BindingDB PrimarySearch

Found 43 hits with Last Name = 'wyman' and Initial = 'b'
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Sodium- and chloride-dependent glycine transporter 1 (Homo sapiens (Human))	BDBM50149871 ((R)-2-((3-(biphenyl-4-yloxy)-3-(4-fluorophenyl)pro...) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	Purchase CHEMBL MCE PC cid PC sid PDB UniChem Patents Similars	Article PubMed	n/a	n/a	26	n/a	n/a	n/a	n/a	n/a	n/a
H. Lundbeck A/S Curated by ChEMBL					Assay Description Inhibition of uptake of [3H]-glycine into cells transfected with human GlyT-1b transporter				Bioorg Med Chem Lett 14: 4027-30 (2004) Checked by Author Article DOI: 10.1016/j.bmcl.2004.05.043 BindingDB Entry DOI: 10.7270/Q2DV1JBF
H. Lundbeck A/S Curated by ChEMBL					More data for this Ligand-Target Pair
Tyrosine-protein kinase JAK3 (Homo sapiens (Human))	BDBM50132421 (3-[1-(1H-Pyrrol-2-yl)-meth-(Z)-ylidene]-5-(thiophe...) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	n/a	n/a	26	n/a	n/a	n/a	n/a	n/a	n/a
Aventis Pharmaceuticals Curated by ChEMBL					Assay Description Inhibitory activity against Janus Kinase 3 protein tyrosine kinase.				Bioorg Med Chem Lett 13: 3105-10 (2003) BindingDB Entry DOI: 10.7270/Q2833RDR
Aventis Pharmaceuticals Curated by ChEMBL					More data for this Ligand-Target Pair
Tyrosine-protein kinase JAK3 (Homo sapiens (Human))	BDBM50132420 (3-((1H-pyrrol-2-yl)methylene)-5-(pyridin-3-yl)indo...) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars	PubMed	n/a	n/a	27	n/a	n/a	n/a	n/a	n/a	n/a
Aventis Pharmaceuticals Curated by ChEMBL					Assay Description Inhibitory activity against Janus Kinase 3 protein tyrosine kinase.				Bioorg Med Chem Lett 13: 3105-10 (2003) BindingDB Entry DOI: 10.7270/Q2833RDR
Aventis Pharmaceuticals Curated by ChEMBL					More data for this Ligand-Target Pair
Tyrosine-protein kinase JAK3 (Homo sapiens (Human))	BDBM50132427 (5-Pyridin-3-yl-3-[1-(1H-pyrrol-2-yl)-meth-(Z)-ylid...) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem	PubMed	n/a	n/a	30	n/a	n/a	n/a	n/a	n/a	n/a
Aventis Pharmaceuticals Curated by ChEMBL					Assay Description Inhibitory activity against Janus Kinase 3 protein tyrosine kinase.				Bioorg Med Chem Lett 13: 3105-10 (2003) BindingDB Entry DOI: 10.7270/Q2833RDR
Aventis Pharmaceuticals Curated by ChEMBL					More data for this Ligand-Target Pair
Sodium- and chloride-dependent glycine transporter 1 (Homo sapiens (Human))	BDBM50149875 (CHEMBL361022 \| {(R)-4-[5-Chloro-2-(4-methoxy-pheny...) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	Purchase CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	150	n/a	n/a	n/a	n/a	n/a	n/a
H. Lundbeck A/S Curated by ChEMBL					Assay Description Inhibition of uptake of [3H]-glycine into cells transfected with human GlyT-1b transporter				Bioorg Med Chem Lett 14: 4027-30 (2004) Checked by Author Article DOI: 10.1016/j.bmcl.2004.05.043 BindingDB Entry DOI: 10.7270/Q2DV1JBF
H. Lundbeck A/S Curated by ChEMBL					More data for this Ligand-Target Pair
