Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Cytosol aminopeptidase (Bos taurus (bovine)) | BDBM23983 (3-amino-N-hydroxy-1,2,3,4-tetrahydronaphthalene-2-...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 1.00E+4 | -29.0 | n/a | n/a | n/a | n/a | n/a | 8.0 | 30 |
ENSCMu | Assay Description Spectrophotometric assays were performed by monitoring hydrolysis of chromogenic substrate. The release of para-nitroaniline at 405 nm was measured t... | Bioorg Med Chem 14: 7241-57 (2006) Article DOI: 10.1016/j.bmc.2006.06.050 BindingDB Entry DOI: 10.7270/Q2N29V73 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytosol aminopeptidase (Bos taurus (bovine)) | BDBM23974 ((3Z)-3-(hydroxyimino)-1,2,3,4-tetrahydronaphthalen...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+6 | n/a | n/a | n/a | n/a | 8.0 | 30 |
ENSCMu | Assay Description Spectrophotometric assays were performed by monitoring hydrolysis of chromogenic substrate. The release of para-nitroaniline at 405 nm was measured t... | Bioorg Med Chem 14: 7241-57 (2006) Article DOI: 10.1016/j.bmc.2006.06.050 BindingDB Entry DOI: 10.7270/Q2N29V73 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytosol aminopeptidase (Bos taurus (bovine)) | BDBM23975 ((3Z)-3-(methoxyimino)-1,2,3,4-tetrahydronaphthalen...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+6 | n/a | n/a | n/a | n/a | 8.0 | 30 |
ENSCMu | Assay Description Spectrophotometric assays were performed by monitoring hydrolysis of chromogenic substrate. The release of para-nitroaniline at 405 nm was measured t... | Bioorg Med Chem 14: 7241-57 (2006) Article DOI: 10.1016/j.bmc.2006.06.050 BindingDB Entry DOI: 10.7270/Q2N29V73 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytosol aminopeptidase (Bos taurus (bovine)) | BDBM23976 ((3Z)-3-[(benzyloxy)imino]-1,2,3,4-tetrahydronaphth...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+6 | n/a | n/a | n/a | n/a | 8.0 | 30 |
ENSCMu | Assay Description Spectrophotometric assays were performed by monitoring hydrolysis of chromogenic substrate. The release of para-nitroaniline at 405 nm was measured t... | Bioorg Med Chem 14: 7241-57 (2006) Article DOI: 10.1016/j.bmc.2006.06.050 BindingDB Entry DOI: 10.7270/Q2N29V73 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytosol aminopeptidase (Bos taurus (bovine)) | BDBM23977 ((3Z)-3-[(2-phenylethoxy)imino]-1,2,3,4-tetrahydron...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | 8.0 | 30 |
ENSCMu | Assay Description Spectrophotometric assays were performed by monitoring hydrolysis of chromogenic substrate. The release of para-nitroaniline at 405 nm was measured t... | Bioorg Med Chem 14: 7241-57 (2006) Article DOI: 10.1016/j.bmc.2006.06.050 BindingDB Entry DOI: 10.7270/Q2N29V73 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytosol aminopeptidase (Bos taurus (bovine)) | BDBM23978 ((3Z)-3-[(3-phenylpropoxy)imino]-1,2,3,4-tetrahydro...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+6 | n/a | n/a | n/a | n/a | 8.0 | 30 |
ENSCMu | Assay Description Spectrophotometric assays were performed by monitoring hydrolysis of chromogenic substrate. The release of para-nitroaniline at 405 nm was measured t... | Bioorg Med Chem 14: 7241-57 (2006) Article DOI: 10.1016/j.bmc.2006.06.050 BindingDB Entry DOI: 10.7270/Q2N29V73 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytosol aminopeptidase (Bos taurus (bovine)) | BDBM23979 ((3Z)-3-[(4-phenylbutoxy)imino]-1,2,3,4-tetrahydron...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | 8.0 | 30 |
ENSCMu | Assay Description Spectrophotometric assays were performed by monitoring hydrolysis of chromogenic substrate. The release of para-nitroaniline at 405 nm was measured t... | Bioorg Med Chem 14: 7241-57 (2006) Article DOI: 10.1016/j.bmc.2006.06.050 BindingDB Entry DOI: 10.7270/Q2N29V73 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytosol aminopeptidase (Bos taurus (bovine)) | BDBM23980 ((3Z)-3-{[(5-phenylpentyl)oxy]imino}-1,2,3,4-tetrah...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | 8.0 | 30 |
