Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
C-C chemokine receptor type 8 (Homo sapiens (Human)) | BDBM50185909 (2-(3-((1-(3-(2-chlorophenoxy)benzyl)piperidin-4-yl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 6 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Millennium Pharmaceuticals Curated by ChEMBL | Assay Description Displacement of [125I]I309 from human CCR8 expressed in L1.2 cells | J Med Chem 49: 2669-72 (2006) Article DOI: 10.1021/jm050965z BindingDB Entry DOI: 10.7270/Q2GH9HJX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-C chemokine receptor type 8 (Homo sapiens (Human)) | BDBM50185912 (2-(4-{1-[3-(2-chloro-phenoxy)-benzyl]-piperidin-4-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 9 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Millennium Pharmaceuticals Curated by ChEMBL | Assay Description Displacement of [125I]I309 from human CCR8 expressed in L1.2 cells | J Med Chem 49: 2669-72 (2006) Article DOI: 10.1021/jm050965z BindingDB Entry DOI: 10.7270/Q2GH9HJX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-C chemokine receptor type 8 (Homo sapiens (Human)) | BDBM50185908 (1-ethyl-4-phenyl-piperidine-4-carboxylic acid {1-[...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 11 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Millennium Pharmaceuticals Curated by ChEMBL | Assay Description Displacement of [125I]I309 from human CCR8 expressed in L1.2 cells | J Med Chem 49: 2669-72 (2006) Article DOI: 10.1021/jm050965z BindingDB Entry DOI: 10.7270/Q2GH9HJX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-C chemokine receptor type 8 (Homo sapiens (Human)) | BDBM50185910 (1-ethyl-4-phenyl-piperidine-4-carboxylic acid {1-[...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 15 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Millennium Pharmaceuticals Curated by ChEMBL | Assay Description Displacement of [125I]I309 from human CCR8 expressed in L1.2 cells | J Med Chem 49: 2669-72 (2006) Article DOI: 10.1021/jm050965z BindingDB Entry DOI: 10.7270/Q2GH9HJX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-C chemokine receptor type 8 (Homo sapiens (Human)) | BDBM50185906 (1-[3-(2-chlorophenoxy)benzyl]-4-{[(1-ethyl-4-pheny...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 23 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Millennium Pharmaceuticals Curated by ChEMBL | Assay Description Displacement of [125I]I309 from human CCR8 expressed in L1.2 cells | J Med Chem 49: 2669-72 (2006) Article DOI: 10.1021/jm050965z BindingDB Entry DOI: 10.7270/Q2GH9HJX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-C chemokine receptor type 8 (Homo sapiens (Human)) | BDBM50185904 ((+/-) 3-phenyl-pyrrolidine-3-carboxylic acid {1-[3...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 27 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Millennium Pharmaceuticals Curated by ChEMBL | Assay Description Displacement of [125I]I309 from human CCR8 expressed in L1.2 cells | J Med Chem 49: 2669-72 (2006) Article DOI: 10.1021/jm050965z BindingDB Entry DOI: 10.7270/Q2GH9HJX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-C chemokine receptor type 8 (Homo sapiens (Human)) | BDBM50185902 (1-[3-(2-methoxy-phenoxy)-benzyl]-4-[(4-phenyl-pipe...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 60 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Millennium Pharmaceuticals Curated by ChEMBL | Assay Description Displacement of [125I]I309 from human CCR8 expressed in L1.2 cells | J Med Chem 49: 2669-72 (2006) Article DOI: 10.1021/jm050965z BindingDB Entry DOI: 10.7270/Q2GH9HJX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-C chemokine receptor type 8 (Homo sapiens (Human)) | BDBM50185905 (4-phenyl-piperidine-4-carboxylic acid {1-[3-(2-met...