Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
B2 bradykinin receptor (RAT) | BDBM50370083 (CHEMBL1907651) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 0.0230 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Novartis Institute for Medical Sciences Curated by ChEMBL | Assay Description Inhibition of specific binding of [3H]-BK (1 nM) to rat Bradykinin receptor B2 by 50% in NG108-15 cell membranes | J Med Chem 45: 2160-72 (2002) BindingDB Entry DOI: 10.7270/Q2X067SG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (RAT) | BDBM50370077 (CHEMBL1907652) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 0.310 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Novartis Institute for Medical Sciences Curated by ChEMBL | Assay Description Inhibition of specific binding of [3H]-BK (1 nM) to rat Bradykinin receptor B2 by 50% in NG108-15 cell membranes | J Med Chem 45: 2160-72 (2002) BindingDB Entry DOI: 10.7270/Q2X067SG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (RAT) | BDBM50113263 ((S)-1-[4-(4-benzhydrylthiosemicarbazido)-3-nitrobe...) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | 0.5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Novartis Institute for Medical Sciences Curated by ChEMBL | Assay Description Inhibition of specific binding of [3H]-BK (1 nM) to rat Bradykinin receptor B2 by 50% in NG108-15 cell membranes | J Med Chem 45: 2160-72 (2002) BindingDB Entry DOI: 10.7270/Q2X067SG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (RAT) | BDBM50409120 (CHEMBL2112044 | CHEMBL2112937) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 0.5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Novartis Institute for Medical Sciences Curated by ChEMBL | Assay Description Inhibition of binding of [3H]-BK to rat bradykinin B2 receptor expressed in NG108-15 neuroblastoma-glioma hybrid cell membranes | J Med Chem 43: 769-71 (2000) BindingDB Entry DOI: 10.7270/Q2XD10W5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (RAT) | BDBM50113263 ((S)-1-[4-(4-benzhydrylthiosemicarbazido)-3-nitrobe...) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | 0.600 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Novartis Institute for Medical Sciences Curated by ChEMBL | Assay Description Inhibition of specific binding of [3H]-BK (1 nM) to rat Bradykinin receptor B2 by 50% in NG108-15 cell membranes | J Med Chem 45: 2160-72 (2002) BindingDB Entry DOI: 10.7270/Q2X067SG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (RAT) | BDBM50409120 (CHEMBL2112044 | CHEMBL2112937) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 0.600 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Novartis Institute for Medical Sciences Curated by ChEMBL | Assay Description Inhibition of binding of [3H]-BK to rat bradykinin B2 receptor expressed in NG108-15 neuroblastoma-glioma hybrid cell membranes | J Med Chem 43: 769-71 (2000) BindingDB Entry DOI: 10.7270/Q2XD10W5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50409527 (CHEMBL2112283) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 0.790 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Novartis Institute for Medical Sciences Curated by ChEMBL | Assay Description Displacement of [3H]BK (1 nM) from human Bradykinin receptor B2 expressed in Cos-7 cells | J Med Chem 45: 2160-72 (2002) BindingDB Entry DOI: 10.7270/Q2X067SG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B1 bradykinin receptor (Homo sapiens (Human)) | BDBM50151885 (1-[4-(2,2-Diphenyl-ethylamino)-3-(morpholine-4-car...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Binding affinity for Bradykinin receptor B1 expressed in HEK293 cells | J Med Chem 47: 4642-4 (2004) Article DOI: 10.1021/jm049747g BindingDB Entry DOI: 10.7270/Q2J965V7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50409529 (CHEMBL2112221) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 1.47 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Novartis Institute for Medical Sciences Curated by ChEMBL | Assay Description Displacement of [3H]BK (1 nM) from human Bradykinin receptor B2 expressed in Cos-7 cells | J Med Chem 45: 2160-72 (2002) BindingDB Entry DOI: 10.7270/Q2X067SG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (RAT) | BDBM50085685 (4-benzhydrylamino(thioxo)methylhydrazine-3-nitrobe...) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | PubMed | 1.80 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Novartis Institute for Medical Sciences Curated by ChEMBL | Assay Description Inhibition of binding of [3H]-BK to rat bradykinin B2 receptor expressed in NG108-15 neuroblastoma-glioma hybrid cell membranes | J Med Chem 43: 769-71 (2000) BindingDB Entry DOI: 10.7270/Q2XD10W5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50409528 (CHEMBL2112220) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 2.79 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Novartis Institute for Medical Sciences Curated by ChEMBL | Assay Description Displacement of [3H]BK (1 nM) from human Bradykinin receptor B2 expressed in Cos-7 cells | J Med Chem 45: 2160-72 (2002) BindingDB Entry DOI: 10.7270/Q2X067SG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (RAT) | BDBM50085684 (4-benzhydrylamino(thioxo)methylhydrazine-3-nitro-1...) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Novartis Institute for Medical Sciences Curated by ChEMBL | Assay Description Inhibition of binding of [3H]-BK to rat bradykinin B2 receptor expressed in NG108-15 neuroblastoma-glioma hybrid cell membranes | J Med Chem 43: 769-71 (2000) BindingDB Entry DOI: 10.7270/Q2XD10W5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50370080 (CHEMBL1907656) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 4.67 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Novartis Institute for Medical Sciences Curated by ChEMBL | Assay Description Displacement of [3H]BK (1 nM) from human Bradykinin receptor B2 expressed in Cos-7 cells | J Med Chem 45: 2160-72 (2002) BindingDB Entry DOI: 10.7270/Q2X067SG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (RAT) | BDBM50370081 (CHEMBL1907654) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 5.46 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Novartis Institute for Medical Sciences Curated by ChEMBL | Assay Description Inhibition of specific binding of [3H]-BK (1 nM) to rat Bradykinin receptor B2 by 50% in NG108-15 cell membranes | J Med Chem 45: 2160-72 (2002) BindingDB Entry DOI: 10.7270/Q2X067SG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (RAT) | BDBM50370078 (CHEMBL1907653) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 7.30 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Novartis Institute for Medical Sciences Curated by ChEMBL | Assay Description Inhibition of specific binding of [3H]-BK (1 nM) to rat Bradykinin receptor B2 by 50% in NG108-15 cell membranes | J Med Chem 45: 2160-72 (2002) BindingDB Entry DOI: 10.7270/Q2X067SG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B1 bradykinin receptor (Homo sapiens (Human)) | BDBM50151884 (CHEMBL185551 | N,N-Bis-(3-dimethylamino-propyl)-3-...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Binding affinity for Bradykinin receptor B1 expressed in HEK293 cells | J Med Chem 47: 4642-4 (2004) Article DOI: 10.1021/jm049747g BindingDB Entry DOI: 10.7270/Q2J965V7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B1 bradykinin receptor (Homo sapiens (Human)) | BDBM50151886 (CHEMBL181695 | {2-(2,2-Diphenyl-ethylamino)-5-[4-(...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Binding affinity for Bradykinin receptor B1 expressed in HEK293 cells | J Med Chem 47: 4642-4 (2004) Article DOI: 10.1021/jm049747g BindingDB Entry DOI: 10.7270/Q2J965V7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B1 bradykinin receptor (Homo sapiens (Human)) | BDBM50151891 (CHEMBL273869 | {2-(2,2-Diphenyl-ethylamino)-5-[4-(...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Binding affinity for Bradykinin receptor B1 expressed in HEK293 cells | J Med Chem 47: 4642-4 (2004) Article DOI: 10.1021/jm049747g BindingDB Entry DOI: 10.7270/Q2J965V7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B1 bradykinin receptor (Homo sapiens (Human)) | BDBM50151894 (1-[4-(2,2-Diphenyl-ethylamino)-3-nitro-benzenesulf...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Binding affinity for Bradykinin receptor B1 expressed in HEK293 cells | J Med Chem 47: 4642-4 (2004) Article DOI: 10.1021/jm049747g BindingDB Entry DOI: 10.7270/Q2J965V7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (RAT) | BDBM50409527 (CHEMBL2112283) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 10.7 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Novartis Institute for Medical Sciences Curated by ChEMBL | Assay Description Inhibition of specific binding of [3H]-BK (1 nM) to rat Bradykinin receptor B2 by 50% in NG108-15 cell membranes | J Med Chem 45: 2160-72 (2002) BindingDB Entry DOI: 10.7270/Q2X067SG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (RAT) | BDBM50370080 (CHEMBL1907656) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 14.5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Novartis Institute