ENSCMu | Assay Description Spectrophotometric assays were performed by monitoring hydrolysis of chromogenic substrate. The release of para-nitroaniline at 405 nm was measured t... | Bioorg Med Chem 14: 7241-57 (2006) Article DOI: 10.1016/j.bmc.2006.06.050 BindingDB Entry DOI: 10.7270/Q2N29V73 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytosol aminopeptidase (Bos taurus (bovine)) | BDBM23981 ((2S)-1,2,3,4-Tetrahydro-naphthalen-2-ylamine | 1,2...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+6 | n/a | n/a | n/a | n/a | 8.0 | 30 |
ENSCMu | Assay Description Spectrophotometric assays were performed by monitoring hydrolysis of chromogenic substrate. The release of para-nitroaniline at 405 nm was measured t... | Bioorg Med Chem 14: 7241-57 (2006) Article DOI: 10.1016/j.bmc.2006.06.050 BindingDB Entry DOI: 10.7270/Q2N29V73 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytosol aminopeptidase (Bos taurus (bovine)) | BDBM23982 (1-(3-amino-1,2,3,4-tetrahydronaphthalen-2-yl)ethan...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >1.00E+6 | n/a | n/a | n/a | n/a | 8.0 | 30 |
ENSCMu | Assay Description Spectrophotometric assays were performed by monitoring hydrolysis of chromogenic substrate. The release of para-nitroaniline at 405 nm was measured t... | Bioorg Med Chem 14: 7241-57 (2006) Article DOI: 10.1016/j.bmc.2006.06.050 BindingDB Entry DOI: 10.7270/Q2N29V73 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytosol aminopeptidase (Bos taurus (bovine)) | BDBM23971 ((2S)-2-[(2S,3R)-3-amino-2-hydroxy-4-phenylbutanami...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | Purchase CHEMBL MCE MMDB PC cid PC sid PDB UniChem Patents Similars | Article PubMed | n/a | n/a | 0.5 | n/a | n/a | n/a | n/a | 8.0 | 30 |
ENSCMu | Assay Description Spectrophotometric assays were performed by monitoring hydrolysis of chromogenic substrate. The release of para-nitroaniline at 405 nm was measured t... | Bioorg Med Chem 14: 7241-57 (2006) Article DOI: 10.1016/j.bmc.2006.06.050 BindingDB Entry DOI: 10.7270/Q2N29V73 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytosol aminopeptidase (Bos taurus (bovine)) | BDBM23973 (3-amino-1,2,3,4-tetrahydronaphthalen-2-one hydroch...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.20E+5 | n/a | n/a | n/a | n/a | 8.0 | 30 |
ENSCMu | Assay Description Spectrophotometric assays were performed by monitoring hydrolysis of chromogenic substrate. The release of para-nitroaniline at 405 nm was measured t... | Bioorg Med Chem 14: 7241-57 (2006) Article DOI: 10.1016/j.bmc.2006.06.050 BindingDB Entry DOI: 10.7270/Q2N29V73 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytosol aminopeptidase (Bos taurus (bovine)) | BDBM23990 (3-amino-1,2,3,4-tetrahydroquinolin-2-one hydrochlo...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+6 | n/a | n/a | n/a | n/a | 8.0 | 30 |
ENSCMu | Assay Description Spectrophotometric assays were performed by monitoring hydrolysis of chromogenic substrate. The release of para-nitroaniline at 405 nm was measured t... | Bioorg Med Chem 14: 7241-57 (2006) Article DOI: 10.1016/j.bmc.2006.06.050 BindingDB Entry DOI: 10.7270/Q2N29V73 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytosol aminopeptidase (Bos taurus (bovine)) | BDBM23989 (1,2,3,4-tetrahydronaphthalen-2-one | CHEMBL191664 ...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents | Article PubMed | n/a | n/a | >1.00E+6 | n/a | n/a | n/a | n/a | 8.0 | 30 |
