Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Ribosomal protein S6 kinase alpha-6 (Homo sapiens (Human)) | BDBM286091 ((R)¿N-(1-(4-aminobenzyl)-1H-pyrazol-4-yl)-9-methyl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.300 | n/a | n/a | n/a | n/a | n/a | n/a |
PHOENIX MOLECULAR DESIGN US Patent | Assay Description Radioisotope assays (SignalChem) were performed for the evaluation of the kinase target profiling and all assays were performed in a designated radio... | US Patent US9771366 (2017) BindingDB Entry DOI: 10.7270/Q2862JK5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ribosomal protein S6 kinase alpha-6 (Homo sapiens (Human)) | BDBM286091 ((R)¿N-(1-(4-aminobenzyl)-1H-pyrazol-4-yl)-9-methyl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.300 | n/a | n/a | n/a | n/a | n/a | n/a |
PHOENIX MOLECULAR DESIGNS US Patent | Assay Description Radioisotope assays were performed for the evaluation of the kinase target profiling and all assays were performed in a designated radioactive workin... | US Patent US10758530 (2020) BindingDB Entry DOI: 10.7270/Q20R9SGD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ribosomal protein S6 kinase alpha-3 (Homo sapiens (Human)) | BDBM286091 ((R)¿N-(1-(4-aminobenzyl)-1H-pyrazol-4-yl)-9-methyl...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 1.70 | n/a | n/a | n/a | n/a | n/a | n/a |
PHOENIX MOLECULAR DESIGN US Patent | Assay Description Radioisotope assays (SignalChem) were performed for the evaluation of the kinase target profiling and all assays were performed in a designated radio... | US Patent US9771366 (2017) BindingDB Entry DOI: 10.7270/Q2862JK5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ribosomal protein S6 kinase alpha-3 (Homo sapiens (Human)) | BDBM286091 ((R)¿N-(1-(4-aminobenzyl)-1H-pyrazol-4-yl)-9-methyl...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 1.70 | n/a | n/a | n/a | n/a | n/a | n/a |
PHOENIX MOLECULAR DESIGNS US Patent | Assay Description Radioisotope assays were performed for the evaluation of the kinase target profiling and all assays were performed in a designated radioactive workin... | US Patent US10758530 (2020) BindingDB Entry DOI: 10.7270/Q20R9SGD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ribosomal protein S6 kinase alpha-1 (Homo sapiens (Human)) | BDBM286091 ((R)¿N-(1-(4-aminobenzyl)-1H-pyrazol-4-yl)-9-methyl...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 2 | n/a | n/a | n/a | n/a | n/a | n/a |
PHOENIX MOLECULAR DESIGN US Patent | Assay Description Radioisotope assays (SignalChem) were performed for the evaluation of the kinase target profiling and all assays were performed in a designated radio... | US Patent US9771366 (2017) BindingDB Entry DOI: 10.7270/Q2862JK5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ribosomal protein S6 kinase alpha-1 (Homo sapiens (Human)) | BDBM286091 ((R)¿N-(1-(4-aminobenzyl)-1H-pyrazol-4-yl)-9-methyl...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 2 | n/a | n/a | n/a | n/a | n/a | n/a |
PHOENIX MOLECULAR DESIGNS US Patent | Assay Description Radioisotope assays were performed for the evaluation of the kinase target profiling and all assays were performed in a designated radioactive workin... | US Patent US10758530 (2020) BindingDB Entry DOI: 10.7270/Q20R9SGD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ribosomal protein S6 kinase alpha-3 (Homo sapiens (Human)) | BDBM342166 ((R)-1-benzyl-N-(9-methyl-6-oxo-6,7,8,9-tetrahydrop...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 6 | n/a | n/a | n/a | n/a | n/a | n/a |
PHOENIX MOLECULAR DESIGN US Patent | Assay Description Radioisotope assays (SignalChem) were performed for the evaluation of the kinase target profiling and all assays were performed in a designated radio... | US Patent US9771366 (2017) BindingDB Entry DOI: 10.7270/Q2862JK5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ribosomal protein S6 kinase alpha-3 (Homo sapiens (Human)) | BDBM458758 ((R)-1-benzyl-N-(9-methyl-6-oxo-6,7,8,9-tetrahydrop...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 6 | n/a | n/a | n/a | n/a | n/a | n/a |
