Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Pyruvate kinase (Staphylococcus aureus (strain MRSA252)) | BDBM50210347 (CHEMBL3921820) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2 | n/a | n/a | n/a | n/a | n/a | n/a |
Simon Fraser University Curated by ChEMBL | Assay Description Inhibition of recombinant N-terminal His-tagged methicillin-resistant Staphylococcus aureus MRSA252 pyruvate kinase expressed in Escherichia coli BL2... | Eur J Med Chem 125: 1-13 (2017) Article DOI: 10.1016/j.ejmech.2016.09.018 BindingDB Entry DOI: 10.7270/Q2CC12P0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Pyruvate kinase (Staphylococcus aureus (strain MRSA252)) | BDBM50210348 (CHEMBL3949603) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3 | n/a | n/a | n/a | n/a | n/a | n/a |
Simon Fraser University Curated by ChEMBL | Assay Description Inhibition of recombinant N-terminal His-tagged methicillin-resistant Staphylococcus aureus MRSA252 pyruvate kinase expressed in Escherichia coli BL2... | Eur J Med Chem 125: 1-13 (2017) Article DOI: 10.1016/j.ejmech.2016.09.018 BindingDB Entry DOI: 10.7270/Q2CC12P0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Pyruvate kinase (Staphylococcus aureus (strain MRSA252)) | BDBM50210352 (CHEMBL3897760) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3 | n/a | n/a | n/a | n/a | n/a | n/a |
Simon Fraser University Curated by ChEMBL | Assay Description Inhibition of recombinant N-terminal His-tagged methicillin-resistant Staphylococcus aureus MRSA252 pyruvate kinase expressed in Escherichia coli BL2... | Eur J Med Chem 125: 1-13 (2017) Article DOI: 10.1016/j.ejmech.2016.09.018 BindingDB Entry DOI: 10.7270/Q2CC12P0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Pyruvate kinase (Staphylococcus aureus (strain MRSA252)) | BDBM50210350 (CHEMBL3898458) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 4 | n/a | n/a | n/a | n/a | n/a | n/a |
Simon Fraser University Curated by ChEMBL | Assay Description Inhibition of recombinant N-terminal His-tagged methicillin-resistant Staphylococcus aureus MRSA252 pyruvate kinase expressed in Escherichia coli BL2... | Eur J Med Chem 125: 1-13 (2017) Article DOI: 10.1016/j.ejmech.2016.09.018 BindingDB Entry DOI: 10.7270/Q2CC12P0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Pyruvate kinase (Staphylococcus aureus (strain MRSA252)) | BDBM50210353 (CHEMBL3933658) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 5 | n/a | n/a | n/a | n/a | n/a | n/a |
Simon Fraser University Curated by ChEMBL | Assay Description Inhibition of recombinant N-terminal His-tagged methicillin-resistant Staphylococcus aureus MRSA252 pyruvate kinase expressed in Escherichia coli BL2... | Eur J Med Chem 125: 1-13 (2017) Article DOI: 10.1016/j.ejmech.2016.09.018 BindingDB Entry DOI: 10.7270/Q2CC12P0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Pyruvate kinase (Staphylococcus aureus (strain MRSA252)) | BDBM50210342 (CHEMBL3925434) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 8 | n/a | n/a | n/a | n/a | n/a | n/a |
Simon Fraser University Curated by ChEMBL | Assay Description Inhibition of recombinant N-terminal His-tagged methicillin-resistant Staphylococcus aureus MRSA252 pyruvate kinase expressed in Escherichia coli BL2... | Eur J Med Chem 125: 1-13 (2017) Article DOI: 10.1016/j.ejmech.2016.09.018 BindingDB Entry DOI: 10.7270/Q2CC12P0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Pyruvate kinase (Staphylococcus aureus (strain MRSA252)) | BDBM50210442 (CHEMBL3926448) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 8 | n/a | n/a | n/a | n/a | n/a | n/a |