for Medical Sciences Curated by ChEMBL | Assay Description Inhibition of specific binding of [3H]-BK (1 nM) to rat Bradykinin receptor B2 by 50% in NG108-15 cell membranes | J Med Chem 45: 2160-72 (2002) BindingDB Entry DOI: 10.7270/Q2X067SG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50370081 (CHEMBL1907654) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 34.1 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Novartis Institute for Medical Sciences Curated by ChEMBL | Assay Description Displacement of [3H]BK (1 nM) from human Bradykinin receptor B2 expressed in Cos-7 cells | J Med Chem 45: 2160-72 (2002) BindingDB Entry DOI: 10.7270/Q2X067SG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (RAT) | BDBM50085698 (CHEMBL164636 | benzhydrylamino-2-nitrobenzylhydraz...) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 38 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Novartis Institute for Medical Sciences Curated by ChEMBL | Assay Description Inhibition of binding of [3H]-BK to rat bradykinin B2 receptor expressed in NG108-15 neuroblastoma-glioma hybrid cell membranes | J Med Chem 43: 769-71 (2000) BindingDB Entry DOI: 10.7270/Q2XD10W5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (RAT) | BDBM50409529 (CHEMBL2112221) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 64.5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Novartis Institute for Medical Sciences Curated by ChEMBL | Assay Description Inhibition of specific binding of [3H]-BK (1 nM) to rat Bradykinin receptor B2 by 50% in NG108-15 cell membranes | J Med Chem 45: 2160-72 (2002) BindingDB Entry DOI: 10.7270/Q2X067SG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50370077 (CHEMBL1907652) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 95 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Novartis Institute for Medical Sciences Curated by ChEMBL | Assay Description Displacement of [3H]BK (1 nM) from human Bradykinin receptor B2 expressed in Cos-7 cells | J Med Chem 45: 2160-72 (2002) BindingDB Entry DOI: 10.7270/Q2X067SG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50370083 (CHEMBL1907651) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 119 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Novartis Institute for Medical Sciences Curated by ChEMBL | Assay Description Displacement of [3H]BK (1 nM) from human Bradykinin receptor B2 expressed in Cos-7 cells | J Med Chem 45: 2160-72 (2002) BindingDB Entry DOI: 10.7270/Q2X067SG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B1 bradykinin receptor (Homo sapiens (Human)) | BDBM50151888 (3-[3-Acetyl-4-(2,2-diphenyl-ethylamino)-benzenesul...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | 130 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Binding affinity for Bradykinin receptor B1 expressed in HEK293 cells | J Med Chem 47: 4642-4 (2004) Article DOI: 10.1021/jm049747g BindingDB Entry DOI: 10.7270/Q2J965V7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B1 bradykinin receptor (Homo sapiens (Human)) | BDBM50151889 (CHEMBL180143 | N,N-Bis-(3-dimethylamino-propyl)-3-...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 140 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Binding affinity for Bradykinin receptor B1 expressed in HEK293 cells | J Med Chem 47: 4642-4 (2004) Article DOI: 10.1021/jm049747g BindingDB Entry DOI: 10.7270/Q2J965V7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (RAT) | BDBM50085696 (1N,1N-di(3-dimethylaminopropyl)-4-benzhydrylamino(...) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 148 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Novartis Institute for Medical Sciences Curated by ChEMBL | Assay Description Inhibition of binding of [3H]-BK to rat bradykinin B2 receptor expressed in NG108-15 neuroblastoma-glioma hybrid cell membranes | J Med Chem 43: 769-71 (2000) BindingDB Entry DOI: 10.7270/Q2XD10W5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (RAT) | BDBM50409528 (CHEMBL2112220) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 176 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Novartis Institute for Medical Sciences Curated by ChEMBL | Assay Description Inhibition of specific binding of [3H]-BK (1 nM) to rat Bradykinin receptor B2 by 50% in NG108-15 cell membranes | J Med Chem 45: 2160-72 (2002) BindingDB Entry DOI: 10.7270/Q2X067SG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B1 bradykinin receptor (Homo sapiens (Human)) | BDBM50151890 (CHEMBL181098 | N,N-Bis-(3-dimethylamino-propyl)-4-...