Sodium- and chloride-dependent glycine transporter 1 (Homo sapiens (Human))	BDBM50149873 (CHEMBL182162 \| {(2R,5S)-4-[2-(4-Methoxy-phenylsulf...) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	160	n/a	n/a	n/a	n/a	n/a	n/a
H. Lundbeck A/S Curated by ChEMBL					Assay Description Inhibition of uptake of [3H]-glycine into cells transfected with human GlyT-1b transporter				Bioorg Med Chem Lett 14: 4027-30 (2004) Checked by Author Article DOI: 10.1016/j.bmcl.2004.05.043 BindingDB Entry DOI: 10.7270/Q2DV1JBF
H. Lundbeck A/S Curated by ChEMBL					More data for this Ligand-Target Pair
Tyrosine-protein kinase JAK3 (Homo sapiens (Human))	BDBM50132422 (5-(Pyridine-3-carbonyl)-3-[1-(1H-pyrrol-2-yl)-meth...) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	n/a	n/a	168	n/a	n/a	n/a	n/a	n/a	n/a
Aventis Pharmaceuticals Curated by ChEMBL					Assay Description Inhibitory activity against Janus Kinase 3 protein tyrosine kinase.				Bioorg Med Chem Lett 13: 3105-10 (2003) BindingDB Entry DOI: 10.7270/Q2833RDR
Aventis Pharmaceuticals Curated by ChEMBL					More data for this Ligand-Target Pair
Tyrosine-protein kinase JAK3 (Homo sapiens (Human))	BDBM50132428 (5-(Hydroxy-thiophen-2-yl-methyl)-3-[1-(1H-pyrrol-2...) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	n/a	n/a	190	n/a	n/a	n/a	n/a	n/a	n/a
Aventis Pharmaceuticals Curated by ChEMBL					Assay Description Inhibitory activity against Janus Kinase 3 protein tyrosine kinase.				Bioorg Med Chem Lett 13: 3105-10 (2003) BindingDB Entry DOI: 10.7270/Q2833RDR
Aventis Pharmaceuticals Curated by ChEMBL					More data for this Ligand-Target Pair
Tyrosine-protein kinase JAK3 (Homo sapiens (Human))	BDBM50132417 (3-[1-(4-Dimethylamino-phenyl)-meth-(Z)-ylidene]-5-...) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	n/a	n/a	200	n/a	n/a	n/a	n/a	n/a	n/a
Aventis Pharmaceuticals Curated by ChEMBL					Assay Description Inhibitory activity against Janus Kinase 3 protein tyrosine kinase.				Bioorg Med Chem Lett 13: 3105-10 (2003) BindingDB Entry DOI: 10.7270/Q2833RDR
Aventis Pharmaceuticals Curated by ChEMBL					More data for this Ligand-Target Pair
Tyrosine-protein kinase JAK3 (Homo sapiens (Human))	BDBM50132423 (2-Oxo-3-[1-(1H-pyrrol-2-yl)-meth-(Z)-ylidene]-2,3-...) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	n/a	n/a	210	n/a	n/a	n/a	n/a	n/a	n/a
Aventis Pharmaceuticals Curated by ChEMBL					Assay Description Inhibitory activity against Janus Kinase 3 protein tyrosine kinase.				Bioorg Med Chem Lett 13: 3105-10 (2003) BindingDB Entry DOI: 10.7270/Q2833RDR
Aventis Pharmaceuticals Curated by ChEMBL					More data for this Ligand-Target Pair
Tyrosine-protein kinase JAK3 (Homo sapiens (Human))	BDBM17032 ((3Z)-2-oxo-3-(1H-pyrrol-2-ylmethylidene)-2,3-dihyd...) Show SMILES OC(=O)c1ccc2NC(=O)\C(=C/c3ccc[nH]3)c2c1 Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	n/a	n/a	213	n/a	n/a	n/a	n/a	n/a	n/a
Aventis Pharmaceuticals Curated by ChEMBL					Assay Description Inhibitory activity against Janus Kinase 3 protein tyrosine kinase.				Bioorg Med Chem Lett 13: 3105-10 (2003) BindingDB Entry DOI: 10.7270/Q2833RDR
Aventis Pharmaceuticals Curated by ChEMBL					More data for this Ligand-Target Pair
