Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Alpha-2A adrenergic receptor (Homo sapiens (Human)) | BDBM50258564 ((S)-6-(2-(pyridin-4-yl)phenyl)-6,7-dihydro-5H-pyrr...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 112 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Inhibition of adrenergic alpha2A receptor (unknown origin) | Bioorg Med Chem Lett 19: 3113-7 (2009) Article DOI: 10.1016/j.bmcl.2009.03.166 BindingDB Entry DOI: 10.7270/Q2WS8T5T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2A adrenergic receptor (Homo sapiens (Human)) | BDBM50258590 ((S)-N-(2'-(6,7-dihydro-5H-pyrrolo[1,2-a]imidazol-6...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | 114 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Inhibition of adrenergic alpha2A receptor (unknown origin) | Bioorg Med Chem Lett 19: 3113-7 (2009) Article DOI: 10.1016/j.bmcl.2009.03.166 BindingDB Entry DOI: 10.7270/Q2WS8T5T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2A adrenergic receptor (Homo sapiens (Human)) | BDBM50258592 ((S)-2'-(6,7-dihydro-5H-pyrrolo[1,2-a]imidazol-6-yl...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | 202 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Inhibition of adrenergic alpha2A receptor (unknown origin) | Bioorg Med Chem Lett 19: 3113-7 (2009) Article DOI: 10.1016/j.bmcl.2009.03.166 BindingDB Entry DOI: 10.7270/Q2WS8T5T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2A adrenergic receptor (Homo sapiens (Human)) | BDBM50258518 ((S)-6-(biphenyl-2-yl)-6,7-dihydro-5H-pyrrolo[1,2-a...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 213 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Inhibition of adrenergic alpha2A receptor (unknown origin) | Bioorg Med Chem Lett 19: 3113-7 (2009) Article DOI: 10.1016/j.bmcl.2009.03.166 BindingDB Entry DOI: 10.7270/Q2WS8T5T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2A adrenergic receptor (Homo sapiens (Human)) | BDBM50258591 ((S)-2-(2-(6,7-dihydro-5H-pyrrolo[1,2-a]imidazol-6-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | 280 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Inhibition of adrenergic alpha2A receptor (unknown origin) | Bioorg Med Chem Lett 19: 3113-7 (2009) Article DOI: 10.1016/j.bmcl.2009.03.166 BindingDB Entry DOI: 10.7270/Q2WS8T5T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2A adrenergic receptor (Homo sapiens (Human)) | BDBM50258565 ((S)-6-(2-(1-methyl-1H-pyrazol-4-yl)phenyl)-6,7-dih...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | 380 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Inhibition of adrenergic alpha2A receptor (unknown origin) | Bioorg Med Chem Lett 19: 3113-7 (2009) Article DOI: 10.1016/j.bmcl.2009.03.166 BindingDB Entry DOI: 10.7270/Q2WS8T5T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2A adrenergic receptor (Homo sapiens (Human)) | BDBM50258640 (2-(2-(6,7-dihydro-5H-pyrrolo[1,2-a]imidazol-6-yl)-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 469 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Inhibition of adrenergic alpha2A receptor (unknown origin) | Bioorg Med Chem Lett 19: 3113-7 (2009) Article DOI: 10.1016/j.bmcl.2009.03.166 BindingDB Entry DOI: 10.7270/Q2WS8T5T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2A adrenergic receptor (Homo sapiens (Human)) | BDBM50258560 ((S)-2-(2-(6,7-dihydro-5H-pyrrolo[1,2-a]imidazol-6-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 805 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Inhibition of adrenergic alpha2A receptor (unknown origin) | Bioorg Med Chem Lett 19: 3113-7 (2009) Article DOI: 10.1016/j.bmcl.2009.03.166 BindingDB Entry DOI: 10.7270/Q2WS8T5T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2A adrenergic receptor (Homo sapiens (Human)) | BDBM50258563 ((S)-6-(2-(pyridin-3-yl)phenyl)-6,7-dihydro-5H-pyrr...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 991 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Inhibition of adrenergic alpha2A receptor (unknown origin) | Bioorg Med Chem Lett 19: 3113-7 (2009) Article DOI: 10.1016/j.bmcl.2009.03.166 BindingDB Entry DOI: 10.7270/Q2WS8T5T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2A adrenergic receptor (Homo sapiens (Human)) | BDBM50258561 ((R)-2-(2-(6,7-dihydro-5H-pyrrolo[1,2-a]imidazol-6-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.02E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Inhibition of adrenergic alpha2A receptor (unknown origin) | Bioorg Med Chem Lett 19: 3113-7 (2009) Article DOI: 10.1016/j.bmcl.2009.03.166 BindingDB Entry DOI: 10.7270/Q2WS8T5T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2A adrenergic receptor (Homo sapiens (Human)) | BDBM50258589 ((S)-6-(2-(1H-pyrazol-1-yl)phenyl)-6,7-dihydro-5H-p...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Inhibition of adrenergic alpha2A receptor (unknown origin) | Bioorg Med Chem Lett 19: 3113-7 (2009) Article DOI: 10.1016/j.bmcl.2009.03.166 BindingDB Entry DOI: 10.7270/Q2WS8T5T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2A adrenergic receptor (Homo sapiens (Human)) | BDBM50258641 (6-(4-fluoro-2-(1H-pyrazol-5-yl)phenyl)-6,7-dihydro...