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 230 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Binding affinity for Bradykinin receptor B1 expressed in HEK293 cells | J Med Chem 47: 4642-4 (2004) Article DOI: 10.1021/jm049747g BindingDB Entry DOI: 10.7270/Q2J965V7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50113264 (1-[4-(4-benzhydrylthiosemicarbazido)-3-nitrobenzen...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 237 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Novartis Institute for Medical Sciences Curated by ChEMBL | Assay Description Displacement of [3H]BK (1 nM) from human Bradykinin receptor B2 expressed in Cos-7 cells | J Med Chem 45: 2160-72 (2002) BindingDB Entry DOI: 10.7270/Q2X067SG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B1 bradykinin receptor (Homo sapiens (Human)) | BDBM50151893 (4-(1-Benzyl-2-phenyl-ethylamino)-N,N-bis-(3-dimeth...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 250 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Binding affinity for Bradykinin receptor B1 expressed in HEK293 cells | J Med Chem 47: 4642-4 (2004) Article DOI: 10.1021/jm049747g BindingDB Entry DOI: 10.7270/Q2J965V7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50409530 (CHEMBL2112219) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 253 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Novartis Institute for Medical Sciences Curated by ChEMBL | Assay Description Displacement of [3H]BK (1 nM) from human Bradykinin receptor B2 expressed in Cos-7 cells | J Med Chem 45: 2160-72 (2002) BindingDB Entry DOI: 10.7270/Q2X067SG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50370082 (CHEMBL1907655) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 299 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Novartis Institute for Medical Sciences Curated by ChEMBL | Assay Description Displacement of [3H]BK (1 nM) from human Bradykinin receptor B2 expressed in Cos-7 cells | J Med Chem 45: 2160-72 (2002) BindingDB Entry DOI: 10.7270/Q2X067SG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (RAT) | BDBM50085689 (1N-benzyl-4-benzylamino(thioxo)methylhydrazine-3-n...) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 310 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Novartis Institute for Medical Sciences Curated by ChEMBL | Assay Description Inhibition of binding of [3H]-BK to rat bradykinin B2 receptor expressed in NG108-15 neuroblastoma-glioma hybrid cell membranes | J Med Chem 43: 769-71 (2000) BindingDB Entry DOI: 10.7270/Q2XD10W5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (RAT) | BDBM50085692 (2-{4-[2-furylmethylamino(thioxo)methylhydrazine]-3...) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | PubMed | 540 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Novartis Institute for Medical Sciences Curated by ChEMBL | Assay Description Inhibition of binding of [3H]-BK to rat bradykinin B2 receptor expressed in NG108-15 neuroblastoma-glioma hybrid cell membranes | J Med Chem 43: 769-71 (2000) BindingDB Entry DOI: 10.7270/Q2XD10W5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50370084 (CHEMBL1907657) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 645 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Novartis Institute for Medical Sciences Curated by ChEMBL | Assay Description Displacement of [3H]BK (1 nM) from human Bradykinin receptor B2 expressed in Cos-7 cells | J Med Chem 45: 2160-72 (2002) BindingDB Entry DOI: 10.7270/Q2X067SG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (RAT) | BDBM50370082 (CHEMBL1907655) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 654 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Novartis Institute for Medical Sciences Curated by ChEMBL | Assay Description Inhibition of specific binding of [3H]-BK (1 nM) to rat Bradykinin receptor B2 by 50% in NG108-15 cell membranes | J Med Chem 45: 2160-72 (2002) BindingDB Entry DOI: 10.7270/Q2X067SG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50113263 ((S)-1-[4-(4-benzhydrylthiosemicarbazido)-3-nitrobe...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | 772 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Novartis Institute for Medical Sciences Curated by ChEMBL | Assay Description Displacement of [3H]BK (1 nM) from human Bradykinin receptor B2 expressed in Cos-7 cells | J Med Chem 45: 2160-72 (2002) BindingDB Entry DOI: 10.7270/Q2X067SG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B1 bradykinin receptor (Homo sapiens (Human)) | BDBM50151892 (3-[3-Chloro-4-(2,2-diphenyl-ethylamino)-benzenesul...