Tyrosine-protein kinase JAK3 (Homo sapiens (Human))	BDBM50132419 (5-Pyridin-3-yl-3-[1-(1H-pyrrol-2-yl)-meth-(Z)-ylid...) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem	PubMed	n/a	n/a	235	n/a	n/a	n/a	n/a	n/a	n/a
Aventis Pharmaceuticals Curated by ChEMBL					Assay Description Inhibitory activity against Janus Kinase 3 protein tyrosine kinase.				Bioorg Med Chem Lett 13: 3105-10 (2003) BindingDB Entry DOI: 10.7270/Q2833RDR
Aventis Pharmaceuticals Curated by ChEMBL					More data for this Ligand-Target Pair
Tyrosine-protein kinase JAK3 (Homo sapiens (Human))	BDBM50132424 (3-[2-Oxo-2-(1H-pyrrol-2-yl)-eth-(Z)-ylidene]-5-(th...) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem	PubMed	n/a	n/a	260	n/a	n/a	n/a	n/a	n/a	n/a
Aventis Pharmaceuticals Curated by ChEMBL					Assay Description Inhibitory activity against Janus Kinase 3 protein tyrosine kinase.				Bioorg Med Chem Lett 13: 3105-10 (2003) BindingDB Entry DOI: 10.7270/Q2833RDR
Aventis Pharmaceuticals Curated by ChEMBL					More data for this Ligand-Target Pair
Sodium- and chloride-dependent glycine transporter 1 (Homo sapiens (Human))	BDBM50149865 (CHEMBL181805 \| {4-[5-Chloro-2-(4-methoxy-phenylsul...) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	290	n/a	n/a	n/a	n/a	n/a	n/a
H. Lundbeck A/S Curated by ChEMBL					Assay Description Inhibition of uptake of [3H]-glycine into cells transfected with human GlyT-1b transporter				Bioorg Med Chem Lett 14: 4027-30 (2004) Checked by Author Article DOI: 10.1016/j.bmcl.2004.05.043 BindingDB Entry DOI: 10.7270/Q2DV1JBF
H. Lundbeck A/S Curated by ChEMBL					More data for this Ligand-Target Pair
Sodium- and chloride-dependent glycine transporter 1 (Homo sapiens (Human))	BDBM50149856 (CHEMBL360052 \| {Methyl-[(R)-3-phenyl-3-(4-trifluor...) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	Purchase CHEMBL MCE PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	320	n/a	n/a	n/a	n/a	n/a	n/a
H. Lundbeck A/S Curated by ChEMBL					Assay Description Inhibition of uptake of [3H]-glycine into cells transfected with human GlyT-1b transporter				Bioorg Med Chem Lett 14: 4027-30 (2004) Checked by Author Article DOI: 10.1016/j.bmcl.2004.05.043 BindingDB Entry DOI: 10.7270/Q2DV1JBF
H. Lundbeck A/S Curated by ChEMBL					More data for this Ligand-Target Pair
Tyrosine-protein kinase JAK3 (Homo sapiens (Human))	BDBM50132418 (5-Pyridin-3-yl-3-[1-(1H-pyrrol-2-yl)-meth-(Z)-ylid...) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem	PubMed	n/a	n/a	350	n/a	n/a	n/a	n/a	n/a	n/a
Aventis Pharmaceuticals Curated by ChEMBL					Assay Description Inhibitory activity against Janus Kinase 3 protein tyrosine kinase.				Bioorg Med Chem Lett 13: 3105-10 (2003) BindingDB Entry DOI: 10.7270/Q2833RDR
Aventis Pharmaceuticals Curated by ChEMBL					More data for this Ligand-Target Pair
Sodium- and chloride-dependent glycine transporter 1 (Homo sapiens (Human))	BDBM50149866 (CHEMBL181643 \| {4-[2-(4-Chloro-phenylsulfanyl)-phe...) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	360	n/a	n/a	n/a	n/a	n/a	n/a