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.47E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Inhibition of adrenergic alpha2A receptor (unknown origin) | Bioorg Med Chem Lett 19: 3113-7 (2009) Article DOI: 10.1016/j.bmcl.2009.03.166 BindingDB Entry DOI: 10.7270/Q2WS8T5T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2A adrenergic receptor (Homo sapiens (Human)) | BDBM50256563 ((R)-2-(5-chloro-4-(methoxymethyl)-2,3-dihydro-1H-i...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | >1.70E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Inhibition of adrenergic alpha2A receptor (unknown origin) | Bioorg Med Chem Lett 19: 3113-7 (2009) Article DOI: 10.1016/j.bmcl.2009.03.166 BindingDB Entry DOI: 10.7270/Q2WS8T5T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2A adrenergic receptor (Homo sapiens (Human)) | BDBM50258562 ((S)-2-(2-(6,7-dihydro-5H-pyrrolo[1,2-a]imidazol-6-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | 1.75E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Inhibition of adrenergic alpha2A receptor (unknown origin) | Bioorg Med Chem Lett 19: 3113-7 (2009) Article DOI: 10.1016/j.bmcl.2009.03.166 BindingDB Entry DOI: 10.7270/Q2WS8T5T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2A adrenergic receptor (Homo sapiens (Human)) | BDBM50258639 (2-(2-(6,7-dihydro-5H-pyrrolo[1,2-a]imidazol-6-yl)-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | >2.16E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Inhibition of adrenergic alpha2A receptor (unknown origin) | Bioorg Med Chem Lett 19: 3113-7 (2009) Article DOI: 10.1016/j.bmcl.2009.03.166 BindingDB Entry DOI: 10.7270/Q2WS8T5T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2A adrenergic receptor (Homo sapiens (Human)) | BDBM50258593 (6-(4-fluoro-2-(pyrimidin-5-yl)phenyl)-6,7-dihydro-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | >2.37E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Inhibition of adrenergic alpha2A receptor (unknown origin) | Bioorg Med Chem Lett 19: 3113-7 (2009) Article DOI: 10.1016/j.bmcl.2009.03.166 BindingDB Entry DOI: 10.7270/Q2WS8T5T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2A adrenergic receptor (Homo sapiens (Human)) | BDBM50258594 (6-(5-fluoro-2-(pyrimidin-5-yl)phenyl)-6,7-dihydro-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | >2.78E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Inhibition of adrenergic alpha2A receptor (unknown origin) | Bioorg Med Chem Lett 19: 3113-7 (2009) Article DOI: 10.1016/j.bmcl.2009.03.166 BindingDB Entry DOI: 10.7270/Q2WS8T5T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2A adrenergic receptor (Homo sapiens (Human)) | BDBM50258644 (6-(4-fluoro-2-(1H-pyrazol-1-yl)phenyl)-6,7-dihydro...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | >3.23E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Inhibition of adrenergic alpha2A receptor (unknown origin) | Bioorg Med Chem Lett 19: 3113-7 (2009) Article DOI: 10.1016/j.bmcl.2009.03.166 BindingDB Entry DOI: 10.7270/Q2WS8T5T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2A adrenergic receptor (Homo sapiens (Human)) | BDBM50258638 (6-(2-fluoro-6-(pyrimidin-5-yl)phenyl)-6,7-dihydro-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | >3.31E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Inhibition of adrenergic alpha2A receptor (unknown origin) | Bioorg Med Chem Lett 19: 3113-7 (2009) Article DOI: 10.1016/j.bmcl.2009.03.166 BindingDB Entry DOI: 10.7270/Q2WS8T5T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2A adrenergic receptor (Homo sapiens (Human)) | BDBM50258559 ((S)-6-(2-(pyrimidin-5-yl)phenyl)-6,7-dihydro-5H-py...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | >3.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Inhibition of adrenergic alpha2A receptor (unknown origin) | Bioorg Med Chem Lett 19: 3113-7 (2009) Article DOI: 10.1016/j.bmcl.2009.03.166 BindingDB Entry DOI: 10.7270/Q2WS8T5T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2A adrenergic receptor (Homo sapiens (Human)) | BDBM50258517 ((S)-2-(6,7-dihydro-5H-pyrrolo[1,2-a]imidazol-6-yl)...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | >4.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Inhibition of adrenergic alpha2A receptor (unknown origin) | Bioorg Med Chem Lett 19: 3113-7 (2009) Article DOI: 10.1016/j.bmcl.2009.03.166 BindingDB Entry DOI: 10.7270/Q2WS8T5T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1D adrenergic receptor (Homo sapiens (Human)) | BDBM50258517 ((S)-2-(6,7-dihydro-5H-pyrrolo[1,2-a]imidazol-6-yl)...) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Agonist activity at human adrenergic alpha1D receptor expressed in CHO cells assessed as calcium mobilization by FLIPR | Bioorg Med Chem Lett 19: 3113-7 (2009) Article DOI: 10.1016/j.bmcl.2009.03.166 BindingDB Entry DOI: 10.7270/Q2WS8T5T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1A adrenergic receptor (Homo sapiens (Human)) | BDBM50258589 ((S)-6-(2-(1H-pyrazol-1-yl)phenyl)-6,7-dihydro-5H-p...