Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Lutropin-choriogonadotropic hormone receptor (Homo sapiens (Human)) | BDBM50335467 (5-amino-N-tert-butyl-2-(methylthio)-4-(3-(2-oxo-2-...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1 | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Agonist activity at human LH receptor expressed in CHO-K1 cells assessed as stimulation of luciferase activity by CRE-driven luciferase reporter gene... | ACS Med Chem Lett 2: 85-89 (2011) Article DOI: 10.1021/ml100229v BindingDB Entry DOI: 10.7270/Q2RV0NZG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lutropin-choriogonadotropic hormone receptor (Homo sapiens (Human)) | BDBM50335473 (5-amino-4-(3-(2-((1-(2-(2-(2-azidoethoxy)ethoxy)et...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 5 | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Agonist activity at human LH receptor expressed in CHO-K1 cells assessed as stimulation of luciferase activity by CRE-driven luciferase reporter gene... | ACS Med Chem Lett 2: 85-89 (2011) Article DOI: 10.1021/ml100229v BindingDB Entry DOI: 10.7270/Q2RV0NZG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lutropin-choriogonadotropic hormone receptor (Homo sapiens (Human)) | BDBM50335468 ((R)-4-(3-(2-((1-(2-(4-((4-(1-acetyl-6-biphenyl-4-y...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 10 | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Agonist activity at human LH receptor expressed in CHO-K1 cells assessed as stimulation of luciferase activity by CRE-driven luciferase reporter gene... | ACS Med Chem Lett 2: 85-89 (2011) Article DOI: 10.1021/ml100229v BindingDB Entry DOI: 10.7270/Q2RV0NZG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lutropin-choriogonadotropic hormone receptor (Homo sapiens (Human)) | BDBM50206401 (CHEMBL246321 | N-((S)-1-amino-3-(4-hydroxyphenyl)-...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 20 | n/a | n/a | n/a | n/a |
Merck Serono Geneva Research Center Curated by ChEMBL | Assay Description Agonist activity at human LH receptor expressed in CHO cells assessed as production of cAMP after 60 mins by SPA | Bioorg Med Chem Lett 17: 2080-5 (2007) Article DOI: 10.1016/j.bmcl.2006.12.062 BindingDB Entry DOI: 10.7270/Q2VQ32B2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lutropin-choriogonadotropic hormone receptor (Homo sapiens (Human)) | BDBM50335474 ((S)-4-(3-(2-((1-(2-(4-((4-(1-acetyl-6-biphenyl-4-y...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 24 | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Agonist activity at human LH receptor expressed in CHO-K1 cells assessed as stimulation of luciferase activity by CRE-driven luciferase reporter gene... | ACS Med Chem Lett 2: 85-89 (2011) Article DOI: 10.1021/ml100229v BindingDB Entry DOI: 10.7270/Q2RV0NZG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lutropin-choriogonadotropic hormone receptor (Homo sapiens (Human)) | BDBM50335469 ((R)-4-(3-(2-((1-(2-(2-(4-((4-(1-acetyl-6-biphenyl-...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 27 | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Agonist activity at human LH receptor expressed in CHO-K1 cells assessed as stimulation of luciferase activity by CRE-driven luciferase reporter gene... | ACS Med Chem Lett 2: 85-89 (2011) Article DOI: 10.1021/ml100229v BindingDB Entry DOI: 10.7270/Q2RV0NZG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lutropin-choriogonadotropic hormone receptor (Homo sapiens (Human)) | BDBM50335478 ((S)-4-(3-(2-((1-(14-(4-((4-(1-acetyl-6-biphenyl-4-...