PHOENIX MOLECULAR DESIGNS US Patent | Assay Description Radioisotope assays were performed for the evaluation of the kinase target profiling and all assays were performed in a designated radioactive workin... | US Patent US10758530 (2020) BindingDB Entry DOI: 10.7270/Q20R9SGD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin-linked protein kinase (Homo sapiens (Human)) | BDBM123945 (US8754233, 2-(5-Amino-3-methyl-1H-pyrazol-4-yl)-5-...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 7 | n/a | n/a | n/a | n/a | n/a | 40 |
Dermira (Canada), Inc. US Patent | Assay Description 5 uL of each compound dilution were robotically pipetted to Costar serocluster plates maintaining the same plate layout. All assay mixtures consisted... | US Patent US8754233 (2014) BindingDB Entry DOI: 10.7270/Q23N2231 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ribosomal protein S6 kinase alpha-6 (Homo sapiens (Human)) | BDBM342166 ((R)-1-benzyl-N-(9-methyl-6-oxo-6,7,8,9-tetrahydrop...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 8 | n/a | n/a | n/a | n/a | n/a | n/a |
PHOENIX MOLECULAR DESIGN US Patent | Assay Description Radioisotope assays (SignalChem) were performed for the evaluation of the kinase target profiling and all assays were performed in a designated radio... | US Patent US9771366 (2017) BindingDB Entry DOI: 10.7270/Q2862JK5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ribosomal protein S6 kinase alpha-6 (Homo sapiens (Human)) | BDBM458758 ((R)-1-benzyl-N-(9-methyl-6-oxo-6,7,8,9-tetrahydrop...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 8 | n/a | n/a | n/a | n/a | n/a | n/a |
PHOENIX MOLECULAR DESIGNS US Patent | Assay Description Radioisotope assays were performed for the evaluation of the kinase target profiling and all assays were performed in a designated radioactive workin... | US Patent US10758530 (2020) BindingDB Entry DOI: 10.7270/Q20R9SGD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin-linked protein kinase (Homo sapiens (Human)) | BDBM123951 (US8754233, 2-(5-Amino-3-methyl-1H-pyrazol-4-yl)-be...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 10 | n/a | n/a | n/a | n/a | n/a | 40 |
Dermira (Canada), Inc. US Patent | Assay Description 5 uL of each compound dilution were robotically pipetted to Costar serocluster plates maintaining the same plate layout. All assay mixtures consisted... | US Patent US8754233 (2014) BindingDB Entry DOI: 10.7270/Q23N2231 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin-linked protein kinase (Homo sapiens (Human)) | BDBM124052 (US8754233, 5-(3-Amino-propyl)-4-benzothiazol-2-yl-...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | Purchase PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 10 | n/a | n/a | n/a | n/a | n/a | 40 |
Dermira (Canada), Inc. US Patent | Assay Description 5 uL of each compound dilution were robotically pipetted to Costar serocluster plates maintaining the same plate layout. All assay mixtures consisted... | US Patent US8754233 (2014) BindingDB Entry DOI: 10.7270/Q23N2231 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ribosomal protein S6 kinase alpha-2 (Homo sapiens (Human)) | BDBM286091 ((R)¿N-(1-(4-aminobenzyl)-1H-pyrazol-4-yl)-9-methyl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 12 | n/a | n/a | n/a | n/a | n/a | n/a |
PHOENIX MOLECULAR DESIGNS US Patent | Assay Description Radioisotope assays were performed for the evaluation of the kinase target profiling and all assays were performed in a designated radioactive workin... | US Patent US10758530 (2020) BindingDB Entry DOI: 10.7270/Q20R9SGD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ribosomal protein S6 kinase alpha-2 (Homo sapiens (Human)) | BDBM286090 ((R)¿N-(1-(2-aminobenzyl)-1H-pyrazol-4-yl)-9-methyl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 14 | n/a | n/a | n/a | n/a | n/a | n/a |
