Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Transient receptor potential protein 5 (Rattus norvegicus) | BDBM50529421 (CHEMBL4530872) | PDB Reactome pathway KEGG UniProtKB/TrEMBL DrugBank GoogleScholar AffyNet | Purchase MCE PC cid PC sid PDB UniChem | Article PubMed | n/a | n/a | 180 | n/a | n/a | n/a | n/a | n/a | n/a |
Goldfinch Bio Inc. Curated by ChEMBL | Assay Description Inhibition of rosiglitazone-activated rat TRPC5 channel expressed in HEK293 cells assessed as reduction in Ca2+ current measured at +80 mV with holdi... | ACS Med Chem Lett 10: 1579-1585 (2019) Article DOI: 10.1021/acsmedchemlett.9b00430 BindingDB Entry DOI: 10.7270/Q2DN48HF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Short transient receptor potential channel 5 (Homo sapiens (Human)) | BDBM50529421 (CHEMBL4530872) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase MCE PC cid PC sid PDB UniChem | Article PubMed | n/a | n/a | 180 | n/a | n/a | n/a | n/a | n/a | n/a |
Goldfinch Bio Inc. Curated by ChEMBL | Assay Description Inhibition of rosiglitazone-activated human TRPC5 channel expressed in HEK293 cells assessed as reduction in Ca2+ current measured at +80 mV with hol... | ACS Med Chem Lett 10: 1579-1585 (2019) Article DOI: 10.1021/acsmedchemlett.9b00430 BindingDB Entry DOI: 10.7270/Q2DN48HF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Short transient receptor potential channel 5 (Homo sapiens (Human)) | BDBM50529421 (CHEMBL4530872) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase MCE PC cid PC sid PDB UniChem | Article PubMed | n/a | n/a | 280 | n/a | n/a | n/a | n/a | n/a | n/a |
Goldfinch Bio Inc. Curated by ChEMBL | Assay Description Inhibition of human TRPC5 channel expressed in HEK293 cells assessed as decrease in current amplitude treated for 3 mins measured between +80 mV and ... | ACS Med Chem Lett 10: 1579-1585 (2019) Article DOI: 10.1021/acsmedchemlett.9b00430 BindingDB Entry DOI: 10.7270/Q2DN48HF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Short transient receptor potential channel 4 (Homo sapiens) | BDBM50529421 (CHEMBL4530872) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase MCE PC cid PC sid PDB UniChem | Article PubMed | n/a | n/a | 290 | n/a | n/a | n/a | n/a | n/a | n/a |
Goldfinch Bio Inc. Curated by ChEMBL | Assay Description Inhibition of Englerin-activated human TRPC4 channel expressed in HEK293 cells by Q-patch clamp assay | ACS Med Chem Lett 10: 1579-1585 (2019) Article DOI: 10.1021/acsmedchemlett.9b00430 BindingDB Entry DOI: 10.7270/Q2DN48HF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Short transient receptor potential channel 5 (Homo sapiens (Human)) | BDBM50529418 (CHEMBL4452948) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 380 | n/a | n/a | n/a | n/a | n/a | n/a |
Goldfinch Bio Inc. Curated by ChEMBL | Assay Description Inhibition of rosiglitazone-activated human TRPC5 channel expressed in HEK293 cells assessed as reduction in Ca2+ current measured at +80 mV with hol... | ACS Med Chem Lett 10: 1579-1585 (2019) Article DOI: 10.1021/acsmedchemlett.9b00430 BindingDB Entry DOI: 10.7270/Q2DN48HF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Short transient receptor potential channel 5 (Homo sapiens (Human)) | BDBM50529427 (CHEMBL4536108) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 490 | n/a | n/a | n/a | n/a | n/a | n/a |
Goldfinch Bio Inc. Curated by ChEMBL | Assay Description Inhibition of rosiglitazone-activated human TRPC5 channel expressed in HEK293 cells assessed as reduction in Ca2+ current measured at +80 mV with hol... | ACS Med Chem Lett 10: 1579-1585 (2019) Article DOI: 10.1021/acsmedchemlett.9b00430 BindingDB Entry DOI: 10.7270/Q2DN48HF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Short transient receptor potential channel 5 (Homo sapiens (Human)) | BDBM50529454 (CHEMBL4440201) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 500 | n/a | n/a | n/a | n/a | n/a | n/a |
Goldfinch Bio Inc. Curated by ChEMBL | Assay Description Inhibition of rosiglitazone-activated human TRPC5 channel expressed in HEK293 cells assessed as reduction in Ca2+ current measured at +80 mV with hol... | ACS Med Chem Lett 10: 1579-1585 (2019) Article DOI: 10.1021/acsmedchemlett.9b00430 BindingDB Entry DOI: 10.7270/Q2DN48HF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Short transient receptor potential channel 5 (Homo sapiens (Human)) | BDBM50529426 (CHEMBL4475970) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 530 | n/a | n/a | n/a | n/a | n/a | n/a |
