Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
2-acylglycerol O-acyltransferase 2 (Homo sapiens (Human)) | BDBM159695 (US9035059, 14-18) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 147 | n/a | n/a | n/a | n/a | n/a | n/a |
Taisho Pharmaceutical Co., Ltd Curated by ChEMBL | Assay Description Inhibition of human recombinant MGAT2 assessed as reduction in enzyme-mediated deacylation of oleoyl-CoA incubated for 20 mins by CPM dye based fluor... | Bioorg Med Chem 23: 5922-31 (2015) Article DOI: 10.1016/j.bmc.2015.06.065 BindingDB Entry DOI: 10.7270/Q2639RJ6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
2-acylglycerol O-acyltransferase 2 (Homo sapiens (Human)) | BDBM159694 (US9035059, 14-16) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 164 | n/a | n/a | n/a | n/a | n/a | n/a |
Taisho Pharmaceutical Co., Ltd Curated by ChEMBL | Assay Description Inhibition of human recombinant MGAT2 assessed as reduction in enzyme-mediated deacylation of oleoyl-CoA incubated for 20 mins by CPM dye based fluor... | Bioorg Med Chem 23: 5922-31 (2015) Article DOI: 10.1016/j.bmc.2015.06.065 BindingDB Entry DOI: 10.7270/Q2639RJ6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
2-acylglycerol O-acyltransferase 2 (Homo sapiens (Human)) | BDBM159693 (US9035059, 14-9) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 168 | n/a | n/a | n/a | n/a | n/a | n/a |
Taisho Pharmaceutical Co., Ltd Curated by ChEMBL | Assay Description Inhibition of human recombinant MGAT2 assessed as reduction in enzyme-mediated deacylation of oleoyl-CoA incubated for 20 mins by CPM dye based fluor... | Bioorg Med Chem 23: 5922-31 (2015) Article DOI: 10.1016/j.bmc.2015.06.065 BindingDB Entry DOI: 10.7270/Q2639RJ6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
2-acylglycerol O-acyltransferase 2 (Homo sapiens (Human)) | BDBM50110678 (CHEMBL3605830) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 547 | n/a | n/a | n/a | n/a | n/a | n/a |
Taisho Pharmaceutical Co., Ltd Curated by ChEMBL | Assay Description Inhibition of human recombinant MGAT2 assessed as reduction in enzyme-mediated deacylation of oleoyl-CoA incubated for 20 mins by CPM dye based fluor... | Bioorg Med Chem 23: 5922-31 (2015) Article DOI: 10.1016/j.bmc.2015.06.065 BindingDB Entry DOI: 10.7270/Q2639RJ6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
2-acylglycerol O-acyltransferase 2 (Homo sapiens (Human)) | BDBM50110581 (CHEMBL3605819) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 594 | n/a | n/a | n/a | n/a | n/a | n/a |
Taisho Pharmaceutical Co., Ltd Curated by ChEMBL | Assay Description Inhibition of human recombinant MGAT2 assessed as reduction in enzyme-mediated deacylation of oleoyl-CoA incubated for 20 mins by CPM dye based fluor... | Bioorg Med Chem 23: 5922-31 (2015) Article DOI: 10.1016/j.bmc.2015.06.065 BindingDB Entry DOI: 10.7270/Q2639RJ6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
2-acylglycerol O-acyltransferase 2 (Homo sapiens (Human)) | BDBM50110697 (CHEMBL3605820) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 685 | n/a | n/a | n/a | n/a | n/a | n/a |
Taisho Pharmaceutical Co., Ltd Curated by ChEMBL | Assay Description Inhibition of human recombinant MGAT2 assessed as reduction in enzyme-mediated deacylation of oleoyl-CoA incubated for 20 mins by CPM dye based fluor... | Bioorg Med Chem 23: 5922-31 (2015) Article DOI: 10.1016/j.bmc.2015.06.065 BindingDB Entry DOI: 10.7270/Q2639RJ6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
2-acylglycerol O-acyltransferase 2 (Homo sapiens (Human)) | BDBM50110688 (CHEMBL3605824) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 733 | n/a | n/a | n/a | n/a | n/a | n/a |
Taisho Pharmaceutical Co., Ltd Curated by ChEMBL | Assay Description Inhibition of human recombinant MGAT2 assessed as reduction in enzyme-mediated deacylation of oleoyl-CoA incubated for 20 mins by CPM dye based fluor... | Bioorg Med Chem 23: 5922-31 (2015) Article DOI: 10.1016/j.bmc.2015.06.065 BindingDB Entry DOI: 10.7270/Q2639RJ6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