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 5 | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Agonist activity at human adrenergic alpha1A receptor expressed in CHO cells assessed as calcium mobilization by FLIPR | Bioorg Med Chem Lett 19: 3113-7 (2009) Article DOI: 10.1016/j.bmcl.2009.03.166 BindingDB Entry DOI: 10.7270/Q2WS8T5T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1D adrenergic receptor (Homo sapiens (Human)) | BDBM50258559 ((S)-6-(2-(pyrimidin-5-yl)phenyl)-6,7-dihydro-5H-py...) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 391 | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Agonist activity at human adrenergic alpha1D receptor expressed in CHO cells assessed as calcium mobilization by FLIPR | Bioorg Med Chem Lett 19: 3113-7 (2009) Article DOI: 10.1016/j.bmcl.2009.03.166 BindingDB Entry DOI: 10.7270/Q2WS8T5T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1A adrenergic receptor (Homo sapiens (Human)) | BDBM50258561 ((R)-2-(2-(6,7-dihydro-5H-pyrrolo[1,2-a]imidazol-6-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 92 | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Agonist activity at human adrenergic alpha1A receptor expressed in CHO cells assessed as calcium mobilization by FLIPR | Bioorg Med Chem Lett 19: 3113-7 (2009) Article DOI: 10.1016/j.bmcl.2009.03.166 BindingDB Entry DOI: 10.7270/Q2WS8T5T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1A adrenergic receptor (Homo sapiens (Human)) | BDBM50258562 ((S)-2-(2-(6,7-dihydro-5H-pyrrolo[1,2-a]imidazol-6-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 3 | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Agonist activity at human adrenergic alpha1A receptor expressed in CHO cells assessed as calcium mobilization by FLIPR | Bioorg Med Chem Lett 19: 3113-7 (2009) Article DOI: 10.1016/j.bmcl.2009.03.166 BindingDB Entry DOI: 10.7270/Q2WS8T5T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1B adrenergic receptor (Homo sapiens (Human)) | BDBM50258639 (2-(2-(6,7-dihydro-5H-pyrrolo[1,2-a]imidazol-6-yl)-...) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Agonist activity at human adrenergic alpha1B receptor expressed in CHO cells assessed as calcium mobilization by FLIPR | Bioorg Med Chem Lett 19: 3113-7 (2009) Article DOI: 10.1016/j.bmcl.2009.03.166 BindingDB Entry DOI: 10.7270/Q2WS8T5T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1A adrenergic receptor (Homo sapiens (Human)) | BDBM50258643 (6-(5-fluoro-2-(1H-pyrazol-1-yl)phenyl)-6,7-dihydro...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 5 | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Agonist activity at human adrenergic alpha1A receptor expressed in CHO cells assessed as calcium mobilization by FLIPR | Bioorg Med Chem Lett 19: 3113-7 (2009) Article DOI: 10.1016/j.bmcl.2009.03.166 BindingDB Entry DOI: 10.7270/Q2WS8T5T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1A adrenergic receptor (Homo sapiens (Human)) | BDBM50258590 ((S)-N-(2'-(6,7-dihydro-5H-pyrrolo[1,2-a]imidazol-6...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 4 | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Agonist activity at human adrenergic alpha1A receptor expressed in CHO cells assessed as calcium mobilization by FLIPR | Bioorg Med Chem Lett 19: 3113-7 (2009) Article DOI: 10.1016/j.bmcl.2009.03.166 BindingDB Entry DOI: 10.7270/Q2WS8T5T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1B adrenergic receptor (Homo sapiens (Human)) | BDBM50258591 ((S)-2-(2-(6,7-dihydro-5H-pyrrolo[1,2-a]imidazol-6-...) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Agonist activity at human adrenergic alpha1B receptor expressed in CHO cells assessed as calcium mobilization by FLIPR | Bioorg Med Chem Lett 19: 3113-7 (2009) Article DOI: 10.1016/j.bmcl.2009.03.166 BindingDB Entry DOI: 10.7270/Q2WS8T5T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1B adrenergic receptor (Homo sapiens (Human)) | BDBM50256563 ((R)-2-(5-chloro-4-(methoxymethyl)-2,3-dihydro-1H-i...) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Agonist activity at human adrenergic alpha1B receptor expressed in CHO cells assessed as calcium mobilization by FLIPR | Bioorg Med Chem Lett 19: 3113-7 (2009) Article DOI: 10.1016/j.bmcl.2009.03.166 BindingDB Entry DOI: 10.7270/Q2WS8T5T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1D adrenergic receptor (Homo sapiens (Human)) | BDBM50258593 (6-(4-fluoro-2-(pyrimidin-5-yl)phenyl)-6,7-dihydro-...) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | >3.40E+3 | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Agonist activity at human adrenergic alpha1D receptor expressed in CHO cells assessed as calcium mobilization by FLIPR | Bioorg Med Chem Lett 19: 3113-7 (2009) Article DOI: 10.1016/j.bmcl.2009.03.166 BindingDB Entry DOI: 10.7270/Q2WS8T5T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1B adrenergic receptor (Homo sapiens (Human)) | BDBM50258589 ((S)-6-(2-(1H-pyrazol-1-yl)phenyl)-6,7-dihydro-5H-p...) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Agonist activity at human adrenergic alpha1B receptor expressed in CHO cells assessed as calcium mobilization by FLIPR | Bioorg Med Chem Lett 19: 3113-7 (2009) Article DOI: 10.1016/j.bmcl.2009.03.166 BindingDB Entry DOI: 10.7270/Q2WS8T5T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1D adrenergic receptor (Homo sapiens (Human)) | BDBM50258590 ((S)-N-(2'-(6,7-dihydro-5H-pyrrolo[1,2-a]imidazol-6...) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Agonist activity at human adrenergic alpha1D receptor expressed in CHO cells assessed as calcium mobilization by FLIPR | Bioorg Med Chem Lett 19: 3113-7 (2009) Article DOI: 10.1016/j.bmcl.2009.03.166 BindingDB Entry DOI: 10.7270/Q2WS8T5T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1A adrenergic receptor (Homo sapiens (Human)) | BDBM50258563 ((S)-6-(2-(pyridin-3-yl)phenyl)-6,7-dihydro-5H-pyrr...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1 | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Agonist activity at human adrenergic alpha1A receptor expressed in CHO cells assessed as calcium mobilization by FLIPR | Bioorg Med Chem Lett 19: 3113-7 (2009) Article DOI: 10.1016/j.bmcl.2009.03.166 BindingDB Entry DOI: 10.7270/Q2WS8T5T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1A adrenergic receptor (Homo sapiens (Human)) | BDBM50258564 ((S)-6-(2-(pyridin-4-yl)phenyl)-6,7-dihydro-5H-pyrr...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 81 | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Agonist activity at human adrenergic alpha1A receptor expressed in CHO cells assessed as calcium mobilization by FLIPR | Bioorg Med Chem Lett 19: 3113-7 (2009) Article DOI: 10.1016/j.bmcl.2009.03.166 BindingDB Entry DOI: 10.7270/Q2WS8T5T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1A adrenergic receptor (Homo sapiens (Human)) | BDBM50258518 ((S)-6-(biphenyl-2-yl)-6,7-dihydro-5H-pyrrolo[1,2-a...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 12 | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Agonist activity at human adrenergic alpha1A receptor expressed in CHO cells assessed as calcium mobilization by FLIPR | Bioorg Med Chem Lett 19: 3113-7 (2009) Article DOI: 10.1016/j.bmcl.2009.03.166 BindingDB Entry DOI: 10.7270/Q2WS8T5T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1A adrenergic receptor (Homo sapiens (Human)) | BDBM50258559 ((S)-6-(2-(pyrimidin-5-yl)phenyl)-6,7-dihydro-5H-py...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 0.400 | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Agonist activity at human adrenergic alpha1A receptor expressed in CHO cells assessed as calcium mobilization by FLIPR | Bioorg Med Chem Lett 19: 3113-7 (2009) Article DOI: 10.1016/j.bmcl.2009.03.166 BindingDB Entry DOI: 10.7270/Q2WS8T5T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1D adrenergic receptor (Homo sapiens (Human)) | BDBM50258560 ((S)-2-(2-(6,7-dihydro-5H-pyrrolo[1,2-a]imidazol-6-...) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 146 | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Agonist activity at human adrenergic alpha1D receptor expressed in CHO cells assessed as calcium mobilization by FLIPR | Bioorg Med Chem Lett 19: 3113-7 (2009) Article DOI: 10.1016/j.bmcl.2009.03.166 BindingDB Entry DOI: 10.7270/Q2WS8T5T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1D adrenergic receptor (Homo sapiens (Human)) | BDBM50258594 (6-(5-fluoro-2-(pyrimidin-5-yl)phenyl)-6,7-dihydro-...) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | >2.60E+3 | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Agonist activity at human adrenergic alpha1D receptor expressed in CHO cells assessed as calcium mobilization by FLIPR | Bioorg Med Chem Lett 19: 3113-7 (2009) Article DOI: 10.1016/j.bmcl.2009.03.166 BindingDB Entry DOI: 10.7270/Q2WS8T5T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1B adrenergic receptor (Homo sapiens (Human)) | BDBM50258641 (6-(4-fluoro-2-(1H-pyrazol-5-yl)phenyl)-6,7-dihydro...) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Agonist activity at human adrenergic alpha1B receptor expressed in CHO cells assessed as calcium mobilization by FLIPR | Bioorg Med Chem Lett 19: 3113-7 (2009) Article DOI: 10.1016/j.bmcl.2009.03.166 BindingDB Entry DOI: 10.7270/Q2WS8T5T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1B adrenergic receptor (Homo sapiens (Human)) | BDBM50258643 (6-(5-fluoro-2-(1H-pyrazol-1-yl)phenyl)-6,7-dihydro...) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Agonist activity at human adrenergic alpha1B receptor expressed in CHO cells assessed as calcium mobilization by FLIPR | Bioorg Med Chem Lett 19: 3113-7 (2009) Article DOI: 10.1016/j.bmcl.2009.03.166 BindingDB Entry DOI: 10.7270/Q2WS8T5T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1B adrenergic receptor (Homo sapiens (Human)) | BDBM50258564 ((S)-6-(2-(pyridin-4-yl)phenyl)-6,7-dihydro-5H-pyrr...) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Agonist activity at human adrenergic alpha1B receptor expressed in CHO cells assessed as calcium mobilization by FLIPR | Bioorg Med Chem Lett 19: 3113-7 (2009) Article DOI: 10.1016/j.bmcl.2009.03.166 BindingDB Entry DOI: 10.7270/Q2WS8T5T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1A adrenergic receptor (Homo sapiens (Human)) | BDBM50258591 ((S)-2-(2-(6,7-dihydro-5H-pyrrolo[1,2-a]imidazol-6-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 12 | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Agonist activity at human adrenergic alpha1A receptor expressed in CHO cells assessed as calcium mobilization by FLIPR | Bioorg Med Chem Lett 19: 3113-7 (2009) Article DOI: 10.1016/j.bmcl.2009.03.166 BindingDB Entry DOI: 10.7270/Q2WS8T5T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1A adrenergic receptor (Homo sapiens (Human)) | BDBM50258560 ((S)-2-(2-(6,7-dihydro-5H-pyrrolo[1,2-a]imidazol-6-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 2 | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Agonist activity at human adrenergic alpha1A receptor expressed in CHO cells assessed as calcium mobilization by FLIPR | Bioorg Med Chem Lett 19: 3113-7 (2009) Article DOI: 10.1016/j.bmcl.2009.03.166 BindingDB Entry DOI: 10.7270/Q2WS8T5T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1B adrenergic receptor (Homo sapiens (Human)) | BDBM50258561 ((R)-2-(2-(6,7-dihydro-5H-pyrrolo[1,2-a]imidazol-6-...) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Agonist activity at human adrenergic alpha1B receptor expressed in CHO cells assessed as calcium mobilization by FLIPR | Bioorg Med Chem Lett 19: 3113-7 (2009) Article DOI: 10.1016/j.bmcl.2009.03.166 BindingDB Entry DOI: 10.7270/Q2WS8T5T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1D adrenergic receptor (Homo sapiens (Human)) | BDBM50258561 ((R)-2-(2-(6,7-dihydro-5H-pyrrolo[1,2-a]imidazol-6-...) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | >3.57E+3 | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Agonist activity at human adrenergic alpha1D receptor expressed in CHO cells assessed as calcium mobilization by FLIPR | Bioorg Med Chem Lett 19: 3113-7 (2009) Article DOI: 10.1016/j.bmcl.2009.03.166 BindingDB Entry DOI: 10.7270/Q2WS8T5T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1B adrenergic receptor (Homo sapiens (Human)) | BDBM50258593 (6-(4-fluoro-2-(pyrimidin-5-yl)phenyl)-6,7-dihydro-...) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Agonist activity at human adrenergic alpha1B receptor expressed in CHO cells assessed as calcium mobilization by FLIPR | Bioorg Med Chem Lett 19: 3113-7 (2009) Article DOI: 10.1016/j.bmcl.2009.03.166 BindingDB Entry DOI: 10.7270/Q2WS8T5T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1D adrenergic receptor (Homo sapiens (Human)) | BDBM50258639 (2-(2-(6,7-dihydro-5H-pyrrolo[1,2-a]imidazol-6-yl)-...) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Agonist activity at human adrenergic alpha1D receptor expressed in CHO cells assessed as calcium mobilization by FLIPR | Bioorg Med Chem Lett 19: 3113-7 (2009) Article DOI: 10.1016/j.bmcl.2009.03.166 BindingDB Entry DOI: 10.7270/Q2WS8T5T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1D adrenergic receptor (Homo sapiens (Human)) | BDBM50258641 (6-(4-fluoro-2-(1H-pyrazol-5-yl)phenyl)-6,7-dihydro...) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 276 | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Agonist activity at human adrenergic alpha1D receptor expressed in CHO cells assessed as calcium mobilization by FLIPR | Bioorg Med Chem Lett 19: 3113-7 (2009) Article DOI: 10.1016/j.bmcl.2009.03.166 BindingDB Entry DOI: 10.7270/Q2WS8T5T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1B adrenergic receptor (Homo sapiens (Human)) | BDBM50258590 ((S)-N-(2'-(6,7-dihydro-5H-pyrrolo[1,2-a]imidazol-6...) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Agonist activity at human adrenergic alpha1B receptor expressed in CHO cells assessed as calcium mobilization by FLIPR | Bioorg Med Chem Lett 19: 3113-7 (2009) Article DOI: 10.1016/j.bmcl.2009.03.166 BindingDB Entry DOI: 10.7270/Q2WS8T5T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1B adrenergic receptor (Homo sapiens (Human)) | BDBM50258563 ((S)-6-(2-(pyridin-3-yl)phenyl)-6,7-dihydro-5H-pyrr...) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 760 | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Agonist activity at human adrenergic alpha1B receptor expressed in CHO cells assessed as calcium mobilization by FLIPR | Bioorg Med Chem Lett 19: 3113-7 (2009) Article DOI: 10.1016/j.bmcl.2009.03.166 BindingDB Entry DOI: 10.7270/Q2WS8T5T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1D adrenergic receptor (Homo sapiens (Human)) | BDBM50258563 ((S)-6-(2-(pyridin-3-yl)phenyl)-6,7-dihydro-5H-pyrr...) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 119 | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Agonist activity at human adrenergic alpha1D receptor expressed in CHO cells assessed as calcium mobilization by FLIPR | Bioorg Med Chem Lett 19: 3113-7 (2009) Article DOI: 10.1016/j.bmcl.2009.03.166 BindingDB Entry DOI: 10.7270/Q2WS8T5T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1B adrenergic receptor (Homo sapiens (Human)) | BDBM50258594 (6-(5-fluoro-2-(pyrimidin-5-yl)phenyl)-6,7-dihydro-...) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Agonist activity at human adrenergic alpha1B receptor expressed in CHO cells assessed as calcium mobilization by FLIPR | Bioorg Med Chem Lett 19: 3113-7 (2009) Article DOI: 10.1016/j.bmcl.2009.03.166 BindingDB Entry DOI: 10.7270/Q2WS8T5T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1B adrenergic receptor (Homo sapiens (Human)) | BDBM50258638 (6-(2-fluoro-6-(pyrimidin-5-yl)phenyl)-6,7-dihydro-...) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Agonist activity at human adrenergic alpha1B receptor expressed in CHO cells assessed as calcium mobilization by FLIPR | Bioorg Med Chem Lett 19: 3113-7 (2009) Article DOI: 10.1016/j.bmcl.2009.03.166 BindingDB Entry DOI: 10.7270/Q2WS8T5T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1A adrenergic receptor (Homo sapiens (Human)) | BDBM50258640 (2-(2-(6,7-dihydro-5H-pyrrolo[1,2-a]imidazol-6-yl)-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 3 | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Agonist activity at human adrenergic alpha1A receptor expressed in CHO cells assessed as calcium mobilization by FLIPR | Bioorg Med Chem Lett 19: 3113-7 (2009) Article DOI: 10.1016/j.bmcl.2009.03.166 BindingDB Entry DOI: 10.7270/Q2WS8T5T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1D adrenergic receptor (Homo sapiens (Human)) | BDBM50258640 (2-(2-(6,7-dihydro-5H-pyrrolo[1,2-a]imidazol-6-yl)-...) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 276 | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Agonist activity at human adrenergic alpha1D receptor expressed in CHO cells assessed as calcium mobilization by FLIPR | Bioorg Med Chem Lett 19: 3113-7 (2009) Article DOI: 10.1016/j.bmcl.2009.03.166 BindingDB Entry DOI: 10.7270/Q2WS8T5T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1A adrenergic receptor (Homo sapiens (Human)) | BDBM50258641 (6-(4-fluoro-2-(1H-pyrazol-5-yl)phenyl)-6,7-dihydro...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 15 | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Agonist activity at human adrenergic alpha1A receptor expressed in CHO cells assessed as calcium mobilization by FLIPR | Bioorg Med Chem Lett 19: 3113-7 (2009) Article DOI: 10.1016/j.bmcl.2009.03.166 BindingDB Entry DOI: 10.7270/Q2WS8T5T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1B adrenergic receptor (Homo sapiens (Human)) | BDBM50258642 (6-(5-fluoro-2-(1H-pyrazol-5-yl)phenyl)-6,7-dihydro...) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Agonist activity at human adrenergic alpha1B receptor expressed in CHO cells assessed as calcium mobilization by FLIPR | Bioorg Med Chem Lett 19: 3113-7 (2009) Article DOI: 10.1016/j.bmcl.2009.03.166 BindingDB Entry DOI: 10.7270/Q2WS8T5T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1D adrenergic receptor (Homo sapiens (Human)) | BDBM50258643 (6-(5-fluoro-2-(1H-pyrazol-1-yl)phenyl)-6,7-dihydro...) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Agonist activity at human adrenergic alpha1D receptor expressed in CHO cells assessed as calcium mobilization by FLIPR | Bioorg Med Chem Lett 19: 3113-7 (2009) Article DOI: 10.1016/j.bmcl.2009.03.166 BindingDB Entry DOI: 10.7270/Q2WS8T5T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1D adrenergic receptor (Homo sapiens (Human)) | BDBM50258564 ((S)-6-(2-(pyridin-4-yl)phenyl)-6,7-dihydro-5H-pyrr...) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 656 | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Agonist activity at human adrenergic alpha1D receptor expressed in CHO cells assessed as calcium mobilization by FLIPR | Bioorg Med Chem Lett 19: 3113-7 (2009) Article DOI: 10.1016/j.bmcl.2009.03.166 BindingDB Entry DOI: 10.7270/Q2WS8T5T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1D adrenergic receptor (Homo sapiens (Human)) | BDBM50258589 ((S)-6-(2-(1H-pyrazol-1-yl)phenyl)-6,7-dihydro-5H-p...) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Agonist activity at human adrenergic alpha1D receptor expressed in CHO cells assessed as calcium mobilization by FLIPR | Bioorg Med Chem Lett 19: 3113-7 (2009) Article DOI: 10.1016/j.bmcl.2009.03.166 BindingDB Entry DOI: 10.7270/Q2WS8T5T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1A adrenergic receptor (Homo sapiens (Human)) | BDBM50258517 ((S)-2-(6,7-dihydro-5H-pyrrolo[1,2-a]imidazol-6-yl)...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 51 | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Agonist activity at human adrenergic alpha1A receptor expressed in CHO cells assessed as calcium mobilization by FLIPR | Bioorg Med Chem Lett 19: 3113-7 (2009) Article DOI: 10.1016/j.bmcl.2009.03.166 BindingDB Entry DOI: 10.7270/Q2WS8T5T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1A adrenergic receptor (Homo sapiens (Human)) | BDBM50258594 (6-(5-fluoro-2-(pyrimidin-5-yl)phenyl)-6,7-dihydro-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1 | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Agonist activity at human adrenergic alpha1A receptor expressed in CHO cells assessed as calcium mobilization by FLIPR | Bioorg Med Chem Lett 19: 3113-7 (2009) Article DOI: 10.1016/j.bmcl.2009.03.166 BindingDB Entry DOI: 10.7270/Q2WS8T5T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1A adrenergic receptor (Homo sapiens (Human)) | BDBM50258642 (6-(5-fluoro-2-(1H-pyrazol-5-yl)phenyl)-6,7-dihydro...