Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Lysophospholipase-like protein 1 (Homo sapiens (Human)) | BDBM195581 ((2R,3R)-2-(3-ethynylphenyl)-1-(3-(4-(2-morpholinop...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 5 | n/a | n/a | n/a | n/a | 7.5 | n/a |
Pfizer Inc. | Assay Description For determination of IC50 values for LYPLAL1 inhibitors, the reactions were carried out in 1.5 mL microcentrifuge tubes in a total reaction volume of... | ACS Chem Biol 11: 2529-40 (2016) Article DOI: 10.1021/acschembio.6b00266 BindingDB Entry DOI: 10.7270/Q24X56K5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Liver carboxylesterase 1 (Homo sapiens (Human)) | BDBM195574 ((R)-(2-phenylpiperidin-1-yl)(3-(4-(pyridin-3-yl)ph...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 5 | n/a | n/a | n/a | n/a | 7.5 | n/a |
Pfizer Inc. | Assay Description For determination of IC50 values for CES1 inhibitors, the reactions were carried out in 1.5 mL microcentrifuge tubes in a total reaction volume of 25... | ACS Chem Biol 11: 2529-40 (2016) Article DOI: 10.1021/acschembio.6b00266 BindingDB Entry DOI: 10.7270/Q24X56K5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Liver carboxylesterase 1 (Homo sapiens (Human)) | BDBM195575 ((R)-(3-(4-(2-morpholinopyrimidin-5-yl)phenyl)-1H-1...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 5 | n/a | n/a | n/a | n/a | 7.5 | n/a |
Pfizer Inc. | Assay Description For determination of IC50 values for CES1 inhibitors, the reactions were carried out in 1.5 mL microcentrifuge tubes in a total reaction volume of 25... | ACS Chem Biol 11: 2529-40 (2016) Article DOI: 10.1021/acschembio.6b00266 BindingDB Entry DOI: 10.7270/Q24X56K5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Liver carboxylesterase 1 (Homo sapiens (Human)) | BDBM195572 ((R)-N,N-dimethyl-4'-(2-(2-phenylpiperidine-1-c...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | <5 | n/a | n/a | n/a | n/a | 7.5 | n/a |
Pfizer Inc. | Assay Description For determination of IC50 values for CES1 inhibitors, the reactions were carried out in 1.5 mL microcentrifuge tubes in a total reaction volume of 25... | ACS Chem Biol 11: 2529-40 (2016) Article DOI: 10.1021/acschembio.6b00266 BindingDB Entry DOI: 10.7270/Q24X56K5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Liver carboxylesterase 1 (Homo sapiens (Human)) | BDBM195571 ((R)-4'-(2-(2-phenylpiperidine-1-carbonyl)-2H-1...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | <5 | n/a | n/a | n/a | n/a | 7.5 | n/a |
Pfizer Inc. | Assay Description For determination of IC50 values for CES1 inhibitors, the reactions were carried out in 1.5 mL microcentrifuge tubes in a total reaction volume of 25... | ACS Chem Biol 11: 2529-40 (2016) Article DOI: 10.1021/acschembio.6b00266 BindingDB Entry DOI: 10.7270/Q24X56K5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Liver carboxylesterase 1 (Homo sapiens (Human)) | BDBM195570 ((S)-4'-(2-(2-phenylpiperidine-1-carbonyl)-2H-1...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | <5 | n/a | n/a | n/a | n/a | 7.5 | n/a |
Pfizer Inc. | Assay Description For determination of IC50 values for CES1 inhibitors, the reactions were carried out in 1.5 mL microcentrifuge tubes in a total reaction volume of 25... | ACS Chem Biol 11: 2529-40 (2016) Article DOI: 10.1021/acschembio.6b00266 BindingDB Entry DOI: 10.7270/Q24X56K5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysophospholipase-like protein 1 (Homo sapiens (Human)) | BDBM195580 ((2R,3R)-1-(3-(4-(2-morpholinopyrimidin-5-yl)phenyl...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | 6 | n/a | n/a | n/a | n/a | 7.5 | n/a |