2-acylglycerol O-acyltransferase 2 (Homo sapiens (Human)) | BDBM50110691 (CHEMBL3605821) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.11E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Taisho Pharmaceutical Co., Ltd Curated by ChEMBL | Assay Description Inhibition of human recombinant MGAT2 assessed as reduction in enzyme-mediated deacylation of oleoyl-CoA incubated for 20 mins by CPM dye based fluor... | Bioorg Med Chem 23: 5922-31 (2015) Article DOI: 10.1016/j.bmc.2015.06.065 BindingDB Entry DOI: 10.7270/Q2639RJ6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
2-acylglycerol O-acyltransferase 2 (Mus musculus) | BDBM50110518 (CHEMBL3605835) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 1.17E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Taisho Pharmaceutical Co., Ltd Curated by ChEMBL | Assay Description Inhibition of mouse recombinant MGAT2 assessed as reduction in enzyme-mediated deacylation of oleoyl-CoA incubated for 20 mins by CPM dye based fluor... | Bioorg Med Chem 23: 5922-31 (2015) Article DOI: 10.1016/j.bmc.2015.06.065 BindingDB Entry DOI: 10.7270/Q2639RJ6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Plasminogen (Homo sapiens (Human)) | BDBM50286441 ((S)-2-((S)-2-Acetylamino-4-(S)-methyl-pentanoylami...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Chiba University Curated by ChEMBL | Assay Description Inhibition of plasmin | J Nat Prod 68: 447-9 (2005) Article DOI: 10.1021/np049622e BindingDB Entry DOI: 10.7270/Q2Z320J8 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
2-acylglycerol O-acyltransferase 2 (Mus musculus) | BDBM50110581 (CHEMBL3605819) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 1.31E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Taisho Pharmaceutical Co., Ltd Curated by ChEMBL | Assay Description Inhibition of mouse recombinant MGAT2 assessed as reduction in enzyme-mediated deacylation of oleoyl-CoA incubated for 20 mins by CPM dye based fluor... | Bioorg Med Chem 23: 5922-31 (2015) Article DOI: 10.1016/j.bmc.2015.06.065 BindingDB Entry DOI: 10.7270/Q2639RJ6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Plasminogen (Homo sapiens (Human)) | BDBM50240897 (2-(3,4-dihydroxyphenyl)-5-hydroxy-3,7-dimethoxy-4H...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE KEGG PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 1.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Chiba University Curated by ChEMBL | Assay Description Inhibition of plasmin | J Nat Prod 68: 447-9 (2005) Article DOI: 10.1021/np049622e BindingDB Entry DOI: 10.7270/Q2Z320J8 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
2-acylglycerol O-acyltransferase 2 (Homo sapiens (Human)) | BDBM50110518 (CHEMBL3605835) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 1.52E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Taisho Pharmaceutical Co., Ltd Curated by ChEMBL | Assay Description Inhibition of human recombinant MGAT2 assessed as reduction in enzyme-mediated deacylation of oleoyl-CoA incubated for 20 mins by CPM dye based fluor... | Bioorg Med Chem 23: 5922-31 (2015) Article DOI: 10.1016/j.bmc.2015.06.065 BindingDB Entry DOI: 10.7270/Q2639RJ6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
2-acylglycerol O-acyltransferase 2 (Homo sapiens (Human)) | BDBM50110679 (CHEMBL3605829) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.98E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Taisho Pharmaceutical Co., Ltd Curated by ChEMBL | Assay Description Inhibition of human recombinant MGAT2 assessed as reduction in enzyme-mediated deacylation of oleoyl-CoA incubated for 20 mins by CPM dye based fluor... | Bioorg Med Chem 23: 5922-31 (2015) Article DOI: 10.1016/j.bmc.2015.06.065 BindingDB Entry DOI: 10.7270/Q2639RJ6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