PHOENIX MOLECULAR DESIGNS US Patent | Assay Description Radioisotope assays were performed for the evaluation of the kinase target profiling and all assays were performed in a designated radioactive workin... | US Patent US10758530 (2020) BindingDB Entry DOI: 10.7270/Q20R9SGD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ribosomal protein S6 kinase alpha-2 (Homo sapiens (Human)) | BDBM286091 ((R)¿N-(1-(4-aminobenzyl)-1H-pyrazol-4-yl)-9-methyl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 18 | n/a | n/a | n/a | n/a | n/a | n/a |
PHOENIX MOLECULAR DESIGNS US Patent | Assay Description Radioisotope assays were performed for the evaluation of the kinase target profiling and all assays were performed in a designated radioactive workin... | US Patent US10758530 (2020) BindingDB Entry DOI: 10.7270/Q20R9SGD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin-linked protein kinase (Homo sapiens (Human)) | BDBM123930 (US8754233, 2-(3-Amino-1H-pyrazol-4-yl)-5-fluoro-be...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 20 | n/a | n/a | n/a | n/a | n/a | 40 |
Dermira (Canada), Inc. US Patent | Assay Description 5 uL of each compound dilution were robotically pipetted to Costar serocluster plates maintaining the same plate layout. All assay mixtures consisted... | US Patent US8754233 (2014) BindingDB Entry DOI: 10.7270/Q23N2231 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ribosomal protein S6 kinase alpha-2 (Homo sapiens (Human)) | BDBM286091 ((R)¿N-(1-(4-aminobenzyl)-1H-pyrazol-4-yl)-9-methyl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 20 | n/a | n/a | n/a | n/a | n/a | n/a |
PHOENIX MOLECULAR DESIGNS US Patent | Assay Description Radioisotope assays were performed for the evaluation of the kinase target profiling and all assays were performed in a designated radioactive workin... | US Patent US10758530 (2020) BindingDB Entry DOI: 10.7270/Q20R9SGD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ribosomal protein S6 kinase alpha-2 (Homo sapiens (Human)) | BDBM286091 ((R)¿N-(1-(4-aminobenzyl)-1H-pyrazol-4-yl)-9-methyl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 20 | n/a | n/a | n/a | n/a | n/a | n/a |
PHOENIX MOLECULAR DESIGN US Patent | Assay Description Radioisotope assays (SignalChem) were performed for the evaluation of the kinase target profiling and all assays were performed in a designated radio... | US Patent US9771366 (2017) BindingDB Entry DOI: 10.7270/Q2862JK5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin-linked protein kinase (Homo sapiens (Human)) | BDBM124067 (US8754233, N3-(2-Amino-ethyl)-4-benzothiazol-2-yl-...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 20 | n/a | n/a | n/a | n/a | n/a | 40 |
Dermira (Canada), Inc. US Patent | Assay Description 5 uL of each compound dilution were robotically pipetted to Costar serocluster plates maintaining the same plate layout. All assay mixtures consisted... | US Patent US8754233 (2014) BindingDB Entry DOI: 10.7270/Q23N2231 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin-linked protein kinase (Homo sapiens (Human)) | BDBM124022 (US8754233, 4-Benzothiazol-2-yl-5-(3-methylamino-pr...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 20 | n/a | n/a | n/a | n/a | n/a | 40 |
Dermira (Canada), Inc. US Patent | Assay Description 5 uL of each compound dilution were robotically pipetted to Costar serocluster plates maintaining the same plate layout. All assay mixtures consisted... | US Patent US8754233 (2014) BindingDB Entry DOI: 10.7270/Q23N2231 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ribosomal protein S6 kinase alpha-2 (Homo sapiens (Human)) | BDBM286089 ((R)¿N-(1-(3-aminobenzyl)-1H-pyrazol-4-yl)-9-methyl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 23 | n/a | n/a | n/a | n/a | n/a | n/a |