Pfizer Inc. | Assay Description For determination of IC50 values for LYPLAL1 inhibitors, the reactions were carried out in 1.5 mL microcentrifuge tubes in a total reaction volume of... | ACS Chem Biol 11: 2529-40 (2016) Article DOI: 10.1021/acschembio.6b00266 BindingDB Entry DOI: 10.7270/Q24X56K5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Liver carboxylesterase 1 (Homo sapiens (Human)) | BDBM195573 ((R)-4'-(1-(2-phenylpiperidine-1-carbonyl)-1H-1...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 7 | n/a | n/a | n/a | n/a | 7.5 | n/a |
Pfizer Inc. | Assay Description For determination of IC50 values for CES1 inhibitors, the reactions were carried out in 1.5 mL microcentrifuge tubes in a total reaction volume of 25... | ACS Chem Biol 11: 2529-40 (2016) Article DOI: 10.1021/acschembio.6b00266 BindingDB Entry DOI: 10.7270/Q24X56K5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysophospholipase-like protein 1 (Homo sapiens (Human)) | BDBM195575 ((R)-(3-(4-(2-morpholinopyrimidin-5-yl)phenyl)-1H-1...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 7 | n/a | n/a | n/a | n/a | 7.5 | n/a |
Pfizer Inc. | Assay Description For determination of IC50 values for LYPLAL1 inhibitors, the reactions were carried out in 1.5 mL microcentrifuge tubes in a total reaction volume of... | ACS Chem Biol 11: 2529-40 (2016) Article DOI: 10.1021/acschembio.6b00266 BindingDB Entry DOI: 10.7270/Q24X56K5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysophospholipase-like protein 1 (Homo sapiens (Human)) | BDBM195578 ((2R, 4R)-1-(3-(4-(2-morpholinopyrimidin-5-yl)pheny...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 11 | n/a | n/a | n/a | n/a | 7.5 | n/a |
Pfizer Inc. | Assay Description For determination of IC50 values for LYPLAL1 inhibitors, the reactions were carried out in 1.5 mL microcentrifuge tubes in a total reaction volume of... | ACS Chem Biol 11: 2529-40 (2016) Article DOI: 10.1021/acschembio.6b00266 BindingDB Entry DOI: 10.7270/Q24X56K5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysophospholipase-like protein 1 (Homo sapiens (Human)) | BDBM195572 ((R)-N,N-dimethyl-4'-(2-(2-phenylpiperidine-1-c...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 21 | n/a | n/a | n/a | n/a | 7.5 | n/a |
Pfizer Inc. | Assay Description For determination of IC50 values for LYPLAL1 inhibitors, the reactions were carried out in 1.5 mL microcentrifuge tubes in a total reaction volume of... | ACS Chem Biol 11: 2529-40 (2016) Article DOI: 10.1021/acschembio.6b00266 BindingDB Entry DOI: 10.7270/Q24X56K5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysophospholipase-like protein 1 (Homo sapiens (Human)) | BDBM195574 ((R)-(2-phenylpiperidin-1-yl)(3-(4-(pyridin-3-yl)ph...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 36 | n/a | n/a | n/a | n/a | 7.5 | n/a |
Pfizer Inc. | Assay Description For determination of IC50 values for LYPLAL1 inhibitors, the reactions were carried out in 1.5 mL microcentrifuge tubes in a total reaction volume of... | ACS Chem Biol 11: 2529-40 (2016) Article DOI: 10.1021/acschembio.6b00266 BindingDB Entry DOI: 10.7270/Q24X56K5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysophospholipase-like protein 1 (Homo sapiens (Human)) | BDBM195573 ((R)-4'-(1-(2-phenylpiperidine-1-carbonyl)-1H-1...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 48 | n/a | n/a | n/a | n/a | 7.5 | n/a |