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 3 | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Agonist activity at human adrenergic alpha1A receptor expressed in CHO cells assessed as calcium mobilization by FLIPR | Bioorg Med Chem Lett 19: 3113-7 (2009) Article DOI: 10.1016/j.bmcl.2009.03.166 BindingDB Entry DOI: 10.7270/Q2WS8T5T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1D adrenergic receptor (Homo sapiens (Human)) | BDBM50256563 ((R)-2-(5-chloro-4-(methoxymethyl)-2,3-dihydro-1H-i...) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | >7.00E+3 | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Agonist activity at human adrenergic alpha1D receptor expressed in CHO cells assessed as calcium mobilization by FLIPR | Bioorg Med Chem Lett 19: 3113-7 (2009) Article DOI: 10.1016/j.bmcl.2009.03.166 BindingDB Entry DOI: 10.7270/Q2WS8T5T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1B adrenergic receptor (Homo sapiens (Human)) | BDBM50258517 ((S)-2-(6,7-dihydro-5H-pyrrolo[1,2-a]imidazol-6-yl)...) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Agonist activity at human adrenergic alpha1B receptor expressed in CHO cells assessed as calcium mobilization by FLIPR | Bioorg Med Chem Lett 19: 3113-7 (2009) Article DOI: 10.1016/j.bmcl.2009.03.166 BindingDB Entry DOI: 10.7270/Q2WS8T5T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1B adrenergic receptor (Homo sapiens (Human)) | BDBM50258559 ((S)-6-(2-(pyrimidin-5-yl)phenyl)-6,7-dihydro-5H-py...) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | >6.50E+3 | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Agonist activity at human adrenergic alpha1B receptor expressed in CHO cells assessed as calcium mobilization by FLIPR | Bioorg Med Chem Lett 19: 3113-7 (2009) Article DOI: 10.1016/j.bmcl.2009.03.166 BindingDB Entry DOI: 10.7270/Q2WS8T5T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1B adrenergic receptor (Homo sapiens (Human)) | BDBM50258592 ((S)-2'-(6,7-dihydro-5H-pyrrolo[1,2-a]imidazol-6-yl...) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Agonist activity at human adrenergic alpha1B receptor expressed in CHO cells assessed as calcium mobilization by FLIPR | Bioorg Med Chem Lett 19: 3113-7 (2009) Article DOI: 10.1016/j.bmcl.2009.03.166 BindingDB Entry DOI: 10.7270/Q2WS8T5T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1A adrenergic receptor (Homo sapiens (Human)) | BDBM50258593 (6-(4-fluoro-2-(pyrimidin-5-yl)phenyl)-6,7-dihydro-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 19 | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Agonist activity at human adrenergic alpha1A receptor expressed in CHO cells assessed as calcium mobilization by FLIPR | Bioorg Med Chem Lett 19: 3113-7 (2009) Article DOI: 10.1016/j.bmcl.2009.03.166 BindingDB Entry DOI: 10.7270/Q2WS8T5T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1A adrenergic receptor (Homo sapiens (Human)) | BDBM50258638 (6-(2-fluoro-6-(pyrimidin-5-yl)phenyl)-6,7-dihydro-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 62 | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Agonist activity at human adrenergic alpha1A receptor expressed in CHO cells assessed as calcium mobilization by FLIPR | Bioorg Med Chem Lett 19: 3113-7 (2009) Article DOI: 10.1016/j.bmcl.2009.03.166 BindingDB Entry DOI: 10.7270/Q2WS8T5T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1B adrenergic receptor (Homo sapiens (Human)) | BDBM50258640 (2-(2-(6,7-dihydro-5H-pyrrolo[1,2-a]imidazol-6-yl)-...) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 990 | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Agonist activity at human adrenergic alpha1B receptor expressed in CHO cells assessed as calcium mobilization by FLIPR | Bioorg Med Chem Lett 19: 3113-7 (2009) Article DOI: 10.1016/j.bmcl.2009.03.166 BindingDB Entry DOI: 10.7270/Q2WS8T5T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1A adrenergic receptor (Homo sapiens (Human)) | BDBM50258644 (6-(4-fluoro-2-(1H-pyrazol-1-yl)phenyl)-6,7-dihydro...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 27 | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Agonist activity at human adrenergic alpha1A receptor expressed in CHO cells assessed as calcium mobilization by FLIPR | Bioorg Med Chem Lett 19: 3113-7 (2009) Article DOI: 10.1016/j.bmcl.2009.03.166 BindingDB Entry DOI: 10.7270/Q2WS8T5T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1D adrenergic receptor (Homo sapiens (Human)) | BDBM50258591 ((S)-2-(2-(6,7-dihydro-5H-pyrrolo[1,2-a]imidazol-6-...) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Agonist activity at human adrenergic alpha1D receptor expressed in CHO cells assessed as calcium mobilization by FLIPR | Bioorg Med Chem Lett 19: 3113-7 (2009) Article DOI: 10.1016/j.bmcl.2009.03.166 BindingDB Entry DOI: 10.7270/Q2WS8T5T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1A adrenergic receptor (Homo sapiens (Human)) | BDBM50256563 ((R)-2-(5-chloro-4-(methoxymethyl)-2,3-dihydro-1H-i...