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 62 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Millennium Pharmaceuticals Curated by ChEMBL | Assay Description Displacement of [125I]I309 from human CCR8 expressed in L1.2 cells | J Med Chem 49: 2669-72 (2006) Article DOI: 10.1021/jm050965z BindingDB Entry DOI: 10.7270/Q2GH9HJX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-C chemokine receptor type 4 (Homo sapiens (Human)) | BDBM50209260 ((S)-1-(5-chloronaphthalen-2-ylsulfonyl)-N-methyl-N...) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 100 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Millennium Pharmaceuticals Curated by ChEMBL | Assay Description Displacement of human TARC from recombinant CCR4 receptor expressed in CHO cells coexpressing Galpha16 by FLIPR assay | Bioorg Med Chem Lett 17: 3141-5 (2007) Article DOI: 10.1016/j.bmcl.2007.03.030 BindingDB Entry DOI: 10.7270/Q2TD9X2P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-C chemokine receptor type 4 (Homo sapiens (Human)) | BDBM50209260 ((S)-1-(5-chloronaphthalen-2-ylsulfonyl)-N-methyl-N...) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 150 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Millennium Pharmaceuticals Curated by ChEMBL | Assay Description Displacement of mouse MDC from recombinant CCR4 receptor expressed in CHO cells coexpressing Galpha16 by FLIPR assay | Bioorg Med Chem Lett 17: 3141-5 (2007) Article DOI: 10.1016/j.bmcl.2007.03.030 BindingDB Entry DOI: 10.7270/Q2TD9X2P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-C chemokine receptor type 4 (Homo sapiens (Human)) | BDBM50209278 ((S)-N-(1-(2-carbamoylphenethyl)piperidin-4-yl)-1-(...) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 240 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Millennium Pharmaceuticals Curated by ChEMBL | Assay Description Displacement of human TARC from recombinant CCR4 receptor expressed in CHO cells coexpressing Galpha16 by FLIPR assay | Bioorg Med Chem Lett 17: 3141-5 (2007) Article DOI: 10.1016/j.bmcl.2007.03.030 BindingDB Entry DOI: 10.7270/Q2TD9X2P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-C chemokine receptor type 8 (Homo sapiens (Human)) | BDBM50185915 (1-(4-chloro-phenyl)-cyclohexanecarboxylic acid {1-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | 250 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Millennium Pharmaceuticals Curated by ChEMBL | Assay Description Displacement of [125I]I309 from human CCR8 expressed in L1.2 cells | J Med Chem 49: 2669-72 (2006) Article DOI: 10.1021/jm050965z BindingDB Entry DOI: 10.7270/Q2GH9HJX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-C chemokine receptor type 8 (Homo sapiens (Human)) | BDBM50185907 (CHEMBL210322 | N-{1-[3-(2-methoxy-phenoxy)-benzyl]...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 250 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Millennium Pharmaceuticals Curated by ChEMBL | Assay Description Displacement of [125I]I309 from human CCR8 expressed in L1.2 cells | J Med Chem 49: 2669-72 (2006) Article DOI: 10.1021/jm050965z BindingDB Entry DOI: 10.7270/Q2GH9HJX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-C chemokine receptor type 4 (Homo sapiens (Human)) | BDBM50209261 ((S)-N-(1-(2-fluorophenethyl)piperidin-4-yl)-1-(5-c...) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 260 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Millennium Pharmaceuticals Curated by ChEMBL | Assay Description Displacement of human TARC from recombinant CCR4 receptor expressed in CHO cells coexpressing Galpha16 by FLIPR assay | Bioorg Med Chem Lett 17: 3141-5 (2007) Article DOI: 10.1016/j.bmcl.2007.03.030 BindingDB Entry DOI: 10.7270/Q2TD9X2P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-C chemokine receptor type 4 (Homo sapiens (Human)) | BDBM50209251 ((S)-N-(1-(2-aminophenethyl)piperidin-4-yl)-1-(5-ch...) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 280 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Millennium Pharmaceuticals Curated by ChEMBL | Assay Description Displacement of human TARC from recombinant CCR4 receptor expressed in CHO cells coexpressing Galpha16 by FLIPR assay | Bioorg Med Chem Lett 17: 3141-5 (2007) Article DOI: 10.1016/j.bmcl.2007.03.030 BindingDB Entry DOI: 10.7270/Q2TD9X2P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-C chemokine receptor type 4 (Homo sapiens (Human)) | BDBM50209257 ((S)-N-(1-(3-chlorophenethyl)piperidin-4-yl)-1-(5-c...) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 400 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Millennium Pharmaceuticals Curated by ChEMBL | Assay Description Displacement of human TARC from recombinant CCR4 receptor expressed in CHO cells coexpressing Galpha16 by FLIPR assay | Bioorg Med Chem Lett 17: 3141-5 (2007) Article DOI: 10.1016/j.bmcl.2007.03.030 BindingDB Entry DOI: 10.7270/Q2TD9X2P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-C chemokine receptor type 4 (Homo sapiens (Human)) | BDBM50209279 ((S)-N-(1-(2-(trifluoromethyl)phenethyl)piperidin-4...) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 420 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Millennium Pharmaceuticals Curated by ChEMBL | Assay Description Displacement of human TARC from recombinant CCR4 receptor expressed in CHO cells coexpressing Galpha16 by FLIPR assay | Bioorg Med Chem Lett 17: 3141-5 (2007) Article DOI: 10.1016/j.bmcl.2007.03.030 BindingDB Entry DOI: 10.7270/Q2TD9X2P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-C chemokine receptor type 4 (Homo sapiens (Human)) | BDBM50209262 ((S)-N-(1-(2-chlorophenethyl)piperidin-4-yl)-1-(5-c...) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 460 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Millennium Pharmaceuticals Curated by ChEMBL | Assay Description Displacement of human TARC from recombinant CCR4 receptor expressed in CHO cells coexpressing Galpha16 by FLIPR assay | Bioorg Med Chem Lett 17: 3141-5 (2007) Article DOI: 10.1016/j.bmcl.2007.03.030 BindingDB Entry DOI: 10.7270/Q2TD9X2P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-C chemokine receptor type 4 (Homo sapiens (Human)) | BDBM50209265 ((S)-N-(1-(3-methoxyphenethyl)piperidin-4-yl)-1-(5-...) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 470 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Millennium Pharmaceuticals Curated by ChEMBL | Assay Description Displacement of human TARC from recombinant CCR4 receptor expressed in CHO cells coexpressing Galpha16 by FLIPR assay | Bioorg Med Chem Lett 17: 3141-5 (2007) Article DOI: 10.1016/j.bmcl.2007.03.030 BindingDB Entry DOI: 10.7270/Q2TD9X2P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-C chemokine receptor type 4 (Homo sapiens (Human)) | BDBM50209260 ((S)-1-(5-chloronaphthalen-2-ylsulfonyl)-N-methyl-N...) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 500 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Millennium Pharmaceuticals Curated by ChEMBL | Assay Description Displacement of human MDC from recombinant CCR4 receptor expressed in CHO cells coexpressing Galpha16 by FLIPR assay | Bioorg Med Chem Lett 17: 3141-5 (2007) Article DOI: 10.1016/j.bmcl.2007.03.030 BindingDB Entry DOI: 10.7270/Q2TD9X2P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-C chemokine receptor type 4 (Homo sapiens (Human)) | BDBM50209253 ((S)-2-(2-(4-(1-(5-chloronaphthalen-2-ylsulfonyl)-N...) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 530 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Millennium Pharmaceuticals Curated by ChEMBL | Assay Description Displacement of human TARC from recombinant CCR4 receptor expressed in CHO cells coexpressing Galpha16 by FLIPR assay | Bioorg Med Chem Lett 17: 3141-5 (2007) Article DOI: 10.1016/j.bmcl.2007.03.030 BindingDB Entry DOI: 10.7270/Q2TD9X2P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-C chemokine receptor type 4 (Homo sapiens (Human)) | BDBM50209268 ((S)-N-methyl-1-(naphthalen-2-ylsulfonyl)-N-(1-phen...) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 590 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Millennium Pharmaceuticals Curated by ChEMBL | Assay Description Displacement of human TARC from recombinant CCR4 receptor expressed in CHO cells coexpressing Galpha16 by FLIPR assay | Bioorg Med Chem Lett 17: 3141-5 (2007) Article DOI: 10.1016/j.bmcl.2007.03.030 BindingDB Entry DOI: 10.7270/Q2TD9X2P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-C chemokine receptor type 4 (Homo sapiens (Human)) | BDBM50209255 ((S)-N-methyl-1-(naphthalen-2-ylsulfonyl)-N-(1-(3-p...) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 620 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Millennium Pharmaceuticals Curated by ChEMBL | Assay Description Displacement of human TARC from recombinant CCR4 receptor expressed in CHO cells coexpressing Galpha16 by FLIPR assay | Bioorg Med Chem Lett 17: 3141-5 (2007) Article DOI: 10.1016/j.bmcl.2007.03.030 BindingDB Entry DOI: 10.7270/Q2TD9X2P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily H member 2 (Homo sapiens (Human)) | BDBM50185905 (4-phenyl-piperidine-4-carboxylic acid {1-[3-(2-met...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 800 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Millennium Pharmaceuticals Curated by ChEMBL | Assay Description Displacement of [3H]dofetilide from hERG expressed in HEK293 cells | J Med Chem 49: 2669-72 (2006) Article DOI: 10.1021/jm050965z BindingDB Entry DOI: 10.7270/Q2GH9HJX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-C chemokine receptor type 4 (Homo sapiens (Human)) | BDBM50209258 ((S)-N-(1-(4-chlorophenethyl)piperidin-4-yl)-1-(5-c...) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 820 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Millennium Pharmaceuticals Curated by ChEMBL | Assay Description Displacement of human TARC from recombinant CCR4 receptor expressed in CHO cells coexpressing Galpha16 by FLIPR assay | Bioorg Med Chem Lett 17: 3141-5 (2007) Article DOI: 10.1016/j.bmcl.2007.03.030 BindingDB Entry DOI: 10.7270/Q2TD9X2P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-C chemokine receptor type 4 (Homo sapiens (Human)) | BDBM50209269 ((S)-1-(5-fluoronaphthalen-2-ylsulfonyl)-N-methyl-N...) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 850 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Millennium Pharmaceuticals Curated by ChEMBL | Assay Description Displacement of human TARC from recombinant CCR4 receptor expressed in CHO cells coexpressing Galpha16 by FLIPR assay | Bioorg Med Chem Lett 17: 3141-5 (2007) Article DOI: 10.1016/j.bmcl.2007.03.030 BindingDB Entry DOI: 10.7270/Q2TD9X2P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-C chemokine receptor type 4 (Homo sapiens (Human)) | BDBM50209263 ((S)-N-(1-benzylpiperidin-4-yl)-N-methyl-1-(naphtha...) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Millennium Pharmaceuticals Curated by ChEMBL | Assay Description Displacement of human TARC from recombinant CCR4 receptor expressed in CHO cells coexpressing Galpha16 by FLIPR assay | Bioorg Med Chem Lett 17: 3141-5 (2007) Article DOI: 10.1016/j.bmcl.2007.03.030 BindingDB Entry DOI: 10.7270/Q2TD9X2P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-C chemokine receptor type 8 (Homo sapiens (Human)) | BDBM50185911 (CHEMBL205692 | N-[1-(3-phenoxy-benzyl)-piperidin-4...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Millennium Pharmaceuticals Curated by ChEMBL | Assay Description Displacement of [125I]I309 from human CCR8 expressed in L1.2 cells | J Med Chem 49: 2669-72 (2006) Article DOI: 10.1021/jm050965z BindingDB Entry DOI: 10.7270/Q2GH9HJX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-C chemokine receptor type 8 (Homo sapiens (Human)) | BDBM50185903 (1-(3-phenoxy-benzyl)-piperidine-4-carboxylic acid ...