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 39 | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Agonist activity at human LH receptor expressed in CHO-K1 cells assessed as stimulation of luciferase activity by CRE-driven luciferase reporter gene... | ACS Med Chem Lett 2: 85-89 (2011) Article DOI: 10.1021/ml100229v BindingDB Entry DOI: 10.7270/Q2RV0NZG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lutropin-choriogonadotropic hormone receptor (Homo sapiens (Human)) | BDBM50335470 ((R)-4-(3-(2-((1-(2-(2-(2-(4-((4-(1-acetyl-6-biphen...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 43 | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Agonist activity at human LH receptor expressed in CHO-K1 cells assessed as stimulation of luciferase activity by CRE-driven luciferase reporter gene... | ACS Med Chem Lett 2: 85-89 (2011) Article DOI: 10.1021/ml100229v BindingDB Entry DOI: 10.7270/Q2RV0NZG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lutropin-choriogonadotropic hormone receptor (Homo sapiens (Human)) | BDBM50335472 ((R)-4-(3-(2-((1-(14-(4-((4-(1-acetyl-6-biphenyl-4-...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 55 | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Agonist activity at human LH receptor expressed in CHO-K1 cells assessed as stimulation of luciferase activity by CRE-driven luciferase reporter gene... | ACS Med Chem Lett 2: 85-89 (2011) Article DOI: 10.1021/ml100229v BindingDB Entry DOI: 10.7270/Q2RV0NZG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lutropin-choriogonadotropic hormone receptor (Homo sapiens (Human)) | BDBM50335477 ((S)-4-(3-(2-((1-(2-(2-(2-(2-(4-((4-(1-acetyl-6-bip...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 57 | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Agonist activity at human LH receptor expressed in CHO-K1 cells assessed as stimulation of luciferase activity by CRE-driven luciferase reporter gene... | ACS Med Chem Lett 2: 85-89 (2011) Article DOI: 10.1021/ml100229v BindingDB Entry DOI: 10.7270/Q2RV0NZG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lutropin-choriogonadotropic hormone receptor (Homo sapiens (Human)) | BDBM50335471 ((R)-4-(3-(2-((1-(2-(2-(2-(2-(4-((4-(1-acetyl-6-bip...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 61 | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Agonist activity at human LH receptor expressed in CHO-K1 cells assessed as stimulation of luciferase activity by CRE-driven luciferase reporter gene... | ACS Med Chem Lett 2: 85-89 (2011) Article DOI: 10.1021/ml100229v BindingDB Entry DOI: 10.7270/Q2RV0NZG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lutropin-choriogonadotropic hormone receptor (Homo sapiens (Human)) | BDBM50335476 ((S)-4-(3-(2-((1-(2-(2-(2-(4-((4-(1-acetyl-6-biphen...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 75 | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Agonist activity at human LH receptor expressed in CHO-K1 cells assessed as stimulation of luciferase activity by CRE-driven luciferase reporter gene... | ACS Med Chem Lett 2: 85-89 (2011) Article DOI: 10.1021/ml100229v BindingDB Entry DOI: 10.7270/Q2RV0NZG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lutropin-choriogonadotropic hormone receptor (Homo sapiens (Human)) | BDBM50335475 ((S)-4-(3-(2-((1-(2-(2-(4-((4-(1-acetyl-6-biphenyl-...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 80 | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Agonist activity at human LH receptor expressed in CHO-K1 cells assessed as stimulation of luciferase activity by CRE-driven luciferase reporter gene... | ACS Med Chem Lett 2: 85-89 (2011) Article DOI: 10.1021/ml100229v BindingDB Entry DOI: 10.7270/Q2RV0NZG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lutropin-choriogonadotropic hormone receptor (Homo sapiens (Human)) | BDBM50206398 (CHEMBL429108 | N-(4-hydroxyphenethyl)-5-(1-(4-tert...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 80 | n/a | n/a | n/a | n/a |