Pfizer Inc. | Assay Description For determination of IC50 values for LYPLAL1 inhibitors, the reactions were carried out in 1.5 mL microcentrifuge tubes in a total reaction volume of... | ACS Chem Biol 11: 2529-40 (2016) Article DOI: 10.1021/acschembio.6b00266 BindingDB Entry DOI: 10.7270/Q24X56K5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysophospholipase-like protein 1 (Homo sapiens (Human)) | BDBM195571 ((R)-4'-(2-(2-phenylpiperidine-1-carbonyl)-2H-1...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 59 | n/a | n/a | n/a | n/a | 7.5 | n/a |
Pfizer Inc. | Assay Description For determination of IC50 values for LYPLAL1 inhibitors, the reactions were carried out in 1.5 mL microcentrifuge tubes in a total reaction volume of... | ACS Chem Biol 11: 2529-40 (2016) Article DOI: 10.1021/acschembio.6b00266 BindingDB Entry DOI: 10.7270/Q24X56K5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysophospholipase-like protein 1 (Homo sapiens (Human)) | BDBM195576 (cis-1-(3-(4-(2-morpholinopyrimidin-5-yl)phenyl)-1H...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 710 | n/a | n/a | n/a | n/a | 7.5 | n/a |
Pfizer Inc. | Assay Description For determination of IC50 values for LYPLAL1 inhibitors, the reactions were carried out in 1.5 mL microcentrifuge tubes in a total reaction volume of... | ACS Chem Biol 11: 2529-40 (2016) Article DOI: 10.1021/acschembio.6b00266 BindingDB Entry DOI: 10.7270/Q24X56K5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysophospholipase-like protein 1 (Homo sapiens (Human)) | BDBM195579 ((2S,3S)-1-(3-(4-(2-morpholinopyrimidin-5-yl)phenyl...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.10E+3 | n/a | n/a | n/a | n/a | 7.5 | n/a |
Pfizer Inc. | Assay Description For determination of IC50 values for LYPLAL1 inhibitors, the reactions were carried out in 1.5 mL microcentrifuge tubes in a total reaction volume of... | ACS Chem Biol 11: 2529-40 (2016) Article DOI: 10.1021/acschembio.6b00266 BindingDB Entry DOI: 10.7270/Q24X56K5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Hexokinase-4 (Rattus norvegicus) | BDBM50444409 (CHEMBL3091581) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.70E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Inc. Curated by ChEMBL | Assay Description Activation of glucokinase in Wistar rat hepatocytes assessed as nuclear to cytosolic translocation of protein by immunofluorescence assay | Bioorg Med Chem Lett 23: 6588-92 (2013) Article DOI: 10.1016/j.bmcl.2013.10.057 BindingDB Entry DOI: 10.7270/Q2QZ2CFX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Liver carboxylesterase 1 (Homo sapiens (Human)) | BDBM195578 ((2R, 4R)-1-(3-(4-(2-morpholinopyrimidin-5-yl)pheny...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.70E+3 | n/a | n/a | n/a | n/a | 7.5 | n/a |
Pfizer Inc. | Assay Description For determination of IC50 values for CES1 inhibitors, the reactions were carried out in 1.5 mL microcentrifuge tubes in a total reaction volume of 25... | ACS Chem Biol 11: 2529-40 (2016) Article DOI: 10.1021/acschembio.6b00266 BindingDB Entry DOI: 10.7270/Q24X56K5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysophospholipase-like protein 1 (Homo sapiens (Human)) | BDBM195577 ((2S,4S)-1-(3-(4-(2-morpholinopyrimidin-5-yl)phenyl...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 6.50E+3 | n/a | n/a | n/a | n/a | 7.5 | n/a |
