Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Delta-type opioid receptor (Homo sapiens (Human)) | BDBM50306288 (4-(1-(cyclopropylmethyl)-3-(3-hydroxyphenyl)piperi...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 0.800 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [125I]diprenorphine from human delta opioid receptor expressed in CHO cells by liquid scintillation counting | Bioorg Med Chem Lett 20: 503-7 (2010) Article DOI: 10.1016/j.bmcl.2009.11.113 BindingDB Entry DOI: 10.7270/Q2C53KX1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Delta-type opioid receptor (Homo sapiens (Human)) | BDBM50306298 (CHEMBL595472 | N,N-diethyl-4-(4-(3-hydroxyphenyl)-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 0.900 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [125I]diprenorphine from human delta opioid receptor expressed in CHO cells by liquid scintillation counting | Bioorg Med Chem Lett 20: 503-7 (2010) Article DOI: 10.1016/j.bmcl.2009.11.113 BindingDB Entry DOI: 10.7270/Q2C53KX1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kappa-type opioid receptor (Homo sapiens (Human)) | BDBM50086359 (CHEMBL147191 | N-Cyclohexylmethyl-2,2-dimethyl-3-m...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 1.20 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Inc Curated by ChEMBL | Assay Description Inhibition of [3H]U-69,593 binding to human Opioid receptor kappa 1 expressed in HEK 293 cells | Bioorg Med Chem Lett 10: 523-6 (2000) BindingDB Entry DOI: 10.7270/Q2BG2N79 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Delta-type opioid receptor (Homo sapiens (Human)) | BDBM50306293 (4-(1-((1H-imidazol-2-yl)methyl)-3-(3-hydroxyphenyl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | 1.20 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [125I]diprenorphine from human delta opioid receptor expressed in CHO cells by liquid scintillation counting | Bioorg Med Chem Lett 20: 503-7 (2010) Article DOI: 10.1016/j.bmcl.2009.11.113 BindingDB Entry DOI: 10.7270/Q2C53KX1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kappa-type opioid receptor (Homo sapiens (Human)) | BDBM50000788 ((morphine)4-methyl-(1S,5R,13R,14S,17R)-12-oxa-4-az...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase DrugBank MCE KEGG PC cid PC sid UniChem Patents Similars | DrugBank PubMed | 1.20 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Inc Curated by ChEMBL | Assay Description Inhibition of [3H]U-69,593 binding to human Opioid receptor kappa 1 expressed in HEK 293 cells | Bioorg Med Chem Lett 10: 523-6 (2000) BindingDB Entry DOI: 10.7270/Q2BG2N79 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kappa-type opioid receptor (Homo sapiens (Human)) | BDBM50086361 (3-(3-Hydroxy-phenyl)-2,2-dimethyl-3-methylamino-N-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | 1.30 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Inc Curated by ChEMBL | Assay Description Inhibition of [3H]U-69,593 binding to human Opioid receptor kappa 1 expressed in HEK 293 cells | Bioorg Med Chem Lett 10: 523-6 (2000) BindingDB Entry DOI: 10.7270/Q2BG2N79 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid receptor (Rattus norvegicus (rat)) | BDBM50086367 (3-(3-Hydroxy-phenyl)-2,2-dimethyl-3-methylamino-N-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | 1.40 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Inc Curated by ChEMBL | Assay Description Inhibition of [3H]-DAMGO binding to rat Opioid receptor mu 1 | Bioorg Med Chem Lett 10: 523-6 (2000) BindingDB Entry DOI: 10.7270/Q2BG2N79 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid receptor (Rattus norvegicus (rat)) | BDBM50000788 ((morphine)4-methyl-(1S,5R,13R,14S,17R)-12-oxa-4-az...