Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Vitamin D3 receptor (Homo sapiens (Human)) | BDBM50388528 (CHEMBL2058272) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid PDB UniChem Similars | Article PubMed | n/a | n/a | 0.0290 | n/a | n/a | n/a | n/a | n/a | n/a |
Showa Pharmaceutical University Curated by ChEMBL | Assay Description Displacement of [3H]1alpha,25-dihydroxyvitamin D3 from human recombinant GST-tagged vitamin D3 receptor LBD expressed in Escherichia coli BL21 after ... | J Med Chem 55: 4373-81 (2012) Article DOI: 10.1021/jm300230a BindingDB Entry DOI: 10.7270/Q25M66R0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Vitamin D3 receptor (Homo sapiens (Human)) | BDBM50200182 ((1S,3R,5Z,7E)-9,10-secocholesta-5,7,10(19)-triene-...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG MMDB PC cid PC sid PDB UniChem Patents Similars | DrugBank Article PubMed | n/a | n/a | 0.0600 | n/a | n/a | n/a | n/a | n/a | n/a |
Showa Pharmaceutical University Curated by ChEMBL | Assay Description Displacement of [3H]-1alpha,25-dihydroxyvitamin D3 from recombinant human VDR LBD expressed in Escherichia coli BL21 (DE3) pLysS after 16 hrs | Bioorg Med Chem 23: 7274-81 (2015) Article DOI: 10.1016/j.bmc.2015.10.026 BindingDB Entry DOI: 10.7270/Q2R78H20 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Vitamin D3 receptor (Homo sapiens (Human)) | BDBM50129805 (CHEMBL3629552) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid PDB UniChem Similars | Article PubMed | n/a | n/a | 0.210 | n/a | n/a | n/a | n/a | n/a | n/a |
Showa Pharmaceutical University Curated by ChEMBL | Assay Description Displacement of [3H]-1alpha,25-dihydroxyvitamin D3 from recombinant human VDR LBD expressed in Escherichia coli BL21 (DE3) pLysS after 16 hrs | Bioorg Med Chem 23: 7274-81 (2015) Article DOI: 10.1016/j.bmc.2015.10.026 BindingDB Entry DOI: 10.7270/Q2R78H20 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Vitamin D3 receptor (Homo sapiens (Human)) | BDBM50388529 (CHEMBL2058273) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.380 | n/a | n/a | n/a | n/a | n/a | n/a |
Showa Pharmaceutical University Curated by ChEMBL | Assay Description Displacement of [3H]1alpha,25-dihydroxyvitamin D3 from human recombinant GST-tagged vitamin D3 receptor LBD expressed in Escherichia coli BL21 after ... | J Med Chem 55: 4373-81 (2012) Article DOI: 10.1021/jm300230a BindingDB Entry DOI: 10.7270/Q25M66R0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Vitamin D3 receptor (Homo sapiens (Human)) | BDBM50388530 (CHEMBL2058274) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid PDB UniChem Similars | Article PubMed | n/a | n/a | 0.410 | n/a | n/a | n/a | n/a | n/a | n/a |
Showa Pharmaceutical University Curated by ChEMBL | Assay Description Displacement of [3H]1alpha,25-dihydroxyvitamin D3 from human recombinant GST-tagged vitamin D3 receptor LBD expressed in Escherichia coli BL21 after ... | J Med Chem 55: 4373-81 (2012) Article DOI: 10.1021/jm300230a BindingDB Entry DOI: 10.7270/Q25M66R0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Vitamin D3 receptor (Homo sapiens (Human)) | BDBM50015318 (CHEMBL3263871) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid PDB UniChem Similars | Article PubMed | n/a | n/a | 0.5 | n/a | n/a | n/a | n/a | n/a | n/a |
Rikkyo University Curated by ChEMBL | Assay Description Displacement of [3H]-1,25(OH)2D3 from GST-fused human VDR-LBD expressed in Escherichia coli BL21 | J Med Chem 57: 4073-87 (2014) Article DOI: 10.1021/jm401989c BindingDB Entry DOI: 10.7270/Q2ZS2Z2G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Vitamin D3 receptor (Homo sapiens (Human)) | BDBM50292705 ((25R)-25-Adamantyl-1alpha,25-dihydroxy-2-methylene...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL MMDB PC cid PC sid PDB UniChem Similars | Article PubMed | n/a | n/a | 3 | n/a | n/a | n/a | n/a | n/a | n/a |