ENSCMu | Assay Description Spectrophotometric assays were performed by monitoring hydrolysis of chromogenic substrate. The release of para-nitroaniline at 405 nm was measured t... | Bioorg Med Chem 14: 7241-57 (2006) Article DOI: 10.1016/j.bmc.2006.06.050 BindingDB Entry DOI: 10.7270/Q2N29V73 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytosol aminopeptidase (Bos taurus (bovine)) | BDBM23988 (2-amino-1,2,3,4-tetrahydroisoquinolin-3-one | N-Su...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | Purchase PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.00E+6 | n/a | n/a | n/a | n/a | 8.0 | 30 |
ENSCMu | Assay Description Spectrophotometric assays were performed by monitoring hydrolysis of chromogenic substrate. The release of para-nitroaniline at 405 nm was measured t... | Bioorg Med Chem 14: 7241-57 (2006) Article DOI: 10.1016/j.bmc.2006.06.050 BindingDB Entry DOI: 10.7270/Q2N29V73 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytosol aminopeptidase (Bos taurus (bovine)) | BDBM23987 (2-hydroxy-1,2,3,4-tetrahydroisoquinolin-3-one | CH...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+6 | n/a | n/a | n/a | n/a | 8.0 | 30 |
ENSCMu | Assay Description Spectrophotometric assays were performed by monitoring hydrolysis of chromogenic substrate. The release of para-nitroaniline at 405 nm was measured t... | Bioorg Med Chem 14: 7241-57 (2006) Article DOI: 10.1016/j.bmc.2006.06.050 BindingDB Entry DOI: 10.7270/Q2N29V73 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytosol aminopeptidase (Bos taurus (bovine)) | BDBM23986 (3,4-dihydro-1H-2-benzothiopyran-3-one | isothiochr...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem Patents | Article PubMed | n/a | n/a | >1.00E+6 | n/a | n/a | n/a | n/a | 8.0 | 30 |
ENSCMu | Assay Description Spectrophotometric assays were performed by monitoring hydrolysis of chromogenic substrate. The release of para-nitroaniline at 405 nm was measured t... | Bioorg Med Chem 14: 7241-57 (2006) Article DOI: 10.1016/j.bmc.2006.06.050 BindingDB Entry DOI: 10.7270/Q2N29V73 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytosol aminopeptidase (Bos taurus (bovine)) | BDBM23985 (3,4-dihydro-1H-2-benzopyran-3-one | isochromanone,...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | Purchase MCE KEGG PC cid PC sid UniChem Patents | Article PubMed | n/a | n/a | >1.00E+6 | n/a | n/a | n/a | n/a | 8.0 | 30 |
ENSCMu | Assay Description Spectrophotometric assays were performed by monitoring hydrolysis of chromogenic substrate. The release of para-nitroaniline at 405 nm was measured t... | Bioorg Med Chem 14: 7241-57 (2006) Article DOI: 10.1016/j.bmc.2006.06.050 BindingDB Entry DOI: 10.7270/Q2N29V73 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytosol aminopeptidase (Bos taurus (bovine)) | BDBM23984 (3-amino-1,2,3,4-tetrahydronaphthalene-2-phosphonic...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >1.00E+6 | n/a | n/a | n/a | n/a | 8.0 | 30 |
ENSCMu | Assay Description Spectrophotometric assays were performed by monitoring hydrolysis of chromogenic substrate. The release of para-nitroaniline at 405 nm was measured t... | Bioorg Med Chem 14: 7241-57 (2006) Article DOI: 10.1016/j.bmc.2006.06.050 BindingDB Entry DOI: 10.7270/Q2N29V73 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytosol aminopeptidase [33-68,L62W] (Sus scrofa (Pig)) | BDBM234297 (Met-ψ[P(O)(OH)CH2]-Ala (5)) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 3.64E+3 | -31.0 | n/a | n/a | n/a | n/a | n/a | 8.4 | 25 |
Academy of Sciences of the Czech Republic | Assay Description LAP was assayed in 75 mM triethanolamine hydrochloride buffer (pH = 8.4, containing 5 mM MgCl2) at 25°C. The substrate (L-leucine-p-nitroanilide) was... | J Enzyme Inhib Med Chem 26: 155-61 (2011) Article DOI: 10.3109/14756366.2010.482047 BindingDB Entry DOI: 10.7270/Q22N515B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytosol aminopeptidase [33-68,L62W] (Sus scrofa (Pig)) | BDBM234295 (Met-PH (2)) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid PDB UniChem | Article PubMed | 2.20E+4 | -26.6 | n/a | n/a | n/a | n/a | n/a | 8.4 | 25 |
