in the synthesis and applications of phosphinic peptide analogs. |
Wroclaw University of Technology |
| 26513642 |
28 |
Highly functionalized tetrahydropyridines are cytotoxic and selective inhibitors of human puromycin sensitive aminopeptidase. |
Csir-Indian Institute of Chemical Technology |
| 7915326 |
28 |
Differential inhibition of aminopeptidase A and aminopeptidase N by new beta-amino thiols. |
University of Paris |
| 29630364 |
63 |
Design of Aminopeptidase N Inhibitors as Anti-cancer Agents. |
Jadavpur University |
| 2738884 |
30 |
New kelatorphan-related inhibitors of enkephalin metabolism: improved antinociceptive properties. |
University of Paris |
| 29202398 |
17 |
Synthesis and biological characterization of ubenimex-fluorouracil conjugates for anti-cancer therapy. |
Shandong University |
| 29859750 |
56 |
Novel leucine ureido derivatives as aminopeptidase N inhibitors using click chemistry. |
Shandong University |
| 28728898 |
3 |
KBE009: An antimalarial bestatin-like inhibitor of the Plasmodium falciparum M1 aminopeptidase discovered in an Ugi multicomponent reaction-derived peptidomimetic library. |
Universidad De La Habana |
Search and Browse