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 31 | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Agonist activity at human adrenergic alpha1A receptor expressed in CHO cells assessed as calcium mobilization by FLIPR | Bioorg Med Chem Lett 19: 3113-7 (2009) Article DOI: 10.1016/j.bmcl.2009.03.166 BindingDB Entry DOI: 10.7270/Q2WS8T5T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1B adrenergic receptor (Homo sapiens (Human)) | BDBM50258518 ((S)-6-(biphenyl-2-yl)-6,7-dihydro-5H-pyrrolo[1,2-a...) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Agonist activity at human adrenergic alpha1B receptor expressed in CHO cells assessed as calcium mobilization by FLIPR | Bioorg Med Chem Lett 19: 3113-7 (2009) Article DOI: 10.1016/j.bmcl.2009.03.166 BindingDB Entry DOI: 10.7270/Q2WS8T5T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1B adrenergic receptor (Homo sapiens (Human)) | BDBM50258560 ((S)-2-(2-(6,7-dihydro-5H-pyrrolo[1,2-a]imidazol-6-...) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.40E+3 | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Agonist activity at human adrenergic alpha1B receptor expressed in CHO cells assessed as calcium mobilization by FLIPR | Bioorg Med Chem Lett 19: 3113-7 (2009) Article DOI: 10.1016/j.bmcl.2009.03.166 BindingDB Entry DOI: 10.7270/Q2WS8T5T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1A adrenergic receptor (Homo sapiens (Human)) | BDBM50258592 ((S)-2'-(6,7-dihydro-5H-pyrrolo[1,2-a]imidazol-6-yl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 19 | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Agonist activity at human adrenergic alpha1A receptor expressed in CHO cells assessed as calcium mobilization by FLIPR | Bioorg Med Chem Lett 19: 3113-7 (2009) Article DOI: 10.1016/j.bmcl.2009.03.166 BindingDB Entry DOI: 10.7270/Q2WS8T5T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1D adrenergic receptor (Homo sapiens (Human)) | BDBM50258592 ((S)-2'-(6,7-dihydro-5H-pyrrolo[1,2-a]imidazol-6-yl...) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Agonist activity at human adrenergic alpha1D receptor expressed in CHO cells assessed as calcium mobilization by FLIPR | Bioorg Med Chem Lett 19: 3113-7 (2009) Article DOI: 10.1016/j.bmcl.2009.03.166 BindingDB Entry DOI: 10.7270/Q2WS8T5T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1D adrenergic receptor (Homo sapiens (Human)) | BDBM50258638 (6-(2-fluoro-6-(pyrimidin-5-yl)phenyl)-6,7-dihydro-...) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Agonist activity at human adrenergic alpha1D receptor expressed in CHO cells assessed as calcium mobilization by FLIPR | Bioorg Med Chem Lett 19: 3113-7 (2009) Article DOI: 10.1016/j.bmcl.2009.03.166 BindingDB Entry DOI: 10.7270/Q2WS8T5T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1A adrenergic receptor (Homo sapiens (Human)) | BDBM50258639 (2-(2-(6,7-dihydro-5H-pyrrolo[1,2-a]imidazol-6-yl)-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 33 | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Agonist activity at human adrenergic alpha1A receptor expressed in CHO cells assessed as calcium mobilization by FLIPR | Bioorg Med Chem Lett 19: 3113-7 (2009) Article DOI: 10.1016/j.bmcl.2009.03.166 BindingDB Entry DOI: 10.7270/Q2WS8T5T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1B adrenergic receptor (Homo sapiens (Human)) | BDBM50258644 (6-(4-fluoro-2-(1H-pyrazol-1-yl)phenyl)-6,7-dihydro...) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Agonist activity at human adrenergic alpha1B receptor expressed in CHO cells assessed as calcium mobilization by FLIPR | Bioorg Med Chem Lett 19: 3113-7 (2009) Article DOI: 10.1016/j.bmcl.2009.03.166 BindingDB Entry DOI: 10.7270/Q2WS8T5T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1D adrenergic receptor (Homo sapiens (Human)) | BDBM50258644 (6-(4-fluoro-2-(1H-pyrazol-1-yl)phenyl)-6,7-dihydro...) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | >4.10E+3 | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Agonist activity at human adrenergic alpha1D receptor expressed in CHO cells assessed as calcium mobilization by FLIPR | Bioorg Med Chem Lett 19: 3113-7 (2009) Article DOI: 10.1016/j.bmcl.2009.03.166 BindingDB Entry DOI: 10.7270/Q2WS8T5T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1A adrenergic receptor (Homo sapiens (Human)) | BDBM50258565 ((S)-6-(2-(1-methyl-1H-pyrazol-4-yl)phenyl)-6,7-dih...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 9 | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Agonist activity at human adrenergic alpha1A receptor expressed in CHO cells assessed as calcium mobilization by FLIPR | Bioorg Med Chem Lett 19: 3113-7 (2009) Article DOI: 10.1016/j.bmcl.2009.03.166 BindingDB Entry DOI: 10.7270/Q2WS8T5T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1D adrenergic receptor (Homo sapiens (Human)) | BDBM50258518 ((S)-6-(biphenyl-2-yl)-6,7-dihydro-5H-pyrrolo[1,2-a...) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 729 | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Agonist activity at human adrenergic alpha1D receptor expressed in CHO cells assessed as calcium mobilization by FLIPR | Bioorg Med Chem Lett 19: 3113-7 (2009) Article DOI: 10.1016/j.bmcl.2009.03.166 BindingDB Entry DOI: 10.7270/Q2WS8T5T | |||||||||||
More data for this Ligand-Target Pair |