Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Histone acetyltransferase KAT2B (Homo sapiens (Human)) | BDBM50234932 (CHEMBL4103402 | US10239861, Example 20) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents | US Patent | n/a | n/a | 12.7 | n/a | n/a | n/a | n/a | n/a | n/a |
GLSynthesis Inc. | Assay Description His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o... | J Med Chem 48: 3919-29 (2005) BindingDB Entry DOI: 10.7270/Q2X06991 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histone acetyltransferase KAT2B (Homo sapiens (Human)) | BDBM371542 (4-chloro-5-(((3R,5S)-1,5-dimethylpiperidin-3-yl)am...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 21.5 | n/a | n/a | n/a | n/a | n/a | n/a |
GLSynthesis Inc. | Assay Description His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o... | J Med Chem 48: 3919-29 (2005) BindingDB Entry DOI: 10.7270/Q2X06991 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histone acetyltransferase KAT2B (Homo sapiens (Human)) | BDBM371577 ((S)-4-chloro-2-methyl-5-((1-methylazepan-3-yl)amin...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 32.9 | n/a | n/a | n/a | n/a | n/a | n/a |
GLSynthesis Inc. | Assay Description His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o... | J Med Chem 48: 3919-29 (2005) BindingDB Entry DOI: 10.7270/Q2X06991 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histone acetyltransferase KAT2B (Homo sapiens (Human)) | BDBM371546 (US10239861, Example 26) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 34.8 | n/a | n/a | n/a | n/a | n/a | n/a |
GLSynthesis Inc. | Assay Description His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o... | J Med Chem 48: 3919-29 (2005) BindingDB Entry DOI: 10.7270/Q2X06991 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histone acetyltransferase KAT2B (Homo sapiens (Human)) | BDBM371541 ((racemic)-4-chloro-5-(((3RS,5SR)-1,5-dimethylpiper...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 36.5 | n/a | n/a | n/a | n/a | n/a | n/a |
GLSynthesis Inc. | Assay Description His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o... | J Med Chem 48: 3919-29 (2005) BindingDB Entry DOI: 10.7270/Q2X06991 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histone acetyltransferase KAT2B (Homo sapiens (Human)) | BDBM371549 (US10239861, Example 29) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 48.5 | n/a | n/a | n/a | n/a | n/a | n/a |
GLSynthesis Inc. | Assay Description His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o... | J Med Chem 48: 3919-29 (2005) BindingDB Entry DOI: 10.7270/Q2X06991 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histone acetyltransferase KAT2B (Homo sapiens (Human)) | BDBM50234932 (CHEMBL4103402 | US10239861, Example 20) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents | US Patent | n/a | n/a | 49.6 | n/a | n/a | n/a | n/a | n/a | n/a |
GLSynthesis Inc. | Assay Description His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o... | J Med Chem 48: 3919-29 (2005) BindingDB Entry DOI: 10.7270/Q2X06991 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histone acetyltransferase KAT2B (Homo sapiens (Human)) | BDBM371533 (4-bromo-2-methyl-5-((1-methylazepan-3-yl)amino)pyr...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 51 | n/a | n/a | n/a | n/a | n/a | n/a |
GLSynthesis Inc. | Assay Description His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o... | J Med Chem 48: 3919-29 (2005) BindingDB Entry DOI: 10.7270/Q2X06991 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histone acetyltransferase KAT2B (Homo sapiens (Human)) | BDBM50234945 (CHEMBL4061142 | US10239861, Example 59) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 51.2 | n/a | n/a | n/a | n/a | n/a | n/a |
GLSynthesis Inc. | Assay Description His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o... | J Med Chem 48: 3919-29 (2005) BindingDB Entry DOI: 10.7270/Q2X06991 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histone acetyltransferase KAT2B (Homo sapiens (Human)) | BDBM371545 (4-chloro-5-((1,6-dimethylpiperidin-3-yl)amino)-2-m...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 60 | n/a | n/a | n/a | n/a | n/a | n/a |
GLSynthesis Inc. | Assay Description His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o... | J Med Chem 48: 3919-29 (2005) BindingDB Entry DOI: 10.7270/Q2X06991 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histone acetyltransferase KAT2B (Homo sapiens (Human)) | BDBM371521 (4-chloro-2-methyl-5-((1-methylazepan-3-yl)amino)py...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 62 | n/a | n/a | n/a | n/a | n/a | n/a |