Goldfinch Bio Inc. Curated by ChEMBL | Assay Description Inhibition of rosiglitazone-activated human TRPC5 channel expressed in HEK293 cells assessed as reduction in Ca2+ current measured at +80 mV with hol... | ACS Med Chem Lett 10: 1579-1585 (2019) Article DOI: 10.1021/acsmedchemlett.9b00430 BindingDB Entry DOI: 10.7270/Q2DN48HF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Short transient receptor potential channel 5 (Homo sapiens (Human)) | BDBM50529447 (CHEMBL4517031) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 530 | n/a | n/a | n/a | n/a | n/a | n/a |
Goldfinch Bio Inc. Curated by ChEMBL | Assay Description Inhibition of rosiglitazone-activated human TRPC5 channel expressed in HEK293 cells assessed as reduction in Ca2+ current measured at +80 mV with hol... | ACS Med Chem Lett 10: 1579-1585 (2019) Article DOI: 10.1021/acsmedchemlett.9b00430 BindingDB Entry DOI: 10.7270/Q2DN48HF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Short transient receptor potential channel 5 (Homo sapiens (Human)) | BDBM50529450 (CHEMBL4563968) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 650 | n/a | n/a | n/a | n/a | n/a | n/a |
Goldfinch Bio Inc. Curated by ChEMBL | Assay Description Inhibition of rosiglitazone-activated human TRPC5 channel expressed in HEK293 cells assessed as reduction in Ca2+ current measured at +80 mV with hol... | ACS Med Chem Lett 10: 1579-1585 (2019) Article DOI: 10.1021/acsmedchemlett.9b00430 BindingDB Entry DOI: 10.7270/Q2DN48HF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Short transient receptor potential channel 5 (Homo sapiens (Human)) | BDBM50529449 (CHEMBL4449727) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 650 | n/a | n/a | n/a | n/a | n/a | n/a |
Goldfinch Bio Inc. Curated by ChEMBL | Assay Description Inhibition of rosiglitazone-activated human TRPC5 channel expressed in HEK293 cells assessed as reduction in Ca2+ current measured at +80 mV with hol... | ACS Med Chem Lett 10: 1579-1585 (2019) Article DOI: 10.1021/acsmedchemlett.9b00430 BindingDB Entry DOI: 10.7270/Q2DN48HF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Short transient receptor potential channel 5 (Homo sapiens (Human)) | BDBM50529430 (CHEMBL4551777) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 660 | n/a | n/a | n/a | n/a | n/a | n/a |
Goldfinch Bio Inc. Curated by ChEMBL | Assay Description Inhibition of rosiglitazone-activated human TRPC5 channel expressed in HEK293 cells assessed as reduction in Ca2+ current measured at +80 mV with hol... | ACS Med Chem Lett 10: 1579-1585 (2019) Article DOI: 10.1021/acsmedchemlett.9b00430 BindingDB Entry DOI: 10.7270/Q2DN48HF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Short transient receptor potential channel 5 (Homo sapiens (Human)) | BDBM50529452 (CHEMBL4458885) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Goldfinch Bio Inc. Curated by ChEMBL | Assay Description Inhibition of rosiglitazone-activated human TRPC5 channel expressed in HEK293 cells assessed as reduction in Ca2+ current measured at +80 mV with hol... | ACS Med Chem Lett 10: 1579-1585 (2019) Article DOI: 10.1021/acsmedchemlett.9b00430 BindingDB Entry DOI: 10.7270/Q2DN48HF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Short transient receptor potential channel 5 (Homo sapiens (Human)) | BDBM50529440 (CHEMBL4467989) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Goldfinch Bio Inc. Curated by ChEMBL | Assay Description Inhibition of rosiglitazone-activated human TRPC5 channel expressed in HEK293 cells assessed as reduction in Ca2+ current measured at +80 mV with hol... | ACS Med Chem Lett 10: 1579-1585 (2019) Article DOI: 10.1021/acsmedchemlett.9b00430 BindingDB Entry DOI: 10.7270/Q2DN48HF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Short transient receptor potential channel 5 (Homo sapiens (Human)) | BDBM50529419 (CHEMBL4434976) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.90E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Goldfinch