Academy of Sciences of the Czech Republic | Assay Description LAP was assayed in 75 mM triethanolamine hydrochloride buffer (pH = 8.4, containing 5 mM MgCl2) at 25°C. The substrate (L-leucine-p-nitroanilide) was... | J Enzyme Inhib Med Chem 26: 155-61 (2011) Article DOI: 10.3109/14756366.2010.482047 BindingDB Entry DOI: 10.7270/Q22N515B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytosol aminopeptidase [33-68,L62W] (Sus scrofa (Pig)) | BDBM234294 (Met-P (1)) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid PDB UniChem | Article PubMed | 2.26E+4 | -26.5 | n/a | n/a | n/a | n/a | n/a | 8.4 | 25 |
Academy of Sciences of the Czech Republic | Assay Description LAP was assayed in 75 mM triethanolamine hydrochloride buffer (pH = 8.4, containing 5 mM MgCl2) at 25°C. The substrate (L-leucine-p-nitroanilide) was... | J Enzyme Inhib Med Chem 26: 155-61 (2011) Article DOI: 10.3109/14756366.2010.482047 BindingDB Entry DOI: 10.7270/Q22N515B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytosol aminopeptidase [33-68,L62W] (Sus scrofa (Pig)) | BDBM50316030 (1-aminopentylphosphonic acid | CHEMBL1089899 | Nle...) | UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid PDB UniChem Patents Similars | Article PubMed | 5.80E+4 | -24.2 | n/a | n/a | n/a | n/a | n/a | 8.4 | 25 |
Academy of Sciences of the Czech Republic | Assay Description LAP was assayed in 75 mM triethanolamine hydrochloride buffer (pH = 8.4, containing 5 mM MgCl2) at 25°C. The substrate (L-leucine-p-nitroanilide) was... | J Enzyme Inhib Med Chem 26: 155-61 (2011) Article DOI: 10.3109/14756366.2010.482047 BindingDB Entry DOI: 10.7270/Q22N515B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytosol aminopeptidase [33-68,L62W] (Sus scrofa (Pig)) | BDBM234296 (Nle-PH (4)) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 7.39E+4 | -23.6 | n/a | n/a | n/a | n/a | n/a | 8.4 | 25 |
Academy of Sciences of the Czech Republic | Assay Description LAP was assayed in 75 mM triethanolamine hydrochloride buffer (pH = 8.4, containing 5 mM MgCl2) at 25°C. The substrate (L-leucine-p-nitroanilide) was... | J Enzyme Inhib Med Chem 26: 155-61 (2011) Article DOI: 10.3109/14756366.2010.482047 BindingDB Entry DOI: 10.7270/Q22N515B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytosol aminopeptidase [33-68,L62W] (Sus scrofa (Pig)) | BDBM234299 (Nle-ψ[P(O)(OH)O]-L-AlaOMe (7)) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 2.19E+5 | -20.9 | n/a | n/a | n/a | n/a | n/a | 8.4 | 25 |
Academy of Sciences of the Czech Republic | Assay Description LAP was assayed in 75 mM triethanolamine hydrochloride buffer (pH = 8.4, containing 5 mM MgCl2) at 25°C. The substrate (L-leucine-p-nitroanilide) was... | J Enzyme Inhib Med Chem 26: 155-61 (2011) Article DOI: 10.3109/14756366.2010.482047 BindingDB Entry DOI: 10.7270/Q22N515B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytosol aminopeptidase [33-68,L62W] (Sus scrofa (Pig)) | BDBM234298 (Nle-ψ[P(O)(OH)O]-L-Ala (6)) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 2.69E+5 | -20.4 | n/a | n/a | n/a | n/a | n/a | 8.4 | 25 |
Academy of Sciences of the Czech Republic | Assay Description LAP was assayed in 75 mM triethanolamine hydrochloride buffer (pH = 8.4, containing 5 mM MgCl2) at 25°C. The substrate (L-leucine-p-nitroanilide) was... | J Enzyme Inhib Med Chem 26: 155-61 (2011) Article DOI: 10.3109/14756366.2010.482047 BindingDB Entry DOI: 10.7270/Q22N515B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aminopeptidase B (Mus musculus) | BDBM50078120 ((R)-1-{[(S)-2-((S)-1-Carboxy-1-methyl-2-phenyl-eth...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | PubMed | >0 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
INSERM Curated by ChEMBL | Assay Description Inhibitory activity was measured on Aminopeptidase B using Arg p.NA as substrate | Bioorg Med Chem Lett 9: 1511-6 (1999) BindingDB Entry DOI: 10.7270/Q2H132JR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aminopeptidase B (Mus musculus) | BDBM50078122 ((R)-1-{[(S)-2-((S)-1-Carboxy-1-methyl-2-phenyl-eth...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | PubMed | >0 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