GLSynthesis Inc. | Assay Description His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o... | J Med Chem 48: 3919-29 (2005) BindingDB Entry DOI: 10.7270/Q2X06991 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histone acetyltransferase KAT2B (Homo sapiens (Human)) | BDBM50234943 (CHEMBL4099456 | US10239861, Example 3) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid PDB UniChem Patents Similars | PDB US Patent | n/a | n/a | 85 | n/a | n/a | n/a | n/a | n/a | n/a |
GLSynthesis Inc. | Assay Description His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o... | J Med Chem 48: 3919-29 (2005) BindingDB Entry DOI: 10.7270/Q2X06991 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Histone acetyltransferase KAT2B (Homo sapiens (Human)) | BDBM371527 ((R)-5-((1-benzylpiperidin-3-yl)amino)-4-chloro-2-m...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | Purchase PC cid PC sid UniChem | US Patent | n/a | n/a | 85.6 | n/a | n/a | n/a | n/a | n/a | n/a |
GLSynthesis Inc. | Assay Description His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o... | J Med Chem 48: 3919-29 (2005) BindingDB Entry DOI: 10.7270/Q2X06991 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histone acetyltransferase KAT2B (Homo sapiens (Human)) | BDBM371564 (4-chloro-5-[[1-[[3-(difluoromethoxy)phenyl]methyl]...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 94.9 | n/a | n/a | n/a | n/a | n/a | n/a |
GLSynthesis Inc. | Assay Description His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o... | J Med Chem 48: 3919-29 (2005) BindingDB Entry DOI: 10.7270/Q2X06991 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histone acetyltransferase KAT2B (Homo sapiens (Human)) | BDBM371559 ((R)-4-chloro-2-methyl-5-((2,3,4,5-tetrahydro-1H-be...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 102 | n/a | n/a | n/a | n/a | n/a | n/a |
GLSynthesis Inc. | Assay Description His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o... | J Med Chem 48: 3919-29 (2005) BindingDB Entry DOI: 10.7270/Q2X06991 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histone acetyltransferase KAT2B (Homo sapiens (Human)) | BDBM371576 (4-chloro-5-[[1-[(4-fluorophenyl)methyl]-3-piperidy...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 139 | n/a | n/a | n/a | n/a | n/a | n/a |
GLSynthesis Inc. | Assay Description His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o... | J Med Chem 48: 3919-29 (2005) BindingDB Entry DOI: 10.7270/Q2X06991 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histone acetyltransferase KAT2B (Homo sapiens (Human)) | BDBM371547 (US10239861, Example 27) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 144 | n/a | n/a | n/a | n/a | n/a | n/a |
GLSynthesis Inc. | Assay Description His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o... | J Med Chem 48: 3919-29 (2005) BindingDB Entry DOI: 10.7270/Q2X06991 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histone acetyltransferase KAT2B (Homo sapiens (Human)) | BDBM371552 (4-chloro-5-((1-isopropylpiperidin-3-yl)amino)-2-me...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 147 | n/a | n/a | n/a | n/a | n/a | n/a |
GLSynthesis Inc. | Assay Description His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o... | J Med Chem 48: 3919-29 (2005) BindingDB Entry DOI: 10.7270/Q2X06991 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histone acetyltransferase KAT2B (Homo sapiens (Human)) | BDBM371560 (4-chloro-2-methyl-5-((1-methylazocan-3-yl)amino)py...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 155 | n/a | n/a | n/a | n/a | n/a | n/a |
GLSynthesis Inc. | Assay Description His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o... | J Med Chem 48: 3919-29 (2005) BindingDB Entry DOI: 10.7270/Q2X06991 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histone acetyltransferase KAT2B (Homo sapiens (Human)) | BDBM371554 (US10239861, Example 34 | racemic-5-((1-benzylpiper...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | Purchase PC cid PC sid UniChem | US Patent | n/a | n/a | 155 | n/a | n/a | n/a | n/a | n/a | n/a |