Bio Inc. Curated by ChEMBL | Assay Description Inhibition of rosiglitazone-activated human TRPC5 channel expressed in HEK293 cells assessed as reduction in Ca2+ current measured at +80 mV with hol... | ACS Med Chem Lett 10: 1579-1585 (2019) Article DOI: 10.1021/acsmedchemlett.9b00430 BindingDB Entry DOI: 10.7270/Q2DN48HF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Short transient receptor potential channel 5 (Homo sapiens (Human)) | BDBM50529444 (CHEMBL4473064) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.90E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Goldfinch Bio Inc. Curated by ChEMBL | Assay Description Inhibition of rosiglitazone-activated human TRPC5 channel expressed in HEK293 cells assessed as reduction in Ca2+ current measured at +80 mV with hol... | ACS Med Chem Lett 10: 1579-1585 (2019) Article DOI: 10.1021/acsmedchemlett.9b00430 BindingDB Entry DOI: 10.7270/Q2DN48HF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Short transient receptor potential channel 5 (Homo sapiens (Human)) | BDBM50529420 (CHEMBL4546342) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Goldfinch Bio Inc. Curated by ChEMBL | Assay Description Inhibition of rosiglitazone-activated human TRPC5 channel expressed in HEK293 cells assessed as reduction in Ca2+ current measured at +80 mV with hol... | ACS Med Chem Lett 10: 1579-1585 (2019) Article DOI: 10.1021/acsmedchemlett.9b00430 BindingDB Entry DOI: 10.7270/Q2DN48HF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Short transient receptor potential channel 5 (Homo sapiens (Human)) | BDBM50529445 (CHEMBL4471419) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Goldfinch Bio Inc. Curated by ChEMBL | Assay Description Inhibition of rosiglitazone-activated human TRPC5 channel expressed in HEK293 cells assessed as reduction in Ca2+ current measured at +80 mV with hol... | ACS Med Chem Lett 10: 1579-1585 (2019) Article DOI: 10.1021/acsmedchemlett.9b00430 BindingDB Entry DOI: 10.7270/Q2DN48HF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Short transient receptor potential channel 5 (Homo sapiens (Human)) | BDBM50529422 (CHEMBL4447753) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase PC cid PC sid UniChem | Article PubMed | n/a | n/a | 4.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Goldfinch Bio Inc. Curated by ChEMBL | Assay Description Inhibition of (-)-Englerin-activated human TRPC5 channel expressed in HEK293 cells measured at holding potential of -60 mV by Q-patch clamp assay | ACS Med Chem Lett 10: 1579-1585 (2019) Article DOI: 10.1021/acsmedchemlett.9b00430 BindingDB Entry DOI: 10.7270/Q2DN48HF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Short transient receptor potential channel 5 (Homo sapiens (Human)) | BDBM50529422 (CHEMBL4447753) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase PC cid PC sid UniChem | Article PubMed | n/a | n/a | 4.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Goldfinch Bio Inc. Curated by ChEMBL | Assay Description Inhibition of lanthanum-activated human TRPC5 channel expressed in HEK293 cells measured at holding potential of -60 mV by Q-patch clamp assay | ACS Med Chem Lett 10: 1579-1585 (2019) Article DOI: 10.1021/acsmedchemlett.9b00430 BindingDB Entry DOI: 10.7270/Q2DN48HF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Short transient receptor potential channel 5 (Homo sapiens (Human)) | BDBM50529422 (CHEMBL4447753) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase PC cid PC sid UniChem | Article PubMed | n/a | n/a | 5.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Goldfinch Bio Inc. Curated by ChEMBL | Assay Description Inhibition of rosiglitazone-activated human TRPC5 channel expressed in HEK293 cells assessed as reduction in Ca2+ current measured at +80 mV with hol... | ACS Med Chem Lett 10: 1579-1585 (2019) Article DOI: 10.1021/acsmedchemlett.9b00430 BindingDB Entry DOI: 10.7270/Q2DN48HF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Short transient receptor potential channel 5 (Homo sapiens (Human)) | BDBM50529422 (CHEMBL4447753) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase PC cid PC sid UniChem | Article PubMed | n/a | n/a | 7.