Simon Fraser University Curated by ChEMBL | Assay Description Inhibition of recombinant N-terminal His-tagged methicillin-resistant Staphylococcus aureus MRSA252 pyruvate kinase expressed in Escherichia coli BL2... | Eur J Med Chem 125: 1-13 (2017) Article DOI: 10.1016/j.ejmech.2016.09.018 BindingDB Entry DOI: 10.7270/Q2CC12P0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Pyruvate kinase (Staphylococcus aureus (strain MRSA252)) | BDBM50210340 (CHEMBL3932602) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 8 | n/a | n/a | n/a | n/a | n/a | n/a |
Simon Fraser University Curated by ChEMBL | Assay Description Inhibition of recombinant N-terminal His-tagged methicillin-resistant Staphylococcus aureus MRSA252 pyruvate kinase expressed in Escherichia coli BL2... | Eur J Med Chem 125: 1-13 (2017) Article DOI: 10.1016/j.ejmech.2016.09.018 BindingDB Entry DOI: 10.7270/Q2CC12P0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Pyruvate kinase (Staphylococcus aureus (strain MRSA252)) | BDBM50210441 (CHEMBL3939774) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 10 | n/a | n/a | n/a | n/a | n/a | n/a |
Simon Fraser University Curated by ChEMBL | Assay Description Inhibition of recombinant N-terminal His-tagged methicillin-resistant Staphylococcus aureus MRSA252 pyruvate kinase expressed in Escherichia coli BL2... | Eur J Med Chem 125: 1-13 (2017) Article DOI: 10.1016/j.ejmech.2016.09.018 BindingDB Entry DOI: 10.7270/Q2CC12P0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Pyruvate kinase (Staphylococcus aureus (strain MRSA252)) | BDBM50210349 (CHEMBL3978020) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 11 | n/a | n/a | n/a | n/a | n/a | n/a |
Simon Fraser University Curated by ChEMBL | Assay Description Inhibition of recombinant N-terminal His-tagged methicillin-resistant Staphylococcus aureus MRSA252 pyruvate kinase expressed in Escherichia coli BL2... | Eur J Med Chem 125: 1-13 (2017) Article DOI: 10.1016/j.ejmech.2016.09.018 BindingDB Entry DOI: 10.7270/Q2CC12P0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Pyruvate kinase (Staphylococcus aureus (strain MRSA252)) | BDBM50210339 (CHEMBL3952026) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents | Article PubMed | n/a | n/a | 11 | n/a | n/a | n/a | n/a | n/a | n/a |
Simon Fraser University Curated by ChEMBL | Assay Description Inhibition of recombinant N-terminal His-tagged methicillin-resistant Staphylococcus aureus MRSA252 pyruvate kinase expressed in Escherichia coli BL2... | Eur J Med Chem 125: 1-13 (2017) Article DOI: 10.1016/j.ejmech.2016.09.018 BindingDB Entry DOI: 10.7270/Q2CC12P0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Pyruvate kinase (Staphylococcus aureus (strain MRSA252)) | BDBM50210346 (CHEMBL3969320) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 12 | n/a | n/a | n/a | n/a | n/a | n/a |
Simon Fraser University Curated by ChEMBL | Assay Description Inhibition of recombinant N-terminal His-tagged methicillin-resistant Staphylococcus aureus MRSA252 pyruvate kinase expressed in Escherichia coli BL2... | Eur J Med Chem 125: 1-13 (2017) Article DOI: 10.1016/j.ejmech.2016.09.018 BindingDB Entry DOI: 10.7270/Q2CC12P0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Pyruvate kinase (Staphylococcus aureus (strain MRSA252)) | BDBM50210457 (CHEMBL3925374) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 14 | n/a | n/a | n/a | n/a | n/a | n/a |
Simon Fraser University Curated by ChEMBL | Assay Description Inhibition of recombinant N-terminal His-tagged methicillin-resistant Staphylococcus aureus MRSA252 pyruvate kinase expressed in Escherichia coli BL2... | Eur J Med Chem 125: 1-13 (2017) Article DOI: 10.1016/j.ejmech.2016.09.018 BindingDB Entry DOI: 10.7270/Q2CC12P0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Pyruvate kinase (Staphylococcus aureus (strain MRSA252)) | BDBM50402636 (CHEMBL2206712) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 15 | n/a | n/a | n/a | n/a | n/a | n/a |