2-acylglycerol O-acyltransferase 2 (Homo sapiens (Human)) | BDBM50110589 (CHEMBL3605833) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.12E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Taisho Pharmaceutical Co., Ltd Curated by ChEMBL | Assay Description Inhibition of human recombinant MGAT2 assessed as reduction in enzyme-mediated deacylation of oleoyl-CoA incubated for 20 mins by CPM dye based fluor... | Bioorg Med Chem 23: 5922-31 (2015) Article DOI: 10.1016/j.bmc.2015.06.065 BindingDB Entry DOI: 10.7270/Q2639RJ6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Plasminogen (Homo sapiens (Human)) | BDBM50240943 (2-(3,4-Dihydroxy-phenyl)-5-hydroxy-7-methoxy-chrom...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid PDB UniChem Similars | Article PubMed | n/a | n/a | 2.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Chiba University Curated by ChEMBL | Assay Description Inhibition of plasmin | J Nat Prod 68: 447-9 (2005) Article DOI: 10.1021/np049622e BindingDB Entry DOI: 10.7270/Q2Z320J8 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
2-acylglycerol O-acyltransferase 2 (Homo sapiens (Human)) | BDBM50110684 (CHEMBL3605825) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Taisho Pharmaceutical Co., Ltd Curated by ChEMBL | Assay Description Inhibition of human recombinant MGAT2 assessed as reduction in enzyme-mediated deacylation of oleoyl-CoA incubated for 20 mins by CPM dye based fluor... | Bioorg Med Chem 23: 5922-31 (2015) Article DOI: 10.1016/j.bmc.2015.06.065 BindingDB Entry DOI: 10.7270/Q2639RJ6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
2-acylglycerol O-acyltransferase 2 (Homo sapiens (Human)) | BDBM50110689 (CHEMBL3605822) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.49E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Taisho Pharmaceutical Co., Ltd Curated by ChEMBL | Assay Description Inhibition of human recombinant MGAT2 assessed as reduction in enzyme-mediated deacylation of oleoyl-CoA incubated for 20 mins by CPM dye based fluor... | Bioorg Med Chem 23: 5922-31 (2015) Article DOI: 10.1016/j.bmc.2015.06.065 BindingDB Entry DOI: 10.7270/Q2639RJ6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
2-acylglycerol O-acyltransferase 2 (Homo sapiens (Human)) | BDBM50110588 (CHEMBL3605834) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.06E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Taisho Pharmaceutical Co., Ltd Curated by ChEMBL | Assay Description Inhibition of human recombinant MGAT2 assessed as reduction in enzyme-mediated deacylation of oleoyl-CoA incubated for 20 mins by CPM dye based fluor... | Bioorg Med Chem 23: 5922-31 (2015) Article DOI: 10.1016/j.bmc.2015.06.065 BindingDB Entry DOI: 10.7270/Q2639RJ6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
2-acylglycerol O-acyltransferase 2 (Homo sapiens (Human)) | BDBM50110683 (CHEMBL3605826) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.16E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Taisho Pharmaceutical Co., Ltd Curated by ChEMBL | Assay Description Inhibition of human recombinant MGAT2 assessed as reduction in enzyme-mediated deacylation of oleoyl-CoA incubated for 20 mins by CPM dye based fluor... | Bioorg Med Chem 23: 5922-31 (2015) Article DOI: 10.1016/j.bmc.2015.06.065 BindingDB Entry DOI: 10.7270/Q2639RJ6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
2-acylglycerol O-acyltransferase 2 (Homo sapiens (Human)) | BDBM50110680 (CHEMBL3605828) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 5.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Taisho Pharmaceutical Co., Ltd Curated by ChEMBL | Assay Description Inhibition of human recombinant MGAT2 assessed as reduction in enzyme-mediated deacylation of oleoyl-CoA incubated for 20 mins by CPM dye based fluor... | Bioorg Med Chem 23: 5922-31 (2015) Article DOI: 10.1016/j.bmc.2015.06.065 BindingDB Entry DOI: 10.7270/Q2639RJ6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
2-acylglycerol O-acyltransferase 2 (Homo sapiens (Human)) | BDBM50110637 (CHEMBL3605832) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 8.07E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Taisho Pharmaceutical Co., Ltd Curated by ChEMBL | Assay Description Inhibition of human recombinant MGAT2 assessed as reduction in enzyme-mediated deacylation of oleoyl-CoA incubated for 20 mins by CPM dye based fluor... | Bioorg Med Chem 23: 5922-31 (2015) Article DOI: 10.1016/j.bmc.2015.06.065 BindingDB Entry DOI: 10.7270/Q2639RJ6 | |||||||||||
More data for this Ligand-Target Pair |