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Goldfinch Bio Inc. Curated by ChEMBL | Assay Description Inhibition of riluzole-activated human TRPC5 channel expressed in HEK293 cells measured at holding potential of -60 mV by Q-patch clamp assay | ACS Med Chem Lett 10: 1579-1585 (2019) Article DOI: 10.1021/acsmedchemlett.9b00430 BindingDB Entry DOI: 10.7270/Q2DN48HF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Short transient receptor potential channel 5 (Homo sapiens (Human)) | BDBM50529457 (CHEMBL4474451) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 8.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Goldfinch Bio Inc. Curated by ChEMBL | Assay Description Inhibition of rosiglitazone-activated human TRPC5 channel expressed in HEK293 cells assessed as reduction in Ca2+ current measured at +80 mV with hol... | ACS Med Chem Lett 10: 1579-1585 (2019) Article DOI: 10.1021/acsmedchemlett.9b00430 BindingDB Entry DOI: 10.7270/Q2DN48HF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Short transient receptor potential channel 5 (Homo sapiens (Human)) | BDBM50529442 (CHEMBL4458766) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 8.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Goldfinch Bio Inc. Curated by ChEMBL | Assay Description Inhibition of rosiglitazone-activated human TRPC5 channel expressed in HEK293 cells assessed as reduction in Ca2+ current measured at +80 mV with hol... | ACS Med Chem Lett 10: 1579-1585 (2019) Article DOI: 10.1021/acsmedchemlett.9b00430 BindingDB Entry DOI: 10.7270/Q2DN48HF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily H member 2 (Homo sapiens (Human)) | BDBM50529421 (CHEMBL4530872) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid PDB UniChem | Article PubMed | n/a | n/a | 8.70E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Goldfinch Bio Inc. Curated by ChEMBL | Assay Description Inhibition of human ERG stably expressed in HEK293 cells measured at holding potential of -90 mV by manual patch clamp assay | ACS Med Chem Lett 10: 1579-1585 (2019) Article DOI: 10.1021/acsmedchemlett.9b00430 BindingDB Entry DOI: 10.7270/Q2DN48HF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Short transient receptor potential channel 5 (Homo sapiens (Human)) | BDBM50529441 (CHEMBL4592027) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 8.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Goldfinch Bio Inc. Curated by ChEMBL | Assay Description Inhibition of rosiglitazone-activated human TRPC5 channel expressed in HEK293 cells assessed as reduction in Ca2+ current measured at +80 mV with hol... | ACS Med Chem Lett 10: 1579-1585 (2019) Article DOI: 10.1021/acsmedchemlett.9b00430 BindingDB Entry DOI: 10.7270/Q2DN48HF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Short transient receptor potential channel 5 (Homo sapiens (Human)) | BDBM50529443 (CHEMBL4442703) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 9.60E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Goldfinch Bio Inc. Curated by ChEMBL | Assay Description Inhibition of rosiglitazone-activated human TRPC5 channel expressed in HEK293 cells assessed as reduction in Ca2+ current measured at +80 mV with hol... | ACS Med Chem Lett 10: 1579-1585 (2019) Article DOI: 10.1021/acsmedchemlett.9b00430 BindingDB Entry DOI: 10.7270/Q2DN48HF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Short transient receptor potential channel 5 (Homo sapiens (Human)) | BDBM50529432 (CHEMBL4473219) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.10E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Goldfinch Bio Inc. Curated by ChEMBL | Assay Description Inhibition of rosiglitazone-activated human TRPC5 channel expressed in HEK293 cells assessed as reduction in Ca2+ current measured at +80 mV with hol... | ACS Med Chem Lett 10: 1579-1585 (2019) Article DOI: 10.1021/acsmedchemlett.9b00430 BindingDB Entry DOI: 10.7270/Q2DN48HF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Short transient receptor potential channel 5 (Homo sapiens (Human)) | BDBM50529424 (CHEMBL4436613) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.12E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Goldfinch Bio Inc. Curated by ChEMBL | Assay Description Inhibition of rosiglitazone-activated human