Pfizer Inc. | Assay Description For determination of IC50 values for LYPLAL1 inhibitors, the reactions were carried out in 1.5 mL microcentrifuge tubes in a total reaction volume of... | ACS Chem Biol 11: 2529-40 (2016) Article DOI: 10.1021/acschembio.6b00266 BindingDB Entry DOI: 10.7270/Q24X56K5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysophospholipase-like protein 1 (Homo sapiens (Human)) | BDBM195570 ((S)-4'-(2-(2-phenylpiperidine-1-carbonyl)-2H-1...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.60E+4 | n/a | n/a | n/a | n/a | 7.5 | n/a |
Pfizer Inc. | Assay Description For determination of IC50 values for LYPLAL1 inhibitors, the reactions were carried out in 1.5 mL microcentrifuge tubes in a total reaction volume of... | ACS Chem Biol 11: 2529-40 (2016) Article DOI: 10.1021/acschembio.6b00266 BindingDB Entry DOI: 10.7270/Q24X56K5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Liver carboxylesterase 1 (Homo sapiens (Human)) | BDBM195577 ((2S,4S)-1-(3-(4-(2-morpholinopyrimidin-5-yl)phenyl...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.90E+4 | n/a | n/a | n/a | n/a | 7.5 | n/a |
Pfizer Inc. | Assay Description For determination of IC50 values for CES1 inhibitors, the reactions were carried out in 1.5 mL microcentrifuge tubes in a total reaction volume of 25... | ACS Chem Biol 11: 2529-40 (2016) Article DOI: 10.1021/acschembio.6b00266 BindingDB Entry DOI: 10.7270/Q24X56K5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Liver carboxylesterase 1 (Homo sapiens (Human)) | BDBM195579 ((2S,3S)-1-(3-(4-(2-morpholinopyrimidin-5-yl)phenyl...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2.90E+4 | n/a | n/a | n/a | n/a | 7.5 | n/a |
Pfizer Inc. | Assay Description For determination of IC50 values for CES1 inhibitors, the reactions were carried out in 1.5 mL microcentrifuge tubes in a total reaction volume of 25... | ACS Chem Biol 11: 2529-40 (2016) Article DOI: 10.1021/acschembio.6b00266 BindingDB Entry DOI: 10.7270/Q24X56K5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Liver carboxylesterase 1 (Homo sapiens (Human)) | BDBM195576 (cis-1-(3-(4-(2-morpholinopyrimidin-5-yl)phenyl)-1H...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.60E+4 | n/a | n/a | n/a | n/a | 7.5 | n/a |
Pfizer Inc. | Assay Description For determination of IC50 values for CES1 inhibitors, the reactions were carried out in 1.5 mL microcentrifuge tubes in a total reaction volume of 25... | ACS Chem Biol 11: 2529-40 (2016) Article DOI: 10.1021/acschembio.6b00266 BindingDB Entry DOI: 10.7270/Q24X56K5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Liver carboxylesterase 1 (Homo sapiens (Human)) | BDBM195581 ((2R,3R)-2-(3-ethynylphenyl)-1-(3-(4-(2-morpholinop...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >5.00E+4 | n/a | n/a | n/a | n/a | 7.5 | n/a |
Pfizer Inc. | Assay Description For determination of IC50 values for CES1 inhibitors, the reactions were carried out in 1.5 mL microcentrifuge tubes in a total reaction volume of 25... | ACS Chem Biol 11: 2529-40 (2016) Article DOI: 10.1021/acschembio.6b00266 BindingDB Entry DOI: 10.7270/Q24X56K5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Liver carboxylesterase 1 (Homo sapiens (Human)) | BDBM195580 ((2R,3R)-1-(3-(4-(2-morpholinopyrimidin-5-yl)phenyl...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | >5.00E+4 | n/a | n/a | n/a | n/a | 7.5 | n/a |
Pfizer Inc. | Assay Description For determination of IC50 values for CES1 inhibitors, the reactions were carried out in 1.5 mL microcentrifuge tubes in a total reaction volume of 25... | ACS Chem Biol 11: 2529-40 (2016) Article DOI: 10.1021/acschembio.6b00266 BindingDB Entry DOI: 10.7270/Q24X56K5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Hexokinase-4 (Rattus norvegicus) | BDBM50444410 (CHEMBL3091580) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 2.60E+4 | n/a | n/a | n/a | n/a |