Merck Serono Geneva Research Center Curated by ChEMBL | Assay Description Agonist activity at human LH receptor expressed in CHO cells assessed as production of cAMP after 60 mins by SPA | Bioorg Med Chem Lett 17: 2080-5 (2007) Article DOI: 10.1016/j.bmcl.2006.12.062 BindingDB Entry DOI: 10.7270/Q2VQ32B2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lutropin-choriogonadotropic hormone receptor (Homo sapiens (Human)) | BDBM50206402 (CHEMBL439392 | N-((S)-1-amino-3-(3-hydroxyphenyl)-...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 150 | n/a | n/a | n/a | n/a |
Merck Serono Geneva Research Center Curated by ChEMBL | Assay Description Agonist activity at human LH receptor expressed in CHO cells assessed as production of cAMP after 60 mins by SPA | Bioorg Med Chem Lett 17: 2080-5 (2007) Article DOI: 10.1016/j.bmcl.2006.12.062 BindingDB Entry DOI: 10.7270/Q2VQ32B2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lutropin-choriogonadotropic hormone receptor (Homo sapiens (Human)) | BDBM50206399 (CHEMBL247700 | N-((S)-2-amino-1-(4-hydroxyphenyl)-...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 170 | n/a | n/a | n/a | n/a |
Merck Serono Geneva Research Center Curated by ChEMBL | Assay Description Agonist activity at human LH receptor expressed in CHO cells assessed as production of cAMP after 60 mins by SPA | Bioorg Med Chem Lett 17: 2080-5 (2007) Article DOI: 10.1016/j.bmcl.2006.12.062 BindingDB Entry DOI: 10.7270/Q2VQ32B2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lutropin-choriogonadotropic hormone receptor (Homo sapiens (Human)) | BDBM50206397 ((S)-N-(4-amino-4-oxo-1-phenylbutan-2-yl)-5-(1-(4-t...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 190 | n/a | n/a | n/a | n/a |
Merck Serono Geneva Research Center Curated by ChEMBL | Assay Description Agonist activity at human LH receptor expressed in CHO cells assessed as production of cAMP after 60 mins by SPA | Bioorg Med Chem Lett 17: 2080-5 (2007) Article DOI: 10.1016/j.bmcl.2006.12.062 BindingDB Entry DOI: 10.7270/Q2VQ32B2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lutropin-choriogonadotropic hormone receptor (Homo sapiens (Human)) | BDBM50189778 (CHEMBL211405 | N-tert-butyl-5-amino-4-(3-methoxyph...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 220 | n/a | n/a | n/a | n/a |
NIH Chemical Genomics Center Curated by ChEMBL | Assay Description Agonist activity at LHCGR (unknown origin) | Medchemcomm 2: 1016-1020 (2011) Article DOI: 10.1039/c1md00145k BindingDB Entry DOI: 10.7270/Q2668H51 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lutropin-choriogonadotropic hormone receptor (Homo sapiens (Human)) | BDBM50206395 ((S)-N-(1-amino-3-(4-hydroxyphenyl)-1-oxopropan-2-y...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 250 | n/a | n/a | n/a | n/a |
Merck Serono Geneva Research Center Curated by ChEMBL | Assay Description Agonist activity at human LH receptor expressed in CHO cells assessed as production of cAMP after 60 mins by SPA | Bioorg Med Chem Lett 17: 2080-5 (2007) Article DOI: 10.1016/j.bmcl.2006.12.062 BindingDB Entry DOI: 10.7270/Q2VQ32B2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lutropin-choriogonadotropic hormone receptor (Homo sapiens (Human)) | BDBM50189778 (CHEMBL211405 | N-tert-butyl-5-amino-4-(3-methoxyph...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 300 | n/a | n/a | n/a | n/a |