PHOENIX MOLECULAR DESIGNS US Patent | Assay Description Radioisotope assays were performed for the evaluation of the kinase target profiling and all assays were performed in a designated radioactive workin... | US Patent US10758530 (2020) BindingDB Entry DOI: 10.7270/Q20R9SGD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ribosomal protein S6 kinase alpha-1 (Homo sapiens (Human)) | BDBM342166 ((R)-1-benzyl-N-(9-methyl-6-oxo-6,7,8,9-tetrahydrop...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 23.6 | n/a | n/a | n/a | n/a | n/a | n/a |
PHOENIX MOLECULAR DESIGN US Patent | Assay Description Radioisotope assays (SignalChem) were performed for the evaluation of the kinase target profiling and all assays were performed in a designated radio... | US Patent US9771366 (2017) BindingDB Entry DOI: 10.7270/Q2862JK5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ribosomal protein S6 kinase alpha-1 (Homo sapiens (Human)) | BDBM458758 ((R)-1-benzyl-N-(9-methyl-6-oxo-6,7,8,9-tetrahydrop...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 23.6 | n/a | n/a | n/a | n/a | n/a | n/a |
PHOENIX MOLECULAR DESIGNS US Patent | Assay Description Radioisotope assays were performed for the evaluation of the kinase target profiling and all assays were performed in a designated radioactive workin... | US Patent US10758530 (2020) BindingDB Entry DOI: 10.7270/Q20R9SGD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin-linked protein kinase (Homo sapiens (Human)) | BDBM124001 (US8754233, 4-(5-Fluoro-benzothiazol-2-yl)-5-methyl...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 40 | n/a | n/a | n/a | n/a | n/a | 40 |
Dermira (Canada), Inc. US Patent | Assay Description 5 uL of each compound dilution were robotically pipetted to Costar serocluster plates maintaining the same plate layout. All assay mixtures consisted... | US Patent US8754233 (2014) BindingDB Entry DOI: 10.7270/Q23N2231 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin-linked protein kinase (Homo sapiens (Human)) | BDBM123992 (US8754233, 4-(5-Fluoro-6-methoxy-benzothiazol-2-yl...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 40 | n/a | n/a | n/a | n/a | n/a | 40 |
Dermira (Canada), Inc. US Patent | Assay Description 5 uL of each compound dilution were robotically pipetted to Costar serocluster plates maintaining the same plate layout. All assay mixtures consisted... | US Patent US8754233 (2014) BindingDB Entry DOI: 10.7270/Q23N2231 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin-linked protein kinase (Homo sapiens (Human)) | BDBM123933 (US8754233, 2-(3-Amino-5-methyl-1H-pyrazol-4-yl)-5-...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 40 | n/a | n/a | n/a | n/a | n/a | 40 |
Dermira (Canada), Inc. US Patent | Assay Description 5 uL of each compound dilution were robotically pipetted to Costar serocluster plates maintaining the same plate layout. All assay mixtures consisted... | US Patent US8754233 (2014) BindingDB Entry DOI: 10.7270/Q23N2231 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin-linked protein kinase (Homo sapiens (Human)) | BDBM123943 (US8754233, 2-(5-Amino-3-methyl-1H-pyrazol-4-yl)-4-...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 40 | n/a | n/a | n/a | n/a | n/a | 40 |
Dermira (Canada), Inc. US Patent | Assay Description 5 uL of each compound dilution were robotically pipetted to Costar serocluster plates maintaining the same plate layout. All assay mixtures consisted... | US Patent US8754233 (2014) BindingDB Entry DOI: 10.7270/Q23N2231 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin-linked protein kinase (Homo sapiens (Human)) | BDBM123965 (US8754233, 2-(5-Amino-3-methyl-1H-pyrazol-4-yl)-be...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 40 | n/a | n/a | n/a | n/a | n/a | 40 |