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase DrugBank MCE KEGG PC cid PC sid UniChem Patents Similars | PubMed | 1.40 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Inc Curated by ChEMBL | Assay Description Inhibition of [3H]-DAMGO binding to rat Opioid receptor mu 1 | Bioorg Med Chem Lett 10: 523-6 (2000) BindingDB Entry DOI: 10.7270/Q2BG2N79 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid receptor (Rattus norvegicus (rat)) | BDBM50086361 (3-(3-Hydroxy-phenyl)-2,2-dimethyl-3-methylamino-N-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | 1.40 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Inc Curated by ChEMBL | Assay Description Inhibition of [3H]-DAMGO binding to rat Opioid receptor mu 1 | Bioorg Med Chem Lett 10: 523-6 (2000) BindingDB Entry DOI: 10.7270/Q2BG2N79 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Delta-type opioid receptor (Homo sapiens (Human)) | BDBM50306299 (CHEMBL595473 | N,N-diethyl-4-(4-(3-hydroxyphenyl)-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.80 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [125I]diprenorphine from human delta opioid receptor expressed in CHO cells by liquid scintillation counting | Bioorg Med Chem Lett 20: 503-7 (2010) Article DOI: 10.1016/j.bmcl.2009.11.113 BindingDB Entry DOI: 10.7270/Q2C53KX1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Delta-type opioid receptor (Homo sapiens (Human)) | BDBM50306297 (4-(1-allyl-4-(3-hydroxyphenyl)piperidin-4-yl)-N,N-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.90 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [125I]diprenorphine from human delta opioid receptor expressed in CHO cells by liquid scintillation counting | Bioorg Med Chem Lett 20: 503-7 (2010) Article DOI: 10.1016/j.bmcl.2009.11.113 BindingDB Entry DOI: 10.7270/Q2C53KX1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Delta-type opioid receptor (Homo sapiens (Human)) | BDBM50306287 (3-(4-(4-(3-hydroxypentan-3-yl)phenyl)-1-(2-methylp...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [125I]diprenorphine from human delta opioid receptor expressed in CHO cells by liquid scintillation counting | Bioorg Med Chem Lett 20: 503-7 (2010) Article DOI: 10.1016/j.bmcl.2009.11.113 BindingDB Entry DOI: 10.7270/Q2C53KX1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Delta-type opioid receptor (Homo sapiens (Human)) | BDBM50306290 (4-(1-(cyclopropylmethyl)-3-(3-hydroxyphenyl)piperi...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 2.20 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [125I]diprenorphine from human delta opioid receptor expressed in CHO cells by liquid scintillation counting | Bioorg Med Chem Lett 20: 503-7 (2010) Article DOI: 10.1016/j.bmcl.2009.11.113 BindingDB Entry DOI: 10.7270/Q2C53KX1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Delta-type opioid receptor (Homo sapiens (Human)) | BDBM50306301 (3-(1-(cyclopropylmethyl)-4-(4-(3-hydroxypentan-3-y...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2.30 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [125I]diprenorphine from human delta opioid receptor expressed in CHO cells by liquid scintillation counting | Bioorg Med Chem Lett 20: 503-7 (2010) Article DOI: 10.1016/j.bmcl.2009.11.113 BindingDB Entry DOI: 10.7270/Q2C53KX1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Delta-type opioid receptor (Homo sapiens (Human)) | BDBM50306291 (CHEMBL595714 | N,N-diethyl-4-(3-(3-hydroxyphenyl)-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2.90 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [125I]diprenorphine from human delta opioid receptor expressed in CHO cells by liquid scintillation counting | Bioorg Med Chem Lett 20: 503-7 (2010) Article DOI: 10.1016/j.bmcl.2009.11.113 BindingDB Entry DOI: 10.7270/Q2C53KX1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kappa-type opioid receptor (Homo sapiens (Human)) | BDBM50086363 (3-(Cyclopropylmethyl-methyl-amino)-3-(3-hydroxy-ph...