H. Lundbeck A/S Curated by ChEMBL					Assay Description Inhibition of uptake of [3H]-glycine into cells transfected with human GlyT-1b transporter				Bioorg Med Chem Lett 14: 4027-30 (2004) Checked by Author Article DOI: 10.1016/j.bmcl.2004.05.043 BindingDB Entry DOI: 10.7270/Q2DV1JBF
H. Lundbeck A/S Curated by ChEMBL					More data for this Ligand-Target Pair
Sodium- and chloride-dependent glycine transporter 1 (Homo sapiens (Human))	BDBM50149862 (CHEMBL182521 \| [2,5-Dimethyl-4-(2-p-tolylsulfanyl-...) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	550	n/a	n/a	n/a	n/a	n/a	n/a
H. Lundbeck A/S Curated by ChEMBL					Assay Description Inhibition of uptake of [3H]-glycine into cells transfected with human GlyT-1b transporter				Bioorg Med Chem Lett 14: 4027-30 (2004) Checked by Author Article DOI: 10.1016/j.bmcl.2004.05.043 BindingDB Entry DOI: 10.7270/Q2DV1JBF
H. Lundbeck A/S Curated by ChEMBL					More data for this Ligand-Target Pair
Sodium- and chloride-dependent glycine transporter 1 (Homo sapiens (Human))	BDBM50149859 (CHEMBL182666 \| {4-[2-(4-Methoxy-phenylsulfanyl)-ph...) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	580	n/a	n/a	n/a	n/a	n/a	n/a
H. Lundbeck A/S Curated by ChEMBL					Assay Description Inhibition of uptake of [3H]-glycine into cells transfected with human GlyT-1b transporter				Bioorg Med Chem Lett 14: 4027-30 (2004) Checked by Author Article DOI: 10.1016/j.bmcl.2004.05.043 BindingDB Entry DOI: 10.7270/Q2DV1JBF
H. Lundbeck A/S Curated by ChEMBL					More data for this Ligand-Target Pair
Tyrosine-protein kinase JAK3 (Homo sapiens (Human))	BDBM50132426 (CHEMBL104062 \| N-{4-[2-Oxo-5-(thiophene-2-carbonyl...) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	n/a	n/a	700	n/a	n/a	n/a	n/a	n/a	n/a
Aventis Pharmaceuticals Curated by ChEMBL					Assay Description Inhibitory activity against Janus Kinase 3 protein tyrosine kinase.				Bioorg Med Chem Lett 13: 3105-10 (2003) BindingDB Entry DOI: 10.7270/Q2833RDR
Aventis Pharmaceuticals Curated by ChEMBL					More data for this Ligand-Target Pair
Tyrosine-protein kinase JAK3 (Homo sapiens (Human))	BDBM50065287 (5-Nitro-3-(1H-pyrrol-2-ylmethylene)-1,3-dihydro-in...) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	n/a	n/a	710	n/a	n/a	n/a	n/a	n/a	n/a
Aventis Pharmaceuticals Curated by ChEMBL					Assay Description Inhibitory activity against Janus Kinase 3 protein tyrosine kinase.				Bioorg Med Chem Lett 13: 3105-10 (2003) BindingDB Entry DOI: 10.7270/Q2833RDR
Aventis Pharmaceuticals Curated by ChEMBL					More data for this Ligand-Target Pair
Tyrosine-protein kinase JAK3 (Homo sapiens (Human))	BDBM50132429 (CHEMBL104409 \| N-{2-Oxo-3-[1-(1H-pyrrol-2-yl)-meth...) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	n/a	n/a	870	n/a	n/a	n/a	n/a	n/a	n/a
Aventis Pharmaceuticals Curated by ChEMBL					Assay Description Inhibitory activity against Janus Kinase 3 protein tyrosine kinase.				Bioorg Med Chem Lett 13: 3105-10 (2003) BindingDB Entry DOI: 10.7270/Q2833RDR
Aventis Pharmaceuticals Curated by ChEMBL					More data for this Ligand-Target Pair