GLSynthesis Inc. | Assay Description His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o... | J Med Chem 48: 3919-29 (2005) BindingDB Entry DOI: 10.7270/Q2X06991 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histone acetyltransferase KAT2B (Homo sapiens (Human)) | BDBM371521 (4-chloro-2-methyl-5-((1-methylazepan-3-yl)amino)py...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 165 | n/a | n/a | n/a | n/a | n/a | n/a |
GLSynthesis Inc. | Assay Description His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o... | J Med Chem 48: 3919-29 (2005) BindingDB Entry DOI: 10.7270/Q2X06991 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histone acetyltransferase KAT2B (Homo sapiens (Human)) | BDBM371544 (4-chloro-2-methyl-5-((1-methyl-5-phenylpiperidin-3...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | Purchase PC cid PC sid UniChem | US Patent | n/a | n/a | 167 | n/a | n/a | n/a | n/a | n/a | n/a |
GLSynthesis Inc. | Assay Description His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o... | J Med Chem 48: 3919-29 (2005) BindingDB Entry DOI: 10.7270/Q2X06991 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histone acetyltransferase KAT2B (Homo sapiens (Human)) | BDBM371578 ((R)-4-chloro-2-methyl-5-((1-methylazepan-3-yl)amin...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 169 | n/a | n/a | n/a | n/a | n/a | n/a |
GLSynthesis Inc. | Assay Description His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o... | J Med Chem 48: 3919-29 (2005) BindingDB Entry DOI: 10.7270/Q2X06991 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histone acetyltransferase KAT2B (Homo sapiens (Human)) | BDBM371548 (US10239861, Example 28) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 175 | n/a | n/a | n/a | n/a | n/a | n/a |
GLSynthesis Inc. | Assay Description His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o... | J Med Chem 48: 3919-29 (2005) BindingDB Entry DOI: 10.7270/Q2X06991 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histone acetyltransferase KAT2B (Homo sapiens (Human)) | BDBM371569 (4-chloro-5-[[1-(1H-imidazol-4-ylmethyl)-3-piperidy...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 178 | n/a | n/a | n/a | n/a | n/a | n/a |
GLSynthesis Inc. | Assay Description His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o... | J Med Chem 48: 3919-29 (2005) BindingDB Entry DOI: 10.7270/Q2X06991 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histone acetyltransferase KAT2B (Homo sapiens (Human)) | BDBM371524 ((racemic)-4-chloro-2-methyl-5-((1-methylazepan-4-y...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 187 | n/a | n/a | n/a | n/a | n/a | n/a |
GLSynthesis Inc. | Assay Description His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o... | J Med Chem 48: 3919-29 (2005) BindingDB Entry DOI: 10.7270/Q2X06991 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histone acetyltransferase KAT2B (Homo sapiens (Human)) | BDBM371561 (Racemic-4-chloro-2-methyl-5-[[1-(3-phenylpropyl)-3...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 232 | n/a | n/a | n/a | n/a | n/a | n/a |
GLSynthesis Inc. | Assay Description His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o... | J Med Chem 48: 3919-29 (2005) BindingDB Entry DOI: 10.7270/Q2X06991 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histone acetyltransferase KAT2B (Homo sapiens (Human)) | BDBM50234944 (CHEMBL4072538 | US10239861, Example 60) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid PDB UniChem Patents Similars | PDB US Patent | n/a | n/a | 235 | n/a | n/a | n/a | n/a | n/a | n/a |
GLSynthesis Inc. | Assay Description His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o... | J Med Chem 48: 3919-29 (2005) BindingDB Entry DOI: 10.7270/Q2X06991 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Histone acetyltransferase KAT2B (Homo sapiens (Human)) | BDBM371566 (4-chloro-5-((1-(3,5-dichlorobenzyl)piperidin-3-yl)...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 278 | n/a | n/a | n/a | n/a | n/a | n/a |
GLSynthesis Inc. | Assay Description His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o... | J Med Chem 48: 3919-29 (2005) BindingDB Entry DOI: 10.7270/Q2X06991 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histone acetyltransferase KAT2B (Homo sapiens (Human)) | BDBM371563 (4-chloro-5-[[1-[(4-dimethylaminophenyl)methyl]-3-p...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 310 | n/a | n/a | n/a | n/a | n/a | n/a |