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2.60E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Millennium Pharmaceuticals Curated by ChEMBL | Assay Description Displacement of [125I]I309 from human CCR8 expressed in L1.2 cells | J Med Chem 49: 2669-72 (2006) Article DOI: 10.1021/jm050965z BindingDB Entry DOI: 10.7270/Q2GH9HJX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-C chemokine receptor type 4 (Homo sapiens (Human)) | BDBM50209281 ((S)-1-(5-chloronaphthalen-2-ylsulfonyl)-N-ethyl-N-...) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Millennium Pharmaceuticals Curated by ChEMBL | Assay Description Displacement of human TARC from recombinant CCR4 receptor expressed in CHO cells coexpressing Galpha16 by FLIPR assay | Bioorg Med Chem Lett 17: 3141-5 (2007) Article DOI: 10.1016/j.bmcl.2007.03.030 BindingDB Entry DOI: 10.7270/Q2TD9X2P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-C chemokine receptor type 4 (Homo sapiens (Human)) | BDBM50209270 ((S)-N-(1-benzylpiperidin-4-yl)-1-(naphthalen-2-yls...) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 4.60E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Millennium Pharmaceuticals Curated by ChEMBL | Assay Description Displacement of human TARC from recombinant CCR4 receptor expressed in CHO cells coexpressing Galpha16 by FLIPR assay | Bioorg Med Chem Lett 17: 3141-5 (2007) Article DOI: 10.1016/j.bmcl.2007.03.030 BindingDB Entry DOI: 10.7270/Q2TD9X2P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-C chemokine receptor type 8 (Homo sapiens (Human)) | BDBM50185916 (1-(3-phenoxy-benzyl)-piperidine-4-carboxylic acid ...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 9.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Millennium Pharmaceuticals Curated by ChEMBL | Assay Description Displacement of [125I]I309 from human CCR8 expressed in L1.2 cells | J Med Chem 49: 2669-72 (2006) Article DOI: 10.1021/jm050965z BindingDB Entry DOI: 10.7270/Q2GH9HJX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-C chemokine receptor type 8 (Homo sapiens (Human)) | BDBM50185913 (CHEMBL381354 | N-[1-(3-phenoxy-benzyl)-piperidin-4...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 9.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Millennium Pharmaceuticals Curated by ChEMBL | Assay Description Displacement of [125I]I309 from human CCR8 expressed in L1.2 cells | J Med Chem 49: 2669-72 (2006) Article DOI: 10.1021/jm050965z BindingDB Entry DOI: 10.7270/Q2GH9HJX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily H member 2 (Homo sapiens (Human)) | BDBM50185909 (2-(3-((1-(3-(2-chlorophenoxy)benzyl)piperidin-4-yl...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Millennium Pharmaceuticals Curated by ChEMBL | Assay Description Displacement of [3H]dofetilide from hERG expressed in HEK293 cells | J Med Chem 49: 2669-72 (2006) Article DOI: 10.1021/jm050965z BindingDB Entry DOI: 10.7270/Q2GH9HJX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-C chemokine receptor type 4 (Homo sapiens (Human)) | BDBM50209246 ((S)-1-(naphthalen-2-ylsulfonyl)-N-(1-(pyridin-3-yl...) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Millennium Pharmaceuticals Curated by ChEMBL | Assay Description Displacement of human TARC from recombinant CCR4 receptor expressed in CHO cells coexpressing Galpha16 by FLIPR assay | Bioorg Med Chem Lett 17: 3141-5 (2007) Article DOI: 10.1016/j.bmcl.2007.03.030 BindingDB Entry DOI: 10.7270/Q2TD9X2P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-C chemokine receptor type 4 (Homo sapiens (Human)) | BDBM50209256 ((S)-N-(1-benzylpiperidin-4-yl)-1-(4-isopropylpheny...) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Millennium Pharmaceuticals Curated by ChEMBL | Assay Description Displacement of human TARC from recombinant CCR4 receptor expressed in CHO cells coexpressing Galpha16 by FLIPR assay | Bioorg Med Chem Lett 17: 3141-5 (2007) Article DOI: 10.1016/j.bmcl.2007.03.030 BindingDB Entry DOI: 10.7270/Q2TD9X2P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-C chemokine receptor type 4 (Homo sapiens (Human)) | BDBM50209248 ((S)-ethyl 2-(1-(naphthalen-2-ylsulfonyl)-N-(1-phen...) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Millennium Pharmaceuticals Curated by ChEMBL | Assay Description Displacement of human TARC from recombinant CCR4 receptor expressed in CHO cells coexpressing Galpha16 by FLIPR assay | Bioorg Med Chem Lett 17: 3141-5 (2007) Article DOI: 10.1016/j.bmcl.2007.03.030 BindingDB Entry DOI: 10.7270/Q2TD9X2P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-C chemokine receptor type 4 (Homo sapiens (Human)) | BDBM50209252 ((S)-1-(5-chloronaphthalen-2-ylsulfonyl)-N-methyl-N...) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Millennium Pharmaceuticals Curated by ChEMBL | Assay Description Displacement of human TARC from recombinant CCR4 receptor expressed in CHO cells coexpressing Galpha16 by FLIPR assay | Bioorg Med Chem Lett 17: 3141-5 (2007) Article DOI: 10.1016/j.bmcl.2007.03.030 BindingDB Entry DOI: 10.7270/Q2TD9X2P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-C chemokine receptor type 4 (Homo sapiens (Human)) | BDBM50209250 ((S)-N-methyl-1-(naphthalen-2-ylsulfonyl)-N-(1-(phe...) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Millennium Pharmaceuticals Curated by ChEMBL | Assay Description Displacement of human TARC from recombinant CCR4 receptor expressed in CHO cells coexpressing Galpha16 by FLIPR assay | Bioorg Med Chem Lett 17: 3141-5 (2007) Article DOI: 10.1016/j.bmcl.2007.03.030 BindingDB Entry DOI: 10.7270/Q2TD9X2P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-C chemokine receptor type 4 (Homo sapiens (Human)) | BDBM50209247 ((S)-1-(5-aminonaphthalen-2-ylsulfonyl)-N-methyl-N-...) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Millennium Pharmaceuticals Curated by ChEMBL | Assay Description Displacement of human TARC from recombinant CCR4 receptor expressed in CHO cells coexpressing Galpha16 by FLIPR assay | Bioorg Med Chem Lett 17: 3141-5 (2007) Article DOI: 10.1016/j.bmcl.2007.03.030 BindingDB Entry DOI: 10.7270/Q2TD9X2P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-C chemokine receptor type 4 (Homo sapiens (Human)) | BDBM50209275 ((S)-N-(1-isobutylpiperidin-4-yl)-1-(naphthalen-2-y...) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Millennium Pharmaceuticals Curated by ChEMBL | Assay Description Displacement of human MDC from recombinant CCR4 receptor expressed in CHO cells coexpressing Galpha16 by FLIPR assay | Bioorg Med Chem Lett 17: 3141-5 (2007) Article DOI: 10.1016/j.bmcl.2007.03.030 BindingDB Entry DOI: 10.7270/Q2TD9X2P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-C chemokine receptor type 4 (Homo sapiens (Human)) | BDBM50209273 ((S)-1-(5-acetamidonaphthalen-2-ylsulfonyl)-N-methy...) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Millennium Pharmaceuticals Curated by ChEMBL | Assay Description Displacement of human TARC from recombinant CCR4 receptor expressed in CHO cells coexpressing Galpha16 by FLIPR assay | Bioorg Med Chem Lett 17: 3141-5 (2007) Article DOI: 10.1016/j.bmcl.2007.03.030 BindingDB Entry DOI: 10.7270/Q2TD9X2P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-C chemokine receptor type 4 (Homo sapiens (Human)) | BDBM50209274 ((S)-N-(2-morpholinoethyl)-1-(naphthalen-2-ylsulfon...) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Millennium Pharmaceuticals Curated by ChEMBL | Assay Description Displacement of human TARC from recombinant CCR4 receptor expressed in CHO cells coexpressing Galpha16 by FLIPR assay | Bioorg Med Chem Lett 17: 3141-5 (2007) Article DOI: 10.1016/j.bmcl.2007.03.030 BindingDB Entry DOI: 10.7270/Q2TD9X2P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily H member 2 (Homo sapiens (Human)) | BDBM50185902 (1-[3-(2-methoxy-phenoxy)-benzyl]-4-[(4-phenyl-pipe...