Tyrosine-protein kinase JAK3 (Homo sapiens (Human))	BDBM17015 ((3Z)-3-(1H-pyrrol-2-ylmethylidene)-2,3-dihydro-1H-...) Show SMILES O=C1Nc2ccccc2\C1=C\c1ccc[nH]1 Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase CHEMBL PC cid PC sid UniChem Patents Similars	PubMed	n/a	n/a	900	n/a	n/a	n/a	n/a	n/a	n/a
Aventis Pharmaceuticals Curated by ChEMBL					Assay Description Inhibitory activity against Janus Kinase 3 protein tyrosine kinase.				Bioorg Med Chem Lett 13: 3105-10 (2003) BindingDB Entry DOI: 10.7270/Q2833RDR
Aventis Pharmaceuticals Curated by ChEMBL					More data for this Ligand-Target Pair
Sodium- and chloride-dependent glycine transporter 1 (Homo sapiens (Human))	BDBM50149872 (CHEMBL182015 \| {4-[2-(Biphenyl-4-ylsulfanyl)-pheny...) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	>1.00E+3	n/a	n/a	n/a	n/a	n/a	n/a
H. Lundbeck A/S Curated by ChEMBL					Assay Description Inhibition of uptake of [3H]-glycine into cells transfected with human GlyT-1b transporter				Bioorg Med Chem Lett 14: 4027-30 (2004) Checked by Author Article DOI: 10.1016/j.bmcl.2004.05.043 BindingDB Entry DOI: 10.7270/Q2DV1JBF
H. Lundbeck A/S Curated by ChEMBL					More data for this Ligand-Target Pair
Sodium- and chloride-dependent glycine transporter 1 (Homo sapiens (Human))	BDBM50149868 (CHEMBL183030 \| {(S)-4-[5-Chloro-2-(4-methoxy-pheny...) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	1.40E+3	n/a	n/a	n/a	n/a	n/a	n/a
H. Lundbeck A/S Curated by ChEMBL					Assay Description Inhibition of uptake of [3H]-glycine into cells transfected with human GlyT-1b transporter				Bioorg Med Chem Lett 14: 4027-30 (2004) Checked by Author Article DOI: 10.1016/j.bmcl.2004.05.043 BindingDB Entry DOI: 10.7270/Q2DV1JBF
H. Lundbeck A/S Curated by ChEMBL					More data for this Ligand-Target Pair
Sodium- and chloride-dependent glycine transporter 1 (Homo sapiens (Human))	BDBM50149853 (CHEMBL181596 \| {4-[2-(4-Methoxy-phenylsulfanyl)-ph...) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	1.50E+3	n/a	n/a	n/a	n/a	n/a	n/a
H. Lundbeck A/S Curated by ChEMBL					Assay Description Inhibition of uptake of [3H]-glycine into cells transfected with human GlyT-1b transporter				Bioorg Med Chem Lett 14: 4027-30 (2004) Checked by Author Article DOI: 10.1016/j.bmcl.2004.05.043 BindingDB Entry DOI: 10.7270/Q2DV1JBF
H. Lundbeck A/S Curated by ChEMBL					More data for this Ligand-Target Pair
Sodium- and chloride-dependent glycine transporter 1 (Homo sapiens (Human))	BDBM50149860 (CHEMBL360501 \| {4-[2-(4-Methoxy-phenylsulfanyl)-5-...) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	1.60E+3	n/a	n/a	n/a	n/a	n/a	n/a
H. Lundbeck A/S Curated by ChEMBL					Assay Description Inhibition of uptake of [3H]-glycine into cells transfected with human GlyT-1b transporter				Bioorg Med Chem Lett 14: 4027-30 (2004) Checked by Author Article DOI: 10.1016/j.bmcl.2004.05.043 BindingDB Entry DOI: 10.7270/Q2DV1JBF
H. Lundbeck A/S Curated by ChEMBL					More data for this Ligand-Target Pair
Sodium- and chloride-dependent glycine transporter 1 (Homo sapiens (Human))	BDBM50149877 (CHEMBL365268 \| {4-[2-(4-Methoxy-phenylsulfanyl)-ph...) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	1.70E+3	n/a	n/a	n/a	n/a	n/a	n/a