INSERM Curated by ChEMBL | Assay Description Inhibitory activity was measured on Aminopeptidase B using Arg p.NA as substrate | Bioorg Med Chem Lett 9: 1511-6 (1999) BindingDB Entry DOI: 10.7270/Q2H132JR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytosol aminopeptidase [33-68,L62W] (Sus scrofa (Pig)) | BDBM50024594 ((R)-1-Ammonium-3-methyl-butane-1-phosphonic acid a...) | UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.230 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Athens Curated by ChEMBL | Assay Description Inhibition of pig recombinant leucine aminopeptidase after 30 to 60 mins by morrison's equation | J Med Chem 57: 8140-51 (2014) Article DOI: 10.1021/jm501071f BindingDB Entry DOI: 10.7270/Q2CF9RQF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytosol aminopeptidase (Homo sapiens (Human)) | BDBM23971 ((2S)-2-[(2S,3R)-3-amino-2-hydroxy-4-phenylbutanami...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE MMDB PC cid PC sid PDB UniChem Patents Similars | Article PubMed | 0.600 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Wroclaw University of Technology Curated by ChEMBL | Assay Description Binding affinity for cytosolic leucine aminopeptidase (LAP) from porcine kidney | J Med Chem 46: 2641-55 (2003) Article DOI: 10.1021/jm030795v BindingDB Entry DOI: 10.7270/Q27P903F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aminopeptidase B (Rattus norvegicus) | BDBM50017480 (5-Amino-8-guanidino-2-(4-hydroxy-benzyl)-4-oxo-oct...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | PubMed | 0.840 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Wisconsin-Madison Curated by ChEMBL | Assay Description Inhibition of aminopeptidase B or arginyl aminopeptidase purified from rat liver | J Med Chem 32: 1378-92 (1989) BindingDB Entry DOI: 10.7270/Q20G3KQ1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aminopeptidase B (Rattus norvegicus) | BDBM50022743 (2,6-Diamino-hexane-1-thiol | CHEMBL68509) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | PubMed | 0.910 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Wisconsin Curated by ChEMBL | Assay Description Inhibitory activity against aminopeptidase B | J Med Chem 31: 2193-9 (1988) BindingDB Entry DOI: 10.7270/Q2Z038RM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aminopeptidase B (Rattus norvegicus) | BDBM50017482 (5-Amino-2-benzyl-8-guanidino-4-oxo-octanoic acid |...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 2.5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Wisconsin-Madison Curated by ChEMBL | Assay Description Inhibition of aminopeptidase B or arginyl aminopeptidase purified from rat liver | J Med Chem 32: 1378-92 (1989) BindingDB Entry DOI: 10.7270/Q20G3KQ1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aminopeptidase B (Rattus norvegicus) | BDBM50017476 (5,9-Diamino-2-benzyl-4-oxo-nonanoic acid | CHEMBL2...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Wisconsin-Madison Curated by ChEMBL | Assay Description Competitive inhibition of aminopeptidase B or arginyl aminopeptidase purified from rat liver; Ki value reporting the slope effect(Kis) | J Med Chem 32: 1378-92 (1989) BindingDB Entry DOI: 10.7270/Q20G3KQ1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytosol aminopeptidase [33-68,L62W] (Sus scrofa (Pig)) | BDBM50316049 (1-amino-3-phenylpropylphosphonic acid | CHEMBL1090...) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid PDB UniChem Patents Similars | Article PubMed | 4.60 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Athens Curated by ChEMBL | Assay Description Inhibition of pig recombinant leucine aminopeptidase after 30 to 60 mins by morrison's equation | J Med Chem 57: 8140-51 (2014) Article DOI: 10.1021/jm501071f BindingDB Entry DOI: 10.7270/Q2CF9RQF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aminopeptidase B (Rattus norvegicus) | BDBM50022751 (2-(3-Amino-2-mercapto-4-phenyl-butyrylamino)-4-met...