Dermira (Canada), Inc. US Patent | Assay Description 5 uL of each compound dilution were robotically pipetted to Costar serocluster plates maintaining the same plate layout. All assay mixtures consisted... | US Patent US8754233 (2014) BindingDB Entry DOI: 10.7270/Q23N2231 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin-linked protein kinase (Homo sapiens (Human)) | BDBM123969 (US8754233, 2-(5-Amino-3-pyridin-4-yl-1H-pyrazol-4-...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 50 | n/a | n/a | n/a | n/a | n/a | 40 |
Dermira (Canada), Inc. US Patent | Assay Description 5 uL of each compound dilution were robotically pipetted to Costar serocluster plates maintaining the same plate layout. All assay mixtures consisted... | US Patent US8754233 (2014) BindingDB Entry DOI: 10.7270/Q23N2231 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin-linked protein kinase (Homo sapiens (Human)) | BDBM123999 (US8754233, 4-(5-Fluoro-6-methyl-benzothiazol-2-yl)...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 50 | n/a | n/a | n/a | n/a | n/a | 40 |
Dermira (Canada), Inc. US Patent | Assay Description 5 uL of each compound dilution were robotically pipetted to Costar serocluster plates maintaining the same plate layout. All assay mixtures consisted... | US Patent US8754233 (2014) BindingDB Entry DOI: 10.7270/Q23N2231 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin-linked protein kinase (Homo sapiens (Human)) | BDBM123946 (US8754233, 2-(5-Amino-3-methyl-1H-pyrazol-4-yl)-5-...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 50 | n/a | n/a | n/a | n/a | n/a | 40 |
Dermira (Canada), Inc. US Patent | Assay Description 5 uL of each compound dilution were robotically pipetted to Costar serocluster plates maintaining the same plate layout. All assay mixtures consisted... | US Patent US8754233 (2014) BindingDB Entry DOI: 10.7270/Q23N2231 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin-linked protein kinase (Homo sapiens (Human)) | BDBM123994 (US8754233, 4-(5-Fluoro-6-methoxy-benzothiazol-2-yl...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 60 | n/a | n/a | n/a | n/a | n/a | 40 |
Dermira (Canada), Inc. US Patent | Assay Description 5 uL of each compound dilution were robotically pipetted to Costar serocluster plates maintaining the same plate layout. All assay mixtures consisted... | US Patent US8754233 (2014) BindingDB Entry DOI: 10.7270/Q23N2231 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin-linked protein kinase (Homo sapiens (Human)) | BDBM124033 (US8754233, 4-Benzothiazol-2-yl-5-piperidin-4-yl-2H...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 60 | n/a | n/a | n/a | n/a | n/a | 40 |
Dermira (Canada), Inc. US Patent | Assay Description 5 uL of each compound dilution were robotically pipetted to Costar serocluster plates maintaining the same plate layout. All assay mixtures consisted... | US Patent US8754233 (2014) BindingDB Entry DOI: 10.7270/Q23N2231 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin-linked protein kinase (Homo sapiens (Human)) | BDBM123932 (US8754233, 2-(3-Amino-5-methyl-1H-pyrazol-4-yl)-5-...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 60 | n/a | n/a | n/a | n/a | n/a | 40 |
Dermira (Canada), Inc. US Patent | Assay Description 5 uL of each compound dilution were robotically pipetted to Costar serocluster plates maintaining the same plate layout. All assay mixtures consisted... | US Patent US8754233 (2014) BindingDB Entry DOI: 10.7270/Q23N2231 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin-linked protein kinase (Homo sapiens (Human)) | BDBM123942 (US8754233, 2-(5-Amino-1H-pyrazol-4-yl)-benzothiazo...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 60 | n/a | n/a | n/a | n/a | n/a | 40 |