H. Lundbeck A/S Curated by ChEMBL					Assay Description Inhibition of uptake of [3H]-glycine into cells transfected with human GlyT-1b transporter				Bioorg Med Chem Lett 14: 4027-30 (2004) Checked by Author Article DOI: 10.1016/j.bmcl.2004.05.043 BindingDB Entry DOI: 10.7270/Q2DV1JBF
H. Lundbeck A/S Curated by ChEMBL					More data for this Ligand-Target Pair
Sodium- and chloride-dependent glycine transporter 1 (Homo sapiens (Human))	BDBM50149876 (CHEMBL184785 \| {4-[5-Chloro-2-(4-methoxy-phenylsul...) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	1.70E+3	n/a	n/a	n/a	n/a	n/a	n/a
H. Lundbeck A/S Curated by ChEMBL					Assay Description Inhibition of uptake of [3H]-glycine into cells transfected with human GlyT-1b transporter				Bioorg Med Chem Lett 14: 4027-30 (2004) Checked by Author Article DOI: 10.1016/j.bmcl.2004.05.043 BindingDB Entry DOI: 10.7270/Q2DV1JBF
H. Lundbeck A/S Curated by ChEMBL					More data for this Ligand-Target Pair
Sodium- and chloride-dependent glycine transporter 1 (Homo sapiens (Human))	BDBM50149861 (CHEMBL182949 \| {4-[2-(4-Fluoro-phenylsulfanyl)-phe...) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	1.90E+3	n/a	n/a	n/a	n/a	n/a	n/a
H. Lundbeck A/S Curated by ChEMBL					Assay Description Inhibition of uptake of [3H]-glycine into cells transfected with human GlyT-1b transporter				Bioorg Med Chem Lett 14: 4027-30 (2004) Checked by Author Article DOI: 10.1016/j.bmcl.2004.05.043 BindingDB Entry DOI: 10.7270/Q2DV1JBF
H. Lundbeck A/S Curated by ChEMBL					More data for this Ligand-Target Pair
Tyrosine-protein kinase JAK3 (Homo sapiens (Human))	BDBM50132431 (3-[1-Phenyl-meth-(Z)-ylidene]-5-(thiophene-2-carbo...) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	n/a	n/a	2.30E+3	n/a	n/a	n/a	n/a	n/a	n/a
Aventis Pharmaceuticals Curated by ChEMBL					Assay Description Inhibitory activity against Janus Kinase 3 protein tyrosine kinase.				Bioorg Med Chem Lett 13: 3105-10 (2003) BindingDB Entry DOI: 10.7270/Q2833RDR
Aventis Pharmaceuticals Curated by ChEMBL					More data for this Ligand-Target Pair
Sodium- and chloride-dependent glycine transporter 1 (Homo sapiens (Human))	BDBM50149874 (CHEMBL363928 \| [2,5-Dimethyl-4-(2-phenylsulfanyl-p...) Show SMILES CC1CN(C(C)CN1CC(O)=O)c1ccccc1Sc1ccccc1 Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	2.90E+3	n/a	n/a	n/a	n/a	n/a	n/a
H. Lundbeck A/S Curated by ChEMBL					Assay Description Inhibition of uptake of [3H]-glycine into cells transfected with human GlyT-1b transporter				Bioorg Med Chem Lett 14: 4027-30 (2004) Checked by Author Article DOI: 10.1016/j.bmcl.2004.05.043 BindingDB Entry DOI: 10.7270/Q2DV1JBF
H. Lundbeck A/S Curated by ChEMBL					More data for this Ligand-Target Pair
Sodium- and chloride-dependent glycine transporter 1 (Homo sapiens (Human))	BDBM50149864 (CHEMBL181698 \| {4-[2-(4-Hydroxy-phenylsulfanyl)-ph...) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	3.60E+3	n/a	n/a	n/a	n/a	n/a	n/a