Tokyo Medical and Dental University Curated by ChEMBL | Assay Description Antagonist activity at VDR expressed in COS7 cells assessed as inhibition of 1,25-Dihydroxyvitamin D3-induced response by transient transcription ass... | J Med Chem 51: 5320-9 (2008) Article DOI: 10.1021/jm8004477 BindingDB Entry DOI: 10.7270/Q28C9W2Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Vitamin D3 receptor (Homo sapiens (Human)) | BDBM50015315 (CHEMBL3263870) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 12 | n/a | n/a | n/a | n/a | n/a | n/a |
Rikkyo University Curated by ChEMBL | Assay Description Displacement of [3H]-1,25(OH)2D3 from GST-fused human VDR-LBD expressed in Escherichia coli BL21 | J Med Chem 57: 4073-87 (2014) Article DOI: 10.1021/jm401989c BindingDB Entry DOI: 10.7270/Q2ZS2Z2G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Vitamin D3 receptor (Homo sapiens (Human)) | BDBM50015316 (CHEMBL3263873) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid PDB UniChem Similars | Article PubMed | n/a | n/a | 12 | n/a | n/a | n/a | n/a | n/a | n/a |
Rikkyo University Curated by ChEMBL | Assay Description Displacement of [3H]-1,25(OH)2D3 from GST-fused human VDR-LBD expressed in Escherichia coli BL21 | J Med Chem 57: 4073-87 (2014) Article DOI: 10.1021/jm401989c BindingDB Entry DOI: 10.7270/Q2ZS2Z2G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Vitamin D3 receptor (Homo sapiens (Human)) | BDBM50015317 (CHEMBL3263872) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid PDB UniChem Similars | Article PubMed | n/a | n/a | 13 | n/a | n/a | n/a | n/a | n/a | n/a |
Rikkyo University Curated by ChEMBL | Assay Description Displacement of [3H]-1,25(OH)2D3 from GST-fused human VDR-LBD expressed in Escherichia coli BL21 | J Med Chem 57: 4073-87 (2014) Article DOI: 10.1021/jm401989c BindingDB Entry DOI: 10.7270/Q2ZS2Z2G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Vitamin D3 receptor (Homo sapiens (Human)) | BDBM50292704 ((1R,3R,7E,17beta)-17-{(1S,2E,5R)-5-hydroxy-1-methy...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL MMDB PC cid PC sid PDB UniChem Similars | Article PubMed | n/a | n/a | 30 | n/a | n/a | n/a | n/a | n/a | n/a |
Tokyo Medical and Dental University Curated by ChEMBL | Assay Description Antagonist activity at VDR expressed in COS7 cells assessed as inhibition of 1,25-Dihydroxyvitamin D3-induced response by transient transcription ass... | J Med Chem 51: 5320-9 (2008) Article DOI: 10.1021/jm8004477 BindingDB Entry DOI: 10.7270/Q28C9W2Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Vitamin D3 receptor (Homo sapiens (Human)) | BDBM50015315 (CHEMBL3263870) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 6.60 | n/a | n/a | n/a | n/a |
Rikkyo University Curated by ChEMBL | Assay Description Transactivation of human VDR expressed in HEK293 cells cotransfected with mouse VDRE, Tk-Sppx3-LUC reporter plasmid measured after 24 hrs by lucifera... | J Med Chem 57: 4073-87 (2014) Article DOI: 10.1021/jm401989c BindingDB Entry DOI: 10.7270/Q2ZS2Z2G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Vitamin D3 receptor (Homo sapiens (Human)) | BDBM50015316 (CHEMBL3263873) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid PDB UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.10 | n/a | n/a | n/a | n/a |
Rikkyo University Curated by ChEMBL | Assay Description Transactivation of human VDR expressed in HEK293 cells cotransfected with mouse VDRE, Tk-Sppx3-LUC reporter plasmid measured after 24 hrs by lucifera... | J Med Chem 57: 4073-87 (2014) Article DOI: 10.1021/jm401989c BindingDB Entry DOI: 10.7270/Q2ZS2Z2G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Vitamin D3 receptor (Homo sapiens (Human)) | BDBM50015317 (CHEMBL3263872) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid PDB UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.5 | n/a | n/a | n/a | n/a |