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Millennium Pharmaceuticals Curated by ChEMBL | Assay Description Displacement of [3H]dofetilide from hERG expressed in HEK293 cells | J Med Chem 49: 2669-72 (2006) Article DOI: 10.1021/jm050965z BindingDB Entry DOI: 10.7270/Q2GH9HJX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-C chemokine receptor type 4 (Homo sapiens (Human)) | BDBM50209271 ((S)-2-(1-(naphthalen-2-ylsulfonyl)-N-(1-phenethylp...) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Millennium Pharmaceuticals Curated by ChEMBL | Assay Description Displacement of human TARC from recombinant CCR4 receptor expressed in CHO cells coexpressing Galpha16 by FLIPR assay | Bioorg Med Chem Lett 17: 3141-5 (2007) Article DOI: 10.1016/j.bmcl.2007.03.030 BindingDB Entry DOI: 10.7270/Q2TD9X2P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-C chemokine receptor type 4 (Homo sapiens (Human)) | BDBM50209272 ((S)-1-(naphthalen-2-ylsulfonyl)-N-(1-(pyridin-2-yl...) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Millennium Pharmaceuticals Curated by ChEMBL | Assay Description Displacement of human TARC from recombinant CCR4 receptor expressed in CHO cells coexpressing Galpha16 by FLIPR assay | Bioorg Med Chem Lett 17: 3141-5 (2007) Article DOI: 10.1016/j.bmcl.2007.03.030 BindingDB Entry DOI: 10.7270/Q2TD9X2P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily H member 2 (Homo sapiens (Human)) | BDBM50185906 (1-[3-(2-chlorophenoxy)benzyl]-4-{[(1-ethyl-4-pheny...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Millennium Pharmaceuticals Curated by ChEMBL | Assay Description Displacement of [3H]dofetilide from hERG expressed in HEK293 cells | J Med Chem 49: 2669-72 (2006) Article DOI: 10.1021/jm050965z BindingDB Entry DOI: 10.7270/Q2GH9HJX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-C chemokine receptor type 4 (Homo sapiens (Human)) | BDBM50209249 ((S)-N-(1-benzylpiperidin-4-yl)-1-(benzylsulfonyl)p...) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.50E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Millennium Pharmaceuticals Curated by ChEMBL | Assay Description Displacement of human MDC from recombinant CCR4 receptor expressed in CHO cells coexpressing Galpha16 by FLIPR assay | Bioorg Med Chem Lett 17: 3141-5 (2007) Article DOI: 10.1016/j.bmcl.2007.03.030 BindingDB Entry DOI: 10.7270/Q2TD9X2P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-C chemokine receptor type 4 (Homo sapiens (Human)) | BDBM50209266 ((S)-N2-(1-benzylpiperidin-4-yl)-N1-(4-tert-butylph...) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | >2.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Millennium Pharmaceuticals Curated by ChEMBL | Assay Description Displacement of human TARC from recombinant CCR4 receptor expressed in CHO cells coexpressing Galpha16 by FLIPR assay | Bioorg Med Chem Lett 17: 3141-5 (2007) Article DOI: 10.1016/j.bmcl.2007.03.030 BindingDB Entry DOI: 10.7270/Q2TD9X2P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-C chemokine receptor type 4 (Homo sapiens (Human)) | BDBM50209277 ((R)-N-(1-benzylpiperidin-4-yl)-1-(naphthalen-2-yls...) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2.02E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Millennium Pharmaceuticals Curated by ChEMBL | Assay Description Displacement of human TARC from recombinant CCR4 receptor expressed in CHO cells coexpressing Galpha16 by FLIPR assay | Bioorg Med Chem Lett 17: 3141-5 (2007) Article DOI: 10.1016/j.bmcl.2007.03.030 BindingDB Entry DOI: 10.7270/Q2TD9X2P | |||||||||||
More data for this Ligand-Target Pair |
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