H. Lundbeck A/S Curated by ChEMBL					Assay Description Inhibition of uptake of [3H]-glycine into cells transfected with human GlyT-1b transporter				Bioorg Med Chem Lett 14: 4027-30 (2004) Checked by Author Article DOI: 10.1016/j.bmcl.2004.05.043 BindingDB Entry DOI: 10.7270/Q2DV1JBF
H. Lundbeck A/S Curated by ChEMBL					More data for this Ligand-Target Pair
Sodium- and chloride-dependent glycine transporter 1 (Homo sapiens (Human))	BDBM50149863 (CHEMBL183508 \| {4-[5-Methoxy-2-(4-methoxy-phenylsu...) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	4.60E+3	n/a	n/a	n/a	n/a	n/a	n/a
H. Lundbeck A/S Curated by ChEMBL					Assay Description Inhibition of uptake of [3H]-glycine into cells transfected with human GlyT-1b transporter				Bioorg Med Chem Lett 14: 4027-30 (2004) Checked by Author Article DOI: 10.1016/j.bmcl.2004.05.043 BindingDB Entry DOI: 10.7270/Q2DV1JBF
H. Lundbeck A/S Curated by ChEMBL					More data for this Ligand-Target Pair
Tyrosine-protein kinase JAK3 (Homo sapiens (Human))	BDBM50132425 (3-[1-(4-Fluoro-phenyl)-meth-(Z)-ylidene]-5-(thioph...) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	n/a	n/a	4.90E+3	n/a	n/a	n/a	n/a	n/a	n/a
Aventis Pharmaceuticals Curated by ChEMBL					Assay Description Inhibitory activity against Janus Kinase 3 protein tyrosine kinase.				Bioorg Med Chem Lett 13: 3105-10 (2003) BindingDB Entry DOI: 10.7270/Q2833RDR
Aventis Pharmaceuticals Curated by ChEMBL					More data for this Ligand-Target Pair
Tyrosine-protein kinase JAK3 (Homo sapiens (Human))	BDBM50132430 (3-[1-(4-Methanesulfonyl-phenyl)-meth-(Z)-ylidene]-...) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	n/a	n/a	7.10E+3	n/a	n/a	n/a	n/a	n/a	n/a
Aventis Pharmaceuticals Curated by ChEMBL					Assay Description Inhibitory activity against Janus Kinase 3 protein tyrosine kinase.				Bioorg Med Chem Lett 13: 3105-10 (2003) BindingDB Entry DOI: 10.7270/Q2833RDR
Aventis Pharmaceuticals Curated by ChEMBL					More data for this Ligand-Target Pair
Sodium- and chloride-dependent glycine transporter 1 (Homo sapiens (Human))	BDBM50149854 (CHEMBL180202 \| {4-[2-(4-Methoxy-phenylsulfanyl)-ph...) Show SMILES COc1ccc(Sc2ccccc2N2CCN(CC(O)=O)CC2C)cc1 Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
H. Lundbeck A/S Curated by ChEMBL					Assay Description Inhibition of uptake of [3H]-glycine into cells transfected with human GlyT-1b transporter				Bioorg Med Chem Lett 14: 4027-30 (2004) Checked by Author Article DOI: 10.1016/j.bmcl.2004.05.043 BindingDB Entry DOI: 10.7270/Q2DV1JBF
H. Lundbeck A/S Curated by ChEMBL					More data for this Ligand-Target Pair
Sodium- and chloride-dependent glycine transporter 1 (Homo sapiens (Human))	BDBM50149858 (CHEMBL184996 \| {4-[2-(4-Methoxy-phenylsulfanyl)-ph...) Show SMILES COc1ccc(Sc2ccccc2N2CCN(CC(O)=O)CC2)cc1 Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
H. Lundbeck A/S Curated by ChEMBL					Assay Description Inhibition of uptake of [3H]-glycine into cells transfected with human GlyT-1b transporter				Bioorg Med Chem Lett 14: 4027-30 (2004) Checked by Author Article DOI: 10.1016/j.bmcl.2004.05.043 BindingDB Entry DOI: 10.7270/Q2DV1JBF