Rikkyo University Curated by ChEMBL | Assay Description Transactivation of human VDR expressed in HEK293 cells cotransfected with mouse VDRE, Tk-Sppx3-LUC reporter plasmid measured after 24 hrs by lucifera... | J Med Chem 57: 4073-87 (2014) Article DOI: 10.1021/jm401989c BindingDB Entry DOI: 10.7270/Q2ZS2Z2G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Vitamin D3 receptor (Homo sapiens (Human)) | BDBM50015318 (CHEMBL3263871) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid PDB UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 0.0700 | n/a | n/a | n/a | n/a |
Rikkyo University Curated by ChEMBL | Assay Description Transactivation of human VDR expressed in HEK293 cells cotransfected with mouse VDRE, Tk-Sppx3-LUC reporter plasmid measured after 24 hrs by lucifera... | J Med Chem 57: 4073-87 (2014) Article DOI: 10.1021/jm401989c BindingDB Entry DOI: 10.7270/Q2ZS2Z2G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Vitamin D3 receptor (Homo sapiens (Human)) | BDBM50015315 (CHEMBL3263870) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 4.40 | n/a | n/a | n/a | n/a |
Rikkyo University Curated by ChEMBL | Assay Description Activation of human VDR expressed in HEK293 cells cotransfected CMX-GAL4-RXRalpha and 4-tk-LUC assessed as heterodimerization with RXRalpha by mammal... | J Med Chem 57: 4073-87 (2014) Article DOI: 10.1021/jm401989c BindingDB Entry DOI: 10.7270/Q2ZS2Z2G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Vitamin D3 receptor (Homo sapiens (Human)) | BDBM50015318 (CHEMBL3263871) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid PDB UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 0.600 | n/a | n/a | n/a | n/a |
Rikkyo University Curated by ChEMBL | Assay Description Activation of human VDR expressed in HEK293 cells cotransfected CMX-GAL4-RXRalpha and 4-tk-LUC assessed as heterodimerization with RXRalpha by mammal... | J Med Chem 57: 4073-87 (2014) Article DOI: 10.1021/jm401989c BindingDB Entry DOI: 10.7270/Q2ZS2Z2G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Vitamin D3 receptor (Homo sapiens (Human)) | BDBM50015317 (CHEMBL3263872) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid PDB UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 2.30 | n/a | n/a | n/a | n/a |
Rikkyo University Curated by ChEMBL | Assay Description Activation of human VDR expressed in HEK293 cells cotransfected CMX-GAL4-RXRalpha and 4-tk-LUC assessed as heterodimerization with RXRalpha by mammal... | J Med Chem 57: 4073-87 (2014) Article DOI: 10.1021/jm401989c BindingDB Entry DOI: 10.7270/Q2ZS2Z2G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Vitamin D3 receptor (Homo sapiens (Human)) | BDBM50015316 (CHEMBL3263873) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid PDB UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 0.800 | n/a | n/a | n/a | n/a |
Rikkyo University Curated by ChEMBL | Assay Description Activation of human VDR expressed in HEK293 cells cotransfected CMX-GAL4-RXRalpha and 4-tk-LUC assessed as heterodimerization with RXRalpha by mammal... | J Med Chem 57: 4073-87 (2014) Article DOI: 10.1021/jm401989c BindingDB Entry DOI: 10.7270/Q2ZS2Z2G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Vitamin D3 receptor (Homo sapiens (Human)) | BDBM50015315 (CHEMBL3263870) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 15 | n/a | n/a | n/a | n/a |
Rikkyo University Curated by ChEMBL | Assay Description Activation of human VDR expressed in HEK293 cells cotransfected CMX-GAL4-SRC1 and 4-tk-LUC assessed as SRC1 interaction with AF2 surface of VDR by ma... | J Med Chem 57: 4073-87 (2014) Article DOI: 10.1021/jm401989c BindingDB Entry DOI: 10.7270/Q2ZS2Z2G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Vitamin D3 receptor (Homo sapiens (Human)) | BDBM50015318 (CHEMBL3263871) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid PDB UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.5 | n/a | n/a | n/a | n/a |
Rikkyo University Curated by ChEMBL | Assay Description Activation of human VDR expressed in HEK293 cells cotransfected CMX-GAL4-SRC1 and 4-tk-LUC assessed as SRC1 interaction with AF2 surface of VDR by ma... | J Med Chem 57: 4073-87 (2014) Article DOI: 10.1021/jm401989c BindingDB Entry DOI: 10.7270/Q2ZS2Z2G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Vitamin D3 receptor (Homo sapiens (Human)) | BDBM50015317 (CHEMBL3263872) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid PDB UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 6.5 | n/a | n/a | n/a | n/a |