National Institute of Diabetes and Digestive and Kidney Diseases Curated by ChEMBL | Assay Description Agonist activity at LHCGR expressed in HEK293 EM cells measured by intracellular cAMP accumulation | J Med Chem 49: 3888-96 (2006) Article DOI: 10.1021/jm060247s BindingDB Entry DOI: 10.7270/Q29886MR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lutropin-choriogonadotropic hormone receptor (Homo sapiens (Human)) | BDBM50206400 (CHEMBL247945 | N-((S)-1-amino-3-(4-hydroxyphenyl)-...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 500 | n/a | n/a | n/a | n/a |
Merck Serono Geneva Research Center Curated by ChEMBL | Assay Description Agonist activity at human LH receptor expressed in CHO cells assessed as production of cAMP after 60 mins by SPA | Bioorg Med Chem Lett 17: 2080-5 (2007) Article DOI: 10.1016/j.bmcl.2006.12.062 BindingDB Entry DOI: 10.7270/Q2VQ32B2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lutropin-choriogonadotropic hormone receptor (Homo sapiens (Human)) | BDBM50189779 (CHEMBL377399 | N-tert-butyl-5-amino-4-(3-methoxyph...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 800 | n/a | n/a | n/a | n/a |
National Institute of Diabetes and Digestive and Kidney Diseases Curated by ChEMBL | Assay Description Agonist activity at LHCGR expressed in HEK293 EM cells measured by intracellular cAMP accumulation | J Med Chem 49: 3888-96 (2006) Article DOI: 10.1021/jm060247s BindingDB Entry DOI: 10.7270/Q29886MR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lutropin-choriogonadotropic hormone receptor (Homo sapiens (Human)) | BDBM50189775 (CHEMBL377769 | N-tert-butyl-5-amino-4-(2,3-dimetho...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 800 | n/a | n/a | n/a | n/a |
National Institute of Diabetes and Digestive and Kidney Diseases Curated by ChEMBL | Assay Description Agonist activity at LHCGR expressed in HEK293 EM cells measured by intracellular cAMP accumulation | J Med Chem 49: 3888-96 (2006) Article DOI: 10.1021/jm060247s BindingDB Entry DOI: 10.7270/Q29886MR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lutropin-choriogonadotropic hormone receptor (Homo sapiens (Human)) | BDBM50189776 (CHEMBL211871 | tert-butyl 5-amino-4-(3-methoxyphen...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 1.10E+3 | n/a | n/a | n/a | n/a |
National Institute of Diabetes and Digestive and Kidney Diseases Curated by ChEMBL | Assay Description Agonist activity at LHCGR expressed in HEK293 EM cells measured by intracellular cAMP accumulation | J Med Chem 49: 3888-96 (2006) Article DOI: 10.1021/jm060247s BindingDB Entry DOI: 10.7270/Q29886MR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lutropin-choriogonadotropic hormone receptor (Homo sapiens (Human)) | BDBM50189777 (CHEMBL212815 | N-tert-butyl-5-amino-4-(3-fluorophe...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.20E+3 | n/a | n/a | n/a | n/a |
National Institute of Diabetes and Digestive and Kidney Diseases Curated by ChEMBL | Assay Description Agonist activity at LHCGR expressed in HEK293 EM cells measured by intracellular cAMP accumulation | J Med Chem 49: 3888-96 (2006) Article DOI: 10.1021/jm060247s BindingDB Entry DOI: 10.7270/Q29886MR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lutropin-choriogonadotropic hormone receptor (Homo sapiens (Human)) | BDBM50189773 (CHEMBL211129 | N-tert-butyl-5-amino-4-(2-fluoro-3-...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.50E+3 | n/a | n/a | n/a | n/a |
National Institute of Diabetes and Digestive and Kidney Diseases Curated by ChEMBL | Assay Description Agonist activity at LHCGR expressed in HEK293 EM cells measured by intracellular cAMP accumulation | J Med Chem 49: 3888-96 (2006) Article DOI: 10.1021/jm060247s BindingDB Entry DOI: 10.7270/Q29886MR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lutropin-choriogonadotropic hormone receptor (Homo sapiens (Human)) | BDBM50256858 (CHEMBL474041 | Cyclopentyl-carbamic acid [1,1',3',...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.60E+3 | n/a | n/a | n/a | n/a |