Simon Fraser University Curated by ChEMBL | Assay Description Inhibition of methicillin-resistant Staphylococcus aureus 252 pyruvate kinase by LDH assay | Bioorg Med Chem 20: 7069-82 (2012) Article DOI: 10.1016/j.bmc.2012.10.002 BindingDB Entry DOI: 10.7270/Q2NZ88ST | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Pyruvate kinase (Staphylococcus aureus (strain MRSA252)) | BDBM50192869 (CIS-3,4-DIHYDROHAMACANTHIN B) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid PDB UniChem Patents Similars | PDB Article PubMed | n/a | n/a | 16 | n/a | n/a | n/a | n/a | n/a | n/a |
Simon Fraser University Curated by ChEMBL | Assay Description Inhibition of recombinant N-terminal His-tagged methicillin-resistant Staphylococcus aureus MRSA252 pyruvate kinase expressed in Escherichia coli BL2... | Eur J Med Chem 125: 1-13 (2017) Article DOI: 10.1016/j.ejmech.2016.09.018 BindingDB Entry DOI: 10.7270/Q2CC12P0 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Pyruvate kinase (Staphylococcus aureus (strain MRSA252)) | BDBM50402630 (CHEMBL2206719) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 17 | n/a | n/a | n/a | n/a | n/a | n/a |
Simon Fraser University Curated by ChEMBL | Assay Description Inhibition of methicillin-resistant Staphylococcus aureus 252 pyruvate kinase by LDH assay | Bioorg Med Chem 20: 7069-82 (2012) Article DOI: 10.1016/j.bmc.2012.10.002 BindingDB Entry DOI: 10.7270/Q2NZ88ST | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Pyruvate kinase (Staphylococcus aureus (strain MRSA252)) | BDBM50402598 (CHEMBL2206157) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 18 | n/a | n/a | n/a | n/a | n/a | n/a |
Simon Fraser University Curated by ChEMBL | Assay Description Inhibition of methicillin-resistant Staphylococcus aureus 252 pyruvate kinase by LDH assay | Bioorg Med Chem 20: 7069-82 (2012) Article DOI: 10.1016/j.bmc.2012.10.002 BindingDB Entry DOI: 10.7270/Q2NZ88ST | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Pyruvate kinase (Staphylococcus aureus (strain MRSA252)) | BDBM50402638 (CHEMBL2206709) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 20 | n/a | n/a | n/a | n/a | n/a | n/a |
Simon Fraser University Curated by ChEMBL | Assay Description Inhibition of methicillin-resistant Staphylococcus aureus 252 pyruvate kinase by LDH assay | Bioorg Med Chem 20: 7069-82 (2012) Article DOI: 10.1016/j.bmc.2012.10.002 BindingDB Entry DOI: 10.7270/Q2NZ88ST | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Pyruvate kinase (Staphylococcus aureus (strain MRSA252)) | BDBM50210439 (CHEMBL3907484) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 23 | n/a | n/a | n/a | n/a | n/a | n/a |
Simon Fraser University Curated by ChEMBL | Assay Description Inhibition of recombinant N-terminal His-tagged methicillin-resistant Staphylococcus aureus MRSA252 pyruvate kinase expressed in Escherichia coli BL2... | Eur J Med Chem 125: 1-13 (2017) Article DOI: 10.1016/j.ejmech.2016.09.018 BindingDB Entry DOI: 10.7270/Q2CC12P0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Pyruvate kinase (Staphylococcus aureus (strain MRSA252)) | BDBM50210356 (CHEMBL3898387) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 24 | n/a | n/a | n/a | n/a | n/a | n/a |
Simon Fraser University Curated by ChEMBL | Assay Description Inhibition of recombinant N-terminal His-tagged methicillin-resistant Staphylococcus aureus MRSA252 pyruvate kinase expressed in Escherichia coli BL2... | Eur J Med Chem 125: 1-13 (2017) Article DOI: 10.1016/j.ejmech.2016.09.018 BindingDB Entry DOI: 10.7270/Q2CC12P0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Pyruvate kinase (Staphylococcus aureus (strain MRSA252)) | BDBM50402639 (CHEMBL2206708) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 24 | n/a | n/a | n/a | n/a | n/a | n/a |