Rikkyo University Curated by ChEMBL | Assay Description Activation of human VDR expressed in HEK293 cells cotransfected CMX-GAL4-SRC1 and 4-tk-LUC assessed as SRC1 interaction with AF2 surface of VDR by ma... | J Med Chem 57: 4073-87 (2014) Article DOI: 10.1021/jm401989c BindingDB Entry DOI: 10.7270/Q2ZS2Z2G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Vitamin D3 receptor (Homo sapiens (Human)) | BDBM50015316 (CHEMBL3263873) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid PDB UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 14 | n/a | n/a | n/a | n/a |
Rikkyo University Curated by ChEMBL | Assay Description Activation of human VDR expressed in HEK293 cells cotransfected CMX-GAL4-SRC1 and 4-tk-LUC assessed as SRC1 interaction with AF2 surface of VDR by ma... | J Med Chem 57: 4073-87 (2014) Article DOI: 10.1021/jm401989c BindingDB Entry DOI: 10.7270/Q2ZS2Z2G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Vitamin D3 receptor (Homo sapiens (Human)) | BDBM50015315 (CHEMBL3263870) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 4 | n/a | n/a | n/a | n/a |
Rikkyo University Curated by ChEMBL | Assay Description Activation of human VDR expressed in HEK293 cells cotransfected CMX-GAL4-N-CoR and 4-tk-LUC assessed as inhibition of N-CoR binding to VDR by mammali... | J Med Chem 57: 4073-87 (2014) Article DOI: 10.1021/jm401989c BindingDB Entry DOI: 10.7270/Q2ZS2Z2G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Vitamin D3 receptor (Homo sapiens (Human)) | BDBM50015318 (CHEMBL3263871) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid PDB UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 0.400 | n/a | n/a | n/a | n/a |
Rikkyo University Curated by ChEMBL | Assay Description Activation of human VDR expressed in HEK293 cells cotransfected CMX-GAL4-N-CoR and 4-tk-LUC assessed as inhibition of N-CoR binding to VDR by mammali... | J Med Chem 57: 4073-87 (2014) Article DOI: 10.1021/jm401989c BindingDB Entry DOI: 10.7270/Q2ZS2Z2G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Vitamin D3 receptor (Homo sapiens (Human)) | BDBM50015317 (CHEMBL3263872) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid PDB UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 3.70 | n/a | n/a | n/a | n/a |
Rikkyo University Curated by ChEMBL | Assay Description Activation of human VDR expressed in HEK293 cells cotransfected CMX-GAL4-N-CoR and 4-tk-LUC assessed as inhibition of N-CoR binding to VDR by mammali... | J Med Chem 57: 4073-87 (2014) Article DOI: 10.1021/jm401989c BindingDB Entry DOI: 10.7270/Q2ZS2Z2G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Vitamin D3 receptor (Homo sapiens (Human)) | BDBM50015316 (CHEMBL3263873) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid PDB UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.80 | n/a | n/a | n/a | n/a |
Rikkyo University Curated by ChEMBL | Assay Description Activation of human VDR expressed in HEK293 cells cotransfected CMX-GAL4-N-CoR and 4-tk-LUC assessed as inhibition of N-CoR binding to VDR by mammali... | J Med Chem 57: 4073-87 (2014) Article DOI: 10.1021/jm401989c BindingDB Entry DOI: 10.7270/Q2ZS2Z2G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Vitamin D3 receptor (Homo sapiens (Human)) | BDBM50015315 (CHEMBL3263870) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 4.10 | n/a | n/a | n/a | n/a |
Rikkyo University Curated by ChEMBL | Assay Description Activation of human VDR expressed in HEK293 cells cotransfected CMX-GAL4-NCoR2 and 4-tk-LUC assessed as inhibition of NCoR2 binding to VDR by mammali... | J Med Chem 57: 4073-87 (2014) Article DOI: 10.1021/jm401989c BindingDB Entry DOI: 10.7270/Q2ZS2Z2G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Vitamin D3 receptor (Homo sapiens (Human)) | BDBM50015318 (CHEMBL3263871) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid PDB UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 0.5 | n/a | n/a | n/a | n/a |