Dermira (Canada), Inc. US Patent | Assay Description 5 uL of each compound dilution were robotically pipetted to Costar serocluster plates maintaining the same plate layout. All assay mixtures consisted... | US Patent US8754233 (2014) BindingDB Entry DOI: 10.7270/Q23N2231 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin-linked protein kinase (Homo sapiens (Human)) | BDBM123931 (US8754233, 2-(3-Amino-5-methyl-1H-pyrazol-4-yl)-4,...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 70 | n/a | n/a | n/a | n/a | n/a | 40 |
Dermira (Canada), Inc. US Patent | Assay Description 5 uL of each compound dilution were robotically pipetted to Costar serocluster plates maintaining the same plate layout. All assay mixtures consisted... | US Patent US8754233 (2014) BindingDB Entry DOI: 10.7270/Q23N2231 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin-linked protein kinase (Homo sapiens (Human)) | BDBM123996 (US8754233, 4-(5-Fluoro-6-methoxy-benzothiazol-2-yl...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 70 | n/a | n/a | n/a | n/a | n/a | 40 |
Dermira (Canada), Inc. US Patent | Assay Description 5 uL of each compound dilution were robotically pipetted to Costar serocluster plates maintaining the same plate layout. All assay mixtures consisted... | US Patent US8754233 (2014) BindingDB Entry DOI: 10.7270/Q23N2231 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin-linked protein kinase (Homo sapiens (Human)) | BDBM123936 (US8754233, 2-(3-Amino-5-methyl-1H-pyrazol-4-yl)-be...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 70 | n/a | n/a | n/a | n/a | n/a | 40 |
Dermira (Canada), Inc. US Patent | Assay Description 5 uL of each compound dilution were robotically pipetted to Costar serocluster plates maintaining the same plate layout. All assay mixtures consisted... | US Patent US8754233 (2014) BindingDB Entry DOI: 10.7270/Q23N2231 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin-linked protein kinase (Homo sapiens (Human)) | BDBM123962 (US8754233, 2-(5-Amino-3-methyl-1H-pyrazol-4-yl)-be...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 90 | n/a | n/a | n/a | n/a | n/a | 40 |
Dermira (Canada), Inc. US Patent | Assay Description 5 uL of each compound dilution were robotically pipetted to Costar serocluster plates maintaining the same plate layout. All assay mixtures consisted... | US Patent US8754233 (2014) BindingDB Entry DOI: 10.7270/Q23N2231 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ribosomal protein S6 kinase alpha-2 (Homo sapiens (Human)) | BDBM458758 ((R)-1-benzyl-N-(9-methyl-6-oxo-6,7,8,9-tetrahydrop...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 94 | n/a | n/a | n/a | n/a | n/a | n/a |
PHOENIX MOLECULAR DESIGNS US Patent | Assay Description Radioisotope assays were performed for the evaluation of the kinase target profiling and all assays were performed in a designated radioactive workin... | US Patent US10758530 (2020) BindingDB Entry DOI: 10.7270/Q20R9SGD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin-linked protein kinase (Homo sapiens (Human)) | BDBM124028 (US8754233, 4-Benzothiazol-2-yl-5-furan-2-yl-2H-pyr...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 100 | n/a | n/a | n/a | n/a | n/a | 40 |
Dermira (Canada), Inc. US Patent | Assay Description 5 uL of each compound dilution were robotically pipetted to Costar serocluster plates maintaining the same plate layout. All assay mixtures consisted... | US Patent US8754233 (2014) BindingDB Entry DOI: 10.7270/Q23N2231 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin-linked protein kinase (Homo sapiens (Human)) | BDBM124024 (US8754233, 4-Benzothiazol-2-yl-5-(4-methylamino-bu...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 100 | n/a | n/a | n/a | n/a | n/a | 40 |
Dermira (Canada), Inc. US Patent | Assay Description 5 uL of each compound dilution were robotically pipetted to Costar serocluster plates maintaining the same plate layout. All assay mixtures consisted... | US Patent US8754233 (2014) BindingDB Entry DOI: 10.7270/Q23N2231 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin-linked protein kinase (Homo sapiens (Human)) | BDBM124053 (US8754233, 5-(4-Amino-phenyl)-4-benzothiazol-2-yl-...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 100 | n/a | n/a | n/a | n/a | n/a | 40 |