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | 2.90 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Inc Curated by ChEMBL | Assay Description Inhibition of [3H]U-69,593 binding to human Opioid receptor kappa 1 expressed in HEK 293 cells | Bioorg Med Chem Lett 10: 523-6 (2000) BindingDB Entry DOI: 10.7270/Q2BG2N79 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Delta-type opioid receptor (Homo sapiens (Human)) | BDBM50306292 (CHEMBL605735 | N,N-diethyl-4-(3-(3-hydroxyphenyl)-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 3.5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [125I]diprenorphine from human delta opioid receptor expressed in CHO cells by liquid scintillation counting | Bioorg Med Chem Lett 20: 503-7 (2010) Article DOI: 10.1016/j.bmcl.2009.11.113 BindingDB Entry DOI: 10.7270/Q2C53KX1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kappa-type opioid receptor (Homo sapiens (Human)) | BDBM50086366 (3-(3-Hydroxy-phenyl)-2,2-dimethyl-3-methylamino-N-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | 3.60 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Inc Curated by ChEMBL | Assay Description Inhibition of [3H]U-69,593 binding to human Opioid receptor kappa 1 expressed in HEK 293 cells | Bioorg Med Chem Lett 10: 523-6 (2000) BindingDB Entry DOI: 10.7270/Q2BG2N79 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid receptor (Rattus norvegicus (rat)) | BDBM50086360 (CHEMBL347531 | N-Cyclohexylmethyl-3-(3-hydroxy-phe...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | 4.40 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Inc Curated by ChEMBL | Assay Description Inhibition of [3H]-DAMGO binding to rat Opioid receptor mu 1 | Bioorg Med Chem Lett 10: 523-6 (2000) BindingDB Entry DOI: 10.7270/Q2BG2N79 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kappa-type opioid receptor (Homo sapiens (Human)) | BDBM50086364 (CHEMBL146750 | N-Benzyl-3-(3-hydroxy-phenyl)-2,2-d...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | 5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Inc Curated by ChEMBL | Assay Description Inhibition of [3H]U-69,593 binding to human Opioid receptor kappa 1 expressed in HEK 293 cells | Bioorg Med Chem Lett 10: 523-6 (2000) BindingDB Entry DOI: 10.7270/Q2BG2N79 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kappa-type opioid receptor (Homo sapiens (Human)) | BDBM50086360 (CHEMBL347531 | N-Cyclohexylmethyl-3-(3-hydroxy-phe...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | 5.70 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Inc Curated by ChEMBL | Assay Description Inhibition of [3H]U-69,593 binding to human Opioid receptor kappa 1 expressed in HEK 293 cells | Bioorg Med Chem Lett 10: 523-6 (2000) BindingDB Entry DOI: 10.7270/Q2BG2N79 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Delta-type opioid receptor (Homo sapiens (Human)) | BDBM50306289 (4-(1-butyl-3-(3-hydroxyphenyl)piperidin-3-yl)-N,N-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 6.20 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [125I]diprenorphine from human delta opioid receptor expressed in CHO cells by liquid scintillation counting | Bioorg Med Chem Lett 20: 503-7 (2010) Article DOI: 10.1016/j.bmcl.2009.11.113 BindingDB Entry DOI: 10.7270/Q2C53KX1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kappa-type opioid receptor (Homo sapiens (Human)) | BDBM50086367 (3-(3-Hydroxy-phenyl)-2,2-dimethyl-3-methylamino-N-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | 6.30 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Inc Curated by ChEMBL | Assay Description Inhibition of [3H]U-69,593 binding to human Opioid receptor kappa 1 expressed in HEK 293 cells | Bioorg Med Chem Lett 10: 523-6 (2000) BindingDB Entry DOI: 10.7270/Q2BG2N79 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Delta-type opioid receptor (Homo sapiens (Human)) | BDBM50306295 (4-(3-(3-carbamoylphenyl)-1-(thiazol-2-ylmethyl)pip...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 7 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [125I]diprenorphine from human delta opioid receptor expressed in CHO cells by liquid scintillation counting | Bioorg Med Chem Lett 20: 503-7 (2010) Article DOI: 10.1016/j.bmcl.2009.11.113 BindingDB Entry DOI: 10.7270/Q2C53KX1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid receptor (Rattus norvegicus (rat)) | BDBM50086364 (CHEMBL146750 | N-Benzyl-3-(3-hydroxy-phenyl)-2,2-d...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | 8.70 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Inc Curated by ChEMBL | Assay Description Inhibition of [3H]-DAMGO binding to rat Opioid receptor mu 1 | Bioorg Med Chem Lett 10: 523-6 (2000) BindingDB Entry DOI: 10.7270/Q2BG2N79 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Delta-type opioid receptor (Homo sapiens (Human)) | BDBM50306296 (4-(1-(cyclopropylmethyl)-4-(3-hydroxyphenyl)piperi...