Rikkyo University Curated by ChEMBL | Assay Description Activation of human VDR expressed in HEK293 cells cotransfected CMX-GAL4-NCoR2 and 4-tk-LUC assessed as inhibition of NCoR2 binding to VDR by mammali... | J Med Chem 57: 4073-87 (2014) Article DOI: 10.1021/jm401989c BindingDB Entry DOI: 10.7270/Q2ZS2Z2G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Vitamin D3 receptor (Homo sapiens (Human)) | BDBM50015317 (CHEMBL3263872) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid PDB UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 2.40 | n/a | n/a | n/a | n/a |
Rikkyo University Curated by ChEMBL | Assay Description Activation of human VDR expressed in HEK293 cells cotransfected CMX-GAL4-NCoR2 and 4-tk-LUC assessed as inhibition of NCoR2 binding to VDR by mammali... | J Med Chem 57: 4073-87 (2014) Article DOI: 10.1021/jm401989c BindingDB Entry DOI: 10.7270/Q2ZS2Z2G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Vitamin D3 receptor (Homo sapiens (Human)) | BDBM50015316 (CHEMBL3263873) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid PDB UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 2.80 | n/a | n/a | n/a | n/a |
Rikkyo University Curated by ChEMBL | Assay Description Activation of human VDR expressed in HEK293 cells cotransfected CMX-GAL4-NCoR2 and 4-tk-LUC assessed as inhibition of NCoR2 binding to VDR by mammali... | J Med Chem 57: 4073-87 (2014) Article DOI: 10.1021/jm401989c BindingDB Entry DOI: 10.7270/Q2ZS2Z2G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Vitamin D3 receptor (Bos taurus) | BDBM50200182 ((1S,3R,5Z,7E)-9,10-secocholesta-5,7,10(19)-triene-...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG MMDB PC cid PC sid PDB UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 0.0500 | n/a | n/a | n/a | n/a |
Showa Pharmaceutical University Curated by ChEMBL | Assay Description Displacement of [3H]1,25-(OH)2D3 from bovine thymus vitamin D receptor | J Med Chem 52: 1438-49 (2010) Article DOI: 10.1021/jm8014348 BindingDB Entry DOI: 10.7270/Q2251J6N | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Vitamin D3 receptor (Bos taurus) | BDBM50293092 (22R-Butyl-1alpha,24-dihydroxy-24,25,26-trinorvitam...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 11 | n/a | n/a | n/a | n/a |
Showa Pharmaceutical University Curated by ChEMBL | Assay Description Displacement of [3H]1,25-(OH)2D3 from bovine thymus vitamin D receptor | J Med Chem 52: 1438-49 (2010) Article DOI: 10.1021/jm8014348 BindingDB Entry DOI: 10.7270/Q2251J6N | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Vitamin D3 receptor (Bos taurus) | BDBM50293093 ((1R,3S,5Z)-5-[(2E)-2-[(1R,3aS,7aR)-1-[(2R,3S)-3-(2...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid PDB UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.20 | n/a | n/a | n/a | n/a |
Showa Pharmaceutical University Curated by ChEMBL | Assay Description Displacement of [3H]1,25-(OH)2D3 from bovine thymus vitamin D receptor | J Med Chem 52: 1438-49 (2010) Article DOI: 10.1021/jm8014348 BindingDB Entry DOI: 10.7270/Q2251J6N | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Vitamin D3 receptor (Bos taurus) | BDBM50293094 ((1R,3S,5Z)-5-[(2E)-2-[(1R,3aS,7aR)-1-[(2S,3S)-3-(2...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid PDB UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 2 | n/a | n/a | n/a | n/a |
Showa Pharmaceutical University Curated by ChEMBL | Assay Description Displacement of [3H]1,25-(OH)2D3 from bovine thymus vitamin D receptor | J Med Chem 52: 1438-49 (2010) Article DOI: 10.1021/jm8014348 BindingDB Entry DOI: 10.7270/Q2251J6N | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Vitamin D3 receptor (Bos taurus) | BDBM50293095 (20S,22R-Butyl-1alpha,24-dihydroxy-24,25,26-trinorv...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 20 | n/a | n/a | n/a | n/a |