TRPC5 channel expressed in HEK293 cells assessed as reduction in Ca2+ current measured at +80 mV with hol... | ACS Med Chem Lett 10: 1579-1585 (2019) Article DOI: 10.1021/acsmedchemlett.9b00430 BindingDB Entry DOI: 10.7270/Q2DN48HF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Short transient receptor potential channel 5 (Homo sapiens (Human)) | BDBM50529428 (CHEMBL4470341) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.45E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Goldfinch Bio Inc. Curated by ChEMBL | Assay Description Inhibition of rosiglitazone-activated human TRPC5 channel expressed in HEK293 cells assessed as reduction in Ca2+ current measured at +80 mV with hol... | ACS Med Chem Lett 10: 1579-1585 (2019) Article DOI: 10.1021/acsmedchemlett.9b00430 BindingDB Entry DOI: 10.7270/Q2DN48HF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Short transient receptor potential channel 5 (Homo sapiens (Human)) | BDBM50529455 (CHEMBL4542897) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.60E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Goldfinch Bio Inc. Curated by ChEMBL | Assay Description Inhibition of rosiglitazone-activated human TRPC5 channel expressed in HEK293 cells assessed as reduction in Ca2+ current measured at +80 mV with hol... | ACS Med Chem Lett 10: 1579-1585 (2019) Article DOI: 10.1021/acsmedchemlett.9b00430 BindingDB Entry DOI: 10.7270/Q2DN48HF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Short transient receptor potential channel 5 (Homo sapiens (Human)) | BDBM50529456 (CHEMBL4524687) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.80E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Goldfinch Bio Inc. Curated by ChEMBL | Assay Description Inhibition of rosiglitazone-activated human TRPC5 channel expressed in HEK293 cells assessed as reduction in Ca2+ current measured at +80 mV with hol... | ACS Med Chem Lett 10: 1579-1585 (2019) Article DOI: 10.1021/acsmedchemlett.9b00430 BindingDB Entry DOI: 10.7270/Q2DN48HF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Short transient receptor potential channel 5 (Homo sapiens (Human)) | BDBM50529438 (CHEMBL4528028) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2.70E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Goldfinch Bio Inc. Curated by ChEMBL | Assay Description Inhibition of rosiglitazone-activated human TRPC5 channel expressed in HEK293 cells assessed as reduction in Ca2+ current measured at +80 mV with hol... | ACS Med Chem Lett 10: 1579-1585 (2019) Article DOI: 10.1021/acsmedchemlett.9b00430 BindingDB Entry DOI: 10.7270/Q2DN48HF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Short transient receptor potential channel 5 (Homo sapiens (Human)) | BDBM50529435 (CHEMBL4594091) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2.70E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Goldfinch Bio Inc. Curated by ChEMBL | Assay Description Inhibition of rosiglitazone-activated human TRPC5 channel expressed in HEK293 cells assessed as reduction in Ca2+ current measured at +80 mV with hol... | ACS Med Chem Lett 10: 1579-1585 (2019) Article DOI: 10.1021/acsmedchemlett.9b00430 BindingDB Entry DOI: 10.7270/Q2DN48HF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Short transient receptor potential channel 5 (Homo sapiens (Human)) | BDBM50529433 (CHEMBL4565194) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2.80E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Goldfinch Bio Inc. Curated by ChEMBL | Assay Description Inhibition of rosiglitazone-activated human TRPC5 channel expressed in HEK293 cells assessed as reduction in Ca2+ current measured at +80 mV with hol... | ACS Med Chem Lett 10: 1579-1585 (2019) Article DOI: 10.1021/acsmedchemlett.9b00430 BindingDB Entry DOI: 10.7270/Q2DN48HF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Short transient receptor potential channel 6 (Homo sapiens (Human)) | BDBM50529422 (CHEMBL4447753) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase PC cid PC sid UniChem | Article PubMed | n/a | n/a | >3.