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 9 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [125I]diprenorphine from human delta opioid receptor expressed in CHO cells by liquid scintillation counting | Bioorg Med Chem Lett 20: 503-7 (2010) Article DOI: 10.1016/j.bmcl.2009.11.113 BindingDB Entry DOI: 10.7270/Q2C53KX1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Delta-type opioid receptor (Homo sapiens (Human)) | BDBM50306300 (4-(4-(3-hydroxyphenyl)-1-(2-methylpentyl)piperidin...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 11 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [125I]diprenorphine from human delta opioid receptor expressed in CHO cells by liquid scintillation counting | Bioorg Med Chem Lett 20: 503-7 (2010) Article DOI: 10.1016/j.bmcl.2009.11.113 BindingDB Entry DOI: 10.7270/Q2C53KX1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid receptor (Rattus norvegicus (rat)) | BDBM50086366 (3-(3-Hydroxy-phenyl)-2,2-dimethyl-3-methylamino-N-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | 12 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Inc Curated by ChEMBL | Assay Description Inhibition of [3H]-DAMGO binding to rat Opioid receptor mu 1 | Bioorg Med Chem Lett 10: 523-6 (2000) BindingDB Entry DOI: 10.7270/Q2BG2N79 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid receptor (Rattus norvegicus (rat)) | BDBM50086357 (2,2-Dimethyl-3-methylamino-N-phenethyl-3-phenyl-pr...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 13 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Inc Curated by ChEMBL | Assay Description Inhibition of [3H]-DAMGO binding to rat Opioid receptor mu 1 | Bioorg Med Chem Lett 10: 523-6 (2000) BindingDB Entry DOI: 10.7270/Q2BG2N79 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kappa-type opioid receptor (Homo sapiens (Human)) | BDBM50306291 (CHEMBL595714 | N,N-diethyl-4-(3-(3-hydroxyphenyl)-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 24 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [125I]diprenorphine from human kappa opioid receptor expressed in CHO cells by liquid scintillation counting | Bioorg Med Chem Lett 20: 503-7 (2010) Article DOI: 10.1016/j.bmcl.2009.11.113 BindingDB Entry DOI: 10.7270/Q2C53KX1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kappa-type opioid receptor (Homo sapiens (Human)) | BDBM50306288 (4-(1-(cyclopropylmethyl)-3-(3-hydroxyphenyl)piperi...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 24 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [125I]diprenorphine from human kappa opioid receptor expressed in CHO cells by liquid scintillation counting | Bioorg Med Chem Lett 20: 503-7 (2010) Article DOI: 10.1016/j.bmcl.2009.11.113 BindingDB Entry DOI: 10.7270/Q2C53KX1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid receptor (Rattus norvegicus (rat)) | BDBM50086365 (3-(Butyl-methyl-amino)-3-(3-hydroxy-phenyl)-2,2-di...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 26 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Inc Curated by ChEMBL | Assay Description Inhibition of [3H]-DAMGO binding to rat Opioid receptor mu 1 | Bioorg Med Chem Lett 10: 523-6 (2000) BindingDB Entry DOI: 10.7270/Q2BG2N79 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid receptor (Rattus norvegicus (rat)) | BDBM50086363 (3-(Cyclopropylmethyl-methyl-amino)-3-(3-hydroxy-ph...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | 28 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Inc Curated by ChEMBL | Assay Description Inhibition of [3H]-DAMGO binding to rat Opioid receptor mu 1 | Bioorg Med Chem Lett 10: 523-6 (2000) BindingDB Entry DOI: 10.7270/Q2BG2N79 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid receptor (Homo sapiens (Human)) | BDBM50306288 (4-(1-(cyclopropylmethyl)-3-(3-hydroxyphenyl)piperi...) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 35 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [125I]diprenorphine from human mu opioid receptor expressed in CHO cells by liquid scintillation counting | Bioorg Med Chem Lett 20: 503-7 (2010) Article DOI: 10.1016/j.bmcl.2009.11.113 BindingDB Entry DOI: 10.7270/Q2C53KX1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Delta-type opioid receptor (Homo sapiens (Human)) | BDBM50306294 (3-(1-(cyclopropylmethyl)-3-(4-(2-hydroxypropan-2-y...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 39 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [125I]diprenorphine from human delta opioid receptor expressed in CHO cells by liquid scintillation counting | Bioorg Med Chem Lett 20: 503-7 (2010) Article DOI: 10.1016/j.bmcl.2009.11.113 BindingDB Entry DOI: 10.7270/Q2C53KX1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Delta-type opioid receptor (Homo sapiens (Human)) | BDBM50000788 ((morphine)4-methyl-(1S,5R,13R,14S,17R)-12-oxa-4-az...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase DrugBank MCE KEGG PC cid PC sid UniChem Patents Similars | DrugBank PubMed | 41 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Inc Curated by ChEMBL | Assay Description Inhibition of [3H]-naltrindole binding to human Opioid receptor delta 1 in CHO cells | Bioorg Med Chem Lett 10: 523-6 (2000) BindingDB Entry DOI: 10.7270/Q2BG2N79 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kappa-type opioid receptor (Homo sapiens (Human)) | BDBM50306294 (3-(1-(cyclopropylmethyl)-3-(4-(2-hydroxypropan-2-y...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 41 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [125I]diprenorphine from human kappa opioid receptor expressed in CHO cells by liquid scintillation counting | Bioorg Med Chem Lett 20: 503-7 (2010) Article DOI: 10.1016/j.bmcl.2009.11.113 BindingDB Entry DOI: 10.7270/Q2C53KX1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kappa-type opioid receptor (Homo sapiens (Human)) | BDBM50306287 (3-(4-(4-(3-hydroxypentan-3-yl)phenyl)-1-(2-methylp...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 45 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [125I]diprenorphine from human kappa opioid receptor expressed in CHO cells by liquid scintillation counting | Bioorg Med Chem Lett 20: 503-7 (2010) Article DOI: 10.1016/j.bmcl.2009.11.113 BindingDB Entry DOI: 10.7270/Q2C53KX1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kappa-type opioid receptor (Homo sapiens (Human)) | BDBM50086357 (2,2-Dimethyl-3-methylamino-N-phenethyl-3-phenyl-pr...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 49 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Inc Curated by ChEMBL | Assay Description Inhibition of [3H]U-69,593 binding to human Opioid receptor kappa 1 expressed in HEK 293 cells | Bioorg Med Chem Lett 10: 523-6 (2000) BindingDB Entry DOI: 10.7270/Q2BG2N79 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid receptor (Homo sapiens (Human)) | BDBM50306290 (4-(1-(cyclopropylmethyl)-3-(3-hydroxyphenyl)piperi...) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 52 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [125I]diprenorphine from human mu opioid receptor expressed in CHO cells by liquid scintillation counting | Bioorg Med Chem Lett 20: 503-7 (2010) Article DOI: 10.1016/j.bmcl.2009.11.113 BindingDB Entry DOI: 10.7270/Q2C53KX1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kappa-type opioid receptor (Homo sapiens (Human)) | BDBM50306290 (4-(1-(cyclopropylmethyl)-3-(3-hydroxyphenyl)piperi...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 66 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [125I]diprenorphine from human kappa opioid receptor expressed in CHO cells by liquid scintillation counting | Bioorg Med Chem Lett 20: 503-7 (2010) Article DOI: 10.1016/j.bmcl.2009.11.113 BindingDB Entry DOI: 10.7270/Q2C53KX1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid receptor (Homo sapiens (Human)) | BDBM50306298 (CHEMBL595472 | N,N-diethyl-4-(4-(3-hydroxyphenyl)-...) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 67 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [125I]diprenorphine from human mu opioid receptor expressed in CHO cells by liquid scintillation counting | Bioorg Med Chem Lett 20: 503-7 (2010) Article DOI: 10.1016/j.bmcl.2009.11.113 BindingDB Entry DOI: 10.7270/Q2C53KX1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kappa-type opioid receptor (Homo sapiens (Human)) | BDBM50086358 (CHEMBL347316 | N-Cyclopropylmethyl-3-(3-hydroxy-ph...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | 75 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Inc Curated by ChEMBL | Assay Description Inhibition of [3H]U-69,593 binding to human Opioid receptor kappa 1 expressed in HEK 293 cells | Bioorg Med Chem Lett 10: 523-6 (2000) BindingDB Entry DOI: 10.7270/Q2BG2N79 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kappa-type opioid receptor (Homo sapiens (Human)) | BDBM50086365 (3-(Butyl-methyl-amino)-3-(3-hydroxy-phenyl)-2,2-di...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 75 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Inc Curated by ChEMBL | Assay Description Inhibition of [3H]U-69,593 binding to human Opioid receptor kappa 1 expressed in HEK 293 cells | Bioorg Med Chem Lett 10: 523-6 (2000) BindingDB Entry DOI: 10.7270/Q2BG2N79 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kappa-type opioid receptor (Homo sapiens (Human)) | BDBM50306301 (3-(1-(cyclopropylmethyl)-4-(4-(3-hydroxypentan-3-y...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 79 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [125I]diprenorphine from human kappa opioid receptor expressed in CHO cells by liquid scintillation counting | Bioorg Med Chem Lett 20: 503-7 (2010) Article DOI: 10.1016/j.bmcl.2009.11.113 BindingDB Entry DOI: 10.7270/Q2C53KX1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid receptor (Rattus norvegicus (rat)) | BDBM50086359 (CHEMBL147191 | N-Cyclohexylmethyl-2,2-dimethyl-3-m...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 85 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Inc Curated by ChEMBL | Assay Description Inhibition of [3H]-DAMGO binding to rat Opioid receptor mu 1 | Bioorg Med Chem Lett 10: 523-6 (2000) BindingDB Entry DOI: 10.7270/Q2BG2N79 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kappa-type opioid receptor (Homo sapiens (Human)) | BDBM50306298 (CHEMBL595472 | N,N-diethyl-4-(4-(3-hydroxyphenyl)-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 95 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [125I]diprenorphine from human kappa opioid receptor expressed in CHO cells by liquid scintillation counting | Bioorg Med Chem Lett 20: 503-7 (2010) Article DOI: 10.1016/j.bmcl.2009.11.113 BindingDB Entry DOI: 10.7270/Q2C53KX1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid receptor (Rattus norvegicus (rat)) | BDBM50086362 (CHEMBL149143 | N-Benzyl-2,2-dimethyl-3-methylamino...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 95 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Inc Curated by ChEMBL | Assay Description Inhibition of [3H]-DAMGO binding to rat Opioid receptor mu 1 | Bioorg Med Chem Lett 10: 523-6 (2000) BindingDB Entry DOI: 10.7270/Q2BG2N79 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid receptor (Homo sapiens (Human)) | BDBM50306294 (3-(1-(cyclopropylmethyl)-3-(4-(2-hydroxypropan-2-y...) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 110 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [125I]diprenorphine from human mu opioid receptor expressed in CHO cells by liquid scintillation counting | Bioorg Med Chem Lett 20: 503-7 (2010) Article DOI: 10.1016/j.bmcl.2009.11.113 BindingDB Entry DOI: 10.7270/Q2C53KX1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kappa-type opioid receptor (Homo sapiens (Human)) | BDBM50306300 (4-(4-(3-hydroxyphenyl)-1-(2-methylpentyl)piperidin...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 150 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [125I]diprenorphine from human kappa opioid receptor expressed in CHO cells by liquid scintillation counting | Bioorg Med Chem Lett 20: 503-7 (2010) Article DOI: 10.1016/j.bmcl.2009.11.113 BindingDB Entry DOI: 10.7270/Q2C53KX1 | |||||||||||
More data for this Ligand-Target Pair |
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