GLSynthesis Inc. | Assay Description His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o... | J Med Chem 48: 3919-29 (2005) BindingDB Entry DOI: 10.7270/Q2X06991 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histone acetyltransferase KAT2B (Homo sapiens (Human)) | BDBM371537 ((E)-2-(but-2-en-1-yl)-4-chloro-5-((1-methylazepan-...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 312 | n/a | n/a | n/a | n/a | n/a | n/a |
GLSynthesis Inc. | Assay Description His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o... | J Med Chem 48: 3919-29 (2005) BindingDB Entry DOI: 10.7270/Q2X06991 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histone acetyltransferase KAT2B (Homo sapiens (Human)) | BDBM371550 (4-chloro-5-((1-(2-methoxyethyl)piperidin-3-yl)amin...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 315 | n/a | n/a | n/a | n/a | n/a | n/a |
GLSynthesis Inc. | Assay Description His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o... | J Med Chem 48: 3919-29 (2005) BindingDB Entry DOI: 10.7270/Q2X06991 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histone acetyltransferase KAT2B (Homo sapiens (Human)) | BDBM371528 ((S)-5-((1-benzylpiperidin-3-yl)amino)-4-chloro-2-m...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | Purchase PC cid PC sid UniChem | US Patent | n/a | n/a | 349 | n/a | n/a | n/a | n/a | n/a | n/a |
GLSynthesis Inc. | Assay Description His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o... | J Med Chem 48: 3919-29 (2005) BindingDB Entry DOI: 10.7270/Q2X06991 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histone acetyltransferase KAT2B (Homo sapiens (Human)) | BDBM371571 (4-chloro-2-methyl-5-[[1-[(1-methylpyrazol-4-yl)met...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 371 | n/a | n/a | n/a | n/a | n/a | n/a |
GLSynthesis Inc. | Assay Description His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o... | J Med Chem 48: 3919-29 (2005) BindingDB Entry DOI: 10.7270/Q2X06991 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histone acetyltransferase KAT2B (Homo sapiens (Human)) | BDBM371568 (4-chloro-5-[[1-(1H-imidazol-2-ylmethyl)-3-piperidy...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 379 | n/a | n/a | n/a | n/a | n/a | n/a |
GLSynthesis Inc. | Assay Description His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o... | J Med Chem 48: 3919-29 (2005) BindingDB Entry DOI: 10.7270/Q2X06991 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histone acetyltransferase KAT2B (Homo sapiens (Human)) | BDBM371565 (4-chloro-5-[[1-[(4-imidazol-1-ylphenyl)methyl]-3-p...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 386 | n/a | n/a | n/a | n/a | n/a | n/a |
GLSynthesis Inc. | Assay Description His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o... | J Med Chem 48: 3919-29 (2005) BindingDB Entry DOI: 10.7270/Q2X06991 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histone acetyltransferase KAT2B (Homo sapiens (Human)) | BDBM371529 (4-chloro-2-methyl-5-((1-(pyridin-2-yl)piperidin-3-...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 403 | n/a | n/a | n/a | n/a | n/a | n/a |
GLSynthesis Inc. | Assay Description His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o... | J Med Chem 48: 3919-29 (2005) BindingDB Entry DOI: 10.7270/Q2X06991 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histone acetyltransferase KAT2B (Homo sapiens (Human)) | BDBM371535 (4-chloro-2-ethyl-5-((1-methylazepan-3-yl)amino)pyr...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 407 | n/a | n/a | n/a | n/a | n/a | n/a |
GLSynthesis Inc. | Assay Description His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o... | J Med Chem 48: 3919-29 (2005) BindingDB Entry DOI: 10.7270/Q2X06991 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histone acetyltransferase KAT2B (Homo sapiens (Human)) | BDBM371536 (4-chloro-2-(cyclopropylmethyl)-5((1-methylazepan-3...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 421 | n/a | n/a | n/a | n/a | n/a | n/a |
GLSynthesis Inc. | Assay Description His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o... | J Med Chem 48: 3919-29 (2005) BindingDB Entry DOI: 10.7270/Q2X06991 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histone acetyltransferase KAT2B (Homo sapiens (Human)) | BDBM371573 (4-chloro-2-methyl-5-[[1-[(5-methyl-3-pyridyl)methy...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 441 | n/a | n/a | n/a | n/a | n/a | n/a |