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Goldfinch Bio Inc. Curated by ChEMBL | Assay Description Inhibition of OAG-activated human TRPC6 channel expressed in HEK293 cells by Q-patch clamp assay | ACS Med Chem Lett 10: 1579-1585 (2019) Article DOI: 10.1021/acsmedchemlett.9b00430 BindingDB Entry DOI: 10.7270/Q2DN48HF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Short transient receptor potential channel 5 (Homo sapiens (Human)) | BDBM50529446 (CHEMBL4436512) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >3.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Goldfinch Bio Inc. Curated by ChEMBL | Assay Description Inhibition of rosiglitazone-activated human TRPC5 channel expressed in HEK293 cells assessed as reduction in Ca2+ current measured at +80 mV with hol... | ACS Med Chem Lett 10: 1579-1585 (2019) Article DOI: 10.1021/acsmedchemlett.9b00430 BindingDB Entry DOI: 10.7270/Q2DN48HF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Short transient receptor potential channel 5 (Homo sapiens (Human)) | BDBM50529448 (CHEMBL4568038) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >3.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Goldfinch Bio Inc. Curated by ChEMBL | Assay Description Inhibition of rosiglitazone-activated human TRPC5 channel expressed in HEK293 cells assessed as reduction in Ca2+ current measured at +80 mV with hol... | ACS Med Chem Lett 10: 1579-1585 (2019) Article DOI: 10.1021/acsmedchemlett.9b00430 BindingDB Entry DOI: 10.7270/Q2DN48HF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium channel protein type 5 subunit alpha (Homo sapiens (Human)) | BDBM50529421 (CHEMBL4530872) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid PDB UniChem | Article PubMed | n/a | n/a | >3.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Goldfinch Bio Inc. Curated by ChEMBL | Assay Description Inhibition of human Nav1.5 stably expressed in CHO cells measured at holding potential of -80 mV by manual patch clamp assay | ACS Med Chem Lett 10: 1579-1585 (2019) Article DOI: 10.1021/acsmedchemlett.9b00430 BindingDB Entry DOI: 10.7270/Q2DN48HF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Short transient receptor potential channel 5 (Homo sapiens (Human)) | BDBM50529425 (CHEMBL4475647) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >3.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Goldfinch Bio Inc. Curated by ChEMBL | Assay Description Inhibition of rosiglitazone-activated human TRPC5 channel expressed in HEK293 cells assessed as reduction in Ca2+ current measured at +80 mV with hol... | ACS Med Chem Lett 10: 1579-1585 (2019) Article DOI: 10.1021/acsmedchemlett.9b00430 BindingDB Entry DOI: 10.7270/Q2DN48HF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Short transient receptor potential channel 5 (Homo sapiens (Human)) | BDBM50529451 (CHEMBL4469449) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >3.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Goldfinch Bio Inc. Curated by ChEMBL | Assay Description Inhibition of rosiglitazone-activated human TRPC5 channel expressed in HEK293 cells assessed as reduction in Ca2+ current measured at +80 mV with hol... | ACS Med Chem Lett 10: 1579-1585 (2019) Article DOI: 10.1021/acsmedchemlett.9b00430 BindingDB Entry DOI: 10.7270/Q2DN48HF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Short transient receptor potential channel 5 (Homo sapiens (Human)) | BDBM50529439 (CHEMBL4590831) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >3.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Goldfinch Bio Inc. Curated by ChEMBL | Assay Description Inhibition of rosiglitazone-activated human TRPC5 channel expressed in HEK293 cells assessed as reduction in Ca2+ current measured at +80 mV with hol... | ACS Med Chem Lett 10: 1579-1585 (2019) Article DOI: 10.1021/acsmedchemlett.9b00430 BindingDB Entry DOI: 10.7270/Q2DN48HF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Short transient receptor potential channel 5 (Homo sapiens (Human)) | BDBM50529453 (CHEMBL4454641) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >3.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Goldfinch Bio Inc. Curated by ChEMBL | Assay Description Inhibition of rosiglitazone-activated human TRPC5 channel expressed in HEK293 cells assessed as reduction in Ca2+ current measured at +80 mV with hol... | ACS Med Chem Lett 10: 1579-1585 (2019) Article DOI: 10.1021/acsmedchemlett.9b00430 BindingDB Entry DOI: 10.7270/Q2DN48HF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Short transient receptor potential channel 6 (Homo sapiens (Human)) | BDBM50529421 (CHEMBL4530872) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid PDB UniChem | Article PubMed | n/a | n/a | >3.