Simon Fraser University Curated by ChEMBL | Assay Description Inhibition of methicillin-resistant Staphylococcus aureus 252 pyruvate kinase by LDH assay | Bioorg Med Chem 20: 7069-82 (2012) Article DOI: 10.1016/j.bmc.2012.10.002 BindingDB Entry DOI: 10.7270/Q2NZ88ST | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Pyruvate kinase (Staphylococcus aureus (strain MRSA252)) | BDBM50402637 (CHEMBL2206710) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 24 | n/a | n/a | n/a | n/a | n/a | n/a |
Simon Fraser University Curated by ChEMBL | Assay Description Inhibition of methicillin-resistant Staphylococcus aureus 252 pyruvate kinase by LDH assay | Bioorg Med Chem 20: 7069-82 (2012) Article DOI: 10.1016/j.bmc.2012.10.002 BindingDB Entry DOI: 10.7270/Q2NZ88ST | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Pyruvate kinase (Staphylococcus aureus (strain MRSA252)) | BDBM50402600 (CHEMBL2206155) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 26 | n/a | n/a | n/a | n/a | n/a | n/a |
Simon Fraser University Curated by ChEMBL | Assay Description Inhibition of methicillin-resistant Staphylococcus aureus 252 pyruvate kinase by LDH assay | Bioorg Med Chem 20: 7069-82 (2012) Article DOI: 10.1016/j.bmc.2012.10.002 BindingDB Entry DOI: 10.7270/Q2NZ88ST | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Pyruvate kinase (Staphylococcus aureus (strain MRSA252)) | BDBM50402599 (CHEMBL2206156) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 31 | n/a | n/a | n/a | n/a | n/a | n/a |
Simon Fraser University Curated by ChEMBL | Assay Description Inhibition of methicillin-resistant Staphylococcus aureus 252 pyruvate kinase by LDH assay | Bioorg Med Chem 20: 7069-82 (2012) Article DOI: 10.1016/j.bmc.2012.10.002 BindingDB Entry DOI: 10.7270/Q2NZ88ST | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Pyruvate kinase (Staphylococcus aureus (strain MRSA252)) | BDBM50402601 (CHEMBL2206154) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 42 | n/a | n/a | n/a | n/a | n/a | n/a |
Simon Fraser University Curated by ChEMBL | Assay Description Inhibition of methicillin-resistant Staphylococcus aureus 252 pyruvate kinase by LDH assay | Bioorg Med Chem 20: 7069-82 (2012) Article DOI: 10.1016/j.bmc.2012.10.002 BindingDB Entry DOI: 10.7270/Q2NZ88ST | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Pyruvate kinase (Staphylococcus aureus (strain MRSA252)) | BDBM50210351 (CHEMBL3916448) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 43 | n/a | n/a | n/a | n/a | n/a | n/a |
Simon Fraser University Curated by ChEMBL | Assay Description Inhibition of recombinant N-terminal His-tagged methicillin-resistant Staphylococcus aureus MRSA252 pyruvate kinase expressed in Escherichia coli BL2... | Eur J Med Chem 125: 1-13 (2017) Article DOI: 10.1016/j.ejmech.2016.09.018 BindingDB Entry DOI: 10.7270/Q2CC12P0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Pyruvate kinase (Staphylococcus aureus (strain MRSA252)) | BDBM50402642 (CHEMBL2206703) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 43 | n/a | n/a | n/a | n/a | n/a | n/a |
Simon Fraser University Curated by ChEMBL | Assay Description Inhibition of methicillin-resistant Staphylococcus aureus 252 pyruvate kinase by LDH assay | Bioorg Med Chem 20: 7069-82 (2012) Article DOI: 10.1016/j.bmc.2012.10.002 BindingDB Entry DOI: 10.7270/Q2NZ88ST | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Pyruvate kinase (Staphylococcus aureus (strain MRSA252)) | BDBM50402607 (CHEMBL2206141) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 49 | n/a | n/a | n/a | n/a | n/a | n/a |
Simon Fraser University Curated by ChEMBL | Assay Description Inhibition of methicillin-resistant Staphylococcus aureus 252 pyruvate kinase by LDH assay | Bioorg Med Chem 20: 7069-82 (2012) Article DOI: 10.1016/j.bmc.2012.10.002 BindingDB Entry DOI: 10.7270/Q2NZ88ST | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Pyruvate kinase (Staphylococcus aureus (strain MRSA252)) | BDBM50402645 (CHEMBL2206725) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 49 | n/a | n/a | n/a | n/a | n/a | n/a |