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | PubMed | 4.60 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Wisconsin Curated by ChEMBL | Assay Description Inhibitory activity against aminopeptidase B | J Med Chem 31: 2193-9 (1988) BindingDB Entry DOI: 10.7270/Q2Z038RM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytosol aminopeptidase [33-68,L62W] (Sus scrofa (Pig)) | BDBM50025048 (CHEMBL3355099) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid PDB UniChem Patents Similars | Article PubMed | 5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Athens Curated by ChEMBL | Assay Description Inhibition of pig recombinant leucine aminopeptidase after 30 to 60 mins by morrison's equation | J Med Chem 57: 8140-51 (2014) Article DOI: 10.1021/jm501071f BindingDB Entry DOI: 10.7270/Q2CF9RQF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aminopeptidase B (Rattus norvegicus) | BDBM50022751 (2-(3-Amino-2-mercapto-4-phenyl-butyrylamino)-4-met...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | PubMed | 6.40 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Wisconsin Curated by ChEMBL | Assay Description Inhibitory activity against aminopeptidase B | J Med Chem 31: 2193-9 (1988) BindingDB Entry DOI: 10.7270/Q2Z038RM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytosol aminopeptidase [33-68,L62W] (Sus scrofa (Pig)) | BDBM50078125 ((1-Amino-3-phenyl-propyl)-phosphinic acid | CHEMBL...) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 7.70 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Athens Curated by ChEMBL | Assay Description Inhibition of pig recombinant leucine aminopeptidase after 30 to 60 mins by morrison's equation | J Med Chem 57: 8140-51 (2014) Article DOI: 10.1021/jm501071f BindingDB Entry DOI: 10.7270/Q2CF9RQF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aminopeptidase B (Rattus norvegicus) | BDBM23971 ((2S)-2-[(2S,3R)-3-amino-2-hydroxy-4-phenylbutanami...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE MMDB PC cid PC sid PDB UniChem Patents Similars | PubMed | 14 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Wisconsin-Madison Curated by ChEMBL | Assay Description Inhibition of aminopeptidase B or arginyl aminopeptidase purified from rat liver | J Med Chem 32: 1378-92 (1989) BindingDB Entry DOI: 10.7270/Q20G3KQ1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytosol aminopeptidase [33-68,L62W] (Sus scrofa (Pig)) | BDBM50025043 (CHEMBL3355104) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 20 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Athens Curated by ChEMBL | Assay Description Inhibition of pig recombinant leucine aminopeptidase after 30 to 60 mins by morrison's equation | J Med Chem 57: 8140-51 (2014) Article DOI: 10.1021/jm501071f BindingDB Entry DOI: 10.7270/Q2CF9RQF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytosol aminopeptidase (Homo sapiens (Human)) | BDBM23971 ((2S)-2-[(2S,3R)-3-amino-2-hydroxy-4-phenylbutanami...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE MMDB PC cid PC sid PDB UniChem Patents Similars | PubMed | 20 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Wisconsin Curated by ChEMBL | Assay Description Inhibitory activity against Leucine aminopeptidase | J Med Chem 31: 2193-9 (1988) BindingDB Entry DOI: 10.7270/Q2Z038RM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytosol aminopeptidase [435-519] (Sus scrofa) | BDBM50022748 (2-Amino-4-methyl-pentane-1-thiol | CHEMBL69349) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 22 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Jadavpur University Curated by ChEMBL | Assay Description Competitive inhibition of LAP in porcine kidney microsomes | J Med Chem 61: 6468-6490 (2018) Article DOI: 10.1021/acs.jmedchem.7b00782 BindingDB Entry DOI: 10.7270/Q28S4SHS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytosol aminopeptidase (Homo sapiens (Human)) | BDBM50017478 (Amastatin | CHEMBL28650 | Leu[1psi,CHOHCONH]ValVal...