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Goldfinch Bio Inc. Curated by ChEMBL | Assay Description Inhibition of OAG-activated human TRPC6 channel expressed in HEK293 cells by Q-patch clamp assay | ACS Med Chem Lett 10: 1579-1585 (2019) Article DOI: 10.1021/acsmedchemlett.9b00430 BindingDB Entry DOI: 10.7270/Q2DN48HF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Short transient receptor potential channel 5 (Homo sapiens (Human)) | BDBM50529437 (CHEMBL4448384) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >3.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Goldfinch Bio Inc. Curated by ChEMBL | Assay Description Inhibition of rosiglitazone-activated human TRPC5 channel expressed in HEK293 cells assessed as reduction in Ca2+ current measured at +80 mV with hol... | ACS Med Chem Lett 10: 1579-1585 (2019) Article DOI: 10.1021/acsmedchemlett.9b00430 BindingDB Entry DOI: 10.7270/Q2DN48HF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Short transient receptor potential channel 5 (Homo sapiens (Human)) | BDBM50529436 (CHEMBL4556467) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >3.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Goldfinch Bio Inc. Curated by ChEMBL | Assay Description Inhibition of rosiglitazone-activated human TRPC5 channel expressed in HEK293 cells assessed as reduction in Ca2+ current measured at +80 mV with hol... | ACS Med Chem Lett 10: 1579-1585 (2019) Article DOI: 10.1021/acsmedchemlett.9b00430 BindingDB Entry DOI: 10.7270/Q2DN48HF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Short transient receptor potential channel 5 (Homo sapiens (Human)) | BDBM50529434 (CHEMBL4518299) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >3.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Goldfinch Bio Inc. Curated by ChEMBL | Assay Description Inhibition of rosiglitazone-activated human TRPC5 channel expressed in HEK293 cells assessed as reduction in Ca2+ current measured at +80 mV with hol... | ACS Med Chem Lett 10: 1579-1585 (2019) Article DOI: 10.1021/acsmedchemlett.9b00430 BindingDB Entry DOI: 10.7270/Q2DN48HF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Short transient receptor potential channel 5 (Homo sapiens (Human)) | BDBM50529429 (CHEMBL4439131) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >3.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Goldfinch Bio Inc. Curated by ChEMBL | Assay Description Inhibition of rosiglitazone-activated human TRPC5 channel expressed in HEK293 cells assessed as reduction in Ca2+ current measured at +80 mV with hol... | ACS Med Chem Lett 10: 1579-1585 (2019) Article DOI: 10.1021/acsmedchemlett.9b00430 BindingDB Entry DOI: 10.7270/Q2DN48HF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Short transient receptor potential channel 5 (Homo sapiens (Human)) | BDBM50529431 (CHEMBL4547350) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >3.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Goldfinch Bio Inc. Curated by ChEMBL | Assay Description Inhibition of rosiglitazone-activated human TRPC5 channel expressed in HEK293 cells assessed as reduction in Ca2+ current measured at +80 mV with hol... | ACS Med Chem Lett 10: 1579-1585 (2019) Article DOI: 10.1021/acsmedchemlett.9b00430 BindingDB Entry DOI: 10.7270/Q2DN48HF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Short transient receptor potential channel 5 (Homo sapiens (Human)) | BDBM50529423 (CHEMBL4454366) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >3.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Goldfinch Bio Inc. Curated by ChEMBL | Assay Description Inhibition of rosiglitazone-activated human TRPC5 channel expressed in HEK293 cells assessed as reduction in Ca2+ current measured at +80 mV with hol... | ACS Med Chem Lett 10: 1579-1585 (2019) Article DOI: 10.1021/acsmedchemlett.9b00430 BindingDB Entry DOI: 10.7270/Q2DN48HF | |||||||||||
More data for this Ligand-Target Pair |