Simon Fraser University Curated by ChEMBL | Assay Description Inhibition of methicillin-resistant Staphylococcus aureus 252 pyruvate kinase by LDH assay | Bioorg Med Chem 20: 7069-82 (2012) Article DOI: 10.1016/j.bmc.2012.10.002 BindingDB Entry DOI: 10.7270/Q2NZ88ST | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Pyruvate kinase (Staphylococcus aureus (strain MRSA252)) | BDBM50402643 (CHEMBL2206702) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 49 | n/a | n/a | n/a | n/a | n/a | n/a |
Simon Fraser University Curated by ChEMBL | Assay Description Inhibition of methicillin-resistant Staphylococcus aureus 252 pyruvate kinase by LDH assay | Bioorg Med Chem 20: 7069-82 (2012) Article DOI: 10.1016/j.bmc.2012.10.002 BindingDB Entry DOI: 10.7270/Q2NZ88ST | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Pyruvate kinase (Staphylococcus aureus (strain MRSA252)) | BDBM50210440 (CHEMBL3960096) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 51 | n/a | n/a | n/a | n/a | n/a | n/a |
Simon Fraser University Curated by ChEMBL | Assay Description Inhibition of recombinant N-terminal His-tagged methicillin-resistant Staphylococcus aureus MRSA252 pyruvate kinase expressed in Escherichia coli BL2... | Eur J Med Chem 125: 1-13 (2017) Article DOI: 10.1016/j.ejmech.2016.09.018 BindingDB Entry DOI: 10.7270/Q2CC12P0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Pyruvate kinase (Staphylococcus aureus (strain MRSA252)) | BDBM50402646 (CHEMBL2206726) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 52 | n/a | n/a | n/a | n/a | n/a | n/a |
Simon Fraser University Curated by ChEMBL | Assay Description Inhibition of methicillin-resistant Staphylococcus aureus 252 pyruvate kinase by LDH assay | Bioorg Med Chem 20: 7069-82 (2012) Article DOI: 10.1016/j.bmc.2012.10.002 BindingDB Entry DOI: 10.7270/Q2NZ88ST | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Pyruvate kinase (Staphylococcus aureus (strain MRSA252)) | BDBM50402594 (CHEMBL2206161) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 52 | n/a | n/a | n/a | n/a | n/a | n/a |
Simon Fraser University Curated by ChEMBL | Assay Description Inhibition of methicillin-resistant Staphylococcus aureus 252 pyruvate kinase by LDH assay | Bioorg Med Chem 20: 7069-82 (2012) Article DOI: 10.1016/j.bmc.2012.10.002 BindingDB Entry DOI: 10.7270/Q2NZ88ST | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Pyruvate kinase (Staphylococcus aureus (strain MRSA252)) | BDBM50402627 (CHEMBL2206722) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 55 | n/a | n/a | n/a | n/a | n/a | n/a |
Simon Fraser University Curated by ChEMBL | Assay Description Inhibition of methicillin-resistant Staphylococcus aureus 252 pyruvate kinase by LDH assay | Bioorg Med Chem 20: 7069-82 (2012) Article DOI: 10.1016/j.bmc.2012.10.002 BindingDB Entry DOI: 10.7270/Q2NZ88ST | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Pyruvate kinase (Staphylococcus aureus (strain MRSA252)) | BDBM50402595 (CHEMBL2206160) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 59 | n/a | n/a | n/a | n/a | n/a | n/a |
Simon Fraser University Curated by ChEMBL | Assay Description Inhibition of methicillin-resistant Staphylococcus aureus 252 pyruvate kinase by LDH assay | Bioorg Med Chem 20: 7069-82 (2012) Article DOI: 10.1016/j.bmc.2012.10.002 BindingDB Entry DOI: 10.7270/Q2NZ88ST | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Pyruvate kinase (Staphylococcus aureus (strain MRSA252)) | BDBM50210344 (BROMODEOXYTOPSENTIN) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 60 | n/a | n/a | n/a | n/a | n/a | n/a |