Leiden University Curated by ChEMBL | Assay Description Agonist activity at human luteinizing hormone receptor expressed in CHOK1 cells assessed as c-AMP-mediated luciferase production | J Med Chem 52: 2036-42 (2009) Article DOI: 10.1021/jm801561h BindingDB Entry DOI: 10.7270/Q2G73DMJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lutropin-choriogonadotropic hormone receptor (Homo sapiens (Human)) | BDBM50189774 (CHEMBL378091 | N-tert-butyl-5-amino-4-(3-hydroxyph...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.90E+3 | n/a | n/a | n/a | n/a |
National Institute of Diabetes and Digestive and Kidney Diseases Curated by ChEMBL | Assay Description Agonist activity at LHCGR expressed in HEK293 EM cells measured by intracellular cAMP accumulation | J Med Chem 49: 3888-96 (2006) Article DOI: 10.1021/jm060247s BindingDB Entry DOI: 10.7270/Q29886MR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lutropin-choriogonadotropic hormone receptor (Homo sapiens (Human)) | BDBM50206405 ((S)-N-(1-amino-3-(4-hydroxyphenyl)-1-oxopropan-2-y...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 2.30E+3 | n/a | n/a | n/a | n/a |
Merck Serono Geneva Research Center Curated by ChEMBL | Assay Description Agonist activity at human LH receptor expressed in CHO cells assessed as production of cAMP after 60 mins by SPA | Bioorg Med Chem Lett 17: 2080-5 (2007) Article DOI: 10.1016/j.bmcl.2006.12.062 BindingDB Entry DOI: 10.7270/Q2VQ32B2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lutropin-choriogonadotropic hormone receptor (Homo sapiens (Human)) | BDBM50206403 (CHEMBL269261 | N-((S)-1-amino-3-(4-tert-butoxyphen...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.21E+4 | n/a | n/a | n/a | n/a |
Merck Serono Geneva Research Center Curated by ChEMBL | Assay Description Agonist activity at human LH receptor expressed in CHO cells assessed as production of cAMP after 60 mins by SPA | Bioorg Med Chem Lett 17: 2080-5 (2007) Article DOI: 10.1016/j.bmcl.2006.12.062 BindingDB Entry DOI: 10.7270/Q2VQ32B2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lutropin-choriogonadotropic hormone receptor (Homo sapiens (Human)) | BDBM50505787 (CHEMBL4537998) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | >1.60E+4 | n/a | n/a | n/a | n/a |
Bayer AG Curated by ChEMBL | Assay Description Agonist activity at human luteinizing hormone receptor incubated for 60 mins by cell based TR-FRET assay | J Med Chem 62: 10321-10341 (2019) Article DOI: 10.1021/acs.jmedchem.9b01382 BindingDB Entry DOI: 10.7270/Q29P34X6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lutropin-choriogonadotropic hormone receptor (Homo sapiens (Human)) | BDBM50206404 ((S)-N-(1-amino-3-(4-hydroxyphenyl)-1-oxopropan-2-y...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a |
Merck Serono Geneva Research Center Curated by ChEMBL | Assay Description Agonist activity at human LH receptor expressed in CHO cells assessed as production of cAMP after 60 mins by SPA | Bioorg Med Chem Lett 17: 2080-5 (2007) Article DOI: 10.1016/j.bmcl.2006.12.062 BindingDB Entry DOI: 10.7270/Q2VQ32B2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lutropin-choriogonadotropic hormone receptor (Homo sapiens (Human)) | BDBM50206396 ((S)-2-{3-[2-(4-tert-butyl-phenyl)-5-pyridin-3-yl-2...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a |
Merck Serono Geneva Research Center Curated by ChEMBL | Assay Description Agonist activity at human LH receptor expressed in CHO cells assessed as production of cAMP after 60 mins by SPA | Bioorg Med Chem Lett 17: 2080-5 (2007) Article DOI: 10.1016/j.bmcl.2006.12.062 BindingDB Entry DOI: 10.7270/Q2VQ32B2 | |||||||||||
More data for this Ligand-Target Pair |