Showa Pharmaceutical University Curated by ChEMBL | Assay Description Displacement of [3H]1,25-(OH)2D3 from bovine thymus vitamin D receptor | J Med Chem 52: 1438-49 (2010) Article DOI: 10.1021/jm8014348 BindingDB Entry DOI: 10.7270/Q2251J6N | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Vitamin D3 receptor (Bos taurus) | BDBM50293096 ((1alpha,22R,24R)-22-Butyl-1,24-dihydroxyvitamin D3...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 16 | n/a | n/a | n/a | n/a |
Showa Pharmaceutical University Curated by ChEMBL | Assay Description Displacement of [3H]1,25-(OH)2D3 from bovine thymus vitamin D receptor | J Med Chem 52: 1438-49 (2010) Article DOI: 10.1021/jm8014348 BindingDB Entry DOI: 10.7270/Q2251J6N | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Vitamin D3 receptor (Bos taurus) | BDBM50293097 ((1alpha,22R,24S)-22-Butyl-1,24-dihydroxyvitamin D3...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 3.40 | n/a | n/a | n/a | n/a |
Showa Pharmaceutical University Curated by ChEMBL | Assay Description Displacement of [3H]1,25-(OH)2D3 from bovine thymus vitamin D receptor | J Med Chem 52: 1438-49 (2010) Article DOI: 10.1021/jm8014348 BindingDB Entry DOI: 10.7270/Q2251J6N | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Vitamin D3 receptor (Bos taurus) | BDBM50293098 ((1R,3S,5Z)-5-[(2E)-2-{(1R,3aS,7aR)-1-[(1R,2S,4R)-2...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid PDB UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 20 | n/a | n/a | n/a | n/a |
Showa Pharmaceutical University Curated by ChEMBL | Assay Description Displacement of [3H]1,25-(OH)2D3 from bovine thymus vitamin D receptor | J Med Chem 52: 1438-49 (2010) Article DOI: 10.1021/jm8014348 BindingDB Entry DOI: 10.7270/Q2251J6N | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Vitamin D3 receptor (Bos taurus) | BDBM50293099 ((1alpha,22S,24S)-22-Butyl-1,24-dihydroxyvitamin D3...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 3.80 | n/a | n/a | n/a | n/a |
Showa Pharmaceutical University Curated by ChEMBL | Assay Description Displacement of [3H]1,25-(OH)2D3 from bovine thymus vitamin D receptor | J Med Chem 52: 1438-49 (2010) Article DOI: 10.1021/jm8014348 BindingDB Entry DOI: 10.7270/Q2251J6N | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Vitamin D3 receptor (Homo sapiens (Human)) | BDBM50292704 ((1R,3R,7E,17beta)-17-{(1S,2E,5R)-5-hydroxy-1-methy...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL MMDB PC cid PC sid PDB UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 24 | n/a | n/a | n/a | n/a |
Tokyo Medical and Dental University Curated by ChEMBL | Assay Description Agonist activity at VDR assessed as receptor transactivation by transient transcription assay | J Med Chem 51: 5320-9 (2008) Article DOI: 10.1021/jm8004477 BindingDB Entry DOI: 10.7270/Q28C9W2Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Vitamin D3 receptor (Homo sapiens (Human)) | BDBM50292705 ((25R)-25-Adamantyl-1alpha,25-dihydroxy-2-methylene...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL MMDB PC cid PC sid PDB UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1 | n/a | n/a | n/a | n/a |
Tokyo Medical and Dental University Curated by ChEMBL | Assay Description Agonist activity at VDR assessed as receptor transactivation by transient transcription assay | J Med Chem 51: 5320-9 (2008) Article DOI: 10.1021/jm8004477 BindingDB Entry DOI: 10.7270/Q28C9W2Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Vitamin D3 receptor (Homo sapiens (Human)) | BDBM50292706 ((1R,3R,7E,17beta)-17-{(1R,2E,4R)-4-hydroxy-1-methy...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL MMDB PC cid PC sid PDB UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 0.0200 | n/a | n/a | n/a | n/a |
Tokyo Medical and Dental University Curated by ChEMBL | Assay Description Agonist activity at VDR assessed as receptor transactivation by transient transcription assay | J Med Chem 51: 5320-9 (2008) Article DOI: 10.1021/jm8004477 BindingDB Entry DOI: 10.7270/Q28C9W2Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Vitamin D3 receptor (Mus musculus) | BDBM50244164 ((20S)-1-alpha-25-Dihydroxy-2-alpha-(2-hydroxyethox...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid PDB UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 0.0270 | n/a | n/a | n/a | n/a |