Simon Fraser University Curated by ChEMBL | Assay Description Inhibition of recombinant N-terminal His-tagged methicillin-resistant Staphylococcus aureus MRSA252 pyruvate kinase expressed in Escherichia coli BL2... | Eur J Med Chem 125: 1-13 (2017) Article DOI: 10.1016/j.ejmech.2016.09.018 BindingDB Entry DOI: 10.7270/Q2CC12P0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Pyruvate kinase (Staphylococcus aureus (strain MRSA252)) | BDBM50402629 (CHEMBL2206720) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 61 | n/a | n/a | n/a | n/a | n/a | n/a |
Simon Fraser University Curated by ChEMBL | Assay Description Inhibition of methicillin-resistant Staphylococcus aureus 252 pyruvate kinase by LDH assay | Bioorg Med Chem 20: 7069-82 (2012) Article DOI: 10.1016/j.bmc.2012.10.002 BindingDB Entry DOI: 10.7270/Q2NZ88ST | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Pyruvate kinase (Staphylococcus aureus (strain MRSA252)) | BDBM50402617 (CHEMBL2206174) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 63 | n/a | n/a | n/a | n/a | n/a | n/a |
Simon Fraser University Curated by ChEMBL | Assay Description Inhibition of methicillin-resistant Staphylococcus aureus 252 pyruvate kinase by LDH assay | Bioorg Med Chem 20: 7069-82 (2012) Article DOI: 10.1016/j.bmc.2012.10.002 BindingDB Entry DOI: 10.7270/Q2NZ88ST | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Pyruvate kinase (Staphylococcus aureus (strain MRSA252)) | BDBM50402615 (CHEMBL2206176) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 64 | n/a | n/a | n/a | n/a | n/a | n/a |
Simon Fraser University Curated by ChEMBL | Assay Description Inhibition of methicillin-resistant Staphylococcus aureus 252 pyruvate kinase by LDH assay | Bioorg Med Chem 20: 7069-82 (2012) Article DOI: 10.1016/j.bmc.2012.10.002 BindingDB Entry DOI: 10.7270/Q2NZ88ST | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Pyruvate kinase (Staphylococcus aureus (strain MRSA252)) | BDBM50402614 (CHEMBL2206177) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 74 | n/a | n/a | n/a | n/a | n/a | n/a |
Simon Fraser University Curated by ChEMBL | Assay Description Inhibition of methicillin-resistant Staphylococcus aureus 252 pyruvate kinase by LDH assay | Bioorg Med Chem 20: 7069-82 (2012) Article DOI: 10.1016/j.bmc.2012.10.002 BindingDB Entry DOI: 10.7270/Q2NZ88ST | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Pyruvate kinase (Staphylococcus aureus (strain MRSA252)) | BDBM50402596 (CHEMBL2206159) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 79 | n/a | n/a | n/a | n/a | n/a | n/a |
Simon Fraser University Curated by ChEMBL | Assay Description Inhibition of methicillin-resistant Staphylococcus aureus 252 pyruvate kinase by LDH assay | Bioorg Med Chem 20: 7069-82 (2012) Article DOI: 10.1016/j.bmc.2012.10.002 BindingDB Entry DOI: 10.7270/Q2NZ88ST | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Pyruvate kinase (Staphylococcus aureus (strain MRSA252)) | BDBM50402644 (CHEMBL2206724) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 85 | n/a | n/a | n/a | n/a | n/a | n/a |
Simon Fraser University Curated by ChEMBL | Assay Description Inhibition of methicillin-resistant Staphylococcus aureus 252 pyruvate kinase by LDH assay | Bioorg Med Chem 20: 7069-82 (2012) Article DOI: 10.1016/j.bmc.2012.10.002 BindingDB Entry DOI: 10.7270/Q2NZ88ST | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Pyruvate kinase (Staphylococcus aureus (strain MRSA252)) | BDBM50402624 (CHEMBL2206164) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid PDB UniChem Similars | PDB Article PubMed | n/a | n/a | 91 | n/a | n/a | n/a | n/a | n/a | n/a |
Simon Fraser University Curated by ChEMBL | Assay Description Inhibition of methicillin-resistant Staphylococcus aureus 252 pyruvate kinase by LDH assay | Bioorg Med Chem 20: 7069-82 (2012) Article DOI: 10.1016/j.bmc.2012.10.002 BindingDB Entry DOI: 10.7270/Q2NZ88ST | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Pyruvate kinase (Staphylococcus aureus (strain MRSA252)) | BDBM50210345 (CHEMBL3903225) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 102 | n/a | n/a | n/a | n/a | n/a | n/a |