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE KEGG MMDB PC cid PC sid UniChem Patents Similars | MMDB Article PubMed | 30 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Wroclaw University of Technology Curated by ChEMBL | Assay Description Binding affinity for cytosolic leucine aminopeptidase (LAP) from porcine kidney | J Med Chem 46: 2641-55 (2003) Article DOI: 10.1021/jm030795v BindingDB Entry DOI: 10.7270/Q27P903F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytosol aminopeptidase [33-68,L62W] (Sus scrofa (Pig)) | BDBM50025041 (CHEMBL3355106) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 39 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Athens Curated by ChEMBL | Assay Description Inhibition of pig recombinant leucine aminopeptidase after 30 to 60 mins by morrison's equation | J Med Chem 57: 8140-51 (2014) Article DOI: 10.1021/jm501071f BindingDB Entry DOI: 10.7270/Q2CF9RQF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytosol aminopeptidase (Homo sapiens (Human)) | BDBM50225458 ((2S)-3-[(R)-[(1S)-1-amino-3-phenylpropyl](hydroxy)...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL MMDB PC cid PC sid UniChem Similars | Article PubMed | 45 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Wroc£?aw University of Technology Curated by ChEMBL | Assay Description Inhibition of pig kidney cytosolic leucine aminopeptidase | Bioorg Med Chem Lett 18: 1550-4 (2008) Article DOI: 10.1016/j.bmcl.2008.01.107 BindingDB Entry DOI: 10.7270/Q28K78TP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytosol aminopeptidase [33-68,L62W] (Sus scrofa (Pig)) | BDBM50025042 (CHEMBL3355105) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid PDB UniChem Patents Similars | Article PubMed | 50 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Athens Curated by ChEMBL | Assay Description Inhibition of pig recombinant leucine aminopeptidase after 30 to 60 mins by morrison's equation | J Med Chem 57: 8140-51 (2014) Article DOI: 10.1021/jm501071f BindingDB Entry DOI: 10.7270/Q2CF9RQF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytosol aminopeptidase (Homo sapiens (Human)) | BDBM50457478 (CHEMBL4208547) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 50 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Jadavpur University Curated by ChEMBL | Assay Description Inhibition of LAP (unknown origin) | J Med Chem 61: 6468-6490 (2018) Article DOI: 10.1021/acs.jmedchem.7b00782 BindingDB Entry DOI: 10.7270/Q28S4SHS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytosol aminopeptidase (Homo sapiens (Human)) | BDBM50129685 (2-Amino-4-methyl-pentanal | CHEMBL88476) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 60 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Wroclaw University of Technology Curated by ChEMBL | Assay Description Binding affinity for cytosolic leucine aminopeptidase (LAP) from porcine kidney | J Med Chem 46: 2641-55 (2003) Article DOI: 10.1021/jm030795v BindingDB Entry DOI: 10.7270/Q27P903F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aminopeptidase B (Rattus norvegicus) | BDBM23971 ((2S)-2-[(2S,3R)-3-amino-2-hydroxy-4-phenylbutanami...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE MMDB PC cid PC sid PDB UniChem Patents Similars | PubMed | 60 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Wisconsin Curated by ChEMBL | Assay Description Inhibitory activity against aminopeptidase B | J Med Chem 31: 2193-9 (1988) BindingDB Entry DOI: 10.7270/Q2Z038RM | |||||||||||
More data for this Ligand-Target Pair |
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