Tokyo Medical and Dental University Curated by ChEMBL | Assay Description Increase in mouse VDR-mediated transcriptional activity in african green monkey COS7 cells after 24 hrs by luciferase assay | Bioorg Med Chem 16: 6949-64 (2008) Article DOI: 10.1016/j.bmc.2008.05.043 BindingDB Entry DOI: 10.7270/Q2Z60NWW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Vitamin D3 receptor (Mus musculus) | BDBM50244268 ((20S)-1-alpha-2-alpha-25-Trihydroxy-2beta-methyl-1...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 0.0170 | n/a | n/a | n/a | n/a |
Tokyo Medical and Dental University Curated by ChEMBL | Assay Description Increase in mouse VDR-mediated transcriptional activity in african green monkey COS7 cells after 24 hrs by luciferase assay | Bioorg Med Chem 16: 6949-64 (2008) Article DOI: 10.1016/j.bmc.2008.05.043 BindingDB Entry DOI: 10.7270/Q2Z60NWW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Vitamin D3 receptor (Mus musculus) | BDBM50244240 ((20S)-(2E)-1-alpha-25-Dihydroxy-2-[2-(hydroxy)-eth...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid PDB UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 0.0850 | n/a | n/a | n/a | n/a |
Tokyo Medical and Dental University Curated by ChEMBL | Assay Description Increase in mouse VDR-mediated transcriptional activity in african green monkey COS7 cells after 24 hrs by luciferase assay | Bioorg Med Chem 16: 6949-64 (2008) Article DOI: 10.1016/j.bmc.2008.05.043 BindingDB Entry DOI: 10.7270/Q2Z60NWW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Vitamin D3 receptor (Mus musculus) | BDBM50412385 (CHEMBL2021488) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 0.0900 | n/a | n/a | n/a | n/a |
Tokyo Medical and Dental University Curated by ChEMBL | Assay Description Increase in mouse VDR-mediated transcriptional activity in african green monkey COS7 cells after 24 hrs by luciferase assay | Bioorg Med Chem 16: 6949-64 (2008) Article DOI: 10.1016/j.bmc.2008.05.043 BindingDB Entry DOI: 10.7270/Q2Z60NWW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Vitamin D3 receptor (Mus musculus) | BDBM50244269 ((20R)-1-alpha-2-alpha-25-Trihydroxy-2-beta-methyl-...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 4.5 | n/a | n/a | n/a | n/a |
Tokyo Medical and Dental University Curated by ChEMBL | Assay Description Increase in mouse VDR-mediated transcriptional activity in african green monkey COS7 cells after 24 hrs by luciferase assay | Bioorg Med Chem 16: 6949-64 (2008) Article DOI: 10.1016/j.bmc.2008.05.043 BindingDB Entry DOI: 10.7270/Q2Z60NWW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Vitamin D3 receptor (Mus musculus) | BDBM50244268 ((20S)-1-alpha-2-alpha-25-Trihydroxy-2beta-methyl-1...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.90 | n/a | n/a | n/a | n/a |
Tokyo Medical and Dental University Curated by ChEMBL | Assay Description Increase in mouse VDR-mediated transcriptional activity in african green monkey COS7 cells after 24 hrs by luciferase assay | Bioorg Med Chem 16: 6949-64 (2008) Article DOI: 10.1016/j.bmc.2008.05.043 BindingDB Entry DOI: 10.7270/Q2Z60NWW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Vitamin D3 receptor (Mus musculus) | BDBM50244165 ((1R,2S,3R,5Z,7E)-17-{(1R)-1-[(2-ethyl-2-hydroxybut...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid PDB UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 0.115 | n/a | n/a | n/a | n/a |
Tokyo Medical and Dental University Curated by ChEMBL | Assay Description Increase in mouse VDR-mediated transcriptional activity in african green monkey COS7 cells after 24 hrs by luciferase assay | Bioorg Med Chem 16: 6949-64 (2008) Article DOI: 10.1016/j.bmc.2008.05.043 BindingDB Entry DOI: 10.7270/Q2Z60NWW | |||||||||||
More data for this Ligand-Target Pair |
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