Dermira (Canada), Inc. US Patent | Assay Description 5 uL of each compound dilution were robotically pipetted to Costar serocluster plates maintaining the same plate layout. All assay mixtures consisted... | US Patent US8754233 (2014) BindingDB Entry DOI: 10.7270/Q23N2231 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin-linked protein kinase (Homo sapiens (Human)) | BDBM124035 (US8754233, 4-Benzothiazol-2-yl-5-pyridin-4-yl-2H-p...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 100 | n/a | n/a | n/a | n/a | n/a | 40 |
Dermira (Canada), Inc. US Patent | Assay Description 5 uL of each compound dilution were robotically pipetted to Costar serocluster plates maintaining the same plate layout. All assay mixtures consisted... | US Patent US8754233 (2014) BindingDB Entry DOI: 10.7270/Q23N2231 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin-linked protein kinase (Homo sapiens (Human)) | BDBM123925 (US8754233, [2-(3-Amino-5-methyl-1H-pyrazol-4-yl)-5...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 100 | n/a | n/a | n/a | n/a | n/a | 40 |
Dermira (Canada), Inc. US Patent | Assay Description 5 uL of each compound dilution were robotically pipetted to Costar serocluster plates maintaining the same plate layout. All assay mixtures consisted... | US Patent US8754233 (2014) BindingDB Entry DOI: 10.7270/Q23N2231 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin-linked protein kinase (Homo sapiens (Human)) | BDBM123993 (US8754233, 4-(5-Fluoro-6-methoxy-benzothiazol-2-yl...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 100 | n/a | n/a | n/a | n/a | n/a | 40 |
Dermira (Canada), Inc. US Patent | Assay Description 5 uL of each compound dilution were robotically pipetted to Costar serocluster plates maintaining the same plate layout. All assay mixtures consisted... | US Patent US8754233 (2014) BindingDB Entry DOI: 10.7270/Q23N2231 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin-linked protein kinase (Homo sapiens (Human)) | BDBM123972 (US8754233, 2-{[2-(5-Amino-3-methyl-1H-pyrazol-4-yl...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 100 | n/a | n/a | n/a | n/a | n/a | 40 |
Dermira (Canada), Inc. US Patent | Assay Description 5 uL of each compound dilution were robotically pipetted to Costar serocluster plates maintaining the same plate layout. All assay mixtures consisted... | US Patent US8754233 (2014) BindingDB Entry DOI: 10.7270/Q23N2231 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ribosomal protein S6 kinase alpha-2 (Homo sapiens (Human)) | BDBM286092 ((R)-1-(3-aminobenzyl)-N-(9-methyl-6-oxo-6,7,8,9-te...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 123 | n/a | n/a | n/a | n/a | n/a | n/a |
PHOENIX MOLECULAR DESIGNS US Patent | Assay Description Radioisotope assays were performed for the evaluation of the kinase target profiling and all assays were performed in a designated radioactive workin... | US Patent US10758530 (2020) BindingDB Entry DOI: 10.7270/Q20R9SGD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ribosomal protein S6 kinase alpha-2 (Homo sapiens (Human)) | BDBM286093 ((R)-9-methyl-N-(1-((1-methylpiperidin-4-yl)methyl)...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 124 | n/a | n/a | n/a | n/a | n/a | n/a |
PHOENIX MOLECULAR DESIGNS US Patent | Assay Description Radioisotope assays were performed for the evaluation of the kinase target profiling and all assays were performed in a designated radioactive workin... | US Patent US10758530 (2020) BindingDB Entry DOI: 10.7270/Q20R9SGD | |||||||||||
More data for this Ligand-Target Pair |
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