Simon Fraser University Curated by ChEMBL | Assay Description Inhibition of recombinant N-terminal His-tagged methicillin-resistant Staphylococcus aureus MRSA252 pyruvate kinase expressed in Escherichia coli BL2... | Eur J Med Chem 125: 1-13 (2017) Article DOI: 10.1016/j.ejmech.2016.09.018 BindingDB Entry DOI: 10.7270/Q2CC12P0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Pyruvate kinase (Staphylococcus aureus (strain MRSA252)) | BDBM50402597 (CHEMBL2206158) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 115 | n/a | n/a | n/a | n/a | n/a | n/a |
Simon Fraser University Curated by ChEMBL | Assay Description Inhibition of methicillin-resistant Staphylococcus aureus 252 pyruvate kinase by LDH assay | Bioorg Med Chem 20: 7069-82 (2012) Article DOI: 10.1016/j.bmc.2012.10.002 BindingDB Entry DOI: 10.7270/Q2NZ88ST | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Pyruvate kinase (Staphylococcus aureus (strain MRSA252)) | BDBM50210464 (CHEMBL3958246) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 116 | n/a | n/a | n/a | n/a | n/a | n/a |
Simon Fraser University Curated by ChEMBL | Assay Description Inhibition of recombinant N-terminal His-tagged methicillin-resistant Staphylococcus aureus MRSA252 pyruvate kinase expressed in Escherichia coli BL2... | Eur J Med Chem 125: 1-13 (2017) Article DOI: 10.1016/j.ejmech.2016.09.018 BindingDB Entry DOI: 10.7270/Q2CC12P0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Pyruvate kinase (Staphylococcus aureus (strain MRSA252)) | BDBM50402609 (CHEMBL2206139) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 126 | n/a | n/a | n/a | n/a | n/a | n/a |
Simon Fraser University Curated by ChEMBL | Assay Description Inhibition of methicillin-resistant Staphylococcus aureus 252 pyruvate kinase by LDH assay | Bioorg Med Chem 20: 7069-82 (2012) Article DOI: 10.1016/j.bmc.2012.10.002 BindingDB Entry DOI: 10.7270/Q2NZ88ST | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Pyruvate kinase (Staphylococcus aureus (strain MRSA252)) | BDBM50210456 (CHEMBL3945342) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 132 | n/a | n/a | n/a | n/a | n/a | n/a |
Simon Fraser University Curated by ChEMBL | Assay Description Inhibition of recombinant N-terminal His-tagged methicillin-resistant Staphylococcus aureus MRSA252 pyruvate kinase expressed in Escherichia coli BL2... | Eur J Med Chem 125: 1-13 (2017) Article DOI: 10.1016/j.ejmech.2016.09.018 BindingDB Entry DOI: 10.7270/Q2CC12P0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Pyruvate kinase (Staphylococcus aureus (strain MRSA252)) | BDBM50402628 (CHEMBL2206721) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 145 | n/a | n/a | n/a | n/a | n/a | n/a |
Simon Fraser University Curated by ChEMBL | Assay Description Inhibition of methicillin-resistant Staphylococcus aureus 252 pyruvate kinase by LDH assay | Bioorg Med Chem 20: 7069-82 (2012) Article DOI: 10.1016/j.bmc.2012.10.002 BindingDB Entry DOI: 10.7270/Q2NZ88ST | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Pyruvate kinase (Staphylococcus aureus (strain MRSA252)) | BDBM50402632 (CHEMBL2206716) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 146 | n/a | n/a | n/a | n/a | n/a | n/a |
Simon Fraser University Curated by ChEMBL | Assay Description Inhibition of methicillin-resistant Staphylococcus aureus 252 pyruvate kinase by LDH assay | Bioorg Med Chem 20: 7069-82 (2012) Article DOI: 10.1016/j.bmc.2012.10.002 BindingDB Entry DOI: 10.7270/Q2NZ88ST | |||||||||||
More data for this Ligand-Target Pair |
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