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | >1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Binding affinity for Bradykinin receptor B1 expressed in HEK293 cells | J Med Chem 47: 4642-4 (2004) Article DOI: 10.1021/jm049747g BindingDB Entry DOI: 10.7270/Q2J965V7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50151887 (4-(Benzhydryl-amino)-N,N-bis-(3-dimethylamino-prop...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Binding affinity for Bradykinin receptor B2 expressed in COS7 cells | J Med Chem 47: 4642-4 (2004) Article DOI: 10.1021/jm049747g BindingDB Entry DOI: 10.7270/Q2J965V7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50113263 ((S)-1-[4-(4-benzhydrylthiosemicarbazido)-3-nitrobe...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | 1.43E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Novartis Institute for Medical Sciences Curated by ChEMBL | Assay Description Displacement of [3H]BK (1 nM) from human Bradykinin receptor B2 expressed in Cos-7 cells | J Med Chem 45: 2160-72 (2002) BindingDB Entry DOI: 10.7270/Q2X067SG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (RAT) | BDBM50085694 (CHEMBL163956 | benzylamino-2-nitrobenzylhydrazinem...) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 1.60E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Novartis Institute for Medical Sciences Curated by ChEMBL | Assay Description Inhibition of binding of [3H]-BK to rat bradykinin B2 receptor expressed in NG108-15 neuroblastoma-glioma hybrid cell membranes | J Med Chem 43: 769-71 (2000) BindingDB Entry DOI: 10.7270/Q2XD10W5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A1 (Homo sapiens (Human)) | BDBM50207120 (3-isobutyl-8-((6-methoxyisoquinolin-4-yl)methyl)-1...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Novartis Institutes of Biomedical Research Curated by ChEMBL | Assay Description Inhibition of adenosine A1 receptor | Bioorg Med Chem Lett 17: 2376-9 (2007) Article DOI: 10.1016/j.bmcl.2006.11.019 BindingDB Entry DOI: 10.7270/Q2X63NSC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B1 bradykinin receptor (Homo sapiens (Human)) | BDBM50151887 (4-(Benzhydryl-amino)-N,N-bis-(3-dimethylamino-prop...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 3.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Binding affinity for Bradykinin receptor B1 expressed in HEK293 cells | J Med Chem 47: 4642-4 (2004) Article DOI: 10.1021/jm049747g BindingDB Entry DOI: 10.7270/Q2J965V7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (RAT) | BDBM50085690 (1-Benzyl-3-(2-nitro-benzyl)-thiourea | CHEMBL16524...) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | PubMed | 7.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Novartis Institute for Medical Sciences Curated by ChEMBL | Assay Description Inhibition of binding of [3H]-BK to rat bradykinin B2 receptor expressed in NG108-15 neuroblastoma-glioma hybrid cell membranes | J Med Chem 43: 769-71 (2000) BindingDB Entry DOI: 10.7270/Q2XD10W5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50075189 (CHEMBL142260 | N-[3-(3-Benzyl-2-oxo-5-phenyl-2,3-d...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 8.90E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Novartis Institute for Medical Sciences Curated by ChEMBL | Assay Description Binding affinity towards human bradykinin B2 receptor (membranes from Cos-7 cells expressing human B2 receptor) using [3H]-BK as radioligand | Bioorg Med Chem Lett 9: 463-8 (1999) BindingDB Entry DOI: 10.7270/Q2PV6JJH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50075187 (CHEMBL442294 | N-[4-(3-Benzyl-2-oxo-5-phenyl-2,3-d...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 9.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Novartis Institute for Medical Sciences Curated by ChEMBL | Assay Description Binding affinity towards human bradykinin B2 receptor (membranes from Cos-7 cells expressing human B2 receptor) using [3H]-BK as radioligand | Bioorg Med Chem Lett 9: 463-8 (1999) BindingDB Entry DOI: 10.7270/Q2PV6JJH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50403721 (CHEMBL2111994) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 1.19E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Novartis Institute for Medical Sciences Curated by ChEMBL | Assay Description Binding affinity towards human bradykinin B2 receptor (membranes from Cos-7 cells expressing human B2 receptor) using [3H]-BK as radioligand | Bioorg Med Chem Lett 9: 463-8 (1999) BindingDB Entry DOI: 10.7270/Q2PV6JJH | |||||||||||
More data for this Ligand-Target Pair |
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