Pfizer Inc. Curated by ChEMBL | Assay Description Activation of glucokinase in rat INS-1 cells assessed as glucose-stimulated insulin secretion | Bioorg Med Chem Lett 23: 6588-92 (2013) Article DOI: 10.1016/j.bmcl.2013.10.057 BindingDB Entry DOI: 10.7270/Q2QZ2CFX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Hexokinase-4 (Homo sapiens (Human)) | BDBM50444411 (CHEMBL3091585) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a |
Pfizer Inc. Curated by ChEMBL | Assay Description Activation of recombinant human glucokinase by G6PDH/NADP coupled assay | Bioorg Med Chem Lett 23: 6588-92 (2013) Article DOI: 10.1016/j.bmcl.2013.10.057 BindingDB Entry DOI: 10.7270/Q2QZ2CFX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Hexokinase-4 (Homo sapiens (Human)) | BDBM50444412 (CHEMBL3091584) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.35E+3 | n/a | n/a | n/a | n/a |
Pfizer Inc. Curated by ChEMBL | Assay Description Activation of recombinant human glucokinase by G6PDH/NADP coupled assay | Bioorg Med Chem Lett 23: 6588-92 (2013) Article DOI: 10.1016/j.bmcl.2013.10.057 BindingDB Entry DOI: 10.7270/Q2QZ2CFX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Hexokinase-4 (Homo sapiens (Human)) | BDBM50444413 (CHEMBL3091583) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 227 | n/a | n/a | n/a | n/a |
Pfizer Inc. Curated by ChEMBL | Assay Description Activation of recombinant human glucokinase by G6PDH/NADP coupled assay | Bioorg Med Chem Lett 23: 6588-92 (2013) Article DOI: 10.1016/j.bmcl.2013.10.057 BindingDB Entry DOI: 10.7270/Q2QZ2CFX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Hexokinase-4 (Homo sapiens (Human)) | BDBM50444414 (CHEMBL3091582) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 113 | n/a | n/a | n/a | n/a |
Pfizer Inc. Curated by ChEMBL | Assay Description Activation of recombinant human glucokinase by G6PDH/NADP coupled assay | Bioorg Med Chem Lett 23: 6588-92 (2013) Article DOI: 10.1016/j.bmcl.2013.10.057 BindingDB Entry DOI: 10.7270/Q2QZ2CFX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Hexokinase-4 (Homo sapiens (Human)) | BDBM50444409 (CHEMBL3091581) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 201 | n/a | n/a | n/a | n/a |
Pfizer Inc. Curated by ChEMBL | Assay Description Activation of recombinant human glucokinase by G6PDH/NADP coupled assay | Bioorg Med Chem Lett 23: 6588-92 (2013) Article DOI: 10.1016/j.bmcl.2013.10.057 BindingDB Entry DOI: 10.7270/Q2QZ2CFX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Hexokinase-4 (Homo sapiens (Human)) | BDBM50444410 (CHEMBL3091580) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 137 | n/a | n/a | n/a | n/a |
Pfizer Inc. Curated by ChEMBL | Assay Description Activation of recombinant human glucokinase by G6PDH/NADP coupled assay | Bioorg Med Chem Lett 23: 6588-92 (2013) Article DOI: 10.1016/j.bmcl.2013.10.057 BindingDB Entry DOI: 10.7270/Q2QZ2CFX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Hexokinase-4 (Rattus norvegicus) | BDBM50444409 (CHEMBL3091581) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.74E+5 | n/a | n/a | n/a | n/a |
Pfizer Inc. Curated by ChEMBL | Assay Description Activation of glucokinase in rat INS-1 cells assessed as glucose-stimulated insulin secretion | Bioorg Med Chem Lett 23: 6588-92 (2013) Article DOI: 10.1016/j.bmcl.2013.10.057 BindingDB Entry DOI: 10.7270/Q2QZ2CFX | |||||||||||
More data for this Ligand-Target Pair |