H. Lundbeck A/S Curated by ChEMBL					More data for this Ligand-Target Pair
Sodium- and chloride-dependent glycine transporter 1 (Homo sapiens (Human))	BDBM50149870 (CHEMBL360768 \| {(2R,5R)-4-[2-(4-Methoxy-phenylsulf...) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	1.60E+4	n/a	n/a	n/a	n/a	n/a	n/a
H. Lundbeck A/S Curated by ChEMBL					Assay Description Inhibition of uptake of [3H]-glycine into cells transfected with human GlyT-1b transporter				Bioorg Med Chem Lett 14: 4027-30 (2004) Checked by Author Article DOI: 10.1016/j.bmcl.2004.05.043 BindingDB Entry DOI: 10.7270/Q2DV1JBF
H. Lundbeck A/S Curated by ChEMBL					More data for this Ligand-Target Pair
Sodium- and chloride-dependent glycine transporter 1 (Homo sapiens (Human))	BDBM50149869 (CHEMBL182917 \| {(2S,5S)-4-[2-(4-Methoxy-phenylsulf...) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	1.80E+4	n/a	n/a	n/a	n/a	n/a	n/a
H. Lundbeck A/S Curated by ChEMBL					Assay Description Inhibition of uptake of [3H]-glycine into cells transfected with human GlyT-1b transporter				Bioorg Med Chem Lett 14: 4027-30 (2004) Checked by Author Article DOI: 10.1016/j.bmcl.2004.05.043 BindingDB Entry DOI: 10.7270/Q2DV1JBF
H. Lundbeck A/S Curated by ChEMBL					More data for this Ligand-Target Pair
Sodium- and chloride-dependent glycine transporter 1 (Homo sapiens (Human))	BDBM50149857 (CHEMBL181745 \| {4-[2-(4-Acetylamino-phenylsulfanyl...) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	2.20E+4	n/a	n/a	n/a	n/a	n/a	n/a
H. Lundbeck A/S Curated by ChEMBL					Assay Description Inhibition of uptake of [3H]-glycine into cells transfected with human GlyT-1b transporter				Bioorg Med Chem Lett 14: 4027-30 (2004) Checked by Author Article DOI: 10.1016/j.bmcl.2004.05.043 BindingDB Entry DOI: 10.7270/Q2DV1JBF
H. Lundbeck A/S Curated by ChEMBL					More data for this Ligand-Target Pair
Sodium- and chloride-dependent glycine transporter 1 (Homo sapiens (Human))	BDBM50149867 (CHEMBL182618 \| {4-[5-Methoxy-2-(4-methoxy-phenylsu...) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	>5.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
H. Lundbeck A/S Curated by ChEMBL					Assay Description Inhibition of uptake of [3H]-glycine into cells transfected with human GlyT-1b transporter				Bioorg Med Chem Lett 14: 4027-30 (2004) Checked by Author Article DOI: 10.1016/j.bmcl.2004.05.043 BindingDB Entry DOI: 10.7270/Q2DV1JBF
H. Lundbeck A/S Curated by ChEMBL					More data for this Ligand-Target Pair
Sodium- and chloride-dependent glycine transporter 1 (Homo sapiens (Human))	BDBM50149855 (CHEMBL182916 \| {(2S,5R)-4-[2-(4-Methoxy-phenylsulf...) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	5.30E+4	n/a	n/a	n/a	n/a	n/a	n/a
H. Lundbeck A/S Curated by ChEMBL					Assay Description Inhibition of uptake of [3H]-glycine into cells transfected with human GlyT-1b transporter				Bioorg Med Chem Lett 14: 4027-30 (2004) Checked by Author Article DOI: 10.1016/j.bmcl.2004.05.043 BindingDB Entry DOI: 10.7270/Q2DV1JBF
H. Lundbeck A/S Curated by ChEMBL					More data for this Ligand-Target Pair