GLSynthesis Inc. | Assay Description His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o... | J Med Chem 48: 3919-29 (2005) BindingDB Entry DOI: 10.7270/Q2X06991 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histone acetyltransferase KAT2B (Homo sapiens (Human)) | BDBM371575 (4-chloro-5-[[1-[[3-(4-chlorophenyl)-1,2,4-oxadiazo...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 466 | n/a | n/a | n/a | n/a | n/a | n/a |
GLSynthesis Inc. | Assay Description His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o... | J Med Chem 48: 3919-29 (2005) BindingDB Entry DOI: 10.7270/Q2X06991 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histone acetyltransferase KAT2B (Homo sapiens (Human)) | BDBM371525 (4-chloro-2-methyl-5-(((1R,3r,5S)-8-methyl-8-azabic...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 480 | n/a | n/a | n/a | n/a | n/a | n/a |
GLSynthesis Inc. | Assay Description His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o... | J Med Chem 48: 3919-29 (2005) BindingDB Entry DOI: 10.7270/Q2X06991 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histone acetyltransferase KAT2B (Homo sapiens (Human)) | BDBM371526 (4-chloro-2-methyl-5-(((1R,3s,5S)-8-methyl-8-azabic...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 492 | n/a | n/a | n/a | n/a | n/a | n/a |
GLSynthesis Inc. | Assay Description His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o... | J Med Chem 48: 3919-29 (2005) BindingDB Entry DOI: 10.7270/Q2X06991 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histone acetyltransferase KAT2B (Homo sapiens (Human)) | BDBM371570 (4-chloro-2-methyl-5-[[1-(pyrimidin-5-ylmethyl)-3-p...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 625 | n/a | n/a | n/a | n/a | n/a | n/a |
GLSynthesis Inc. | Assay Description His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o... | J Med Chem 48: 3919-29 (2005) BindingDB Entry DOI: 10.7270/Q2X06991 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histone acetyltransferase KAT2B (Homo sapiens (Human)) | BDBM371556 (4-chloro-2-methyl-5-((1-((S)-1-phenylethyl)piperid...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 631 | n/a | n/a | n/a | n/a | n/a | n/a |
GLSynthesis Inc. | Assay Description His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o... | J Med Chem 48: 3919-29 (2005) BindingDB Entry DOI: 10.7270/Q2X06991 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histone acetyltransferase KAT2B (Homo sapiens (Human)) | BDBM371555 (4-chloro-2-methyl-5-((1-((R)-1-phenylethyl)piperid...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 671 | n/a | n/a | n/a | n/a | n/a | n/a |
GLSynthesis Inc. | Assay Description His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o... | J Med Chem 48: 3919-29 (2005) BindingDB Entry DOI: 10.7270/Q2X06991 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histone acetyltransferase KAT2B (Homo sapiens (Human)) | BDBM371543 (4-chloro-5-(((3S,5R)-1,5-dimethylpiperidin-3-yl)am...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 902 | n/a | n/a | n/a | n/a | n/a | n/a |
GLSynthesis Inc. | Assay Description His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o... | J Med Chem 48: 3919-29 (2005) BindingDB Entry DOI: 10.7270/Q2X06991 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histone acetyltransferase KAT2B (Homo sapiens (Human)) | BDBM371567 (4-chloro-2-methyl-5-[[1-[(2-morpholinophenyl)methy...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 921 | n/a | n/a | n/a | n/a | n/a | n/a |
GLSynthesis Inc. | Assay Description His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o... | J Med Chem 48: 3919-29 (2005) BindingDB Entry DOI: 10.7270/Q2X06991 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histone acetyltransferase KAT2B (Homo sapiens (Human)) | BDBM371557 (US10239861, Example 37) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 972 | n/a | n/a | n/a | n/a | n/a | n/a |
GLSynthesis Inc. | Assay Description His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o... | J Med Chem 48: 3919-29 (2005) BindingDB Entry DOI: 10.7270/Q2X06991 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histone acetyltransferase KAT2B (Homo sapiens (Human)) | BDBM371530 ((racemic)-4-chloro-2-methyl-5-(quinuclidin-3-ylami...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 975 | n/a | n/a | n/a | n/a | n/a | n/a |
GLSynthesis Inc. | Assay Description His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o... | J Med Chem 48: 3919-29 (2005) BindingDB Entry DOI: 10.7270/Q2X06991 | |||||||||||
More data for this Ligand-Target Pair |
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